Riham F. George

发表

Synthesis, Bioassay, and Molecular Field Topology Analysis of Diverse Vasodilatory Heterocycles

Polina V. Oliferenko, Alexander A. Oliferenko, Girinath G. Pillai, 2014, J. Chem. Inf. Model..

Synthesis of some N-aroyl-2-oxindole benzenesulfonamide conjugates with carbonic anhydrase inhibitory activity.

Riham F. George, C. Supuran, F. Awadallah, 2020, Bioorganic chemistry.

Synthesis and selective inhibitory effects of some 2-oxindole benzenesulfonamide conjugates on human carbonic anhydrase isoforms CA I, CA II, CA IX and CAXII.

Riham F. George, C. Supuran, Silvia Bua, 2019, Bioorganic chemistry.

Synthesis, vasorelaxant activity and 2D-QSAR study of some novel pyridazine derivatives.

Dalia O. Saleh, Riham F. George, D. Saleh, 2016, European journal of medicinal chemistry.

Rational design, synthesis and 2D-QSAR studies of antiproliferative tropane-based compounds

Adel S. Girgis, Riham F. George, Fady N. Baselious, 2016 .

Synthesis of some tropane-based compounds targeting colon cancer.

Riham F. George, J. Plaisier, N. Demitri, 2020, Future medicinal chemistry.

Synthesis, antiproliferative activity and 2D-QSAR study of some 8-alkyl-2,4-bisbenzylidene-3-nortropinones.

Riham F. George, N. Demitri, M. Wink, 2018, Future medicinal chemistry.

Design, synthesis and QSAR studies of dispiroindole derivatives as new antiproliferative agents.

Riham F. George, A. S. Girgis, N. S. Ismail, 2013, European journal of medicinal chemistry.

Design and synthesis of 1,2,4‐triazolo[1,5‐a]pyrimidine derivatives as PDE 4B inhibitors endowed with bronchodilator activity

Amr A. Kamel, Riham F. George, G. Piazza, 2019, Archiv der Pharmazie.

Synthesis, antitumor and antibacterial activities of some novel tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidine derivatives.

Riham F. George, Nagwa M. Abdel Gawad, S. Abbas, 2013, European journal of medicinal chemistry.

Microwave assisted synthesis and QSAR study of novel NSAID acetaminophen conjugates with amino acid linkers.

Aladdin M. Srour, Riham F. George, A. Katritzky, 2014, Organic & biomolecular chemistry.

Facile synthesis of some pyrazoline-based compounds with promising anti-inflammatory activity.

Riham F. George, N. M. Eid, 2018, Future medicinal chemistry.

Synthesis, bioassay, and QSAR study of bronchodilatory active 4H-pyrano[3,2-c]pyridine-3-carbonitriles.

Aladdin M. Srour, Riham F. George, C. S. Panda, 2015, European journal of medicinal chemistry.

Stereoselective Synthesis, Structural and Spectroscopic Study of 4,5,11‐Triazatricyclo[6.2.1.0*2,6*]Undec‐5‐ene

Riham F. George, Fady N. Baselious, ElSayed M Shalaby, 2016 .

Design and synthesis of some new 6-bromo-2-(pyridin-3-yl)-4-substituted quinazolines as multi tyrosine kinase inhibitors.

Riham F. George, S. Abbas, A. Farouk, 2022, Bioorganic chemistry.

Synthesis, analgesic and anti-inflammatory activities evaluation of some bi-, tri- and tetracyclic condensed pyrimidines.

Riham F. George, K. Amin, M. M. Hanna, 2009, European journal of medicinal chemistry.

Synthesis of some tropane derivatives of anticipated activity on the reuptake of norepinephrine and/or serotonin.

Riham F. George, M. M. Hanna, N. M. Eid, 2007, Bioorganic & medicinal chemistry.

Synthesis and vasodilator activity of some pyridazin-3(2H)-one based compounds.

Amr A. Kamel, Riham F. George, M. El-Daly, 2019, Future medicinal chemistry.

Some 2-(4-bromophenoxymethyl)-6-iodo-3-substituted quinazolin-4(3H)ones: Synthesis, cytotoxic activity, EGFR inhibition and molecular docking

Riham F. George, S. Abbas, Mohamed K. El-Ashrey, 2022, Journal of Molecular Structure.

Synthesis & molecular modeling studies of bronchodilatory active indole-pyridine conjugates.

Aladdin M. Srour, Riham F. George, A. Fitch, 2018, Future medicinal chemistry.

Design and synthesis of novel imidazo[4,5-b]pyridine based compounds as potent anticancer agents with CDK9 inhibitory activity.

Riham F. George, Faten Farouk, S. Abbas, 2018, Bioorganic chemistry.

Design, synthesis, antimicrobial, and DNA gyrase inhibitory properties of fluoroquinolone–dichloroacetic acid hybrids

Riham F. George, W. Fayad, S. Panda, 2020, Chemical biology & drug design.

Design and synthesis of novel benzimidazole derivatives as potential Pseudomonas aeruginosa anti-biofilm agents inhibiting LasR: Evidence from comprehensive molecular dynamics simulation and in vitro investigation.

Riham F. George, Hanan H. Georgey, A. Sayed, 2022, European journal of medicinal chemistry.

Synthesis, antitumor activity evaluation, and DNA‐binding study of coumarin‐based agents

Riham F. George, K. Amin, Nada M. Mohamed, 2018, Archiv der Pharmazie.

Exploration of thiazolidine‐2,4‐diones as tyrosine kinase inhibitors: Design, synthesis, ADMET, docking, and antiproliferative evaluations

Riham F. George, Khaled El-Adl, Walaa R Mahmoud, 2022, Archiv der Pharmazie.

Synthesis and anti-proliferative activity of some new quinoline based 4,5-dihydropyrazoles and their thiazole hybrids as EGFR inhibitors.

Riham F. George, H. Abdel‐Aziz, E. Samir, 2019, Bioorganic chemistry.

New 1-phthalazinone Scaffold based Compounds: Design, Synthesis, Cytotoxicity and Protein Kinase Inhibition Activity.

Riham F. George, Reem K. Arafa, Nehad E Abo-Elmagd, 2018, Mini-Reviews in Medical Chemistry.

Synthesis and cytotoxic activities of some pyrazoline derivatives bearing phenyl pyridazine core as new apoptosis inducers.

Riham F. George, M. Fouad, I. Gomaa, 2016, European journal of medicinal chemistry.

Synthesis and QSAR study of novel anti-inflammatory active mesalazine-metronidazole conjugates.

Riham F. George, A. Katritzky, S. Panda, 2015, Bioorganic & medicinal chemistry letters.

Synthesis of 1,2,4-triazolo[1,5-a]pyrimidine derivatives: Antimicrobial activity, DNA Gyrase inhibition and molecular docking.

Riham F. George, G. S. Hassan, H. Abdel-Rahman, 2019, Bioorganic chemistry.

Mechanistic selectivity investigation and 2D-QSAR study of some new antiproliferative pyrazoles and pyrazolopyridines as potential CDK2 inhibitors.

Esraa Z. Mohammed, Riham F. George, G. S. Hassan, 2021, European journal of medicinal chemistry.

Synthesis, in vitro anticancer activity and in silico studies of certain pyrazole-based derivatives as potential inhibitors of cyclin dependent kinases (CDKs).

Esraa Z. Mohammed, Riham F. George, G. S. Hassan, 2021, Bioorganic chemistry.

Synthesis and molecular modeling studies of indole-based antitumor agents

Aladdin M. Srour, Riham F. George, ElSayed M Shalaby, 2016 .

Design, Synthesis and QSAR Studies of Dispiroindole Derivatives as New Antiproliferative Agents.

Riham F. George, A. S. Girgis, N. S. Ismail, 2014 .

Synthesis, hypnotic properties and molecular modeling studies of 1,2,7,9-tetraaza-spiro[4.5]dec-2-ene-6,8,10-triones.

Riham F. George, A. S. Girgis, N. S. Ismail, 2011, European journal of medicinal chemistry.

Synthesis and biological evaluation of 2-aminothiazole-thiazolidinone conjugates as potential antitubercular agents.

Riham F. George, Wagdy M. Eldehna, S. M. Abou-Seri, 2018, Future medicinal chemistry.

Stereoselective synthesis and QSAR study of cytotoxic 2-(4-oxo-thiazolidin-2-ylidene)-2-cyano-N-arylacetamides.

Riham F. George, 2012, European journal of medicinal chemistry.

New quinazolinone‐based derivatives as DHFR/EGFR‐TK inhibitors: Synthesis, molecular modeling simulations, and anticancer activity

Riham F. George, Ahmed M. El Kerdawy, Hanan H. Georgey, 2022, Archiv der Pharmazie.

Synthesis and anticancer activity of some pyrido[2,3-d]pyrimidine derivatives as apoptosis inducers and cyclin-dependent kinase inhibitors.

Riham F. George, H. Abdel‐Aziz, E. Samir, 2019, Future medicinal chemistry.

Novel indole-thiazolidinone conjugates: Design, synthesis and whole-cell phenotypic evaluation as a novel class of antimicrobial agents.

Riham F. George, S. Bhakta, Wagdy M. Eldehna, 2018, European journal of medicinal chemistry.

Synthesis of new ibuprofen hybrid conjugates as potential anti-inflammatory and analgesic agents.

Aladdin M. Srour, Riham F. George, S. Panda, 2020, Future medicinal chemistry.

Synthesis and DFT studies of an antitumor active spiro-oxindole

Riham F. George, ElSayed M Shalaby, A. S. Girgis, 2015 .

New benzimidazole derivatives targeting LasR with antibiofilm efficacy against Pseudomonas aeruginosa: An integrated in vitro and molecular dynamics simulation- based investigation.

Riham F. George, Hanan H. Georgey, A. Sayed, 2022, Journal of Molecular Structure.

Facile synthesis of simple 2-oxindole-based compounds with promising antiproliferative activity.

Riham F. George, 2018, Future medicinal chemistry.

Fluoroquinolone-3-carboxamide amino acid conjugates: Synthesis, antibacterial properties and molecular modeling studies.

Riham F. George, W. Fayad, Riham M Bokhtia, 2019, Medicinal chemistry (Shariqah (United Arab Emirates)).

Design, synthesis and in silico insights of new 7,8-disubstituted-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione derivatives with potent anticancer and multi-kinase inhibitory activities.

Riham F. George, Nagwa M. Abdel Gawad, Ahmed M. El Kerdawy, 2020, Bioorganic chemistry.

Bacterial virulence factors: a target for heterocyclic compounds to combat bacterial resistance

Riham F. George, Hanan H. Georgey, H. Abdel-Rahman, 2021, RSC advances.

Aurones and furoaurones: Biological activities and synthesis

Riham F. George, G. S. Hassan, Hanan H. Georgey, 2018, Bulletin of Faculty of Pharmacy, Cairo University.

Construction of some cytotoxic agents with aurone and furoaurone scaffolds.

Riham F. George, G. S. Hassan, Hanan H. Georgey, 2018, Future medicinal chemistry.

Identification of some benzoxazepines as anticancer agents inducing cancer cell apoptosis.

Riham F. George, Hanan H. Georgey, N. Abdel-Gawad, 2018, Future medicinal chemistry.

Synthesis of new phenolic compounds and biological evaluation as antiproliferative agents

Riham F. George, Samir M. El-Moghazy, S. M. Abou-Seri, 2020 .

Synthesis, molecular modelling and QSAR study of new N-phenylacetamide-2-oxoindole benzensulfonamide conjugates as carbonic anhydrase inhibitors with antiproliferative activity

Riham F. George, C. Supuran, Nada M. Mohamed, 2022, Journal of enzyme inhibition and medicinal chemistry.

Synthesis, X-ray powder diffraction and DFT-D studies of indole-based compounds

Aladdin M. Srour, Riham F. George, A. Fitch, 2017 .

Synthesis, pharmacological profile and 2D-QSAR studies of curcumin-amino acid conjugates as potential drug candidates.

Riham F. George, S. Panda, A. S. Girgis, 2020, European journal of medicinal chemistry.

Staquorsin: A Novel Staphylococcus aureus Agr-Mediated Quorum Sensing Inhibitor Impairing Virulence in vivo Without Notable Resistance Development

A. S. Attia, Riham F. George, Ahmed S. Attia, 2021, Frontiers in Microbiology.

Identification of some novel xanthine-based derivatives with bronchodilator activity.

Riham F. George, Nagwa M. Abdel Gawad, Hanan H. Georgey, 2017, Future medicinal chemistry.

Some 1,3,5-trisubstituted pyrazoline derivatives targeting breast cancer: Design, synthesis, cytotoxic activity, EGFR inhibition and molecular docking.

Riham F. George, Ahmed M. El Kerdawy, M. Kandeel, 2020, Bioorganic chemistry.

Novel pyrazolo[3,4-d]pyrimidines as dual Src-Abl inhibitors active against mutant form of Abl and the leukemia K-562 cell line.

Riham F. George, E. Crespan, G. Maga, 2016, European journal of medicinal chemistry.

Design and synthesis of some barbituric and 1,3-dimethylbarbituric acid derivatives: A non-classical scaffold for potential PARP1 inhibitors.

Riham F. George, Samir M. El-Moghazy, Essam Eldin A Osman, 2020, Bioorganic chemistry.

Design, synthesis, in silico docking, ADMET and anticancer evaluations of thiazolidine-2,4-diones bearing heterocyclic rings as dual VEGFR-2/EGFRT790M tyrosine kinase inhibitors

Riham F. George, Khaled El-Adl, Walaa R Mahmoud, 2022, RSC advances.

Synthesis, Antitumor and Antibacterial Activities of Some Novel Tetrahydrobenzo[4,5]thieno[2,3‐d]pyrimidine Derivatives.

Riham F. George, S. Abbas, Yahya A. Akar, 2013 .

New 2-aminobenzothiazole derivatives: Design, synthesis, anti-inflammatory and ulcerogenicity evaluation

Riham F. George, Hanan H. Georgey, T. Nasr, 2023, Journal of Molecular Structure.

3-Methyl-imidazo[2,1-b]thiazole derivatives as a new class of antifolates: Synthesis, in vitro/in vivo bio-evaluation and molecular modeling simulations.

Riham F. George, Hanan H. Georgey, H. El-Subbagh, 2021, Bioorganic chemistry (Print).

Nanomolar potency of imidazo[2,1‐b]thiazole analogs as indoleamine 2,3‐dioxygenase inhibitors

Riham F. George, Hanan H. Georgey, H. El-Subbagh, 2021, Archiv der Pharmazie.

HER2 Kinase-Targeted Breast Cancer Therapy: Design, Synthesis, and In Vitro and In Vivo Evaluation of Novel Lapatinib Congeners as Selective and Potent HER2 Inhibitors with Favorable Metabolic Stability.

Hamed I. Ali, Riham F. George, Z. A. Abd Elmageed, 2020, Journal of medicinal chemistry.

Synthesis, analgesic and anti-inflammatory activities evaluation of some bi-, tri- and tetracyclic condensed pyrimidines.

Riham F. George, K. Amin, Hanan E. Abo-Youssef, 2009, European journal of medicinal chemistry.

Design, synthesis, and pharmacological characterization of some 2‐substituted‐3‐phenyl‐quinazolin‐4(3H)‐one derivatives as phosphodiesterase inhibitors

Riham F. George, K. Amin, Nada M. Mohamed, 2021, Archiv der Pharmazie.