Margot Ernst

SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the α1+/γ2- Benzodiazepine Site

Thierry Langer, Lars Richter, Stefan Boresch, 2018, J. Chem. Inf. Model..

Accelerated discovery of novel benzodiazepine ligands by experiment-guided virtual screening.

Erwin Sigel, Margot Ernst, E. Sigel, 2014, ACS chemical biology.

Affinity of various benzodiazepine site ligands in mice with a point mutation in the GABA(A) receptor gamma2 subunit.

William Wisden, Peer Wulff, Werner Sieghart, 2004, Biochemical pharmacology.

Comparative Models of GABAA Receptor Extracellular and Transmembrane Domains: Important Insights in Pharmacology and Functions⃞

Stefan Boresch, Werner Sieghart, Margot Ernst, 2005, Molecular Pharmacology.

Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands.

Chris de Graaf, Lars Richter, Iwan J P de Esch, 2012, Nature chemical biology.