Michael J. Ardolino

发表

Process Safety Considerations for the Supply of a High-Energy Oxadiazole IDO1-Selective Inhibitor

Lu Chen, Theodore A. Martinot, Michael J. Ardolino, 2019, Organic Process Research & Development.

Development of Scalable Routes to 1-Bicyclo[1.1.1]pentylpyrazoles

Michael J. Ardolino, Matthew L. Maddess, Kaitlyn M. Logan, 2020 .

Construction of 1,5-enynes by stereospecific Pd-catalyzed allyl-propargyl cross-couplings.

Michael J. Ardolino, J. Morken, 2012, Journal of the American Chemical Society.

Diastereocontrol in asymmetric allyl-allyl cross-coupling: stereocontrolled reaction of prochiral allylboronates with prochiral allyl chlorides.

Michael J. Ardolino, J. Morken, L. A. Brozek, 2011, Journal of the American Chemical Society.

Discovery of Amino-cyclobutarene-derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors for Cancer Immunotherapy.

Theodore A. Martinot, Michael J. Ardolino, Xiao Wang, 2019, ACS medicinal chemistry letters.

Surprising Reactivity in NiXantphos/Palladium-Catalyzed α-Arylation of Substituted Cyclopropyl Nitriles.

Michael J. Ardolino, B. Wright, B. A. Wright, 2018, The Journal of organic chemistry.

Branched/linear selectivity in palladium-catalyzed allyl-allyl cross-couplings: The role of ligands.

Michael J. Ardolino, J. Morken, 2015, Tetrahedron.

Congested C-C bonds by Pd-catalyzed enantioselective allyl-allyl cross-coupling, a mechanism-guided solution.

Michael J. Ardolino, J. Morken, 2014, Journal of the American Chemical Society.

Stereocontrol in Palladium-Catalyzed Propargylic Substitutions: Kinetic Resolution to give Enantioenriched 1,5-Enynes and Propargyl Acetates.

Michael J. Ardolino, J. Morken, Meredith S Eno, 2013, Advanced synthesis & catalysis.

Structure-Guided Discovery of Aminoquinazolines as Brain-Penetrant and Selective LRRK2 Inhibitors.

Michael J. Ardolino, Karin M. Otte, M. Kennedy, 2021, Journal of medicinal chemistry.

Discovery and Optimization of Potent, Selective, and Brain-Penetrant 1-Heteroaryl-1H-Indazole LRRK2 Kinase Inhibitors for the Treatment of Parkinson's Disease.

Theodore A. Martinot, Michael J. Ardolino, Matthew L. Maddess, 2022, Journal of medicinal chemistry.

Directed Evolution to Reverse Epoxide Hydrolase Enantioselectivity for meso‐3,4‐Epoxytetrahydrofuran

Michael J. Ardolino, K. Hiraga, T. Itoh, 2023, ChemCatChem.

Diastereocontrol in asymmetric allyl-allyl cross-coupling: stereocontrolled reaction of prochiral allylboronates with prochiral allyl chlorides.

Michael J. Ardolino, J. Morken, L. A. Brozek, 2011, Journal of the American Chemical Society.