Shane W. Krska

发表

Heterocyclic Regioisomer Enumeration (HREMS): A Cheminformatics Design Tool

Edward C. Sherer, Zhengwei Peng, Sriram Tyagarajan, 2015, J. Chem. Inf. Model..

Chemistry informer libraries: a chemoinformatics enabled approach to evaluate and advance synthetic methods† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c5sc04751j

Bing Li, Peter S. Kutchukian, Ian W. Davies, 2016, Chemical science.

Asymmetric Alkene Hydrogenation Catalysts Cobalt Precursors for High-Throughput Discovery of Base Metal

Michael Shevlin, Shane W. Krska, Paul J. Chirik, 2014 .

Cobalt Precursors for High‐Throughput Discovery of Base Metal Asymmetric Alkene Hydrogenation Catalysts.

Michael Shevlin, Shane W. Krska, Paul J. Chirik, 2014 .

Synthesis of Sitagliptin

Feng Xu, Edward J. J. Grabowski, Shane W. Krska, 2009 .

Enabling Efficient Late‐Stage Functionalization of Drug‐Like Molecules with LC‐MS and Reaction‐Driven Data Processing

Shane W. Krska, L. Goracci, I. Zamora, 2017 .

Silyl Phosphorus and Nitrogen Donor Chelates for Homogeneous Ortho Borylation Catalysis

Shane W. Krska, Sean M. Preshlock, Milton R. Smith, 2014, Journal of the American Chemical Society.

A traceless directing group for C-H borylation.

Shane W. Krska, Sean M. Preshlock, Milton R. Smith, 2013, Angewandte Chemie.

The medicinal chemist's toolbox for late stage functionalization of drug-like molecules.

Shane W. Krska, P. Váchal, T. Cernak, 2016, Chemical Society reviews.

Site-selective 18F fluorination of unactivated C–H bonds mediated by a manganese porphyrin

Shane W. Krska, J. Groves, J. Hooker, 2017, Chemical science.

Emerging fluorination methods in organic chemistry relevant for life science application

Shane W. Krska, S. Krska, P. Richardson, 2019, Fluorine in Life Sciences: Pharmaceuticals, Medicinal Diagnostics, and Agrochemicals.

High-throughput optimization of Ir-catalyzed C-H borylation: a tutorial for practical applications.

Shane W. Krska, Sean M. Preshlock, Milton R. Smith, 2013, Journal of the American Chemical Society.

Late-stage functionalization of biologically active heterocycles through photoredox catalysis.

Shane W. Krska, P. Váchal, S. Krska, 2014, Angewandte Chemie.

Cu-Mediated C–H 18F-Fluorination of Electron-Rich (Hetero)arenes

Allen F. Brooks, Shane W. Krska, M. Sanford, 2017, Organic letters.

An approach to heterodiarylmethanes via sp2–sp3 Suzuki−Miyaura cross-coupling

Jeremy P. Scott, Shane W. Krska, S. Krska, 2016 .

Copper-catalysed benzylic C–H coupling with alcohols via radical relay enabled by redox buffering

Shane W. Krska, C. Cramer, S. Stahl, 2020, Nature Catalysis.

Protecting group free radical C–H trifluoromethylation of peptides† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8sc00368h

Shane W. Krska, Xiaohong Zhu, S. Krska, 2018, Chemical science.

Highly efficient asymmetric synthesis of sitagliptin.

Feng Xu, Andrew Clausen, Shane W. Krska, 2009, Journal of the American Chemical Society.

Understanding the Origin of Unusual Stepwise Hydrogenation Kinetics in the Synthesis of the 3-(4-Fluorophenyl)morpholine Moiety of NK1 Receptor Antagonist Aprepitant

Shane W. Krska, E. Corley, R. Reamer, 2006 .

Merging Late-Stage Diversification with Solid-Phase Peptide Synthesis Enabled by High-Throughput On-Resin Reaction Screening

Shane W. Krska, Shasha Li, Michael Wleklinski, 2022, ACS Catalysis.

Discovery of MK-4409, a Novel Oxazole FAAH Inhibitor for the Treatment of Inflammatory and Neuropathic Pain.

Shane W. Krska, R. DeVita, R. Nargund, 2014, ACS medicinal chemistry letters.

Synthesis and Hydrogenation Activity of Iron Dialkyl Complexes with Chiral Bidentate Phosphines

Shane W. Krska, P. Chirik, Grant W. Margulieux, 2014 .

Synthesis of antifungal glucan synthase inhibitors from enfumafungin.

Shane W. Krska, R. Ball, M. McLaughlin, 2012, The Journal of organic chemistry.

Enantioselective hydrogenation of alpha-aryloxy alpha,beta-unsaturated acids. Asymmetric synthesis of alpha-aryloxycarboxylic acids.

Shane W. Krska, G. Humphrey, S. Krska, 2004, Organic letters.

Highly enantioselective synthesis of anti aryl β-hydroxy α-amino esters via DKR transfer hydrogenation

Shane W. Krska, James F Cuff, E. Sherer, 2011 .

Application of High-Throughput Competition Experiments in the Development of Aspartate-Directed Site-Selective Modification of Tyrosine Residues in Peptides.

Scott J. Miller, Shane W. Krska, Byoungmoo Kim, 2020, The Journal of organic chemistry.

Cobalt Precursors for High-Throughput Discovery of Base Metal Asymmetric Alkene Hydrogenation Catalysts

Shane W. Krska, P. Chirik, S. Krska, 2013, Science.

Highly efficient synthesis of beta-amino acid derivatives via asymmetric hydrogenation of unprotected enamines.

Shane W. Krska, E. Njolito, F. Wang, 2004, Journal of the American Chemical Society.

Protecting group free radical C–H trifluoromethylation of peptides

Shane W. Krska, Xiaohong Zhu, S. Krska, 2018, Chemical science.

C(sp3)–H methylation enabled by peroxide photosensitization and Ni-mediated radical coupling

Shane W. Krska, S. Stahl, S. Krska, 2021, Science.