Y. Fall

发表

QSAR and complex network study of the chiral HMGR inhibitor structural diversity.

E. Uriarte, C. Munteanu, H. González-Díaz, 2009, Bioorganic & medicinal chemistry.

An application of two MIFs-based tools (Volsurf+ and Pentacle) to binary QSAR: the case of a palinurin-related data set of non-ATP competitive glycogen synthase kinase 3β (GSK-3β) inhibitors.

Y. Fall, G. Gómez, G. Caron, 2011, European journal of medicinal chemistry.

A topological sub-structural approach to the mutagenic activity in dental monomers. 3. Heterogeneous set of compounds

Maykel Pérez González, Aliuska Morales Helguera, Yagamare Fall, 2005 .

Using Topological Indices to Predict Anti-Alzheimer and Anti-Parasitic GSK-3 Inhibitors by Multi-Target QSAR in Silico Screening

I. García, Y. Fall, G. Gómez, 2010, Molecules.

Synthesis and structure–activity relationships of new arylpiperazines: para substitution with electron-withdrawing groups decrease binding to 5-HT1A and D2A receptors

L. Santana, E. Uriarte, Y. Fall, 2002 .

The first enantioselective synthesis of palinurin.

Y. Fall, G. Gómez, M. Perez, 2009, Chemical communications.

Synthesis and characterization of some coumarins with two hydroxy or methoxy substituents

L. Santana, E. Uriarte, Y. Fall, 2001 .

Novel calcitriol analogue with an oxolane group: In vitro, in vivo, and in silico studies

Y. Fall, G. Gómez, M. M. Facchinetti, 2019, Archiv der Pharmazie.

Synthesis of a novel analog of calcitriol and its biological evaluation as antitumor agent

Y. Fall, G. Gómez, M. M. Facchinetti, 2019, The Journal of Steroid Biochemistry and Molecular Biology.

Rapid access to a series of calcitriol analogues with restricted side chain conformation

Y. Fall, G. Gómez, Carlos Fernandez, 2016 .

Synthesis of new triazolium-based ionic liquids and their use in the Morita–Baylis–Hillman reaction

Y. Fall, G. Gómez, O. Diouf, 2015 .

Vitamin D and click chemistry. Part 1: A stereoselective route to vitamin D analogues with triazole rings in their side chains

Y. Fall, G. Gómez, Z. Gándara, 2004 .

Easy Access to Polyfunctionalized Chiral Decalins

Y. Fall, G. Gómez, Z. Gándara, 2020, ACS omega.

An efficient synthesis of the 25-hydroxy Windaus–Grundmann ketone

Y. Fall, C. Vitale, A. Mouriño, 2000 .

Copper-mediated alkylation of vitamin D C-ring. Synthesis of C11-functionalized 1α,25-dihydroxyvitamin D3

Y. Fall, L. Castedo, A. Mouriño, 1997 .

The furan approach to azacyclic compounds

I. García, Y. Fall, G. Gómez, 2008 .

The thioacetate approach to vitamin D analogues. Part 2: Synthesis of (25S)-23-thia-1α,25,26-trihydroxyvitamin D3

Y. Fall, G. Gómez, O. Diouf, 2007 .

The thioacetate approach to the synthesis of the side chain of vitamin D metabolites and analogues

Y. Fall, G. Gómez, O. Diouf, 2003 .

An efficient route to 1α,25-dihydroxyvitamin D3 functionalized at C-11

Y. Fall, L. Castedo, A. Mouriño, 1992 .

Synthesis and properties of novel chiral imidazolium-based ionic liquids derived from carvone

Y. Fall, M. Vilas, E. Tojo, 2016 .

Synthesis of a New Type of Trans-Decalin Vitamin D Analogue through a Dyotropic Ring Expansion

Y. Fall, Hugo Santalla, Uxía Gómez-Bouzó, 2021, Journal of Chemistry.

Vitamin D Analogue: Potent Antiproliferative Effects on Cancer Cell Lines and Lack of Hypercalcemic Activity

Y. Fall, G. Gómez, M. M. Facchinetti, 2015, Archiv der Pharmazie.

Synthesis and biological evaluation of a new vitamin D2 analogue.

Y. Fall, G. Gómez, M. M. Facchinetti, 2012, Bioorganic & medicinal chemistry letters.

Review of synthesis, biological assay, and QSAR studies of HMGR inhibitors.

I. García, Y. Fall, G. Gómez, 2012, Current topics in medicinal chemistry.

Novel alkynylphosphonate analogue of calcitriol with potent antiproliferative effects in cancer cells and lack of calcemic activity.

Y. Fall, M. M. Facchinetti, M. Perez, 2011, ACS medicinal chemistry letters.

An Efficient Stereoselective Synthesis of 1α,24(R)- Dihydroxyvitamin D3 by the Dienyne Route.

Y. Fall, L. Castedo, A. Mouriño, 1997 .

A nitrile approach to the synthesis of the side chain of vitamin D metabolites and analogues

Y. Fall, L. Castedo, A. Mouriño, 1992 .

d- and l-Serine, useful synthons for the synthesis of 24-hydroxyvitamin D3 metabolites. A formal synthesis of 1α,24R,25-(OH)3-D3, 24R,25-(OH)2-D3 and 24S,25-(OH)2-D3

Y. Fall, G. Gómez, Z. Gándara, 2007 .

Vitamin D heterocyclic analogues. Part 1: A stereoselective route to CD systems with pyrazole rings in their side chains

Y. Fall, A. Mouriño, Carlos Fernandez, 2002 .

A NEW APPROACH TO THE SYNTHESIS OF THE 25-HYDROXY-22-OXA-VITAMIN D3 SIDE CHAIN

Y. Fall, 1997 .

Stereoselective synthesis of vitamin D3 analogues with cyclic side chains

Y. Fall, C. Vitale, A. Mouriño, 2000 .

Phenylpiperazine derivatives with strong affinity for 5HT1A, D2A and D3 receptors.

L. Santana, E. Uriarte, Y. Fall, 1998, Bioorganic & medicinal chemistry letters.

Enantiodivergent synthesis of (+)- and (−)-isolaurepan

Y. Fall, G. Gómez, M. Perez, 2012 .

A new, enantioselective synthesis of (+)-isolaurepan

Y. Fall, G. Gómez, M. Perez, 2009 .

A Convenient Synthesis of Benzofuran-3-acetic Acids.

L. Santana, E. Uriarte, Y. Fall, 1995 .

Solvent-free synthesis of some N4O2, N4S2 and N6 Schiff-base ligands assisted by microwave irradiation

Y. Fall, M. Rezaeivala, H. Keypour, 2009 .

Total synthesis of (+)-decytospolides A and B

Y. Fall, G. Gómez, M. Perez, 2015 .

Efficient and rapid experimental procedure for the synthesis of furan diol from D-glucal using ionic liquid

Marta Teijeira, Yagamare Fall, Y. Fall, 2007 .

From Hydrindane to Decalin: A Mild Transformation through a Dyotropic Ring Expansion.

Y. Fall, G. Gómez, O. N. Faza, 2017, Organic letters.

Alkylation of diene allylic tertiary amines with grignard reagents. In situ activation with alkyl chloroformates.

Y. Fall, Y. Langlois, N. V. Bac, 1985 .

The furan approach to carbocyclic systems. Synthesis of cyclohexane derivatives from butenolides through an intramolecular Michael addition

I. García, Y. Fall, G. Gómez, 2005 .

Synthesis of the pheromone of the comstock mealybug via a sila-cope elimination

Y. Fall, Y. Langlois, N. V. Bac, 1986 .

The Methoxyallene Approach to Oxacycles, Part 2: Stereoselective Synthesis of 2,3-Disubstituted Oxepanes

Y. Fall, G. Gómez, M. Teijeira, 2005 .

The furan approach to oxacycles: synthesis of medium-size 2,3-disubstituted oxacycles

Y. Fall, G. Gómez, M. Perez, 2004 .

Stereoselective synthesis of 2,3,4-trisubstituted tetrahydrothiophenes

Y. Fall, G. Gómez, M. Perez, 2009 .

The furan approach to oxacycles. Part 3: Stereoselective synthesis of 2,3-disubstituted tetrahydropyrans

Y. Fall, G. Gómez, M. Perez, 2005 .

Synthesis of seven-membered oxacycles. Part 2: The furan approach

Y. Fall, G. Gómez, D. Alonso, 2003 .

METHOXYALLENE, A BUILDING BLOCK FOR THE SYNTHESIS OF SEVEN-MEMBERED OXACYCLES

Y. Fall, G. Gómez, Carlos Fernandez, 1999 .

The furan approach to oxacycles. Part 6: From THF to fused polyoxepanes

Y. Fall, G. Gómez, M. Perez, 2007 .

Ionic liquid-supported TEMPO as catalyst in the oxidation of alcohols to aldehydes and ketones

Y. Fall, G. Gómez, A. Fall, 2010 .

Stereoselective synthesis of polytetrahydropyrans

Y. Fall, G. Gómez, M. Perez, 2008 .

Total synthesis of (−)-muricatacin

Y. Fall, G. Gómez, Z. Gándara, 2011 .

Synthesis of (4S, 5S, 11R) and (4S, 5S, 11S)-iso-cladospolide B

Y. Fall, G. Gómez, Z. Gándara, 2013 .

Synthesis of (+)-Muricatacin and a Formal Synthesis of CMI-977 from l-Malic Acid

Y. Fall, G. Gómez, Z. Gándara, 2013 .

Synthesis of (–)-Muricatacin from Tri-O-acetyl-d-glucal

Y. Fall, G. Gómez, Z. Gándara, 2013 .

Synthesis of a chiral building block for highly functionalized polycyclic ethers.

Y. Fall, G. Gómez, Z. Gándara, 2014, Organic & biomolecular chemistry.

The furan approach to the synthesis of natural products having highly substituted cyclic ether moieties

Y. Fall, G. Gómez, O. Diouf, 2017 .

Access To A Library Of 1,3-Disubstituted-1,2,3-Triazenes And Evaluation Of Their Antimicrobial Properties.

Y. Fall, G. Gómez, A. Diop, 2020, Current topics in medicinal chemistry.

First total synthesis of 6-epi-phomonol

Y. Fall, G. Gómez, Hugo Santalla, 2016 .

The alkynylphosphonate analogue of calcitriol EM1 has potent anti-metastatic effects in breast cancer

Y. Fall, M. M. Facchinetti, E. Alonso, 2015, The Journal of Steroid Biochemistry and Molecular Biology.

The furan approach to thiacyclic compounds. Stereoselective synthesis of 2,3-disubstituted tetrahydrothiopyrans

Y. Fall, G. Gómez, M. Perez, 2008 .

The furan approach to oxacycles. Part 4: A synthesis of (+)-decarestrictine L

I. García, Y. Fall, G. Gómez, 2006 .

The UVB1 Vitamin D analogue inhibits colorectal carcinoma progression

Y. Fall, G. Gómez, M. M. Facchinetti, 2016, The Journal of Steroid Biochemistry and Molecular Biology.

Theoretical study of GSK−3α: neural networks QSAR studies for the design of new inhibitors using 2D descriptors

Yagamare Fall, Isela García, Xerardo García-Mera, 2011, Molecular Diversity.

Comparative Analysis of the Neurochemical Profile and MAO Inhibition Properties of N-(Furan-2-ylmethyl)-N-methylprop-2-yn-1-amine.

Yagamare Fall, José Marco-Contelles, P. De Deurwaerdère, 2017, ACS chemical neuroscience.

Antitumoral effects of the alkynylphosphonate analogue of calcitriol EM1 on glioblastoma multiforme cells

Y. Fall, M. M. Facchinetti, E. Alonso, 2017, The Journal of Steroid Biochemistry and Molecular Biology.

Vitamin D receptor exhibits different pharmacodynamic features in tumoral and normal microenvironments: A molecular modeling study

Sergio R. Ribone, Y. Fall, M. M. Facchinetti, 2020, The Journal of Steroid Biochemistry and Molecular Biology.

Synthetic studies toward zoapatanol

I. García, Y. Fall, G. Gómez, 2008 .

1,2,3-triazenes and 1,2,3-triazoles as antileishmanial, antitrypanosomal, and antiplasmodial agents

Y. Fall, G. Gómez, S. Cojean, 2022, Medicinal Chemistry Research.

Synthesis of a Greek tobacco lactonic natural product and its analogues

Y. Fall, P. Besada, G. Pazos, 2012 .

Synthesis of New Triazolium‐Based Ionic Liquids and Their Use in the Morita—Baylis—Hillman Reaction.

Y. Fall, G. Gómez, O. Diouf, 2015 .

Use of surface plasmon resonance in the binding study of vitamin D, metabolites and analogues with vitamin D binding protein

Y. Fall, G. Gómez, J. Popplewell, 2017, Analytical and Bioanalytical Chemistry.

First computational chemistry multi-target model for anti-Alzheimer, anti-parasitic, anti-fungi, and anti-bacterial activity of GSK-3 inhibitors in vitro, in vivo, and in different cellular lines

Humberto González-Díaz, Yagamare Fall, Isela García, 2011, Molecular Diversity.

Synthesis of a trans-Hydrindanone, Precursor for the Preparation of Vitamin D Analogues†

Y. Fall, G. Gómez, M. Perez, 2013 .

[3,3]-Sigmatropic rearrangement mediated synthesis of chiral building blocks for the preparation of Gemini and its analogs

Y. Fall, G. Gómez, M. Perez, 2016 .

Synthesis of a trans‐Hydrindanone, Precursor for the Preparation of Vitamin D Analogues.

Y. Fall, G. Gómez, M. Perez, 2014 .

New Synthetic Strategies to Vitamin D Analogues Modified at the Side Chain and D Ring. Synthesis of 1alpha,25-Dihydroxy-16-ene-vitamin D(3) and C-20 Analogues(1).

Y. Fall, J. Granja, K. Halkes, 1999, The Journal of organic chemistry.

N‐(furan‐2‐ylmethyl)‐N‐methylprop‐2‐yn‐1‐amine (F2MPA): A Potential Cognitive Enhancer with MAO Inhibitor Properties

P. De Deurwaerdère, I. García, Y. Fall, 2014, CNS neuroscience & therapeutics.

A more reliable synthesis of a Gemini vitamin D analog, a potentially effective chemotherapeutic agent for the treatment of colorectal carcinomas

Y. Fall, G. Gómez, Hugo Santalla, 2018 .

An improved methodology for the synthesis of 1α,25-dihydroxy-20-epi-vitamin D3 (MC 1288) and Gemini analog Ro-438-3582

Y. Fall, G. Gómez, Andrea R. Martinez, 2017 .

New Synthetic Strategies to Vitamin D Analogues Modified at the Side Chain and D Ring. Synthesis of 1α,25-Dihydroxy-16-ene-vitamin D3 and C-20 Analogues.

Y. Fall, J. Granja, K. Halkes, 1999 .

Structural analysis and biological activities of C25-amino and C25-nitro vitamin D analogs.

Y. Fall, G. Gómez, N. Rochel, 2023, Bioorganic chemistry.

Quantitative structure-activity relationship studies of HIV-1 integrase inhibition. 1. GETAWAY descriptors.

Maykel Pérez González, Yagamare Fall, Y. Fall, 2007, European journal of medicinal chemistry.

Modified Julia olefination and α aminoxylation reactions mediated convergent synthesis of 1α, 24 (R)-dihydroxyvitamin D3 (tacalcitol)

Y. Fall, G. Gómez, Andrea R. Martinez, 2017 .

Synthesis of the Pheromone of the Comstock Mealybug via a Sila-Cope Elimination.

Y. Fall, Y. Langlois, N. V. Bac, 1986 .

Structure-activity relationship study of vitamin D analogs with oxolane group in their side chain.

Andrea Martínez, Yagamare Fall, Natacha Rochel, 2017, European journal of medicinal chemistry.

In silico studies using Radial Distribution Function approach for predicting affinity of 1α,25-dihydroxyvitamin D3 analogues for Vitamin D receptor

Maykel Pérez González, Yagamare Fall, Y. Fall, 2006, Steroids.

Quantitative structure-activity relationship studies of vitamin D receptor affinity for analogues of 1alpha,25-dihydroxyvitamin D3. 1: WHIM descriptors.

Maykel Pérez González, Yagamare Fall, Y. Fall, 2005, Bioorganic & medicinal chemistry letters.

New Experimental and Computational Tools for Drug Discovery. From Old Way to New Series - Part-X.

Humbert González-Díaz, Matthew M Montemore, Ricardo Santana, 2020, Current topics in medicinal chemistry.

The furan approach to oxacycles. Part 5: Synthesis of a chiral butenolide, building block towards biologically interesting natural products

Y. Fall, G. Gómez, M. Teijeira, 2005 .

An Efficient Synthesis of the 25-Hydroxy Windaus—Grundmann Ketone.

Y. Fall, C. Vitale, A. Mouriño, 2000 .

Stereoselective Synthesis of (22R)- and (22S)-22-Methyl-1α,25-Dihydroxyvitamin D3

Y. Fall, A. Mouriño, Carlos Fernandez, 2001 .

Stereoselective synthesis of (22Z)-25-hydroxyvitamin D2 and (22Z)-1α,25-dihydroxyvitamin D2

Y. Fall, G. Gómez, M. Perez, 2009 .

A key intermediate for the convenient synthesis of series of vitamin D 3 analogues with modified side chains

Y. Fall, A. Mouriño, Carlos Fernandez, 2001 .

Pd-allylic substitution mediated synthesis of 25-amino vitamin D3 derivatives

Y. Fall, G. Gómez, M. Perez, 2013 .

Synthesis of new calcitriol analogues with an oxolane moiety in their side chains

Y. Fall, G. Gómez, Z. Gándara, 2013 .

Radial Distribution Function descriptors for predicting affinity for vitamin D receptor.

Maykel Pérez González, Yagamare Fall, Y. Fall, 2008, European journal of medicinal chemistry.

The UVB1 Vitamin D analogue inhibits colorectal carcinoma progression

Y. Fall, M. M. Facchinetti, E. Alonso, 2016, The Journal of Steroid Biochemistry and Molecular Biology.

A radial distribution function approach to predict A(2B) agonist effect of adenosine analogues.

Maykel Pérez González, Marta Teijeira, Yagamare Fall, 2005, Bioorganic & medicinal chemistry.

QSAR and complex network study of the chiral HMGR inhibitor structural diversity.

E. Uriarte, C. Munteanu, H. González-Díaz, 2009, Bioorganic & medicinal chemistry.

Antitumoral effects of the alkynylphosphonate analogue of calcitriol EM1 on glioblastoma multiforme cells

Y. Fall, M. M. Facchinetti, E. Alonso, 2017, The Journal of Steroid Biochemistry and Molecular Biology.

Vitamin D analogues exhibit antineoplastic activity in breast cancer patient-derived xenograft cells

Y. Fall, J. Arribas, M. M. Facchinetti, 2020, The Journal of Steroid Biochemistry and Molecular Biology.

Synthesis of Seven-Membered Oxacycles. Part 2. The Furan Approach.

Y. Fall, D. Alonso, Beatriz Vidal, 2003 .