D. Brittelli

发表

Simple selection criteria for drug-like chemical matter.

I. Muegge, S. Heald, D. Brittelli, 2001, Journal of medicinal chemistry.

Synthesis and structure activity relationships of novel small molecule cathepsin D inhibitors.

D. Brittelli, J. Dumas, J. Chen, 1999, Bioorganic & medicinal chemistry letters.

Phosphite-mediated in situ carboxyvinylation: a new general acrylic acid synthesis

D. Brittelli, 1981 .

Omega-carboxypyridyl substituted ureas as Raf kinase inhibitors: SAR of the amide substituent.

Xiao-Gao Liu, Barbara Hibner, Joel Renick, 2004, Bioorganic & medicinal chemistry letters.

Synthesis of conformationally-restricted boropeptide thrombin inhibitors

D. Brittelli, P. Weber, R. Knabb, 1996 .

Design and synthesis of ring-constrained boropeptide thrombin inhibitors

M. Abelman, D. Brittelli, P. Weber, 1996 .

Perturbed [12]annulenes. Synthesis of pyracylenes

B. Trost, D. Brittelli, C. Frihart, 1971 .

Protocols for amide high-speed analoging. Preparation of novel, small molecule cathepsin D inhibitors

D. Brittelli, J. Chen, R. DixonBrian, 1999 .

Phosphine-and phosphite- mediated difluorocarbene exchange reactions of (bromodifluoromethyl)phosphonium salts: evidence for facile dissociation of (difluoromethylene)triphenylphosphorane

D. Brittelli, B. Smart, R. M. Flynn, 1983 .

Antibacterials. Synthesis and structure-activity studies of 3-aryl-2-oxooxazolidines. 2. The "A" group.

D. Brittelli, M. A. Wuonola, C. Park, 1989, Journal of medicinal chemistry.

An automated pulse labelling method for structure-activity relationship studies with antibacterial oxazolidinones.

D. Brittelli, L. Brown, P. Feldman, 1990, Drugs under experimental and clinical research.

Antibacterials. synthesis and structure-activity studies of 3-aryl-2-oxooxazolidines. 4. Multiply-substituted aryl derivatives.

D. Brittelli, A. Slee, M. A. Wuonola, 1992, Journal of medicinal chemistry.

A study of the reaction of 2-haloacyl halides with trialkyl phosphites. Synthesis of (2-substituted acyl)phosphonates

D. Brittelli, 1985 .

New furoxan chemistry. 2. Chemistry of acyl nitrile oxides generated in situ by thermolysis of diacylfuroxans

D. Brittelli, G. A. Boswell, D. R. Brittelli, 1981 .

1,2‐Bis(Dichlorophosphino)Ethane

D. Brittelli, R. Henderson, W. Hussain, 2007 .

Twisted internal charge transfer emission in B,B‐bis(mesityl) pyrroloboranes

D. Brittelli, D. F. Eaton, 1989 .

NEW FUROXAN CHEMISTRY. 1. SYNTHESIS OF DIACYLFUROXANS BY REACTION OF ETHYNYL ACETATES WITH NITROSYL FLUORIDE NITROSONIUM TETRAFLUOROBORATE

D. Brittelli, G. A. Boswell, 2002 .

Imidazo[1,2-a]pyrazine diaryl ureas: inhibitors of the receptor tyrosine kinase EphB4.

D. Brittelli, R. Desimone, K. Currie, 2009, Bioorganic & medicinal chemistry letters.

Abstract 17: Preclinical and phase 1 trial results of JI-101, a novel, oral tyrosine kinase inhibitor that selectively targets VEGFR2, EphB4, and PDGFRβ

D. Brittelli, L. Miller, M. Velleca, 2010 .

Acetylcholine-releasing agents as cognition enhancers. Structure-activity relationships of pyridinyl pendant groups on selected core structures.

D. Brittelli, R. Earl, M. A. Wuonola, 1992 .

Abstract B11: Preclinical and preliminary phase 1 trial results of JI‐101: A novel, oral tyrosine kinase inhibitor that selectively targets VEGFR2, EphB4, and PDGFR

D. Brittelli, L. Miller, M. Velleca, 2009 .

Antibacterials. Synthesis and structure-activity studies of 3-aryl-2-oxooxazolidines. 1. The "B" group.

D. Brittelli, M. A. Wuonola, W. A. Gregory, 1989, Journal of medicinal chemistry.

The halogenation of acenaphthene derivatives

B. Trost, D. Brittelli, 1967 .