M. Giulianotti

发表

Shifting from the single to the multitarget paradigm in drug discovery.

J. Medina-Franco, M. Giulianotti, G. Welmaker, 2013, Drug discovery today.

Towards a systematic characterization of the antiprotozoal activity landscape of benzimidazole derivatives.

Jaime Pérez-Villanueva, Rafael Castillo, Radleigh Santos, 2010, Bioorganic & medicinal chemistry.

Identification, structure-activity relationships and molecular modeling of potent triamine and piperazine opioid ligands.

Austin B. Yongye, Karina Martínez-Mayorga, Adel Nefzi, 2009, Bioorganic & medicinal chemistry.

Expanding the medicinally relevant chemical space with compound libraries.

J. Medina-Franco, M. Giulianotti, R. Houghten, 2012, Drug discovery today.

Integrating virtual screening and combinatorial chemistry for accelerated drug discovery.

Fabian López-Vallejo, Karina Martínez-Mayorga, Adel Nefzi, 2011, Combinatorial chemistry & high throughput screening.

Glycosylation of a disintegrin and metalloprotease 17 affects its activity and inhibition.

M. Giulianotti, R. Houghten, G. Fields, 2014, Analytical biochemistry.

SAR Studies of Exosite-Binding Substrate-Selective Inhibitors of A Disintegrin And Metalloprotease 17 (ADAM17) and Application as Selective in Vitro Probes.

M. Giulianotti, R. Houghten, R. Fridman, 2015, Journal of medicinal chemistry.

A Novel Probe for Spliceosomal Proteins that Induces Autophagy and Death of Melanoma Cells Reveals New Targets for Melanoma Drug Discovery

M. Giulianotti, R. Houghten, G. Fields, 2020, Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology.

Direct Phenotypic Screening in Mice: Identification of Individual, Novel Antinociceptive Compounds from a Library of 734 821 Pyrrolidine Bis-piperazines

Radleigh G. Santos, M. Giulianotti, G. Welmaker, 2015, ACS combinatorial science.

Identification of Two Novel, Potent, Low-Liability Antinociceptive Compounds from the Direct In Vivo Screening of a Large Mixture-Based Combinatorial Library

Adel Nefzi, M. Giulianotti, R. Houghten, 2010, The AAPS Journal.

Identification of Tetrapeptides from a Mixture Based Positional Scanning Library That Can Restore nM Full Agonist Function of the L106P, I69T, I102S, A219V, C271Y, and C271R Human Melanocortin-4 Polymorphic Receptors (hMC4Rs)

Clemencia Pinilla, Michael A. Walters, Richard A. Houghten, 2014, Journal of medicinal chemistry.

Discovery of Novel Inhibitors of a Disintegrin and Metalloprotease 17 (ADAM17) Using Glycosylated and Non-glycosylated Substrates*

M. Giulianotti, R. Houghten, Nina Bionda, 2012, The Journal of Biological Chemistry.

Highly Selective and Potent α4β2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats.

M. Giulianotti, G. Welmaker, R. Houghten, 2017, Journal of medicinal chemistry.

Fluorescent mu selective opioid ligands from a mixture based cyclic peptide library.

M. Giulianotti, R. Houghten, C. Dooley, 2012, ACS combinatorial science.

Use and implications of the harmonic mean model on mixtures for basic research and drug discovery.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2011, ACS combinatorial science.

Synthesis of 2,3,4-trisubstituted pyrroles via a facile reaction of vinyl azides and tosylmethyl isocyanide

M. Giulianotti, Wenteng Chen, Yongping Yu, 2012 .

Scaffold ranking and positional scanning utilized in the discovery of nAChR-selective compounds suitable for optimization studies.

Radleigh G. Santos, M. Giulianotti, G. Welmaker, 2013, Journal of medicinal chemistry.

Solid-phase synthesis of bis-heterocyclic compounds from resin-bound orthogonally protected lysine.

M. Giulianotti, R. Houghten, A. Nefzi, 2001, Journal of combinatorial chemistry.

Inhibition of Aminoglycoside 6′-N-acetyltransferase Type Ib (AAC(6′)-Ib): Structure–Activity Relationship of Substituted Pyrrolidine Pentamine Derivatives as Inhibitors

Radleigh G. Santos, M. Giulianotti, C. Pinilla, 2021, Biomedicines.

Inhibition of Aminoglycoside 6’-N-Acetyltransferase Type Ib [Aac(6′)-Ib]: Structure-Activity Relationship of Substituted Pyrrolidine Pentamine Derivatives as Inhibitors

Radleigh G. Santos, M. Giulianotti, C. Pinilla, 2021 .

A Robust and Cost-Effective Luminescent-Based High-Throughput Assay for Fructose-1,6-Bisphosphate Aldolase A

M. Giulianotti, R. Houghten, G. Powis, 2020, SLAS discovery : advancing life sciences R & D.

Identification of beryllium-dependent peptides recognized by CD4+ T cells in chronic beryllium disease

Radleigh G. Santos, P. Marrack, M. Giulianotti, 2013, The Journal of experimental medicine.

Identi fi cation of Small Molecule Inhibitors of Human As ( III ) S ‐ Adenosylmethionine Methyltransferase ( AS 3 MT )

M. Giulianotti, R. Houghten, A. Nefzi, 2019 .

Identification of Small Molecule Inhibitors of Human As(III) S-Adenosylmethionine Methyltransferase (AS3MT)

M. Giulianotti, R. Houghten, A. Nefzi, 2015, Chemical research in toxicology.

Discovery of Polypharmacological Melanocortin-3 and -4 Receptor Probes and Identification of a 100-Fold Selective nM MC3R Agonist versus a μM MC4R Partial Agonist.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2019, Journal of medicinal chemistry.

Selective agonists and antagonists of formylpeptide receptors: duplex flow cytometry and mixture-based positional scanning libraries

Susan M. Young, Radleigh G. Santos, J. Medina-Franco, 2013 .

Functional Mixture-Based Positional Scan Identifies a Library of Antagonist Tetrapeptide Sequences (LAtTeS) with Nanomolar Potency for the Melanocortin-4 Receptor and Equipotent with the Endogenous AGRP(86-132) Antagonist.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2021, Journal of medicinal chemistry.

A novel method for the determination of isokinetic ratios and its application in the synthesis of two new positional scanning libraries.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2012, ACS combinatorial science.

Solid phase synthesis of heterocyclic combinatorial libraries derived from peptides

Michael J. Kurth, M. Giulianotti, R. Houghten, 2002 .

Identification of Protein Palmitoylation Inhibitors from a Scaffold Ranking Library

Radleigh G. Santos, R. Deschenes, M. Giulianotti, 2016, Combinatorial chemistry & high throughput screening.

Interaction Fingerprints and Their Applications to Identify Hot Spots.

J. Medina-Franco, M. Giulianotti, K. Martínez-Mayorga, 2015, Methods in molecular biology.

Multiple Sclerosis-Associated HLA-DR2 of the HLA-DR and -DQ Molecules in the Redundancy in Antigen-Presenting Function

M. Giulianotti, C. Pinilla, M. Sospedra, 2006 .

Differential regulation of alcohol taking and seeking by antagonism at α4β2 and α3β4 nAChRs

M. Giulianotti, G. Welmaker, Gloria Brunori, 2018, Psychopharmacology.

Identification of small molecules by screening a mixture-based scaffold compound library for treatment of alpha-1 antitrypsin deficiency.

Radleigh G. Santos, M. Giulianotti, Chen Liu, 2020, Biochemical and biophysical research communications.

Traceless solid-phase synthesis of N-substituted 3,5-bis(substituted-idene)piperidin-4-one derivatives

J. Medina-Franco, M. Giulianotti, R. Houghten, 2010 .

The value of antimicrobial peptides in the age of resistance.

Andrew L. Ferguson, Steven B. Bradfute, A. Ferguson, 2020, The Lancet. Infectious diseases.

Synthesis and biological evaluation of 2-indolinone derivatives as potential antitumor agents.

M. Giulianotti, Yongping Yu, Liang Zhang, 2011, European journal of medicinal chemistry.

Novel T cell driven approach leads to the identification of immunoprevalent antigens

Radleigh G. Santos, M. Giulianotti, C. Pinilla, 2012 .

HTS by NMR of combinatorial libraries: a fragment-based approach to ligand discovery.

M. Giulianotti, R. Houghten, C. Pinilla, 2013, Chemistry & biology.

Combinatorial Libraries As a Tool for the Discovery of Novel, Broad-Spectrum Antibacterial Agents Targeting the ESKAPE Pathogens.

Radleigh G. Santos, J. Medina-Franco, M. Giulianotti, 2015, Journal of medicinal chemistry.

The Use of Synthetic Mixture Based Libraries to Identify Hit Compounds for ESKAPE Pathogens, Leishmaniasis, and Inhibitors of Palmitoylation

M. Giulianotti, 2016 .

Solid phase synthesis of 1,4-benzothiazepin-5-one derivatives

Richard A. Houghten, Marc A. Giulianotti, Adel Nefzi, 1999 .

Strategies for the use of mixture-based synthetic combinatorial libraries: scaffold ranking, direct testing in vivo, and enhanced deconvolution by computational methods.

Clemencia Pinilla, Yongping Yu, Adel Nefzi, 2008, Journal of combinatorial chemistry.

Solid‐Phase Synthesis of Heterocycles from Peptides and Amino Acids

M. Giulianotti, R. Houghten, Wenteng Chen, 2011 .

Palladium-catalyzed C-H functionalization using guanidine as a directing group: ortho arylation and olefination of arylguanidines.

M. Giulianotti, R. Houghten, Wenteng Chen, 2012, Organic letters.

A facile approach to polysubstituted pyrazoles from hydrazonyl chlorides and vinyl azides

M. Giulianotti, Wenteng Chen, Yongping Yu, 2011 .

A Facile Approach to the Synthesis of 3,4-Disubstituted-2-Aminothiazolium Derivatives through the Use of A "Volatilizable" Support.

M. Giulianotti, R. Houghten, Yangmei Li, 2010, Tetrahedron letters.

Solid-phase synthesis of N-substituted 3,4-dihydroquinazolinone derivatives

M. Giulianotti, R. Houghten, Zhang Liu, 2011 .

Solid-phase synthesis of linear ureas tethered to hydantoins and thiohydantoins.

M. Giulianotti, R. Houghten, L. Truong, 2002, Journal of combinatorial chemistry.

Solid-phase synthesis of branched thiohydantoin benzimidazolinethiones and branched thiohydantoin tetrahydroquinoxalinediones

M. Giulianotti, R. Houghten, A. Nefzi, 2000 .

Efficient solid phase synthesis of 3,5-disubstituted hydantoins

M. Giulianotti, R. Houghten, A. Nefzi, 1998 .

Solid-phase synthesis of 2-alkylidene-6-alkyl-imidazo[2,1-b]thiazole-3,5[2H,6H]-dione derivatives

M. Giulianotti, R. Houghten, Yangmei Li, 2009 .

Parallel synthesis of novel antitumor agents: 1,2,3-triazoles bearing biologically active sulfonamide moiety and their 3D-QSAR

J. Medina-Franco, M. Giulianotti, Bo Yang, 2011, Molecular Diversity.

A one-pot multicomponent approach to a new series of morphine derivatives and their biological evaluation.

M. Giulianotti, R. Houghten, C. Dooley, 2017, Organic & biomolecular chemistry.

Conformation-opioid activity relationships of bicyclic guanidines from 3D similarity analysis.

Clemencia Pinilla, Karina Martínez-Mayorga, Marc A Giulianotti, 2008, Bioorganic & medicinal chemistry.

High throughput synthesis of peptide alpha-thioesters through the use of "volatilizable" support.

Yongping Yu, Yangmei Li, Richard A Houghten, 2008, Journal of combinatorial chemistry.

High Throughput Synthesis of 2,3,6-Trisubstituted-5,6-Dihydroimidazo[2,1-b]thiazole Derivatives.

Yangmei Li, Richard A Houghten, M. Giulianotti, 2011, Tetrahedron letters.

A traceless approach to amide and peptide construction from thioacids and dithiocarbamate-terminal amines

M. Giulianotti, R. Houghten, Wenteng Chen, 2013 .

Solid phase synthesis of 1,6-disubstituted 2,3-diketopiperazines and 1,2-disubstituted piperazines from N-acylated amino acids

M. Giulianotti, R. Houghten, A. Nefzi, 1999 .

Synthesis and biological evaluations of novel endomorphin analogues containing α-hydroxy-β-phenylalanine (AHPBA) displaying mixed μ/δ opioid receptor agonist and δ opioid receptor antagonist activities.

Austin B. Yongye, Radleigh G. Santos, M. Giulianotti, 2015, European journal of medicinal chemistry.

Synthesis of 2,3,4-Trisubstituted Pyrroles via a Facile Reaction of Vinyl Azides and Tosylmethyl Isocyanide.

M. Giulianotti, Wenteng Chen, Yongping Yu, 2012 .

Synthesis of cyclic peptides through direct aminolysis of peptide thioesters catalyzed by imidazole in aqueous organic solutions.

M. Giulianotti, R. Houghten, A. Yongye, 2009, Journal of combinatorial chemistry.

Efficient approach for the diversity-oriented synthesis of macro-heterocycles on solid-support

M. Giulianotti, A. Nefzi, 2003 .

Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries

Clemencia Pinilla, Susan M. Young, Bruce S Edwards, 2013, Molecular Pharmacology.

Identification of a Novel Polyamine Scaffold With Potent Efflux Pump Inhibition Activity Toward Multi-Drug Resistant Bacterial Pathogens

Radleigh G. Santos, M. Giulianotti, G. Welmaker, 2018, Front. Microbiol..

Solid-Phase Synthesis of 2,3,5,6-Tetrahydro-1H-imidazo[1,2-a]benzo[d]-[1,3]diazepinesvia Pd(OAc)2/Cu(OAc)2-CocatalyzedCyclization

M. Giulianotti, R. Houghten, Wenteng Chen, 2011 .

Identification of SARS-CoV-2 Spike Palmitoylation Inhibitors That Results in Release of Attenuated Virus with Reduced Infectivity

R. Deschenes, M. Giulianotti, B. Chandran, 2022, Viruses.

Inhibition of SARS-CoV-2 spike protein palmitoylation reduces virus infectivity

R. Deschenes, M. Giulianotti, B. Chandran, 2021, bioRxiv.

SOLID PHASE SYNTHESIS OF 2,4,5-TRISUBSTITUTED THIOMORPHOLIN-3-ONES

M. Giulianotti, R. Houghten, A. Nefzi, 1998 .

Redundancy in Antigen-Presenting Function of the HLA-DR and -DQ Molecules in the Multiple Sclerosis-Associated HLA-DR2 Haplotype1

R. Simon, M. Giulianotti, C. Pinilla, 2006, The Journal of Immunology.

Haplotype Multiple Sclerosis-Associated HLA-DR 2 of the HLA-DR and-DQ Molecules in the Redundancy in Antigen-Presenting Function

R. Simon, M. Giulianotti, C. Pinilla, 2006 .

Chemoinformatic Analysis of Combinatorial Libraries, Drugs, Natural Products, and Molecular Libraries Small Molecule Repository

Rajarshi Guha, José L. Medina-Franco, Richard A. Houghten, 2009, J. Chem. Inf. Model..

Small-Molecule Inhibitors Targeting Topoisomerase I as Novel Antituberculosis Agents

M. Giulianotti, G. Welmaker, R. Houghten, 2016, Antimicrobial Agents and Chemotherapy.

GM-CSF Production Allows the Identification of Immunoprevalent Antigens Recognized by Human CD4+ T Cells Following Smallpox Vaccination

Radleigh G. Santos, D. Douek, M. Giulianotti, 2011, PloS one.

Ligand/kappa-opioid receptor interactions: insights from the X-ray crystal structure.

Karina Martinez-Mayorga, Austin B Yongye, Marc A Giulianotti, 2013, European journal of medicinal chemistry.

Characterization of a comprehensive flavor database

Austin B. Yongye, José L. Medina-Franco, Marc A. Giulianotti, 2011 .

Combining positional scanning peptide libraries, HLA-DR transfectants and bioinformatics to dissect the epitope spectrum of HLA class II cross-restricted CD4+ T cell clones.

R. Simon, M. Giulianotti, C. Pinilla, 2010, Journal of immunological methods.

Structure–activity relationships of benzimidazole derivatives as antiparasitic agents: Dual activity-difference (DAD) maps

José L. Medina-Franco, Jaime Pérez-Villanueva, Rafael Castillo, 2011 .

Pharmaceutical Research Enabled Through Microgravity: Perspectives on the Use of the International Space Station U.S. National Laboratory

Lucie A. Low, Marc A. Giulianotti, M. Giulianotti, 2019, Pharmaceutical Research.

Scaffold Ranking and Positional Scanning Identify Novel Neurite Outgrowth Promoters with Nanomolar Potency.

Radleigh G. Santos, J. Bixby, M. Giulianotti, 2018, ACS medicinal chemistry letters.

Identification of B Cell and T Cell Epitopes Using Synthetic Peptide Combinatorial Libraries

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2022, Current protocols.

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput "Unbiased" Screening Campaign.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2021, Journal of medicinal chemistry.

Identification of a Small Molecule Inhibitor of the Aminoglycoside 6’-N-Acetyltransferase Type Ib [AAC(6’)-Ib] Using Mixture-Based Combinatorial Libraries

Radleigh G. Santos, M. Giulianotti, C. Pinilla, 2017, bioRxiv.

Discovery of Mixed Pharmacology Melanocortin-3 Agonists and Melanocortin-4 Receptor Tetrapeptide Antagonist Compounds (TACOs) Based on the Sequence Ac-Xaa1-Arg-(pI)DPhe-Xaa4-NH2.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2017, Journal of medicinal chemistry.

Novel Pyrrolidine Diketopiperazines Selectively Inhibit Melanoma Cells via Induction of Late-Onset Apoptosis

M. Giulianotti, R. Houghten, G. Kaushik, 2014, Journal of medicinal chemistry.

High-throughput parallel synthesis of 3,4-disubstituted 1-(ω-hydroxyalkyl) imidazolin-2-ones on ‘volatilizable’ supports

M. Giulianotti, R. Houghten, Yongping Yu, 2008 .

Combinatorial libraries: Equimolar incorporation of benzaldehyde mixtures in reductive alkylation reactions

Michael J. Kurth, M. Giulianotti, R. Houghten, 2002 .

Solid-Phase Synthesis of Substituted 2,3-Diketopiperazines from Reduced Polyamides

Richard A. Houghten, Marc A. Giulianotti, Adel Nefzi, 2000 .

Tissue Chips in Space: Modeling Human Diseases in Microgravity

M. Giulianotti, L. Low, 2019, Pharmaceutical Research.

Activity of ADAM17 (a Disintegrin and Metalloprotease 17) Is Regulated by Its Noncatalytic Domains and Secondary Structure of its Substrates*

M. Giulianotti, R. Houghten, G. Fields, 2013, The Journal of Biological Chemistry.

Docking of Protein Kinase B Inhibitors: Implications in the Structure‐Based Optimization of a Novel Scaffold

J. Medina-Franco, M. Giulianotti, R. Castillo, 2010, Chemical biology & drug design.

Opportunities for Biomanufacturing in Low Earth Orbit: Current Status and Future Directions

G. Rodrigue, Michael Roberts, A. Grodzinsky, 2021 .

Potent antimicrobial small molecules screened as inhibitors of tyrosine recombinases and Holliday junction-resolving enzymes

P. Salamon, A. Segall, M. Giulianotti, 2011, Molecular Diversity.

Solid-phase synthesis of bis-2-imidazolidinethiones from resin-bound tripeptides.

N. A. Ong, M. Giulianotti, R. Houghten, 2000, Organic letters.

Modeling of peptides containing D-amino acids: implications on cyclization

Austin B. Yongye, Richard A. Houghten, Yongping Yu, 2009, J. Comput. Aided Mol. Des..

Biomanufacturing in low Earth orbit for regenerative medicine

Nicole L. Wagner, D. L. Taylor, A. Grodzinsky, 2021, Stem cell reports.

Visualization of the Chemical Space in Drug Discovery

José L. Medina-Franco, Karina Martinez-Mayorga, Marc A. Giulianotti, 2008 .

Libraries from Libraries: A Series of Sulfonamide Linked Heterocycles Derived from the Same Scaffold.

M. Giulianotti, R. Houghten, Wenteng Chen, 2013, Tetrahedron letters.

Parallel synthesis of 1,6-disubstituted-1,2,4-triazin-3-ones on solid-phase.

M. Giulianotti, R. Houghten, Yongping Yu, 2013, ACS combinatorial science.

Rapid Scanning Structure-Activity Relationships in Combinatorial Data Sets: Identification of Activity Switches

Clemencia Pinilla, Bruce S. Edwards, Larry A. Sklar, 2013, J. Chem. Inf. Model..

The Mathematics of a Successful Deconvolution: A Quantitative Assessment of Mixture-Based Combinatorial Libraries Screened Against Two Formylpeptide Receptors

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2013, Molecules.

Integrating computational and mixture-based screening of combinatorial libraries

Clemencia Pinilla, Austin B. Yongye, Richard A. Houghten, 2011, Journal of molecular modeling.

Conformational landscape of platinum(II)-tetraamine complexes: DFT and NBO studies

Austin B. Yongye, Richard A. Houghten, Karina Martínez-Mayorga, 2010, J. Comput. Aided Mol. Des..

Characterization of Activity Landscapes Using 2D and 3D Similarity Methods: Consensus Activity Cliffs

José L. Medina-Franco, Andreas Bender, Richard A. Houghten, 2009, J. Chem. Inf. Model..

A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation.

M. Giulianotti, R. Houghten, T. Kaoud, 2019, ACS chemical biology.

Identification and characterization of an atypical Gαs-biased β2AR agonist that fails to evoke airway smooth muscle cell tachyphylaxis

W. Goddard, M. Giulianotti, S. Liggett, 2021, Proceedings of the National Academy of Sciences.

Antigen discovery for the identification of vaccine candidates and biomarkers using a T cell driven approach in combination with positional scanning peptide libraries

Radleigh G. Santos, M. Giulianotti, C. Pinilla, 2015 .

Combinatorial chemistry: Solid-phase synthesis of heterocyclic compounds from C α -functionalized amino acids

N. A. Ong, M. Giulianotti, R. Houghten, 2002 .

Peptides as precursors in the synthesis of heterocyclic positional scanning combinatorial libraries

M. Giulianotti, R. Houghten, A. Nefzi, 2002 .

The Parallel Structure–Activity Relationship Screening of Three Compounds Identifies the Common Agonist Pharmacophore of Pyrrolidine Bis-Cyclic Guanidine Melanocortin-3 Receptor (MC3R) Small-Molecule Ligands

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2023, International journal of molecular sciences.

Discovery of a novel protein kinase B inhibitor by structure-based virtual screening.

Yongping Yu, Marc A Giulianotti, J. Medina-Franco, 2009, Bioorganic & medicinal chemistry letters.

Clemencia Pinilla, José L Medina-Franco, Gerald M Maggiora, 2007, Chemical biology & drug design.

Glycosylation of A Disintegrin And Metalloprotease 17 (ADAM17) Affects its Activity and Inhibition

M. Giulianotti, R. Houghten, G. Fields, 2015 .

Activity of ADAM17 (a Disintegrin and Metalloprotease 17) Is Regulated by Its Noncatalytic Domains and Secondary Structure of its Substrates*

M. Giulianotti, R. Houghten, G. Fields, 2013, Journal of Biological Chemistry.

Conformational landscape of platinum(II)-tetraamine complexes: DFT and NBO studies

Austin B. Yongye, M. Giulianotti, R. Houghten, 2010, J. Comput. Aided Mol. Des..

Conditional Probabilistic Analysis for Prediction of the Activity Landscape and Relative Compound Activities

José L. Medina-Franco, Richard A. Houghten, Marc A. Giulianotti, 2013, J. Chem. Inf. Model..

Characterization of Activity Landscapes Using 2D and 3D Similarity Methods: Consensus Activity Cliffs

Ray M. Marín, J. Medina-Franco, A. Bender, 2009, J. Chem. Inf. Model..

Solid-phase synthesis of 2,3,4,5-tetrahydro-1 H-benzo[ e][1,4]diazepine derivatives

M. Giulianotti, R. Houghten, Wenteng Chen, 2011 .

Potent antimicrobial small molecules screened as inhibitors of tyrosine recombinases and Holliday junction-resolving enzymes

P. Salamon, A. Segall, M. Giulianotti, 2011, Molecular Diversity.

Identi ﬁ cation and characterization of an atypical G α s-biased β 2 AR agonist that fails to evoke airway smooth muscle cell tachyphylaxis

W. Goddard, M. Giulianotti, S. Liggett, 2022 .

Amphiphilic Cell-Penetrating Peptides Containing Arginine and Amphiphilic Cell-Penetrating Peptides Containing Arginine and Hydrophobic Residues as Protein Delivery Agents Hydrophobic Residues as Protein Delivery Agents

M. Giulianotti, K. Parang, R. Tiwari, 2022 .

Identification of a Hit Series of Antileishmanial Compounds through the Use of Mixture-Based Libraries.

D. Kyle, M. Giulianotti, R. Houghten, 2017, ACS medicinal chemistry letters.