G. Welmaker

发表

Shifting from the single to the multitarget paradigm in drug discovery.

J. Medina-Franco, M. Giulianotti, G. Welmaker, 2013, Drug discovery today.

Antiobesity-like effects of the 5-HT2C receptor agonist WAY-161503

J. Barrett, B. Harrison, G. Welmaker, 2006, Brain Research.

Direct Phenotypic Screening in Mice: Identification of Individual, Novel Antinociceptive Compounds from a Library of 734 821 Pyrrolidine Bis-piperazines

Radleigh G. Santos, M. Giulianotti, G. Welmaker, 2015, ACS combinatorial science.

Highly Selective and Potent α4β2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats.

M. Giulianotti, G. Welmaker, R. Houghten, 2017, Journal of medicinal chemistry.

Scaffold ranking and positional scanning utilized in the discovery of nAChR-selective compounds suitable for optimization studies.

Radleigh G. Santos, M. Giulianotti, G. Welmaker, 2013, Journal of medicinal chemistry.

Synthesis and 5-hydroxytryptamine (5-HT) activity of 2,3,4,4a-tetrahydro-1H-pyrazino[1,2-a]quinoxalin-5-(6H)ones and 2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-a]quinoxalines.

G. Welmaker, J. Nelson, S. Rosenzweig-Lipson, 2000, Bioorganic & medicinal chemistry letters.

Differential regulation of alcohol taking and seeking by antagonism at α4β2 and α3β4 nAChRs

M. Giulianotti, G. Welmaker, Gloria Brunori, 2018, Psychopharmacology.

Modulation of Wnt signaling through inhibition of secreted frizzled-related protein I (sFRP-1) with N-substituted piperidinyl diphenylsulfonyl sulfonamides.

G. Welmaker, R. Bhat, P. Bodine, 2009, Journal of medicinal chemistry.

Combinatorial Libraries As a Tool for the Discovery of Novel, Broad-Spectrum Antibacterial Agents Targeting the ESKAPE Pathogens.

Radleigh G. Santos, J. Medina-Franco, M. Giulianotti, 2015, Journal of medicinal chemistry.

Chiral γ-silyloxy allylstannanes as synthetic reagents. Proof of absolute configuration

G. Welmaker, J. A. Marshall, 1991 .

ON THE 1,3-ISOMERIZATION OF NONRACEMIC ALPHA -(ALKOXY)ALLYL STANNANES

G. Welmaker, J. A. Marshall, B. W. Gung, 1991 .

A microwave-assisted, green procedure for the synthesis of N-aryl sulfonyl and N-aryl pyrroles

G. Welmaker, Matthew A. Wilson, G. Filzen, 2009 .

Mannich Biscyclizations. Total Synthesis of (-)-Ajmalicine

L. Overman, G. Welmaker, M. Loegers, 1995 .

Enantioselective Synthesis of (+)- and (-)-Muricatacin through SE2' Addition of Nonracemic .gamma.-Silyloxy Allylic Stannanes to Aldehydes

G. Welmaker, J. A. Marshall, 1994 .

(Z)- and (E)-.gamma.-silyloxy allylic stannanes. Highly syn selective reagents for SE' additions to aldehydes

G. Welmaker, J. A. Marshall, 1992 .

On the 1,3‐Isomerization of Nonracemic α‐(Alkoxy)allyl Stannanes.

G. Welmaker, J. A. Marshall, B. W. Gung, 1991 .

The Aza‐Cope/Mannich Reaction

L. Overman, G. Welmaker, P. Humphreys, 2011 .

Chiral γ-Siloxyallylstannanes as Synthetic Reagents. Proof of Absolute Configuration.

G. Welmaker, J. A. Marshall, 1992 .

A process for the preparation of 1,2,3,4,8,9,10,10a-octahydro-7bH-cyclopenta[b][1,4]diazepino[6,7,1-hi]indole

G. Welmaker, J. Sabalski, 2004 .

Identification of a Novel Polyamine Scaffold With Potent Efflux Pump Inhibition Activity Toward Multi-Drug Resistant Bacterial Pathogens

Radleigh G. Santos, M. Giulianotti, G. Welmaker, 2018, Front. Microbiol..

A small molecule inhibitor of the Wnt antagonist secreted frizzled-related protein-1 stimulates bone formation.

B. Komm, G. Welmaker, R. Bhat, 2009, Bone.

Small-Molecule Inhibitors Targeting Topoisomerase I as Novel Antituberculosis Agents

M. Giulianotti, G. Welmaker, R. Houghten, 2016, Antimicrobial Agents and Chemotherapy.

Cycloalkyl[b][1,4]benzodiazepinoindoles are agonists at the human 5-HT2C receptor.

B. Harrison, G. Welmaker, S. Rosenzweig-Lipson, 2004, Bioorganic & Medicinal Chemistry Letters.

Cycloalkyl[b][1,4]benzodiazepinoindoles Are Agonists at the Human 5‐HT2C Receptor.

B. Harrison, G. Welmaker, S. Rosenzweig-Lipson, 2004 .