A. di Pietro

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Multidrug resistance phenotype mediated by the P-glycoprotein-like transporter in Leishmania: a search for reversal agents.

J. M. Pérez-Victoria, A. di Pietro, D. Barron, 2002, Current drug targets.

Multidrug resistance ABC transporter structure predictions by homology modeling approaches.

A. di Pietro, C. Dumontet, Myléne Honorat, 2011, Current drug metabolism.

A 3D linear solvation energy model to quantify the affinity of flavonoid derivatives toward P-glycoprotein.

P. Carrupt, S. Rudaz, F. Bajot, 2009, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Inhibitors of cancer cell multidrug resistance mediated by breast cancer resistance protein (BCRP/ABCG2)

A. di Pietro, S. Macalou, A. Boumendjel, 2006, Anti-cancer drugs.

Evaluation of Jatrophane Esters from Euphorbia spp. as Modulators of Candida albicans Multidrug Transporters.

Julien Paolini, Marc Litaudon, Louis-Félix Nothias, 2017, Journal of natural products.

Structural mapping of catalytic site with respect to alpha-subunit and noncatalytic site in yeast mitochondrial F1-ATPase using fluorescence resonance energy transfer.

R. Goody, A. di Pietro, G. Divita, 1993, The Journal of biological chemistry.

Discovery of a new series of jatrophane and lathyrane diterpenes as potent and specific P-glycoprotein modulators.

A. di Pietro, E. Barile, C. Fattorusso, 2008, Organic & biomolecular chemistry.

MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts

A. di Pietro, A. Puisieux, C. Rioufol, 2014, Oncotarget.

Iodination of verapamil for a stronger induction of death, through GSH efflux, of cancer cells overexpressing MRP1.

A. di Pietro, Doriane Lorendeau, H. Baubichon-Cortay, 2010, Bioorganic & medicinal chemistry.

Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

Mathieu Marchivie, Joachim Jose, Jean Guillon, 2015, Drug design, development and therapy.

Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2.

A. di Pietro, B. Sarkadi, P. Falson, 2020, European journal of medicinal chemistry.

The acridone derivative MBLI-87 sensitizes breast cancer resistance protein-expressing xenografts to irinotecan.

S. Bates, A. di Pietro, E. Matera, 2011, European journal of cancer.

Targeting the multidrug ABCG2 transporter with flavonoidic inhibitors: in vitro optimization and in vivo validation.

P. Carrupt, A. di Pietro, P. Falson, 2011, Current medicinal chemistry.

Methoxy stilbenes as potent, specific, untransported, and noncytotoxic inhibitors of breast cancer resistance protein.

A. di Pietro, Luciana Pereira Rangel, J. Guitton, 2012, ACS chemical biology.

Sequence requirements of the ATP-binding site within the C-terminal nucleotide-binding domain of mouse P-glycoprotein: structure-activity relationships for flavonoid binding.

T. Krell, A. di Pietro, D. Barron, 2001, Biochemistry.

Binding of the polyflavane P13 on various pig myocardial membranes--effects on protein release and on Ca2+ and Mg2+ movements.

A. di Pietro, D. Gautheron, C. Godinot, 1977, Biochemical pharmacology.

ABCG2 is not able to catalyze glutathione efflux and does not contribute to GSH-dependent collateral sensitivity

G. Szakács, A. di Pietro, B. Sarkadi, 2013, Front. Pharmacol..

Selective modulation of P-glycoprotein activity by steroidal saponines from Paris polyphylla.

A. di Pietro, C. Dumontet, D. Guilet, 2009, Fitoterapia.

Overexpression of homogeneous and active ABCG2 in insect cells.

J. M. Pérez-Victoria, A. di Pietro, A. Pozza, 2009, Protein expression and purification.

Jatrophane diterpenes from Euphorbia spp. as modulators of multidrug resistance in cancer therapy

A. di Pietro, C. Dumontet, G. Corea, 2009, Phytochemistry Reviews.

The "catalytic" triad of isocitrate dehydrogenase kinase/phosphatase from E. coli and its relationship with that found in eukaryotic protein kinases.

C. Blanchet, A. di Pietro, A. Cozzone, 2001, Biochemistry.

GTP binding to elongation factor eEF-2 unmasks a tryptophan residue required for biological activity.

F. Penin, A. di Pietro, J. Lavergne, 1993, The Journal of biological chemistry.

Isoprenoid flavonoids are new leads in the modulation of chemoresistance

A. di Pietro, D. Barron, C. Dumontet, 2002, Phytochemistry Reviews.

Pig heart mitochondrial ATPase : properties of purified and membrane-bound enzyme. Effects of flavonoids.

A. di Pietro, D. Gautheron, C. Godinot, 1975, Biochimie.

(R)- and (S)-Verapamil Differentially Modulate the Multidrug-resistant Protein MRP1*

A. di Pietro, X. Chang, H. Baubichon-Cortay, 2007, Journal of Biological Chemistry.

Flavonoid dimers are highly potent killers of multidrug resistant cancer cells overexpressing MRP1

L. Chow, A. di Pietro, P. Falson, 2017, Biochemical pharmacology.

ABCG2: recent discovery of potent and highly selective inhibitors.

A. di Pietro, Evelyn Winter, L. Payen, 2013, Future medicinal chemistry.

Jatrophane diterpenes as modulators of multidrug resistance. Advances of structure-activity relationships and discovery of the potent lead pepluanin A.

A. di Pietro, C. Dumontet, G. Corea, 2004, Journal of medicinal chemistry.

Jatrophane diterpenes as P-glycoprotein inhibitors. First insights of structure-activity relationships and discovery of a new, powerful lead.

A. di Pietro, C. Dumontet, G. Appendino, 2003, Journal of medicinal chemistry.

The Q-loop Disengages from the First Intracellular Loop during the Catalytic Cycle of the Multidrug ABC Transporter BmrA*

C. Geourjon, A. di Pietro, J. Jault, 2005, Journal of Biological Chemistry.

Impairment of oxidative phosphorylation increases the toxicity of SYD-1 on hepatocarcinoma cells (HepG2).

A. di Pietro, G. Martinez, A. Echevarria, 2016, Chemico-biological interactions.

Anticancer multidrug resistance mediated by MRP1: Recent advances in the discovery of reversal agents

A. di Pietro, A. Boumendjel, H. Baubichon-Cortay, 2005, Medicinal research reviews.

Prenyl-flavonoids as potent inhibitors of the Pdr5p multidrug ABC transporter from Saccharomyces cerevisiae.

A. Goffeau, A. di Pietro, D. Barron, 2000, Biochemistry.

An Open Randomized Controlled Study on the Efficacy of Low-Sodium Water Intake Evaluated by Non-Invasive Methods in Patients with Cellulite

A. di Pietro, P. Puddu, O. De Pità, 2003 .

Transfer of the Cystic Fibrosis Transmembrane Conductance Regulator to Human Cystic Fibrosis Cells Mediated by Extracellular Vesicles.

A. di Pietro, M. Chanson, P. Boulanger, 2016, Human gene therapy.

"Hysteric" behavior and nucleotide binding sites of pig heart mitochondrial F1 adenosine 5'-triphosphatase.

F. Penin, A. di Pietro, D. Gautheron, 1980, Biochemistry.

Conformational change induced by ATP binding in the multidrug ATP-binding cassette transporter BmrA.

A. di Pietro, A. Durand, P. Gros, 2008, Biochemistry.

Characterization of YvcC (BmrA), a multidrug ABC transporter constitutively expressed in Bacillus subtilis.

F. Denizot, A. di Pietro, J. Jault, 2004, Biochemistry.

Role of magnesium on kinetic parameters of soluble F1-ATPase from pig heart mitochondria.

A. di Pietro, D. Gautheron, C. Godinot, 1980, Biochimie.

Lathyrol and epoxylathyrol derivatives: Modulation of Cdr1p and Mdr1p drug-efflux transporters of Candida albicans in Saccharomyces cerevisiae model.

Maria-José U. Ferreira, A. di Pietro, R. Prasad, 2017, Bioorganic & medicinal chemistry.

Highly efficient over-production in E. coli of YvcC, a multidrug-like ATP-binding cassette transporter from Bacillus subtilis.

F. Penin, A. di Pietro, B. Miroux, 2002, Biochimica et biophysica acta.

Maraviroc intensification for HIV-1-positive immunological non-responders (INRs) despite virological suppression during HAART

A. di Pietro, G. d’Ettorre, P. Vitiello, 2010, Journal of the International AIDS Society.

Essential arginyl residues in the H+-translocating ATPase of plasma membrane from the yeast Schizosaccharomyces pombe.

A. Goffeau, A. di Pietro, 1985, European journal of biochemistry.

Abolition of anion‐activation of mitochondrial F1‐ATPase by the partial ADP‐induced hysteretic inhibition

A. di Pietro, D. Gautheron, C. Godinot, 1982, FEBS letters.

Structure-function relationships of mitochondrial ATPase-ATPsynthase using Schizosaccharomyces pombe yeast mutants with altered F1 subunits.

A. di Pietro, G. Divita, J. Jault, 1989, Biochimie.

Purification from a yeast mutant of mitochondrial F1 with modified beta-subunit. High affinity for nucleotides and high negative cooperativity of ATPase activity.

A. di Pietro, J. Jault, P. Falson, 1989, Biochimica et biophysica acta.

A yeast strain with mutated beta-subunits of mitochondrial ATPase-ATPsynthase: high azide and bicarbonate sensitivity of the ATPase activity.

A. Goffeau, A. di Pietro, J. Jault, 1989, Biochemical and biophysical research communications.

Revertant of the yeast Schizosaccharomyces pombe with modified alpha subunits of mitochondrial ATPase-ATPsynthase: impaired nucleotide interactions with soluble and membrane-bound enzyme.

A. Goffeau, A. di Pietro, J. Jault, 1987, Biochemical and biophysical research communications.

New structure–activity relationships of chalcone inhibitors of breast cancer resistance protein: polyspecificity toward inhibition and critical substitutions against cytotoxicity

A. di Pietro, A. Mascarello, L. D. Chiaradia-Delatorre, 2013, Drug design, development and therapy.

Jatrophanes from Euphorbia squamosa as potent inhibitors of Candida albicans multidrug transporters.

Y. Shokoohinia, A. di Pietro, G. Appendino, 2014, Journal of natural products.

Correlation between the affinity of flavonoids binding to the cytosolic site of Leishmania tropica multidrug transporter and their efficiency to revert parasite resistance to daunomycin.

J. M. Pérez-Victoria, A. di Pietro, D. Barron, 1999, Biochemistry.

Synthesis and Anticancer Cytotoxicity of Azaaurones Overcoming Multidrug Resistance

G. Szakács, A. di Pietro, B. Sarkadi, 2020, Molecules.

Verapamil and Its Derivative Trigger Apoptosis through Glutathione Extrusion by Multidrug Resistance Protein MRP1

A. di Pietro, X. Chang, H. Baubichon-Cortay, 2004, Cancer Research.

Alteration of apparent negative cooperativity of ATPase activity by alpha-subunit glutamine 173 mutation in yeast mitochondrial F1. Correlation with impaired nucleotide interaction at a regulatory site.

A. di Pietro, J. Jault, P. Falson, 1991, The Journal of biological chemistry.

Isolation and sequence of an endochitinase-encoding gene from a cDNA library of Trichoderma harzianum.

A. di Pietro, M. Lorito, J. P. Nakas, 1994, Gene.

Natural and synthetic benzophenones: interaction with the cytosolic binding domain of P-glycoprotein.

A. Chaboud, A. di Pietro, D. Barron, 2001, Phytochemistry.

C-Isoprenylation of flavonoids enhances binding affinity toward P-glycoprotein and modulation of cancer cell chemoresistance.

A. di Pietro, D. Barron, C. Dumontet, 2001, Journal of medicinal chemistry.

Prenylated xanthones as potential P-glycoprotein modulators.

A. di Pietro, D. Barron, G. Conseil, 2000, Bioorganic & medicinal chemistry letters.

Flavonoids: a class of modulators with bifunctional interactions at vicinal ATP- and steroid-binding sites on mouse P-glycoprotein.

A. di Pietro, D. Barron, J. Jault, 1998, Proceedings of the National Academy of Sciences of the United States of America.

Anticancer multidrug resistance mediated by MRP1: Recent advances in the discovery of reversal agents

A. di Pietro, A. Boumendjel, H. Baubichon-Cortay, 2005, Medicinal research reviews.

B-ring substituted 5,7-dihydroxyflavonols with high-affinity binding to P-glycoprotein responsible for cell multidrug resistance.

A. di Pietro, F. Bois, A. Boumendjel, 2001, Bioorganic & medicinal chemistry letters.

Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2.

Joachim Jose, Jean Guillon, A. di Pietro, 2015, Journal of medicinal chemistry.

Symmetric bis-chalcones as a new type of breast cancer resistance protein inhibitors with a mechanism different from that of chromones.

A. di Pietro, L. D. Chiaradia-Delatorre, R. Yunes, 2014, Journal of medicinal chemistry.

Halogenated chalcones with high-affinity binding to P-glycoprotein: potential modulators of multidrug resistance.

A. di Pietro, F. Bois, A. Boumendjel, 1998, Journal of medicinal chemistry.

Investigation of chalcones as selective inhibitors of the breast cancer resistance protein: critical role of methoxylation in both inhibition potency and cytotoxicity.

Raphaël Terreux, Xavier Ronot, A. di Pietro, 2012, Journal of medicinal chemistry.

Targeting the Achilles Heel of Multidrug-Resistant Cancer by Exploiting the Fitness Cost of Resistance

M. Gottesman, G. Szakács, M. Hall, 2014, Chemical reviews.

Cytotoxicity of η6-areneruthenium-based molecules to glioblastoma cells and their recognition by multidrug ABC transporters.

A. di Pietro, H. Winnischofer, G. Martinez, 2018, European journal of medicinal chemistry.

Selective Cytotoxicity of 1,3,4-Thiadiazolium Mesoionic Derivatives on Hepatocarcinoma Cells (HepG2)

A. di Pietro, G. Martinez, A. Echevarria, 2015, PloS one.

Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein.

Jérôme Guitton, Raphaël Terreux, A. di Pietro, 2012, Journal of medicinal chemistry.

Ferrocene-embedded flavonoids targeting the Achilles heel of multidrug-resistant cancer cells through collateral sensitivity.

A. di Pietro, A. Boumendjel, Malik Zarioh, 2017, European journal of medicinal chemistry.

Azaindole derivatives are inhibitors of microtubule dynamics, with anti‐cancer and anti‐angiogenic activities

Laurence Lafanechère, Caroline Barette, Anne Martinez, 2013, British journal of pharmacology.

Structuring Detergents for Extracting and Stabilizing Functional Membrane Proteins

A. di Pietro, D. Ficheux, R. Kahn, 2011, PloS one.

Breast cancer resistance protein (BCRP/ABCG2): new inhibitors and QSAR studies by a 3D linear solvation energy approach.

Julien Boccard, Pierre-Alain Carrupt, P. Carrupt, 2009, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Nonprenylated rotenoids, a new class of potent breast cancer resistance protein inhibitors.

Francesca Borrelli, Raffaele Capasso, R. Capasso, 2007, Journal of medicinal chemistry.

Acridone derivatives: design, synthesis, and inhibition of breast cancer resistance protein ABCG2.

A. di Pietro, S. Macalou, A. Boumendjel, 2007, Bioorganic & medicinal chemistry.

Competition between ADP and nucleotide analogues to occupy regulatory sites(s) related to hysteretic inhibition of mitochondrial F1-ATPase.

A. di Pietro, D. Gautheron, C. Godinot, 1981, Biochemical and biophysical research communications.

High-Affinity Binding of Silybin Derivatives to the Nucleotide-Binding Domain of a Leishmania tropicaP-Glycoprotein-Like Transporter and Chemosensitization of a Multidrug-Resistant Parasite to Daunomycin

J. M. Pérez-Victoria, A. di Pietro, D. Barron, 2001, Antimicrobial Agents and Chemotherapy.

Recent advances in the discovery of flavonoids and analogs with high‐affinity binding to P‐glycoprotein responsible for cancer cell multidrug resistance

A. di Pietro, D. Barron, C. Dumontet, 2002, Medicinal research reviews.

Chemical modification of thiol groups of mitochondrial F1-ATPase from the yeast Schizosaccharomyces pombe. Involvement of alpha- and gamma-subunits in the enzyme activity.

A. di Pietro, P. Falson, D. Gautheron, 1986, The Journal of biological chemistry.

The Conserved Glutamate Residue Adjacent to the Walker-B Motif Is the Catalytic Base for ATP Hydrolysis in the ATP-binding Cassette Transporter BmrA*

A. di Pietro, P. Gros, J. Jault, 2003, Journal of Biological Chemistry.

The flavanolignan silybin and its hemisynthetic derivatives, a novel series of potential modulators of P-glycoprotein.

A. di Pietro, D. Barron, K. El Kirat, 2000, Bioorganic & medicinal chemistry letters.

Effects of P13, a polyflavane compound, on pig myocardium ATP-synthesis, ATPases and creatine kinase.

A. di Pietro, D. Gautheron, C. Godinot, 1977, Biochemical pharmacology.

Time-resolved fluorescence resonance energy transfer shows that the bacterial multidrug ABC half-transporter BmrA functions as a homodimer.

A. di Pietro, M. R. Lugo, J. Jault, 2005, Biochemistry.

The ABC transporter BmrA from Bacillus subtilis is a functional dimer when in a detergent-solubilized state.

A. di Pietro, R. Haser, C. Ebel, 2006, The Biochemical journal.

4-Hydroxy-6-methoxyaurones with high-affinity binding to cytosolic domain of P-glycoprotein.

A. di Pietro, N. Deka, A. Boumendjel, 2002, Chemical & pharmaceutical bulletin.

Chemical modification of alpha-subunit tryptophan residues in Schizosaccharomyces pombe mitochondrial F1 adenosine 5'-triphosphatase: differential reactivity and role in activity.

A. di Pietro, G. Divita, J. Jault, 1993, Biochemistry.

Quinoxaline-substituted chalcones as new inhibitors of breast cancer resistance protein ABCG2: polyspecificity at B-ring position

Ricardo José Nunes, A. di Pietro, A. Mascarello, 2014, Drug design, development and therapy.

Synthesis of new piperazinyl-pyrrolo[1,2-a]quinoxaline derivatives as inhibitors of Candida albicans multidrug transporters by a Buchwald–Hartwig cross-coupling reaction

A. di Pietro, R. Prasad, M. Marchivie, 2020, RSC advances.

Structure and function of the ATPase-ATP synthase complex of mitochondria as compared to chloroplasts and bacteria.

A. di Pietro, C. Godinot, 1986, Biochimie.

Structure-activity relationships of chromone derivatives toward the mechanism of interaction with and inhibition of breast cancer resistance protein ABCG2.

G. Szakács, A. di Pietro, Evelyn Winter, 2013, Journal of medicinal chemistry.

Dicer-Mediated Upregulation of BCRP Confers Tamoxifen Resistance in Human Breast Cancer Cells

S. Fuqua, I. Barone, S. Andò, 2011, Clinical Cancer Research.

The ATP-binding Site in the 2-Kinase Domain of Liver 6-Phosphofructo-2-kinase/Fructose-2,6-bisphosphatase

D. Vertommen, A. di Pietro, L. Bertrand, 1996, The Journal of Biological Chemistry.

Multiple flavonoid-binding sites within multidrug resistance protein MRP1

J. Riordan, A. di Pietro, D. Barron, 2003, Cellular and Molecular Life Sciences CMLS.

Dual properties of hispidulin: antiproliferative effects on HepG2 cancer cells and selective inhibition of ABCG2 transport activity

A. di Pietro, G. Martinez, G. Valdameri, 2015, Molecular and Cellular Biochemistry.

Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds

A. di Pietro, S. Døskeland, L. Herfindal, 2015, Journal of Enzyme Inhibition and Medicinal Chemistry.

New, highly potent and non-toxic, chromone inhibitors of the human breast cancer resistance protein ABCG2.

A. di Pietro, Evelyn Winter, A. Boumendjel, 2016, European journal of medicinal chemistry.

Collateral sensitivity of resistant MRP1-overexpressing cells to flavonoids and derivatives through GSH efflux.

P. Carrupt, A. di Pietro, R. Terreux, 2014, Biochemical pharmacology.

Flavonoid structure-activity studies identify 6-prenylchrysin and tectochrysin as potent and specific inhibitors of breast cancer resistance protein ABCG2.

Francisco Gamarro, Francisco Muñoz-Martínez, S. Bates, 2005, Cancer research.

The linker region of breast cancer resistance protein ABCG2 is critical for coupling of ATP-dependent drug transport

S. Bates, A. di Pietro, R. Robey, 2015, Cellular and Molecular Life Sciences.

Pharmacokinetic interactions in mice between irinotecan and MBL‐II‐141, an ABCG2 inhibitor

A. di Pietro, J. Guitton, Myléne Honorat, 2017, Biopharmaceutics & drug disposition.

Dexamethasone down-regulates ABCG2 expression levels in breast cancer cells.

A. di Pietro, C. Dumontet, Myléne Honorat, 2008, Biochemical and biophysical research communications.

Mutations in the chloride-bicarbonate exchanger gene AE1 cause autosomal dominant but not autosomal recessive distal renal tubular acidosis.

A. di Pietro, R. Lifton, A. Nayır, 1998, Proceedings of the National Academy of Sciences of the United States of America.

A common mechanism for ATP hydrolysis in ABC transporter and helicase superfamilies.

G. Deléage, C. Geourjon, C. Blanchet, 2001, Trends in biochemical sciences.

RU49953: a non-hormonal steroid derivative that potently inhibits P-glycoprotein and reverts cellular multidrug resistance

J. M. Pérez-Victoria, A. di Pietro, S. Castanys, 2003, Cellular and Molecular Life Sciences CMLS.

Understanding polyspecificity within the substrate‐binding cavity of the human multidrug resistance P‐glycoprotein

A. di Pietro, G. Chang, Qinghai Zhang, 2014, The FEBS journal.

ABCG2 Transports and Transfers Heme to Albumin through Its Large Extracellular Loop*

A. di Pietro, P. Falson, O. Arnaud, 2010, The Journal of Biological Chemistry.

MRP8/ABCC11 Expression Is Regulated by Dexamethasone in Breast Cancer Cells and Is Associated to Progesterone Receptor Status in Breast Tumors

A. di Pietro, C. Dumontet, Myléne Honorat, 2011, International journal of breast cancer.

A Two-complementary Method Assay for Screening New Reversal Agents of Cancer Cell Multidrug Resistance

A. Chaboud, A. di Pietro, D. Barron, 2003 .

Three-dimensional structure by cryo-electron microscopy of YvcC, an homodimeric ATP-binding cassette transporter from Bacillus subtilis.

A. di Pietro, M. Chami, J. Jault, 2002, Journal of molecular biology.

Modulation by flavonoids of cell multidrug resistance mediated by P-glycoprotein and related ABC transporters

A. Goffeau, J. M. Pérez-Victoria, A. di Pietro, 2002, Cellular and Molecular Life Sciences CMLS.

P-glycoprotein-mediated resistance to chemotherapy in cancer cells: using recombinant cytosolic domains to establish structure-function relationships.

T. Krell, A. di Pietro, J. Jault, 1999, Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas.

Localization of putative binding sites for cyclic guanosine monophosphate and the anti-cancer drug 5-fluoro-2′-deoxyuridine-5′-monophosphate on ABCC11 in silico models

A. di Pietro, C. Dumontet, Myléne Honorat, 2013, BMC Structural Biology.

Pharmacological inhibition of LIM kinase stabilizes microtubules and inhibits neoplastic growth.

S. Knapp, A. di Pietro, C. Nguyen, 2012, Cancer research.

Use of trypsin to monitor conformational changes of mitochondrial adenosinetriphosphatase induced by nucleotides and phosphate.

A. di Pietro, D. Gautheron, C. Godinot, 1983, Biochemistry.

Role of phosphate on the ADP-induced hysteretic inhibition of mitochondrial adenosine 5'-triphosphatase. Effects of the natural protein inhibitor.

A. di Pietro, D. Gautheron, C. Godinot, 1986, Biochimica et biophysica acta.

Identification of specific reversal agents for Leishmania ABCI4-mediated antimony resistance by flavonoid and trolox derivative screening.

A. di Pietro, S. Castanys, F. Gamarro, 2014, The Journal of antimicrobial chemotherapy.

P-Glycoprotein 1 Affects Chemoactivities of Resveratrol against Human Colorectal Cancer Cells

D. Colin, A. di Pietro, Y. Artur, 2019, Nutrients.

Combination of Suboptimal Doses of Inhibitors Targeting Different Domains of LtrMDR1 Efficiently Overcomes Resistance of Leishmania spp. to Miltefosine by Inhibiting Drug Efflux

Maria Paola Costi, J. M. Pérez-Victoria, A. di Pietro, 2006, Antimicrobial Agents and Chemotherapy.

IF1 inhibition of mitochondrial F1-ATPase is correlated to entrapment of four adenine- or guanine-nucleotides including at least one triphosphate.

F. Penin, A. di Pietro, D. Gautheron, 1988, Biochemical and biophysical research communications.

Fate of nucleotides bound to reconstituted Fo-F1 during adenosine 5'-triphosphate synthesis activation or hydrolysis: role of protein inhibitor and hysteretic inhibition.

F. Penin, A. di Pietro, D. Gautheron, 1988, Biochemistry.

Functional nucleotide-binding domain in the F0F1-ATPsynthase alpha subunit from the yeast Schizosaccharomyces pombe.

F. Penin, R. Goody, A. di Pietro, 1993, Biochemistry.

The HPr Kinase from Bacillus subtilis Is a Homo-oligomeric Enzyme Which Exhibits Strong Positive Cooperativity for Nucleotide and Fructose 1,6-Bisphosphate Binding*

A. di Pietro, J. Deutscher, P. Gonzalo, 2000, The Journal of Biological Chemistry.

Structure-activity relationships for euphocharacins A-L, a new series of jatrophane diterpenes, as inhibitors of cancer cell P-glycoprotein.

A. di Pietro, C. Dumontet, G. Corea, 2004, Planta medica.

Modified jatrophane diterpenes as modulators of multidrug resistance from Euphorbia dendroides L.

A. di Pietro, C. Dumontet, G. Appendino, 2003, Bioorganic & medicinal chemistry.

The RNA polymerase I initiation site and the external transcribed spacer of the fission yeast Schizosaccharomyces pombe ribosomal RNA genes.

A. Goffeau, E. Balzi, A. di Pietro, 1985, Gene.

Glutamine 170 to tyrosine substitution in yeast mitochondrial F1 beta-subunit increases catalytic site interaction with GDP and IDP and produces negative cooperativity of GTP and ITP hydrolysis.

A. di Pietro, G. Divita, J. Jault, 1993, The Journal of biological chemistry.

Intrinsic tryptophan fluorescence of Schizosaccharomyces pombe mitochondrial F1-ATPase. A powerful probe for phosphate and nucleotide interactions.

G. Deléage, A. di Pietro, G. Divita, 1991, Biochemistry.

Overcoming Multidrug Resistance in Candida albicans: Macrocyclic Diterpenes from Euphorbia Species as Potent Inhibitors of Drug Efflux Pumps

Maria-José U. Ferreira, A. di Pietro, R. Prasad, 2016, Planta Medica.

A synthetic chalcone as a potent inducer of glutathione biosynthesis.

A. di Pietro, B. Day, A. Boumendjel, 2012, Journal of medicinal chemistry.

The multidrug resistance half-transporter ABCG2 is purified as a tetramer upon selective extraction from membranes.

A. di Pietro, S. Marco, P. Falson, 2010, Biochimica et biophysica acta.

Chemical modification of essential carboxyl group and histidine residue in the plasma-membrane 5'-nucleotidase.

A. di Pietro, J. Harb, D. Gautheron, 1986, Biochimica et biophysica acta.

Intrinsic tryptophan fluorescence of rat liver elongation factor eEF-2 to monitor the interaction with guanylic and adenylic nucleotides and related conformational changes.

A. di Pietro, G. Divita, D. Guillot, 1993, Biochemistry.

Microparticle-Mediated Transfer of the Viral Receptors CAR and CD46, and the CFTR Channel in a CHO Cell Model Confers New Functions to Target Cells

A. di Pietro, M. Chanson, P. Boulanger, 2012, PloS one.

A new P-glycoprotein inhibitor from the caper spurge (Euphorbia lathyris).

A. di Pietro, C. Dumontet, G. Appendino, 2003, Journal of natural products.

Potent competitive inhibition of drug binding to the Saccharomyces cerevisiae ABC exporter Pdr5p by the hydrophobic estradiol-derivative RU49953.

A. Goffeau, J. M. Pérez-Victoria, A. di Pietro, 2003, Biochimica et biophysica acta.

Protein kinase C effectors bind to multidrug ABC transporters and inhibit their activity.

A. Goffeau, J. M. Pérez-Victoria, A. di Pietro, 2001, Biochemistry.

Prenylated xanthones as potential P-glycoprotein modulators.

A. di Pietro, D. Barron, G. Conseil, 2000, Bioorganic & medicinal chemistry letters.

Binding of steroid modulators to recombinant cytosolic domain from mouse P-glycoprotein in close proximity to the ATP site.

A. di Pietro, E. Baulieu, P. Gros, 1997, Biochemistry.

Overexpression and purification of the carboxyl-terminal nucleotide-binding domain from mouse P-glycoprotein. Strategic location of a tryptophan residue.

A. di Pietro, L. Baggetto, H. Baubichon-Cortay, 1994, The Journal of biological chemistry.

Potent and fully noncompetitive peptidomimetic inhibitor of multidrug resistance P-glycoprotein.

A. di Pietro, C. Dumontet, P. Falson, 2010, Journal of medicinal chemistry.

Insect cell versus bacterial overexpressed membrane proteins: an example, the human ABCG2 transporter.

J. M. Pérez-Victoria, A. di Pietro, A. Pozza, 2010, Methods in molecular biology.

Masking of co‐operativity of nucleotide sites in pig heart mitochondrial ATPase (F1) by heating

A. di Pietro, D. Gautheron, C. Godinot, 1975, FEBS letters.

Metronomic administration of pegylated liposomal-doxorubicin in extensively pre-treated metastatic breast cancer patients: a mono-institutional case-series report.

D. Radice, A. di Pietro, A. Goldhirsch, 2010, Breast.