D. Barawkar

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Discovery of 3-hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles as potent MEK1 inhibitors.

C. Varaprasad, D. Barawkar, Hassan El Abdellaoui, 2006, Bioorganic & medicinal chemistry letters.

Identification of isothiazole-4-carboxamidines derivatives as a novel class of allosteric MEK1 inhibitors.

Shunqi Yan, C. Varaprasad, D. Barawkar, 2006, Bioorganic & medicinal chemistry letters.

A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives.

G. Bedse, S. Menon, A. Chugh, 2017, European journal of medicinal chemistry.

Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors.

S. Menon, D. Barawkar, Vishal V Pathade, 2012, Bioorganic & medicinal chemistry letters.

Triplex formation at physiological pH by oligonucleotides incorporating 5-Me-dC-(N4-spermine).

D. Barawkar, V. A. Kumar, K. Ganesh, 1994, Biochemical and biophysical research communications.

Modulation of DNA Triplex Stability Through Nucleobase Modifications

K. G. Rajeev, D. Barawkar, K. Ganesh, 1997 .

Effect of C5-amino substituent on 2′-deoxyuridine base pairing with 2′-deoxyadenosine: investigation by 1H and 13C NMR spectroscopy

D. Barawkar, K. Ganesh, R. K. Kumar, 1992 .

Synthesis, biophysical properties, and nuclease resistance properties of mixed backbone oligodeoxynucleotides containing cationic internucleoside guanidinium linkages: deoxynucleic guanidine/DNA chimeras.

D. Barawkar, T. C. Bruice, 1998, Proceedings of the National Academy of Sciences of the United States of America.

Synthesis of protected guanidinium linked dinucleoside incorporable into an oligonucleotide using solid phase DNA methodology.

D. Barawkar, T. C. Bruice, B. Linkletter, 1998, Bioorganic & medicinal chemistry letters.

Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain L-2-hydroxy acid oxidase.

A. Chugh, J. Vacca, D. Barawkar, 2012, Bioorganic & medicinal chemistry letters.

Highly efficient one-pot amination of carboxylate-substituted nitrogen-containing heteroaryl chlorides via Staudinger reaction

D. Barawkar, D. Bhuniya, P. Ramaiah, 2013 .

Dinucleotide Analogues as Novel Inhibitors of RNA-Dependent RNA Polymerase of Hepatitis C Virus

D. Barawkar, Z. Hong, W. Zhong, 2003, Antimicrobial Agents and Chemotherapy.

Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression.

A. Chugh, S. Chaudhary, D. Barawkar, 2017, ACS medicinal chemistry letters.

Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2's-hydroxy-3's-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors.

D. Barawkar, K. Mookhtiar, A. Raje, 2017, Bioorganic & medicinal chemistry.

Synthetic Control of DNA Triplex Structure through Chemical Modifications

D. Barawkar, K. Ganesh, Vaijayanti A. Kumar, 2007 .

Fluorescent d(CGCGAATTCGCG): characterization of major groove polarity and study of minor groove interactions through a major groove semantophore conjugate

Dinesh A. Barawkar, Krishna N. Ganesh, D. Barawkar, 1995, Nucleic Acids Res..

Synthesis of site-specific oligonucleotide-polyamine conjugates

D. Barawkar, T. P. Prakash, K. Ganesh, 1994 .

Triplex formation at physiological pH by 5-Me-dC-N4-(spermine) [X] oligodeoxynucleotides: non protonation of N3 in X of X*G:C triad and effect of base mismatch/ionic strength on triplex stabilities.

K. G. Rajeev, D. Barawkar, K. Ganesh, 1996, Nucleic acids research.

Exploring DNA minor groove interactions through a probe conjugate in major groove: fluorescence studies on netropsin complexation with dU-5-aminodansyl-DNA.

D. Barawkar, K. Ganesh, 1994, Biochemical and biophysical research communications.

5-Amido-(carboxyfluorescein)-2′-dU-oligonucloetides: Novel Primers for Fluorescent Detection of PCR Amplified DNA

D. Barawkar, V. Jadhav, K. Ganesh, 1997 .

Molecular Recognition of 5-Amino-dU in the Central Strand of a DNA Triplex: Formation of Triads AU(#):A in Parallel and GU(#):A in Antiparallel Motif(,).

D. Barawkar, K. Ganesh, V. S. Rana, 1996, The Journal of organic chemistry.

Solid phase synthesis of DNA containing 5-NH2-2′-deoxyuridine☆

D. Barawkar, K. Ganesh, 1993 .

Synthesis of substituted esters of imidazoles, oxazoles, thiazoles, and diethyl pyrazine-2,5-dicarboxylate from a common acyclic precursor employing C-formylation strategy

Santoshkumar N. Patil, D. Barawkar, R. Kulkarni, 2014 .

Discovery of 3-hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles as potent MEK1 inhibitors.

C. Varaprasad, D. Barawkar, Hassan El Abdellaoui, 2006, Bioorganic & medicinal chemistry letters.

Synthesis of Substituted Esters of Imidazoles, Oxazoles, Thiazoles, and Diethylpyrazine-2,5-dicarboxylate from a Common Acyclic Precursor Employing C-Formylation Strategy.

Santoshkumar N. Patil, D. Barawkar, R. Kulkarni, 2014 .

Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation.

G. Bedse, S. Menon, A. Chugh, 2017, Bioorganic & medicinal chemistry.

Potent and Selective Inhibitors of Long Chain l-2-Hydroxy Acid Oxidase Reduced Blood Pressure in DOCA Salt-Treated Rats.

A. Chugh, S. Chaudhary, J. Vacca, 2011, ACS medicinal chemistry letters.

Deoxynucleic Guanidines/PNA (DNG/PNA) Chimeras: Oligonucleoside Analogue Containing Cationic Guanidinium and Neutral Amide Linkages

D. Barawkar, T. C. Bruice, 1999 .

Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation.

S. Menon, S. Chaudhary, D. Barawkar, 2017, Journal of medicinal chemistry.

Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases.

S. Menon, A. Chugh, V. Karande, 2017, European journal of medicinal chemistry.

Polarity Sensing by Fluorescent Oligonucleotides: First Demonstration of Sequence-Dependent Microenvironmental Changes in the DNA Major Groove

D. Barawkar, V. Jadhav, K. Ganesh, 1999 .