V. Kauss

发表

Virtual Screening for Selective Allosteric mGluR1 Antagonists and Structure–Activity Relationship Investigations for Coumarine Derivatives

G. Schneider, Tobias Noeske, C. Parsons, 2007, ChemMedChem.

Positive and negative modulation of group I metabotropic glutamate receptors.

Ilya Pyatkin, Steffen Renner, Tanja Weil, 2008, Journal of medicinal chemistry.

Synergism of virtual screening and medicinal chemistry: identification and optimization of allosteric antagonists of metabotropic glutamate receptor 1.

G. Schneider, Tobias Noeske, C. Parsons, 2009, Bioorganic & medicinal chemistry.

Synthesis of 3,4-dihydro-2H-1,2-benzothiazine-3-carboxylic acid 1,1-dioxides and their evaluation as ligands for NMDA receptor glycine binding site

V. Kauss, U. Abel, Meik Sladek, 2016, Journal of enzyme inhibition and medicinal chemistry.

Application of the heck reaction for the synthesis of 1-alkoxyisoquinoline- 3-carboxylic acids esters

V. Kauss, K. Rubina, A. Ture, 2011 .

A Practical Synthesis of tert-Alkylamines via the Ritter Reaction with Chloroacetonitrile

A. Jirgensons, V. Kauss, I. Kalvinsh, 2000 .

Synthesis and structure-affinity relationships of 1,3, 5-alkylsubstituted cyclohexylamines binding at NMDA receptor PCP site.

C. Parsons, W. Danysz, A. Jirgensons, 2000, European journal of medicinal chemistry.

Evaluation of an enantioselective synthesis of 6-chloro-3,4-dihydro-2H-1,2-benzothiazine-3-carboxylic acid 1,1-dioxide and its derivatives

V. Kauss, U. Abel, Meik Sladek, 2015, Chemistry of Heterocyclic Compounds.

The synthesis of potential Neramexane metabolites: cis- and trans-3-amino-1,3,5,5-tetramethylcyclohexanecarboxylic acids

A. Jirgensons, D. Trifanova, V. Kauss, 2004 .

Pharmacological approaches to tackle NCLs.

V. Kauss, D. Medina, M. Dambrova, 2020 .

A convenient synthesis of 5β-cholestan-26-oic and 5β-cholestan-26,27-dioic acids

V. Kauss, P. Trapencieris, G. Jas, 2000, Steroids.

Spirocyclic betaines or 2-amino-Δ2-1,3,4-thiadiazoline-5-acetic acid and their rearrangement in acetic anhydride

V. Kauss, I. Kalvin'sh, 1993 .

Reactions of 1,1-dialkylthiosemicarbazides with propiolic acid and its esters

V. Kauss, A. Mishnev, I. Kalvin'sh, 1992 .

2-Amino-4,4-disubstituted-5-carboxymethyl-Δ2-1,3,4-oxadiazolin-4-ium chlorides and their recyclization in acetic anhydride

V. Kauss, I. Kalvin'sh, 1992 .

Structure of products of addition of thiosemicarbazides and thiosemicarbazones to acetylenedicarboxylic acid and its dimethyl ester

V. Kauss, É. Lukevits, É. Liepin'sh, 1990, Chemistry of Heterocyclic Compounds.

Amino-alkyl-cyclohexanes as a novel class of uncompetitive NMDA receptor antagonists.

C. Parsons, W. Danysz, A. Jirgensons, 2002, Current pharmaceutical design.

A Convenient Reagent for N-hydroxyguanylation

A. Jirgensons, V. Kauss, I. Kalvins, 1997 .

A novel class of amino-alkylcyclohexanes as uncompetitive, fast, voltage-dependent, N-methyl-D-aspartate (NMDA) receptor antagonists – in vitro characterization

C. Parsons, C. Jatzke, A. Jirgensons, 2007, Journal of Neural Transmission.

Unnatural Amino Acids. 1. A Facile Synthesis of the Methyl Ester of Aziridine-2-carboxylic Acid

V. Kauss, P. Trapencieris, I. Kalvins, 1997 .

Unnatural Amino Acids. Part 1. A Facile Synthesis of the Methyl Ester of Aziridine‐2‐carboxylic Acid.

V. Kauss, P. Trapencieris, I. Kalvins, 1997 .

Application of the heck reaction for the synthesis of 1-alkoxyisoquinoline- 3-carboxylic acids esters

V. Kauss, K. Rubina, A. Ture, 2011 .

Electron impact mass spectra of 2-hydrazono-1,3-thiazolidin-4-one derivatives

V. Kauss, É. Lukevits, I. Mazheika, 1990 .

Discovery, synthesis, and structure-activity relationships of 2-aminoquinazoline derivatives as a novel class of metabotropic glutamate receptor 5 negative allosteric modulators.

Bjoern A. Krueger, M. Hechenberger, V. Kauss, 2013, Bioorganic & medicinal chemistry letters.

A Practical Synthesis of tert-Alkylamines via the Ritter Reaction with Chloroacetonitrile

A. Jirgensons, V. Kauss, I. Kalvinsh, 2001 .