A. Vasella

发表

The structures of Salmonella typhimurium LT2 neuraminidase and its complexes with three inhibitors at high resolution.

S. Crennell, E. Garman, C. Philippon, 1996, Journal of molecular biology.

Oligosaccharide Analogues of Polysaccharides. Part 5. Studies on the cross‐coupling of alkynes and haloalkynes

A. Vasella, Chengzhi Cai, 1995 .

A sialic acid-derived phosphonate analog inhibits different strains of influenza virus neuraminidase with different efficiencies.

W G Laver, G. Air, M. Luo, 1995, Journal of molecular biology.

Deoxy‐nitrosugars. 16th Communication. Synthesis of N‐acetyl‐4‐deoxyneuraminic acid

A. Vasella, F. Baumberger, 1986 .

Orthogonally protected dialkynes

A. Vasella, A. Ernst, L. Gobbi, 1996 .

Synthesis, antiribosomal and antibacterial activity of 4′-O-glycopyranosyl paromomycin aminoglycoside antibiotics

H. Boukari, A. Vasella, E. Böttger, 2014 .

Influence of 4'-O-Glycoside Constitution and Configuration on Ribosomal Selectivity of Paromomycin.

A. Vasella, E. Böttger, Takahiko Matsushita, 2015, Journal of the American Chemical Society.

Synthesis of Spiropyrimidodiazepines and Spirodiazepinopurines by Tandem Nitroso-ene/Diels–Alder Reactions

A. Vasella, Fang-Li Zhang, 2007 .

A New Synthesis of Pteridines Substituted with Branched and Linear Alkenyl Groups at C(6). The Nitroso‐Ene Reaction of 4‐(Alkenoylamino)‐5‐nitrosopyrimidines

A. Vasella, W. Schweizer, Fang-Li Zhang, 2007 .

I Hydroxyl and Amino Groups Kanamycin Aminoglycosides: Role of Ring Structure-Activity Relationships among the

E. Westhof, A. Vasella, R. Akbergenov, 2014 .

Glycosylidene Carbenes. Part 21. Synthesis of N-tosylglycono-1,4-lactone hydrazones as precursors of glycofuranosylidene carbenes

A. Vasella, S. Mangholz, 1995 .

N-acetylglucosaminono-1,5-lactone oxime and the corresponding (phenylcarbamoyl)oxime. Novel and potent inhibitors of beta-N-acetylglucosaminidase.

M. Horsch, A. Vasella, D. Rast, 1991, European journal of biochemistry.

Determination of the gauche effect of 3-acetamido- and 3-acetoxy-piperidine and -tetrahydropyran by 1H-n.m.r. spectroscopy

A. Vasella, U. Piantini, B. Bernet, 1990 .

Identification and Evaluation of Improved 4′-O-(Alkyl) 4,5-Disubstituted 2-Deoxystreptamines as Next-Generation Aminoglycoside Antibiotics

H. Boukari, J. Schacht, A. Vasella, 2014, mBio.

Synthesis of paromomycin derivatives modified at C(5'') to selectively target bacterial rRNA.

A. Vasella, E. Böttger, Iwona Kudyba, 2007, Carbohydrate research.

Design and Synthesis of Aminoglycoside Antibiotics to Selectively Target 16S Ribosomal RNA Position 1408

A. Vasella, E. Böttger, R. Pathak, 2005 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 20

Fabio De Giacomo, A. Vasella, M. Peifer, 2009 .

Synthesis of Glycaro‐1,5‐lactams and Tetrahydrotetrazolopyridine‐5‐carboxylates: Inhibitors of β‐D‐Glucuronidase and α‐L‐Iduronidase

S. Withers, A. Vasella, B. Rempel, 2006 .

Synthesis of d-gluco-, l-ido-, d-galacto-, and l-altro-configured glycaro-1,5-lactams from tartaric acid

A. Vasella, Jagadish Pabba, 2005 .

6-(Diazomethyl)-1,3-bis(methoxymethyl)uracil, Synthesis and Transformation into Annulated Pyrimidinediones

A. Vasella, S. Rani, Fuyi Zhang, 2008 .

Interaction ofN-acetyl-4-, 7-, 8- or 9-deoxyneuraminic acids andN-acetyl-4-, 7- or 8-mono-epi- and-7,8-di-epineuraminic acids withN-acetylneuraminate lyase

E. Schreiner, A. Vasella, E. Zbiral, 1987, Glycoconjugate Journal.

Biological action of phosphonate analogs of fructose 2,6‐bisphosphate on enzymes from higher plants

M. Stitt, A. Vasella, 1988 .

Predictive Analysis of the Side Chain Conformation of the Higher Carbon Sugars: Application to the Preorganization of the Aminoglycoside Ring 1 Side Chain for Binding to the Bacterial Ribosomal Decoding A Site.

A. Vasella, S. Hobbie, M. G. Pirrone, 2020, The Journal of organic chemistry.

Stereospecific synthesis of methyl 2-amino-2-deoxy-(6S)-deuterio-α,β-d-glucopyranoside and methyl 2,6-diamino-2,6-dideoxy-(6R)-deuterio-α,β-d-glucopyranoside: Side chain conformations of the 2-amino-2-deoxy and 2,6-diamino-2,6-dideoxyglucopyranosides.

A. Vasella, Takayuki Kato, D. Crich, 2017, Carbohydrate research.

2‐Azido‐2‐deoxycellulose: Synthesis and 1,3‐Dipolar Cycloaddition

O. Dangles, A. Vasella, V. Bonnet, 2008 .

High Resolution X-ray Crystallography Shows That Ascorbate Is a Cofactor for Myrosinase and Substitutes for the Function of the Catalytic Base*

Bernard Henrissat, Wilhelm Pascal Burmeister, B. Henrissat, 2000, The Journal of Biological Chemistry.

Configurationally selective transition state analogue inhibitors of glycosidases. A study with nojiritetrazoles, a new class of glycosidase inhibitors

S. Withers, A. Vasella, K. Rupitz, 1993 .

Synthesis of a Glucose-Derived Tetrazole as a New β-Glucosidase Inhibitor. A New Synthesis of 1-Deoxynojirimycin

A. Vasella, P. Ermert, 1991 .

Effects of the 1- N-(4-Amino-2 S-hydroxybutyryl) and 6'- N-(2-Hydroxyethyl) Substituents on Ribosomal Selectivity, Cochleotoxicity, and Antibacterial Activity in the Sisomicin Class of Aminoglycoside Antibiotics.

J. Schacht, A. Vasella, E. Böttger, 2018, ACS infectious diseases.

Inhibition of O-GlcNAcase by a gluco-configured nagstatin and a PUGNAc-imidazole hybrid inhibitor.

A. Vasella, G. Davies, D. Vocadlo, 2006, Chemical communications.

Synthesis and Evaluation of Indolizine‐Type Inhibitors of N‐acetyl‐β‐D‐glucosaminidases

A. Vasella, T. Granier, Narendra Panday, 1998 .

Synthesis of Allosamidin

B. Trost, A. Vasella, D. Vranken, 1992 .

Inhibition of O‐GlcNAcase by a gluco‐Configured Nagstatin and a PUGNAc—Imidazole Hybrid Inhibitor.

A. Vasella, G. Davies, D. Vocadlo, 2007 .

Glycosylidene Carbenes. Part 22. α-D-Selectivity in the Glycosidation by Carbenes Derived from 2-Acetamido-hexoses

A. Vasella, C. Witzig, 1995 .

Temporary Protection and Activation in the Regioselective Synthesis of Saccharide Sulfates

A. Vasella, B. Bernet, S. Langston, 1994 .

Glycosylidene Carbenes. Part 14. Glycosidation of partially protected galactopyranose-, glucopyranose-, and mannopyranose-derived vicinal diols

A. Vasella, É. Bozó, B. Bernet, 1994 .

Glycosylidene Carbenes. Part 15. Synthesis of disaccharides from allopyranose-derived vicinal 1,2-diols. Evidence for the protonation by a H-bonded hydroxy group in the σ-plane of the intermediate carbene, followed by attack on the oxycarbenium ion in the π-plane

A. Vasella, B. Bernet, Pulla Reddy Muddasani, 1994 .

Synthesis of 1,2‐cis‐Configurated Glycosylphosphonates

A. Vasella, R. Meuwly, 1986 .

Synthesis of 2‐Acetamido‐2‐deoxy‐D‐gluconhydroximolactone‐ and Chitobionhydroximolactone‐Derived N‐Phenylcarbamates, Potential Inhibitors of β‐N‐Acetylglucosaminidase

A. Vasella, D. Rast, J. Maloisel, 1990 .

Synthesis of 1,2,3‐Triazole Analogues of Lincomycin

A. Vasella, S. Hobbie, E. Böttger, 2008 .

Synthesis and Antiribosomal Activities of 4'-O-, 6'-O-, 4″-O-, 4',6'-O- and 4″,6″-O-Derivatives in the Kanamycin Series Indicate Differing Target Selectivity Patterns between the 4,5- and 4,6-Series of Disubstituted 2-Deoxystreptamine Aminoglycoside Antibiotics.

A. Vasella, Takayuki Kato, Guanyu Yang, 2015, ACS infectious diseases.

Structure‐Activity Relationships for 5′′ Modifications of 4,5‐Aminoglycoside Antibiotics

A. Vasella, S. Hobbie, E. Böttger, 2022, ChemMedChem.

Synthesis of Benzimidazoles by Phosphine-Mediated Reductive Cyclisation of ortho-Nitro-anilides

A. Vasella, J. Duchek, 2011 .

Synthesis of Fused Triazoles as Probes for the Active Site of Retaining β‐Glycosidases: From Which Direction Is the Glycoside Protonated?

A. Vasella, T. Heightman, M. Locatelli, 1996 .

Importance of the 6′‐Hydroxy Group and Its Configuration for Apramycin Activity

A. Vasella, E. Böttger, D. Crich, 2014, ChemMedChem.

Design, Multigram Synthesis, and in Vitro and in Vivo Evaluation of Propylamycin: A Semisynthetic 4,5-Deoxystreptamine Class Aminoglycoside for the Treatment of Drug-Resistant Enterobacteriaceae and Other Gram-Negative Pathogens.

J. Schacht, A. Vasella, Takayuki Kato, 2019, Journal of the American Chemical Society.

Synthesis of glycosylphosphine oxides and related compounds

A. Vasella, A. Linden, B. Bernet, 1993 .

Glycosylidene Carbenes part 26. The intramolecular F…︁HO hydrogen bond of 1,3‐diaxial 3‐fluorocyclohexanols

A. Vasella, M. Biamonte, 1998 .

Mutagenesis of 16 S rRNA C 1409-G 1491 Base-pair Differentiates Between 6 0 OH and 6 0 NH 3 C Aminoglycosides

E. Westhof, A. Vasella, S. Hobbie, 2005 .

4‐Methylumbelliferyl 5‐Acetamido‐3,4,5‐trideoxy‐α‐D‐manno‐2‐nonulopyranosidonic Acid: Synthesis and Resistance to Bacterial Sialidases

A. Vasella, R. Schauer, F. Baumberger, 1986 .

SYNTHESIS OF A FULLERENE[60] CRYPTATE AND SYSTEMATIC LANGMUIR-BLODGETT AND THIN-FILM INVESTIGATIONS OF AMPHIPHILIC FULLERENE DERIVATIVES

F. Diederich, H. Ringsdorf, E. Harth, 1995 .

Synthesis of glycosyl phosphonates and related compounds

A. Vasella, L. Panza, G. Baudin, 1991 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 32: Thiomethylene- and Aminomethylene-Linked GG Dinucleosides of the ONIB Type: Formation of Quadruplexes

A. Vasella, D. Touboul, Daniel H. Egli, 2014 .

Oligonucleotide Analogues with Integrated Bases and Backbones. Part 26

A. Vasella, B. Bernet, Katja Chiesa, 2010 .

Glycosylidene Carbenes. Part 20. Synthesis of deprotected, spiro‐linked C‐glycosides of C60

E. Harth, A. Vasella, P. Uhlmann, 1994 .

Glycosylidene Carbenes. Part 9. Fullerene Sugars: Preparation of Enantiomerically Pure, Spiro-Linked C-Glycosides of C60.

F. Diederich, A. Vasella, C. Thilgen, 1993 .

Fullerene Sugars: Preparation of Enantiomerically Pure, Spiro‐Linked C‐Glycosides of C60

F. Diederich, A. Vasella, C. Thilgen, 1992 .

Oligosaccharide Analogues of Polysaccharides Part 23. Synthesis of a Dimeric Acetyleno Cyclodextrin from a Mannopyranose-Derived Dialkyne

A. Vasella, Jürgen Stichler-Bonaparte, 2001 .

Oligosaccharide Analogues of Polysaccharides. Part 4. Synthesis of a monosaccharide-derived octamer†

A. Vasella, J. Alzeer, 1995 .

Oligosaccharide Analogues of Polysaccharides. Part 3. A new protecting group for alkynes: Orthogonally protected dialkynes

A. Vasella, Chengzhi Cai, 1995 .

A Synthesis of 1D- and 1L-myo-Inositol 1,3,4,5,-Tetraphosphate

K. S. Swaminathan, A. Vasella, B. I. Glänzer, 1988 .

Glycosylidene Carbenes. Part 27. Glucosidation of titanium dioxide with 1-aziglucoses: Preparation and characterization of modified titanium-dioxide surfaces†

M. Textor, N. Spencer, A. Vasella, 1998 .

A structural view of the action of Escherichia coli (lacZ) beta-galactosidase.

B. Matthews, S. Withers, J. McCarter, 2001, Biochemistry.

Synthesis of Stable Dolichylphosphomannose Analogues

M. Aebi, A. Vasella, C. Frank, 2004 .

Synthesis and reactivity of a new glycosyl donor: O-(1-phenyltetrazol-5-yl) glucoside.

A. Vasella, M. Palme, 1994, Bioorganic & medicinal chemistry.

Probing the Interaction of the Hydroxy Group at C(4) of Lactone‐Type Inhibitors with β‐Glucosidases and β‐Galactosidases

A. Vasella, Jagadish Pabba, 2006 .

Synthesis of N‐Acetylglucosamine‐Derived Nagstatin Analogues and Their Evaluation as Glycosidase Inhibitors

A. Vasella, M. Terinek, 2005 .

Synthesis of Tetrahydropyridoimidazole‐2‐acetates: Effect of Carboxy and Methoxycarbonyl Groups at C(2) on the Inhibition of Some β‐ and α‐Glycosidases

A. Vasella, M. Terinek, 2004 .

Structure‐Activity Relations for Imidazo‐pyridine‐Type Inhibitors of β‐D‐Glucosidases

A. Vasella, T. Granier, Narendra Panday, 1997 .

d-Glyconhydroximolactams strongly inhibit α-glycosidases

S. Withers, A. Vasella, K. Rupitz, 1997 .

Synthesis and Enzymatic Evaluation of Substrates and Inhibitors of β‐Glucuronidases

A. Vasella, P. Weiss, R. Hoos, 1996 .

Synthesis of New Sialidase Inhibitors, 6‐Amino‐6‐Deoxysialic Acids

A. Vasella, R. Schauer, F. Baumberger, 1988 .

Deoxy‐nitrosugars. 17th communication. Synthesis of ketose‐derived nucleosides from 1‐deoxy‐1‐nitroribose

A. Vasella, K. Mahmood, B. Bernet, 1991 .

Inhibition of Emulsin by D‐Gluconhydroximo‐1,5‐lactone and Related Compounds

A. Vasella, Dieter Beer, 1986 .

Oligosaccharide analogues of polysaccharides. Part 14:. Carbocyclic cyclodextrin analogues. Synthesis of all trimeric and tetrameric isomers by homo‐ and heterocoupling of 1,4‐cis‐diethynylated 1,5‐anhydroglucitols

R. Bürli, A. Vasella, 1997 .

Cyclic “Acetylenosaccharides”—Novel Cyclodextrin Analogues

R. Bürli, A. Vasella, 1997 .

Oligosaccharide Analogues of Polysaccharides. Part 12. Synthesis of ‘acetyleno‐saccharide’‐derived cyclodextrin analogues

R. Bürli, A. Vasella, 1997 .

Oligosaccharide Analogues of Polysaccharides. Part 6. Orthogonal protecting/activating groups in an improved binomial synthesis of ‘acetyleno‐oligosaccharides’

A. Vasella, Chengzhi Cai, 1996 .

Deoxy‐nitrosugars. 5th Communication. The anomeric effect of the nitro group

A. Vasella, B. Aebischer, R. Hollenstein, 1983 .

Fragmentation of 6-deoxy-6-halo-hexono-1,5-ortholactones: a concerted, nonstereospecific process

A. Vasella, B. Bernet, 1984 .

Apralogs: Apramycin 5-O-Glycosides and Ethers with Improved Antibacterial Activity and Ribosomal Selectivity and Reduced Susceptibility to the Aminoacyltranserferase (3)-IV Resistance Determinant.

J. Schacht, A. Vasella, S. Hobbie, 2019, Journal of the American Chemical Society.

Crystal Structure of Glucooligosaccharide Oxidase from Acremonium strictum

A. Vasella, Y. Tsai, Chun-Hsiang Huang, 2005, Journal of Biological Chemistry.

Glycosylidene Carbenes. Part 9. Regioselective glycosidation of diols and triols: Intra‐ and intermolecular hydrogen bonds

A. Vasella, P. Uhlmann, 1992 .

Synthesis and evaluation in asymmetric hydrogenation of carbohydrate-derived 1,3-bisphosphines

A. Vasella, Chunbao Li, B. Bernet, 1992 .

Aldehyde‐Promoted Addition of 2‐(Trimethylsilyl)thiazole to α,α′‐Dialkoxy Ketones: A new way to branched‐chain monosaccharides

A. Vasella, M. Carcano, 1998 .

Regioselective synthesis of 1I,1II,5I,5II,6I,6I,6II,6II-2H8-cellobiose.

A. Vasella, Fuyi Zhang, 2007, Carbohydrate research.

Synthesis of anL-Fucose-Derived Cyclic Nitrone and its Conversion toα-L-Fucosidase Inhibitors

A. Vasella, Andreas Peer, 1999 .

Nucleophilic additions to N‐glycosylnitrones part IV Asymmetric synthesis of N‐hydroxy‐α‐aminophosphonic and α‐aminophosphonic acids

A. Vasella, R. Huber, 1987 .

Diastereoselectivity in the Reaction of N-Glycosyl-nitrones: 1,3-Dipolar Cycloaddition and Addition of Phosphite Anion

A. Vasella, B. Bernet, E. Krawczyk, 1985 .

4,5,6‐Trisubstituted Piperidinones as Conformationally Restricted Ceramide Analogues: Synthesis and Evaluation as Inhibitors of Sphingosine and Ceramide Kinases and as NKT Cell‐Stimulatory Antigens

A. Vasella, P. Nussbaumer, A. Billich, 2009, Chemistry & biodiversity.

Towards stable di-carba analogues of guanofosfocins

A. Vasella, J. Duchek, Mu-Hua Huang, 2011 .

Oligonucleotide Analogues with Integrated Bases and Backbones. Part 24

A. Vasella, B. Bernet, Katja Chiesa, 2010 .

Analogues of Sialic Acids as Potential Sialidase Inhibitors. Synthesis of C6 and C7 Analogues of N‐Acetyl‐6‐amino‐2,6‐dideoxyneuraminic Acid

A. Vasella, Z. Györgydeák, B. Bernet, 1991 .

Synthesis of New Sialidase Inhibitors, 6-Amino-6-deoxysialic Acids.

A. Vasella, R. Schauer, F. Baumberger, 1988 .

Synthesis of (2R,4S,5S)-5-Acetamido-4-hydroxypipecolinic Acid (II) as a Potential Inhibitor of Sialidases.

A. Vasella, R. Schauer, K. Clinch, 1988 .

Glyconothio‐O‐lactones. Part 2. Cycloaddition to Dienes, Diazomethane, and Carbenoids.

A. Vasella, B. Bernet, T. Maeder, 2010 .

Glyconothio-O-lactones Part II. Cycloaddition to Dienes, Diazomethane, and Carbenoids

A. Vasella, B. Bernet, T. Mäder, 1993 .

Intramolecular addition of nucleophilic carbenes to acceptor-substituted alkenyl groups : synthesis and transformation of homobenzofurans and synthesis of a homoindole

A. Vasella, Chunbao Li, 1993 .

Thermal Rearrangement of Azido Ketones into Oxazoles via Azirines: One-Pot, Metal-Free Heteroannulation to Functionalized 1,3-Oxazoles†

Amol G. Dikundwar, A. Vasella, T. Row, 2013 .

Deoxy‐nitrosugars. 11th Communication. Reactions of 1‐C‐nitroglycosyl halides and 1‐C‐nitroglycosyl sulfones with dialkyl‐phosphite anions: Nucleophilic attack vs. single‐electron transfer

A. Vasella, R. Meuwly, 1985 .

Fluorine-Decoupled Carbon Spectroscopy for the Determination of Configuration at Fully Substituted, Trifluoromethyl- and Perfluoroalkyl-Bearing Carbons: Comparison with 19F–1H Heteronuclear Overhauser Effect Spectroscopy

A. Vasella, Takayuki Kato, E. Böttger, 2015, The Journal of organic chemistry.

Synthesis, ribosomal selectivity, and antibacterial activity of netilmicin 4'-derivatives.

A. Vasella, E. Böttger, D. Crich, 2019, MedChemComm.

Substrate specificity engineering of beta-mannosidase and beta-glucosidase from Pyrococcus by exchange of unique active site residues.

W. D. de Vos, A. Vasella, J. van der Oost, 2002, Biochemistry.

Glycosidase mechanisms.

A. Vasella, G. Davies, M. Böhm, 2002, Current opinion in chemical biology.

Structural studies of the beta-glycosidase from Sulfolobus solfataricus in complex with covalently and noncovalently bound inhibitors.

A. Vasella, M. Rossi, G. Davies, 2004, Biochemistry.

Regioselective Benzoylation of 6-O-Protected and 4,6-O-Diprotected Hexopyranosides as Promoted by Chiral and Achiral Ditertiary 1,2-Diamines

A. Vasella, Guixian Hu, 2002 .

INHIBITION OF GLYCOSIDASES BY LACTAM OXIMES : INFLUENCE OF THE AGLYCON IN DISACCHARIDE ANALOGUES

A. Vasella, T. Heightman, S. Vonhoff, 1998 .

Deoxy‐nitrosugars 12th communication Synthesis of isosteric mono‐phosphonate analogues of β‐and α‐D‐fructose 2,6‐bisphosphate

A. Vasella, R. Meuwly, 1986 .

Carbasaccharides via Ring‐Closing Alkene Metathesis. A Synthesis of (+)‐Valienamine from D‐Glucose

A. Vasella, F. Sarabia, Peter Kapferer, 1999 .

Oligosaccharide Analogues of Polysaccharides. Part 7. Synthesis of a monosaccharide‐derived monomer for amylose and cyclodextrin analogues

R. Bürli, A. Vasella, 1996 .

Synthesis of a non-isosteric, isopolar monophosphonate analogue of β-d-fructose 2,6-bisphosphate

A. Vasella, A. Dessinges, 1988 .

Deoxy‐nitrosugars. 10th Communication. Synthesis of Isosteric Phosphonate Analogues of Ulose‐1‐Phosphates

A. Vasella, R. Julina, 1985 .

Synthesis of the 6‐C‐Methyl and 6‐C‐(Hydroxymethyl) Analogues of N‐Acetylneuraminic Acid and of N‐Acetyl‐2,3‐didehydro‐2‐deoxyneuraminic Acid

A. Vasella, R. Wyler, 1990 .

Deoxy‐Nitrosugars. Part 12. Synthesis of Isosteric Mono‐Phosphonate Analogues of β‐ and α‐D‐Fructose 2,6‐Bisphosphate,

A. Vasella, R. Meuwly, 1986 .

Deoxy‐nitrosugars. 6th communication. Stereoelectronic control in the reductive denitration of tertiary nitro ethers. A synthesis of ‘C‐glycosides’

A. Vasella, F. Baumberger, 1983 .

A new synthesis of N‐acetylneuraminic acid

A. Vasella, M. Hugener, R. Csuk, 1988 .

Synthesis of Enantiomerically Pure Carbohydrate‐Derived Annulated Cyclopentadienes and Ferrocenes

Zhi Li, A. Vasella, 1996 .

Nucleophilic Additions to N-Glycosylnitrones. Asymmetric Synthesis of α-Aminophosphonic Acids†‡

A. Vasella, J. Obrecht, A. Knierzinger, 1985 .

A laser flash photolysis derived study of a glycosylidene carbene

K. Briner, A. Vasella, M. Platz, 1991 .

The kinetic anomeric effect. Additions of nucleophiles and of dipolarophiles to N-glycosylnitrones and to N-pseudoglycosylnitrones

A. Vasella, R. Huber, 1990 .

Monocyclic, substituted imidazoles as glycosidase inhibitors

A. Vasella, P. Magdolen, 2005 .

Synthesis and Some Transformations of 2‐Acetamido‐5‐amino‐3,4,6‐tri‐O‐benzyl‐2,5‐dideoxy‐D‐glucono‐1,5‐lactam

A. Vasella, T. Granier, 1998 .

Synthesis of Naphtho[2,3‐b]pyrandiones: (−)‐Cryptosporin

A. Vasella, W. Brade, 1989 .

Enantioselective Synthesis of D‐erythro‐Sphingosine and of Ceramide

A. Vasella, T. Herzig, B. Bernet, 1986 .

Recent Insights into Inhibition, Structure, and Mechanism of Configuration-Retaining Glycosidases.

A. Vasella, T. Heightman, Tom D Heightman, 1999, Angewandte Chemie.

Functionalised Monocyclic Five- to Seven-Membered exo-Glycals by Alkynol Cycloisomerisation of Hydroxy Buta-1,3-diynes and 1-Haloalkynols

A. Vasella, Zhiwei Miao, Ming Xu, 2005 .

Convenient Synthesis of 2‐Azido‐2‐deoxy‐aldoses by Diazo Transfer

A. Vasella, J. L. Chiara, C. Witzig, 1991 .

Enantioselective synthesis of D-erythro-sphingosine

A. Vasella, B. Bernet, 1984 .

SYNTHESIS AND ENZYMATIC PHOSPHORYLATION OF A PHOTOACTIVATABLE DOLICHOL ANALOGUE

M. Aebi, A. Vasella, D. Grassi, 1997 .

Asymmetric synthesis of a new proline analogue

A. Vasella, R. Voeffray, 1981 .

Oligosaccharide Analogues of Polysaccharides. Part 15. Oligomers of Cellobiose-Derived Dialkynes and First Crystal Structure of an Anomeric Pair of Trichloroacetimidates.

A. Vasella, W. Schweizer, A. Ernst, 1999 .

An approach to the synthesis of polysaccharide analogues

A. Vasella, 1998 .

Oligosaccharide Analogues of Polysaccharides. Part 9. Synthesis and Thermolysis of Acetylenosaccharide‐Derived 1,2‐Dialkynylbenzenes

A. Vasella, B. Bernet, Jinwang Xu, 1996 .

Oligosaccharide Analogues of Polysaccharides. Part 2. Regioselective deprotection of monosaccharide‐derived monomers and dimers

A. Vasella, Andrea Vasella, Jawad Alzeer, 1995 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 13

A. Vasella, Xiaomin Zhang, B. Bernet, 2006 .

Synthesis of Enantiomerically Pure Ferrocenes from Glycofuranosyl‐cyclopentadienes, synthetic equivalents of (alkoxyalkyl)fulvenes

Zhi Li, A. Vasella, R. Chauvin, 1994 .

Synthesis of a Fusion‐Isomeric Cellobionoimidazole and Its Evaluation against the syn‐Protonating Glycosidase Cel7A

A. Vasella, B. Bernet, Narinder Mohal, 2005 .

Functionalised bicyclic exo-glycals by alkynol cycloisomerisation of hydroxy 1,3-diynes and hydroxy haloalkynes

A. Vasella, Zhiwei Miao, Ming Xu, 2005 .

The ‘t‐Amino Effect’ of ortho‐Nitroso Amines. Synthesis of 2,6‐Diaminoadenine Derivatives from 6‐(Dialkylamino)‐5‐nitrosopyrimidines

A. Vasella, M. D. Ruiz, 2011 .

Oligonucleotide Analogues with Integrated Bases and Backbone

A. Vasella, B. Bernet, A. Ritter, 2008 .

7‐Oxanorbornane and Norbornane Mimics of a Distorted β‐D‐Mannopyranoside: Synthesis and Evaluation as β‐Mannosidase Inhibitors

A. Vasella, Stephan Buser, 2005 .

Electrophilic bromination of N-acylated cyclohex-3-en-1-amines: Synthesis of 7-azanorbornanes

A. Vasella, Peter Kapferer, 2004 .

Synthesis of Galactose‐ and N‐Acetylglucosamine‐Derived Tetrazoles and their evaluation as β‐glycosidase inhibitors

A. Vasella, T. Heightman, P. Ermert, 1995 .

Oxidation of aldose oximes. Formation and structure of hydroxydiazene oxide acetals and preparation of hydroximolactones. X-Ray crystal structure of 2,3:5,6-di-O-isopropylidene-α-D-mannofuranosyl-ONN-azoxy 2,3:5,6-di-O-isopropylidene-α-D-mannofuranoside

A. Vasella, W. Schweizer, B. Aebischer, 1982 .

1H‐NMR Analysis of Intra‐ and Intermolecular H‐Bonds of Alcohols in DMSO: Chemical Shift of Hydroxy Groups and Aspects of Conformational Analysis of Selected Monosaccharides, Inositols, and Ginkgolides

A. Vasella, B. Bernet, 2000 .

Oligosaccharide Analogues of Polysaccharides

A. Vasella, B. Bernet, B. Hoffmann, 1998 .

β-Lactams fromD-Erythrose-Derived Imines: A Convenient Synthesis of 2,3-Diamino-2,3-dideoxy-D-mannonic-Acid Derivatives

A. Vasella, B. Bernet, T. Storz, 1999 .

Oligosaccharide Analogues of Polysaccharides. Part 3. A new protecting group for alkynes: Orthogonally protected dialkynes

A. Vasella, Chengzhi Cai, 1995 .

Synthesis of Monosaccharide-Derived Spirocyclic Cyclopropylamines and Their Evaluation as Glycosidase Inhibitors

A. Vasella, C. Ramana, Christian Blüchel, 2003 .

Conformationally Biased Mimics of Mannopyranosylamines: Inhibitors of β‐Mannosidases?

A. Vasella, L. Remeň, 2002 .

Synthesis, Antibacterial and Antiribosomal Activity of the 3C-Aminoalkyl Modification in the Ribofuranosyl Ring of Apralogs (5-O-Ribofuranosyl Apramycins)

A. Vasella, S. Hobbie, Dmitrijs Lubriks, 2022, Antibiotics.

Synthesis of N-Acetylallosamine-Derived Disaccharides

A. Vasella, Jean-Luc Maloisel, 1992 .

Glyconothio‐O‐lactones. Part III. Thermolysis of a 4,5‐Dihydro‐1,2,3‐ and a 2,5‐Dihydro‐1,3,4‐thiadiazole

A. Vasella, B. Bernet, T. Mäder, 1997 .

A New Synthesis of Pteridines

A. Vasella, Ming Xu, 2006 .

Glycosylidene Carbenes. Part 7. Neighbouring‐group participation by the 2‐benzyloxy group in the glycosidation of strongly acidic hydroxy compounds

A. Vasella, Yoshikazu Takahashi, 1992 .

Synthesis and evaluation of two mannosamine-derived lactone-type inhibitors of snail β-mannosidase

A. Vasella, M. Terinek, 2005 .

Sugar‐Derived Di‐ and Tetrahydropyridazinones: Synthesis of New Glycosidase Inhibitors

A. Vasella, C. Ramana, 2000 .

Preparation and Transmetallation of a Triphenylstannyl β-D-Glucopyranoside: A highly stereoselective route to β-D-C-glycosides via glycosyl dianions

A. Vasella, H. Kessler, V. Wittmann, 1994 .

Glycosylidene Carbenes. Part 3. Synthesis of Spirocyclopropanes

A. Vasella, Christian A. A. Waldraff, 1991 .

Diastereoselectivity and Reactivity in the Diels‐Alder Reactions of α‐Chloronitroso Ethers

A. Vasella, G. Kresze, R. Prewo, 1986 .

Asymmetric diels - alder reacrions with α-chloronitroso compounds- II. The use of a carbohydrate derived α-chloro-α-nitroso ether

A. Vasella, G. Kresze, H. Braun, 1984 .

A New Synthesis of Benzylidene Acetals

A. Vasella, Chunbao Li, 1993 .

Synthesis of glycosyl boranes and glycosyl borinates

A. Vasella, T. Rajamannar, W. Wenger, 1999 .

Glycosylidene Carbenes a new approach to glycoside synthesis. Part 1. Preparation of glycosylidene-derived diaziridines and diazirines†

K. Briner, A. Vasella, 1989 .

N-Monoalkylation of Tetra-O-benzyl-D-arabinonamide: Synthesis of Some Open-Chain Analogues ofN-Acetylneuraminic Acid and Their Evaluation as Sialidase Inhibitors

A. Vasella, T. Storz, 1998 .

Aldonhydroximo‐lactones. Preparation and Determination of Configuration

A. Vasella, Dieter Beer, 1985 .

Glyconothio-O-lactones. Part I. Preparation and reactions with nucleophiles

A. Vasella, B. Bernet, M. Hürzeler, 1993 .

Glycosylphosphonates of 2‐Amino‐2‐deoxy‐aldoses. Synthesis of a Phosphonate Analogue of Lipid X

K. Briner, A. Vasella, 1987 .

An improved procedure for the preparation of 8-substituted guanines.

A. Vasella, T. G. George, Ming Xu, 2003, Chemical communications.

Synthesis of (2R,4S,5S)-5-acetamido-4-hydroxy-pipecolinic acid as a potential inhibitor of sialidases

A. Vasella, R. Schauer, K. Clinch, 1987 .

Hydrogen Bonding of Fluorinated Saccharides in Solution: F Acting as H-Bond Acceptor in a Bifurcated H-Bond of 4-Fluorinated Levoglucosans†

A. Vasella, B. Bernet, 2007 .

Preparation of an Advanced Intermediate for the Synthesis of Stable Analogues of Guanofosfocin

A. Vasella, T. G. George, Y. Isshiki, 2004 .

Glycosylidene Carbenes. Part 13. Synthesis and thermolysis of representative 1‐azi‐glycoses

K. Briner, A. Vasella, L. Panza, 1993 .

Oligosaccharide Analogues of Polysaccharides. Part 1. Concept and synthesis of monosaccharide‐derived monomers

A. Vasella, Chengzhi Cai, J. Alzeer, 1995 .

A new approach to 5-thiosugars : 5-thio-D-gluconhydroximo-1,5-lactone, synthesis and evaluation as β-glucosidase inhibitor

A. Vasella, P. Ermert, 1993 .

Synthesis of N,N‐Disubstituted Lactone Hydrazones via (Sulfonylimino)‐ethers

A. Vasella, Stephan P. Fritschi, 1991 .

A Convenient Procedure for he Synthesis o 2,3,4,6-Tetra-O-benzyl-D-gluconolactam and D-Nojirilactam

A. Vasella, R. Hoos, Andrew B. J. Naughton, 1993 .

Synthesis of a Pseudodisaccharide α-C-Glycosidically Linked to an 8-Alkylated Guanine

A. Vasella, J. Duchek, Mu-Hua Huang, 2013, Molecules.

Oligosaccharide analogues of polysaccharides Part 26 Mimics of cellulose I and cellulose II : Di- and monoalkynyl c-cellosides of 1,8-disubstituted anthraquinones

A. Vasella, Tong Xie, B. Bernet, 2006 .

The structural basis of glycosidase inhibition by five-membered iminocyclitols: the clan a glycoside hydrolase endoglycoceramidase as a model system.

S. Withers, A. Vasella, N. Strynadka, 2007, Angewandte Chemie.

Synthesis of D‐ and L‐5‐Oxaproline and of a New Captopril Analogue

A. Vasella, R. Huguenin, J. Pless, 1983 .

Deoxy-nitrosugars. 4th communication†. Convenient synthesis of 1-deoxy-1-nitroaldoses

A. Vasella, B. Aebischer, 1983 .

Deoxy-nitrosugars, 7th communication Synthesis of methyl shikimate and of diethyl phosphashikimate from D-ribose†

A. Vasella, S. Mirza, 1984 .

Synthesis of a Glyoxalase I Inhibitor from Streptomyces griseosporeus NIIDAet OGASAWARA

A. Vasella, L. Molleyres, S. Mirza, 1985 .

Carbasaccharides via Ring-Closing Alkene Metathesis. A Synthesis of (+)-Valienamine from D-Glucose.

A. Vasella, F. Sarabia, Peter Kapferer, 1999 .

Synthesis of Fusion-Isomeric Imidazopyridines and Their Evaluation as Inhibitors of syn- and anti-Protonating Glycosidases

A. Vasella, Narinder Mohal, 2005 .

Glycosylidene Carbenes. Part 17. Glycosidation of benzyl β‐D‐ and β‐L‐ribopyranosides. Further evidence for the effect of stereoelectronic control on the regioselectivity of glycosidation

A. Vasella, P. Uhlmann, 1994 .

Structure-Based Design and Synthesis of Apramycin-Paromomycin Analogues: Importance of the Configuration at the 6'-Position and Differences between the 6'-Amino and Hydroxy Series.

A. Vasella, Takayuki Kato, S. Hobbie, 2017, Journal of the American Chemical Society.

A synthesis of N-acetylneuraminic acid and [6-2H]-N-acetylneuraminic acid from N-acetyl-D-glucosamine.

A. Vasella, R. Wyler, I. Müller, 1987, Carbohydrate research.

Deoxy‐nitrosugars 15th communication Synthesis of N‐acetylneuraminic acid and N‐acetyl‐4‐epineuraminic Acid

A. Vasella, F. Baumberger, 1986 .

DEOXY-NITROSUGARS. 10TH COMMUNICATION. SYNTHESIS OF ISOSTERIC PHOSPHONATE ANALOGS OF ULOSE-1-PHOSPHATES

A. Vasella, R. Julina, 1985 .

DEOXYNITROSUGARS. 7TH COMMUNICATION. SYNTHESIS OF METHYL SHIKIMATE AND OF DIETHYL PHOSPHASHIKIMATE FROM D-RIBOSE

A. Vasella, S. Mirza, 1984 .

N‐Acetylgucosaminono‐1,5‐lactone oxime and the corresponding (phenylcarbamoyl)oxime

M. Horsch, A. Vasella, D. Rast, 1991 .

Oligosaccharide Analogues of Polysaccharides. Part 8. Orthogonally Protected Cellobiose‐Derived Dialkynes. A Convenient Method for the Regioselective Bromo‐ and Protodegermylation of Trimethylgermyl‐ and Trimethylsilyl‐protected Dialkynes

A. Vasella, A. Ernst, 1996 .

Oligosaccharide Analogues of Polysaccharides. Part 7. Synthesis of a Monosaccharide-Derived Monomer for Amylose and Cyclodextrin Analogues.

A. Vasella, R. Buerli, 2010 .

Oligosaccharide Analogues of Polysaccharides Part 25

A. Vasella, B. Bernet, Jürgen Stichler-Bonaparte, 2002 .

O-(1-Phenyl-1H-tetrazol-5-yl) Glycosides: Alternative synthesis and transformation into glycosyl fluorides

A. Vasella, M. Palme, 1995 .

Synthesis and Evaluation of Paromomycin Derivatives Modified at C(4

A. Vasella, E. Böttger, R. Pathak, 2008 .

Phosphonic‐Acid Analogues of the N‐Acetyl‐2‐deoxyneiiraniinic Acids: Synthesis and Inhibition of Vibrio cholerae Sialidase

A. Vasella, K. Wallimann, 1990 .

Glycosylidene Carbenes. Part 16. Glycosidation of methyl 6‐O‐trityl‐α‐D‐altropyranoside

A. Vasella, E. Bozo, 1994 .

Analogues of Sialic Acids as Potential Sialidase Inhibitors Synthesis of 2‐C‐Hydroxymethyl Derivatives of N‐Acetyl‐6‐amino‐2,6‐dideoxy‐neuraminic Acid

A. Vasella, B. Bernet, A. B. Murty, 1990 .

Synthesis and Evaluation as Irreversible Glycosidase Inhibitors of Mono‐ and Oligo(glycosylthio)benzoquinones

S. Withers, A. Vasella, M. Schnabelrauch, 1994 .

Glycosylidene Carbenes. Part 18. Insertion of glycosylidene carbenes into the SnH bond of tributyl- and triphenylstannane: A synthesis of stannoglycosides

D. Nanz, A. Vasella, É. Bozó, 1994 .

Glycosylidene Carbenes Part 12. A new synthesis and some reactions of spirooxiranes

A. Vasella, P. Dhar, C. Witzig, 1993 .

Glycosylidene Carbenes. Part 10. Regioselective Glycosidation of 4,6‐O‐Benzylidene‐D‐altropyranosides

A. Vasella, É. Bozó, E. Bozo, 1992 .

Towards the Synthesis of 1‐Deoxy‐1‐nitropiperidinoses

A. Vasella, Marie-Pierre Collin, 2010 .

Synthesis and Evaluation of S- and C(1)-Substituted Analogues of Lincomycin

A. Vasella, S. Hobbie, E. Böttger, 2009 .

N-(4-nitrophenyl)oxamic acid and related N-acylanilines are non-competitive inhibitors of Vibrio cholerae sialidase but do not inhibit Trypanosoma cruzi or trypanosoma brucei trans-sialidases

A. Vasella, M. Engstler, A. Parodi, 1994 .

Synthesis of a phosphonic acid analogue of N-acetyl-2,3-didehydro-2-deoxyneuraminic acid, an inhibitor of Vibrio cholerae sialidase

A. Vasella, R. Wyler, 1991 .

Synthesis of the 6-C-Methyl and 6-C-(Hydroxymethyl) Analogues of N-Acetylneuraminic Acid and of N-Acetyl-2,3-didehydro-2-deoxyneuraminic Acid.

A. Vasella, R. Wyler, 1990 .

Synthesis of Pyrano(3,2-b)(1)benzopyrans from 1-Nitroglycals.

A. Vasella, W. Brade, 1991 .

Deoxynitro Sugars. Part 13. Preparation of Unprotected and Partially Protected 1-Deoxy-1-nitro-D-aldoses and Some Representative X-Ray Structure Analyses.

A. Vasella, I. Macher, R. Prewo, 1986 .

Glycosylidene Carbenes. Part 6. Synthesis of alkyl and fluoroalkyl glycosides

K. Briner, A. Vasella, 1992 .

DEOXYNITROSUGARS. PART 3. SYNTHESIS OF KETOSES BY CHAIN ELONGATION OF 1-DEOXY-1-NITROALDOSES. NUCLEOPHILIC ADDITIONS AND SOLVOLYSIS OF NITRO ETHERS

A. Vasella, B. Aebischer, R. Prewo, 1983 .

DEOXYNITROSUGARS. 9TH COMMUNICATION. CHAIN ELONGATION OF 1-C-NITROGLYCOSYL HALIDES BY SUBSTITUTION WITH SOME WEAKLY BASIC CARBANIONS

A. Vasella, B. Aebischer, R. Meuwly, 1985 .

Deoxy‐nitrosugars 8th communication Convenient preparation of 1‐C‐nitroglycosyl chlorides. Halonitro ethers from hydroxy oximes

A. Vasella, R. Meuwly, 1984 .

A Comparison of Glucose- and Glucosamine-Related Inhibitors: Probing the Interaction of the 2-Hydroxy Group with Retaining beta-Glucosidases

A. Vasella, M. Meyyappan, Narendra Panday, 2000 .

Synthesis ofgluco-Configured Tetrahydroimidazopyridine-2phosphonate-Derived Lipids, Potential Glucosyl Transferase Inhibitors

A. Vasella, I. Billault, 1999 .

DEOXYNITROSUGARS. THE 6TH COMMUNICATION. STEREOELECTRONIC CONTROL IN THE REDUCTIVE DENITRATION OF TERTIARY NITRO ETHERS. A SYNTHESIS OF ′C-GLYCOSIDES′

A. Vasella, F. Baumberger, 1984 .

Glycosylidene Carbenes, Part 29 , Insertion into B−C and Al−C Bonds: Glycosylborinates, ‐boranes, and ‐alanes

A. Vasella, W. Wenger, 2000 .

Synthesis and Evaluation as Glycosidase Inhibitors of 1H‐Imidazol‐2‐yl C‐Glycopyranosides

A. Vasella, T. Granier, 1995 .

A New Synthesis of N-Acetylneuraminic Acid.

A. Vasella, M. Hugener, R. Csuk, 1988 .

Synthesis of 7‐Aza‐ and 7‐Thiasphingosines, and Evaluation of Their Interaction with Sphingosine Kinases and with T‐Cells

A. Vasella, P. Nussbaumer, A. Billich, 2009, Chemistry & biodiversity.

Synthesis of 7‐Oxasphingosine and ‐ceramide Analogues and Their Evaluation in a Model for Apoptosis

A. Vasella, P. Canonico, R. Rajan, 2004, Chemistry & biodiversity.

Synthesis of Potential Glucosidase‐Inhibitors: D‐Xylopyranoside‐5‐spiro‐l′‐cyclopropanes

A. Vasella, L. Molleyres, R. Huber, 1990 .

Oligonucleotide Analogues with a Nucleobase-Including Backbone. Part 5. 2'-Deoxy-8-(hydroxymethyl)adenosine- and 2'-Deoxy-6-(hydroxymethyl)uridine-Derived Phosphoramidites: Synthesis and Incorporation into 14-Mer DNA Strands

A. Vasella, Werngard Czechtizky, 2001 .

Synthesis of Enantiomerically Pure Carbohydrate‐Derived Annulated Cyclopentadienes and of a Ferrocene.

A. Vasella, B. Bernet, Christoph Widauer, 2010 .

SYNTHESIS OF ENANTIOMERICALLY PURE CARBOHYDRATE DERIVED ANNULATED CYCLOPENTADIENES AND OF A FERROCENE

A. Vasella, B. Bernet, Christoph Widauer, 1998 .

Nucleophilic Additions to N‐Glycosylnitrones. Part 4. Asymmetric Synthesis of N‐Hydroxy‐α‐aminophosphonic and α‐Aminophosphonic Acids.

A. Vasella, R. Huber, 1987 .

NUCLEOPHILIC ADDITIONS TO N-GLYCOSYLNITRONES. ASYMMETRIC SYNTHESIS OF α-AMINOPHOSPHONIC ACIDS

A. Vasella, J. Obrecht, A. Knierzinger, 1985 .

L‐Erythruronic Acid Derivatives as Building Blocks for Nucleoside Analogs. Synthesis of 4′‐C‐Aryl‐D‐ribonucleosides

A. Vasella, R. Meuwly, Dieter Beer, 1982 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 27

A. Vasella, R. Kälin, B. Bernet, 2011 .

Synthesis and Incorporation of C(5′)-Ethynylated Uracil-Derived Phosphoramidites into RNA

A. Vasella, M. Christen, S. Eppacher, 2004 .

A MULTICOMPONENT ONE-POT REACTION INTEGRATING A BIS-FUNCTIONAL CARBOHYDRATE DERIVATIVE

A. Vasella, H. Wessel, Michael Justus, 1999 .

Oligonucleotide Analogues with Integrated Bases and Backbones. Part 23

A. Vasella, N. Bogliotti, B. Bernet, 2010 .

Synthesis and Evaluation of N‐Acetyl‐2‐amino‐2‐deoxy‐α‐D‐galactosyl 1‐Thio‐7‐oxaceramide, a New Analogue of α‐D‐Galactosyl Ceramide

A. Vasella, P. Nussbaumer, G. Libero, 2009 .

Synthesis and Evaluation of Sphingolipid Analogues

A. Vasella, P. Nussbaumer, A. Billich, 2009, Chemistry & biodiversity.

Oligonucleotide Analogues with Integrated Bases and Backbones. Part 19.: Gelation of Organic Solvents by Self-Complementary A*[s]U(*)Dinucleosides

A. Vasella, N. Bogliotti, Séverine Hebbe, 2008 .

Intra- and intermolecular H-bonds of alcohols in DMSO. 1H-NMR analysis of inter-residue H-bonds in selected oligosaccharides: cellobiose, lactose, N,N′-diacetylchitobiose, maltose, sucrose, agarose, and hyaluronates.

A. Vasella, B. Bernet, 2000 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 17

A. Vasella, Daniel H. Egli, B. Bernet, 2008 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 14

A. Vasella, Xiaomin Zhang, B. Bernet, 2007 .

Oligonucleosides with a nucleobase-including backbone; synthesis and self-association of novel dinucleotide analogues.

A. Vasella, P. Bhardwaj, A. J. Matthews, 2003, Chemical communications.

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 30

A. Vasella, Siji Thomas, B. Bernet, 2013 .

Oligonucleotide Analogues with Integrated Bases and Backbone (ONIB). Part 31

A. Vasella, D. Touboul, B. Bernet, 2014 .

Oligonucleotide analogues with integrated bases and backbone Part 15 Synthesis and association of ethenylene-linked self-complementary dimers

A. Vasella, Xiaomin Zhang, B. Bernet, 2007 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 16

A. Vasella, Xiaomin Zhang, B. Bernet, 2007 .

Oligonucleotide Analogues with Integrated Bases and Backbones. Part 25

A. Vasella, N. Bogliotti, 2010 .

Stereoselectivity of Ins(1,3,4,5)P4 recognition sites: implications for the mechanism of the Ins(1,3,4,5)P4-induced Ca2+ mobilization.

A. Vasella, R. Challiss, B. Potter, 1993, The Biochemical journal.

Selenium dioxide oxidations of olefins. Trapping of the allylic seleninic acid intermediate as a seleninolactone

A. Vasella, K. Sharpless, D. Arigoni, 1973 .

Synthesis and Reactivity in [3+2] Cycloadditions of Isoxanthopterin N(5)-Oxides – A New Synthesis of 6-Substituted Pteridinediones

A. Vasella, T. Steinlin, Tiziana Sonati, 2008 .

Synthesis and Enzyme-Inhibition Studies of Phenylsemicarbazones derived from D-glucono-1,5-lactone and 2-acetamido-2-deoxy-D-glucono-1,5-lactone

A. Vasella, M. Peter, F. Schweikart, 1992 .

Selenium dioxide oxidations of olefins. Trapping of the allylic seleninic acid intermediate as a seleninolactone

A. Vasella, D. Arigoni, K. B. Sharpless, 1973 .

Mechanism of the Reductive Half-reaction in Cellobiose Dehydrogenase*

C. Divne, G. Pettersson, A. Vasella, 2003, The Journal of Biological Chemistry.

An Advanced Apralog with Increased in vitro and in vivo Activity toward Gram‐negative Pathogens and Reduced ex vivo Cochleotoxicity

J. Schacht, A. Vasella, S. Hobbie, 2020, ChemMedChem.

Modification at the 2′-Position of the 4,5-Series of 2-Deoxystreptamine Aminoglycoside Antibiotics To Resist Aminoglycoside Modifying Enzymes and Increase Ribosomal Target Selectivity

A. Vasella, S. Hobbie, S. Mondal, 2019, ACS infectious diseases.

Synthesis of saccharocin from apramycin and evaluation of its ribosomal selectivity.

A. Vasella, S. Hobbie, D. Crich, 2019, MedChemComm.

D-gluconhydroximo-1,5-lactam and related N-arylcarbamates : theoretical calculations, structure, synthesis, and inhibitory effect on β-glucosidases

S. Withers, A. Vasella, W. Thiel, 1993 .

Very Strong Inhibition of Glucosidases by C(2)‐Substituted Tetrahydroimidazopyridines.

A. Vasella, Y. Canac, Narendra Panday, 2000 .

Very Strong Inhibition of Glucosidases by C(2)-Substituted Tetrahydroimidazopyridines

A. Vasella, Y. Canac, Narendra Panday, 2000 .

Glycosidase inhibition: an assessment of the binding of 18 putative transition-state mimics.

David Zechel, A. Vasella, G. Davies, 2007, Journal of the American Chemical Society.

Structural, kinetic, and thermodynamic analysis of glucoimidazole-derived glycosidase inhibitors.

A. Vasella, M. Rossi, G. Davies, 2006, Biochemistry.

Cyclopentanes from N-amino-glyconolactams. A synthesis of mannostatin A.

A. Vasella, C. Ramana, M. Zimmermann, 2003, Chemical communications.

Synthesis via a Carbohydrate‐Derived Münchnone of Pyrrolopyridines (Indolizines) and imidazopyridines, and their evaluation as inhibitors of β‐D‐glucosidases

A. Vasella, Lukas Hintermann, T. Granier, 1997 .

A Comparison of Glucose‐ and Glucosamine‐Related Inhibitors. Probing the Interaction of the 2‐Hydroxy Group with Retaining ‐Glucosidases.

A. Vasella, M. Meyyappan, Narendra Panday, 2000 .

Synthesis of Pyrrolidine Analogues of N-Acetylneuraminic Acid as Potential Sialidase Inhibitors

A. Vasella, L. Czollner, J. Kuszmann, 1990 .

Lateral Protonation of a Glycosidase Inhibitor. Structure of the Bacillus agaradhaerens Cel5A in Complex with a Cellobiose-Derived Imidazole at 0.97 A Resolution

A. Vasella, G. Davies, M. Schülein, 1999 .

Glycosylidene Carbenes. Part 4. Synthesis of Spirocyclopropanes from Acetamidoglycosylidene-Derived Diazirines

A. Vasella, C. Witzig, R. Husi, 1991 .

Synthesis of 2-azabicyclo[3.2.2]nonane-derived monosaccharide mimics and their evaluation as glycosidase inhibitors

A. Vasella, Stephan Buser, 2006 .

Synthesis of Pyrrolidine Analogues of N-Acetylneuraminic Acid as Potential Sialidase Inhibitors.

A. Vasella, L. Czollner, J. Kuszmann, 1990 .

Synthesis of Glucuronic, Mannuronic, and Galacturonic Acid‐Derived Imidazoles as Inhibitors of Bovine Liver β‐Glucuronidase

A. Vasella, Jagadish Pabba, Narinder Mohal, 2006 .

Synthesis and Oxidation of N‐Aminoglyconolactams: A Synthesis of Mannostatin A

A. Vasella, Guixian Hu, 2004 .

Three-dimensional Structure of the Barley β-d-Glucan Glucohydrolase in Complex with a Transition State Mimic*

Brian J. Smith, J. Varghese, A. Vasella, 2004, Journal of Biological Chemistry.

Structural and biochemical evidence for a boat-like transition state in beta-mannosidases.

Claire Dumon, A. Vasella, L. Tailford, 2008, Nature chemical biology.

CARBOCYCLIC COMPOUNDS FROM MONOSACCHARIDES. I. TRANSFORMATIONS IN THE GLUCOSE E SERIES

A. Vasella, B. Bernet, 1979 .

Synthesis of New C(2)-Substituted gluco-Configured Tetrahydroimidazopyridines and Their Evaluation as Glucosidase Inhibitors

A. Vasella, Bhagavathy Shanmugasundaram, 2005 .

Structures of Phanerochaete chrysosporium Cel7D in complex with product and inhibitors

J. Ståhlberg, A. Vasella, I. Muñoz, 2005, The FEBS journal.

β-Glycosidase inhibitors mimicking the pyranoside boat conformation

A. Vasella, E. Lorthiois, M. Meyyappan, 2000 .

Stereospecific synthesis of methyl 2-amino-2,4-dideoxy-6S-deuterio-α-D-xylo-hexopyranoside and methyl 2-amino-2,4-dideoxy-6S-deuterio-4-propyl-α-d-glucopyranoside: Side chain conformation of the novel aminoglycoside antibiotic propylamycin.

A. Vasella, Takahiko Matsushita, D. Crich, 2020, Carbohydrate research.

A 1H-NMR SPECTROSCOPIC INVESTIGATION OF THE CONFORMATION OF THE ACETAMIDO GROUP IN SOME DERIVATIVES OF N-ACETYL-D-ALLOSAMINE AND -D-GLUCOSAMINE

A. Vasella, P. Fowler, B. Bernet, 1996 .

Glycosylidene Carbenes. Part 24 Reactivity modulation by protecting groups of the addition of glycosylidene carbenes to electron‐rich alkenes

A. Vasella, B. Bernet, Christian A. A. Waldraff, 1997 .

Glycosylidene Carbenes. Part 8. Crystal Structure of a Cyclic, N‐Acetylallosamine‐Derived Alkoxy‐alkyl‐diazirine

A. Vasella, A. Linden, C. Witzig, 1992 .

New reactions and intermediates involving the anomeric center

A. Vasella, 1991 .

Glycosylidene Carbenes. Part 2. Synthesis of O‐Aryl Glycosides

K. Briner, A. Vasella, 1990 .

AN ADVANTAGEOUS SYNTHESIS OF 1D- AND 1L-1,2,3,5/4-CYCLOHEXANEPENTOL

A. Vasella, M. Biamonte, 1998 .

Norbornane Mimics of Distorted β‐D‐Glucopyranosides – Inhibitors of β‐D‐Glucopyranosidases?

A. Vasella, Stephan Buser, 2006 .

The active site of cellobiohydrolase Cel6A from Trichoderma reesei: the roles of aspartic acids D221 and D175.

G. Kleywegt, T. Reinikainen, J. Zou, 2002, Journal of the American Chemical Society.

Glycosylidene Carbenes. Part 23. Regioselective glycosidation of deoxy- and fluorodeoxy-myo-inositol derivatives†

A. Vasella, B. Bernet, A. Zapata, 1996 .

Glycosylidene Carbenes. Part 19. Regioselective glycosidation of allyl 2-deoxy-2-phthalimido-D-allopyranosides

K. Briner, A. Vasella, B. Bernet, 1994 .

Cooperative Interactions of the Catalytic Nucleophile and the Catalytic Acid in the Inhibition of β-Glycosidases. Calculations and their validation by comparative kinetic and structural studies of the inhibition of glycogen phosphorylase b

Spyros E. Zographos, Katerina E. Tsitsanou, S. Zographos, 1998 .

Diastereoselektive Diels-Alder-Reaktionen mit α-Chlornitrososacchariden

A. Vasella, F. Schmidtchen, G. Kresze, 1993 .

Synthesis via a Carbohydrate‐Derived Muenchnone of Pyrrolopyridines ( Indolizines) and Imidazopyridines, and Their Evaluation as Inhibitors of β‐D‐Glucosidases.

A. Vasella, Lukas Hintermann, T. Granier, 1997 .

Diastereoselective Diels‐Alder Reactions with α‐Chloronitroso Saccharides.

A. Vasella, F. Schmidtchen, R. Prewo, 1993 .

Structural determinants of substrate specificity in family 1 beta-glucosidases: novel insights from the crystal structure of sorghum dhurrinase-1, a plant beta-glucosidase with strict specificity, in complex with its natural substrate.

B. Henrissat, A. Vasella, D. Bevan, 2004, The Journal of biological chemistry.

An Improved Synthesis of 2-Acetamido-2-deoxy-D-gluconohydroximolactone (PUGNAc), A Strong Inhibitor ofβ-N-Acetylglucosaminidases

A. Vasella, Halasyam Mohan, 2000 .

4′-O-substitutions determine selectivity of aminoglycoside antibiotics

H. Boukari, V. Ramakrishnan, A. Vasella, 2014, Nature Communications.

Influence of ring size in conformationally restricted ring I analogs of paromomycin on antiribosomal and antibacterial activity.

A. Vasella, S. Hobbie, E. Böttger, 2021, RSC medicinal chemistry.

Oligonucleosides with a nucleobase-including backbone. Part 12: Synthesis of mixed ethynylene-linked uridine- and adenosine-derived tetramers

T. Knöpfel, A. Vasella, P. Bhardwaj, 2004 .

An Improved Synthesis of 2‐Acetamido‐2‐deoxy‐D‐gluconohydroximolactone (PUGNAc), a Strong Inhibitor of β‐N‐Acetylglucosaminidases.

A. Vasella, Halasyam Mohan, 2000 .

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 22

B. Jaun, A. Vasella, B. Bernet, 2009 .

N6', N6''', and O4' Modifications to Neomycin Affect Ribosomal Selectivity without Compromising Antibacterial Activity.

A. Vasella, S. Hobbie, E. Böttger, 2017, ACS infectious diseases.

Dissociation of antibacterial activity and aminoglycoside ototoxicity in the 4-monosubstituted 2-deoxystreptamine apramycin

J. Xie, J. Schacht, V. Ramakrishnan, 2012, Proceedings of the National Academy of Sciences.

Engineering the rRNA decoding site of eukaryotic cytosolic ribosomes in bacteria

A. Vasella, S. Hobbie, E. Böttger, 2007, Nucleic acids research.

Synthesis of a Pseudotrisaccharide Suitable for Synthesis of Ring I Modified 4,5-2-Deoxystreptamine Type Aminoglycoside Antibiotics.

A. Vasella, D. Crich, A. Sonousi, 2020, The Journal of organic chemistry.

Oligonucleosides with a Nucleobase-Including Backbone. Part 12

A. Vasella, P. Bhardwaj, 2002 .

Acylation of a 6-(Methylamino)-5-nitrosopyrimidine and 1,3-Dipolar Cycloaddition of an 8-Methylisoxanthopterin N(5)-Oxide. Synthesis of C(6) ,N(8)-Disubstituted Isoxanthopterins

A. Vasella, T. Steinlin, 2009 .

Synthesis of Tetrahydropyridoimidazole-2-acetates: Effect of Carboxy and Methoxycarbonyl Groups at C(2) on the Inhibition of Some β- and α-Glycosidases.

A. Vasella, M. Terinek, 2005 .

Improved Access to Imidazole-phosphonic Acids: Synthesis of D-manno-Tetrahydroimidazopyridine-2-phosphonates†

A. Vasella, M. Terinek, 2004 .

Ene reactions with α‐chloronitroso compounds: Asymmetric synthesis of N‐allylhydroxylamines

A. Vasella, A. Ritter, G. Kresse, 2010 .

Carbocyclic Analogues of N-Acetyl-2,3-didehydro-2-deoxy-D-neuraminic Acid (Neu5Ac2en, DANA): Synthesis and Inhibition of Viral and Bacterial Neuraminidases.

A. Vasella, S. Vorwerk, 1998, Angewandte Chemie.

Aggregation of yeast cells: direct measurement of discrete lectin-carbohydrate interactions.

A. Vasella, A. Touhami, Y. Dufrêne, 2003, Microbiology.

Oligosaccharide Analogues of Polysaccharides, Part 16, Cross‐Coupling of Partially Protected Dialkynyl Monosaccharides

R. Beaudegnies, A. Vasella, Tanja Verena Bohner, 1999 .

Oligonucleosides with a Nucleobase‐Including Backbone, Part 3, Synthesis of Acetyleno‐Linked Adenosine Dimers

A. Vasella, H. Gunji, 2000 .

A New Synthesis of Ciliapterin and Dictyopterin. Ene Reactions of (Alkenylamino)-nitroso-pyrimidines

A. Vasella, Fang-Li Zhang, 2008 .

Probing the Conformational Changes in the Enzymatic Hydrolysis of 2‐Acetamido‐2‐deoxy‐β‐D‐glucopyranosides

A. Vasella, M. Böhm, 2004 .

Structure-Activity Relationships among the Kanamycin Aminoglycosides: Role of Ring I Hydroxyl and Amino Groups

E. Westhof, A. Vasella, E. Böttger, 2012, Antimicrobial Agents and Chemotherapy.

Channels at the catalytic site of glycogen phosphorylase b: binding and kinetic studies with the beta-glycosidase inhibitor D-gluconohydroximo-1,5-lactone N-phenylurethane.

J. Hajdu, L. Johnson, D. Barford, 1988, Biochemistry.

Membrane Topography of the Coupling Ion Binding Site in Na+-translocating F1F0 ATP Synthase*

A. Vasella, P. Dimroth, J. Brunner, 2002, The Journal of Biological Chemistry.

Oligonucleotide Analogues with Integrated Bases and Backbone. Part 28: Hydrazide- and Amide-Linked Analogues. 2. Di-, Tetra-, Octa-, and Decamers: Synthesis and Association

Fabio De Giacomo, A. Vasella, M. Peifer, 2011 .

Oligosaccharide Analogues of Polysaccharides, Part 19, Synthesis of 2‐(Naphthalen‐1‐yl)ethyl Cellooligoglycosides and [(Naphthalene‐1,8‐diyl)di(ethane‐2,1‐diyl)] Bis[cellooligoglycosides]

A. Vasella, Jinwang Xu, 1999 .

Structural rationale for low-nanomolar binding of transition state mimics to a family GH3 beta-D-glucan glucohydrolase from barley.

Brian J. Smith, J. Varghese, A. Vasella, 2005, Biochemistry.

Oligonucleotide Analogues with a `Nucleobase-Including Backbone' Part 10. Design, Synthesis, and Association of Ether-Linked Dimers

A. Vasella, P. Bhardwaj, A. J. Matthews, 2004 .

Interactions of a Family 18 Chitinase with the Designed Inhibitor HM508 and Its Degradation Product, Chitobiono-δ-lactone*

B. Synstad, D. V. van Aalten, A. Vasella, 2004, Journal of Biological Chemistry.

An Advantageous Synthesis of 5,6,7,8-Tetra-Hydrotetrazolo[1,5-a]Pyridines

A. Vasella, S. Vonhoff, 1999 .

Novel Type of Rigid C-Linked Glycosylacetylene−Phenylalanine Building Blocks for Combinatorial Synthesis of C-linked Glycopeptides

A. Vasella, M. Meldal, T. Lowary, 1998 .

Probing specific lectin-carbohydrate interactions using atomic force microscopy imaging and force measurements

A. Vasella, A. Touhami, Y. Dufrêne, 2003 .

Synthesis of C(2)-substituted manno-configured tetrahydroimidazopyridines and their evaluation as inhibitors of snail β-mannosidase

A. Vasella, M. Terinek, 2003 .

Ternary complex crystal structures of glycogen phosphorylase with the transition state analogue nojirimycin tetrazole and phosphate in the T and R states.

S. Withers, L. Johnson, E. Mitchell, 1996, Biochemistry.

Mutagenesis of 16S rRNA C1409-G1491 base-pair differentiates between 6'OH and 6'NH3+ aminoglycosides.

E. Westhof, A. Vasella, S. Hobbie, 2005, Journal of molecular biology.

Decoding and deafness: Two sides of a coin

A. Vasella, E. Böttger, R. Pathak, 2011 .

Specific photoaffinity inactivation of the D-glucose transporter in small intestinal brush border membrane using new phlorizin analogues.

G. Semenza, A. Vasella, M. Hosang, 1981, Biochemistry.

Structural Determinants of Substrate Specificity in Family 1 β-Glucosidases

B. Henrissat, A. Vasella, D. Bevan, 2004, Journal of Biological Chemistry.

B. Henrissat, A. Vasella, D. Bevan, 2004, The Journal of biological chemistry.

Importance of the 6′‐Hydroxy Group and Its Configuration for Apramycin Activity

A. Vasella, E. Böttger, D. Crich, 2014, ChemMedChem.

Recent Insights into Inhibition, Structure, and Mechanism of Configuration-Retaining Glycosidases.

A. Vasella, T. Heightman, 1999, Angewandte Chemie.

Glycosidase mechanisms.

A. Vasella, G. Davies, M. Böhm, 2002, Current opinion in chemical biology.

Inhibition of cellobiohydrolases from Trichoderma reesei. Synthesis and evaluation of some glucose-, cellobiose-, and cellotriose-derived hydroximolactams and imidazoles.

A. Vasella, S. Vonhoff, M. Claeyssens, 1999 .

A Synthesis of 1D- and 1L-myo-Inositol 1,3,4,5,-Tetraphosphate

K. S. Swaminathan, A. Vasella, B. I. Glänzer, 1988 .

The binding of D-gluconohydroximo-1,5-lactone to glycogen phosphorylase. Kinetic, ultracentrifugation and crystallographic studies.

N. Oikonomakos, A. Vasella, D. Leonidas, 1991, The Biochemical journal.