J. Miyashiro

发表

1,2‐Diarylpyrroles as Potent and Selective Inhibitors of Cyclooxygenase‐2.

C. Koboldt, K. Seibert, P. Isakson, 1997 .

Synthesis and biological evaluation of the 1,5-diarylpyrazole class of cyclooxygenase-2 inhibitors: identification of 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benze nesulfonamide (SC-58635, celecoxib).

R. S. Rogers, C. Koboldt, K. Seibert, 1997, Journal of medicinal chemistry.

Structural basis for selective inhibition of cyclooxygenase-2 by anti-inflammatory agents

R. Kurumbail, W. Stallings, J. Gierse, 1997, Nature.

Synthesis and SAR of novel tricyclic quinoxalinone inhibitors of poly(ADP-ribose)polymerase-1 (PARP-1).

Eric F. Johnson, X. Liu, V. Giranda, 2009, Bioorganic & medicinal chemistry letters.

Synthesis of imidazopyridines and purines as potent inhibitors of leukotriene A4 hydrolase.

J. Gierse, J. Miyashiro, T. Penning, 2003, Bioorganic & medicinal chemistry letters.

Discovery of Diphenylmethanepropionic and Dihydrostilbeneacetic Acids as Antagonists of the Integrin αvβ3

D. Griggs, J. Miyashiro, V. Engleman, 2006 .

Enantioselective total synthesis and pharmacologic profile of 12-deoxy-12(S)-methyl leukotriene B4

J. Miyashiro, T. Penning, S. Djurić, 1991 .

Structure−Activity Relationship Studies on 1-[2-(4-Phenylphenoxy)ethyl]pyrrolidine (SC-22716), a Potent Inhibitor of Leukotriene A4 (LTA4) Hydrolase

J. Gierse, J. Miyashiro, T. Penning, 2000 .

Improved Procedure for the Reduction of N-Acyloxazolidinones

J. Miyashiro, T. Penning, V. Kalish, 1990 .

Synthesis of potent leukotriene A(4) hydrolase inhibitors. Identification of 3-[methyl[3-[4-(phenylmethyl)phenoxy]propyl]amino]propanoic acid.

J. Gierse, J. Miyashiro, T. Penning, 2002, Journal of medicinal chemistry.

1,2-Diarylpyrroles as potent and selective inhibitors of cyclooxygenase-2.

C. Koboldt, K. Seibert, P. Isakson, 1997, Journal of medicinal chemistry.

Aminopyrimidinone cdc7 kinase inhibitors.

Eric F. Johnson, N. Soni, J. Miyashiro, 2012, Bioorganic & medicinal chemistry letters.

Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors: Identification of 4-(5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1-yl)benzenesulfonamide (SC-58635, Celecoxib).

P. Collins, J. Miyashiro, T. Penning, 2010 .

SC-41930 inhibits neutrophil infiltration of the cavine dermis induced by 12(R)-hydroxyeicosatetraenoic acid.

J. Miyashiro, T. Penning, S. Djurić, 1989, Prostaglandins, leukotrienes, and essential fatty acids.

12(R)-hydroxyeicosatetraenoic acid is a neutrophil chemoattractant in the cavine, lapine, murine and canine dermis.

J. Miyashiro, T. Penning, S. Djurić, 1989, Prostaglandins, leukotrienes, and essential fatty acids.

Second-generation leukotriene B4 receptor antagonists related to SC-41930: heterocyclic replacement of the methyl ketone pharmacophore.

J. Snyder, J. Miyashiro, T. Penning, 1995, Journal of Medicinal Chemistry.