T. Kuntzweiler

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Rapid assessment of ligand actions with nicotinic acetylcholine receptors using calcium dynamics and FLIPR

D. Donnelly-roberts, S. Arneric, T. Kuntzweiler, 1998 .

Synthesis and structure-activity relationships of pyridine-modified analogs of 3-[2-((S)-pyrrolidinyl)methoxy]pyridine, A-84543, a potent nicotinic acetylcholine receptor agonist.

D. Donnelly-roberts, S. Arneric, J. Sullivan, 1998, Bioorganic & medicinal chemistry letters.

Amino acid substitutions in the rat Na+, K(+)‐ATPase alpha 2‐subunit alter the cation regulation of pump current expressed in HeLa cells.

T. Kuntzweiler, S. Yamamoto, N. Sperelakis, 1996, The Journal of physiology.

Amino Acid Replacement of Asp369 in the Sheep α1 Isoform Eliminates ATP and Phosphate Stimulation of [3]H Ouabain Binding to the Na+,K+-ATPase without Altering the Cation Binding Properties of the Enzyme (*)

Carl L. Johnson, C. L. Johnson, J. Lingrel, 1995, The Journal of Biological Chemistry.

ABT-594 [(R)-5-(2-azetidinylmethoxy)-2-chloropyridine]: a novel, orally effective analgesic acting via neuronal nicotinic acetylcholine receptors: I. In vitro characterization.

D. Donnelly-roberts, D. Mckenna, S. Arneric, 1998, The Journal of pharmacology and experimental therapeutics.

Novel 2-(2'-furo[3,2-b]pyridinyl) pyrrolidines : Potent neuronal nicotinic acetylcholine receptor ligands

D. Donnelly-roberts, S. Arneric, T. Kuntzweiler, 1997 .

Na+,K(+)-ATPase.

J. Lingrel, T. Kuntzweiler, J B Lingrel, 1994, The Journal of biological chemistry.

Identification and initial structure-activity relationships of (R)-5-(2-azetidinylmethoxy)-2-chloropyridine (ABT-594), a potent, orally active, non-opiate analgesic agent acting via neuronal nicotinic acetylcholine receptors.

D. Donnelly-roberts, S. Arneric, C. Briggs, 1998, Journal of medicinal chemistry.

Structure-activity studies related to ABT-594, a potent nonopioid analgesic agent: effect of pyridine and azetidine ring substitutions on nicotinic acetylcholine receptor binding affinity and analgesic activity in mice.

D. Donnelly-roberts, S. Arneric, J. Sullivan, 1998, Bioorganic & medicinal chemistry letters.

The role of neuronal nicotinic acetylcholine receptors in antinociception: Effects of ABT-594

D. Donnelly-roberts, S. Arneric, C. Briggs, 1998, Journal of Physiology-Paris.

Inactivation and phosphorylation of sarcoplasmic reticulum Ca(2+)-ATPase by Mg.ATP analogues Rh(III)-ATP and Co(III)-ATP.

T. Kuntzweiler, C. Grisham, 1992, Archives of biochemistry and biophysics.

Mono- and disubstituted-3,8-diazabicyclo[3.2.1]octane derivatives as analgesics structurally related to epibatidine: synthesis, activity, and modeling.

D. Anderson, T. Kuntzweiler, D. Colombo, 1998, Journal of medicinal chemistry.

Glutamic Acid 327 in the Sheep 1 Isoform of Na,K-ATPase Stabilizes a K-induced Conformational Change *

J. Lingrel, T. Kuntzweiler, E. Wallick, 1995, The Journal of Biological Chemistry.

A Solid Supported Membrane-Based Technology for Electrophysical Screening of B0AT1-Modulating Compounds

G. Hessler, T. Kuntzweiler, T. Licher, 2021, SLAS discovery : advancing life sciences R & D.

Ouabain Interactions with the H5-H6 Hairpin of the Na,K-ATPase Reveal a Possible Inhibition Mechanism via the Cation Binding Domain*

J. Lingrel, T. Kuntzweiler, J. Argüello, 1996, The Journal of Biological Chemistry.

Cation and Cardiac Glycoside Binding Sites of the Na,K‐ATPase a

J. Lingrel, T. Kuntzweiler, J. Argüello, 1997, Annals of the New York Academy of Sciences.

Identification and Characterization of Inhibitors of a Neutral Amino Acid Transporter, SLC6A19, Using Two Functional Cell-Based Assays

T. Kuntzweiler, B. Liang, Kristen L. Randall, 2019, SLAS discovery : advancing life sciences R & D.

Synthesis and structure–activity relationships of 5-substituted pyridine analogues of 3-[2-((S)-pyrrolidinyl)methoxy]pyridine, A-84543: A potent nicotinic receptor ligand

S. Arneric, T. Kuntzweiler, N. Lin, 2001 .

Critical effects on catalytic function produced by amino acid substitutions at Asp804 and Asp808 of the al isoform of Na,K‐ATPase

J. Lingrel, T. Kuntzweiler, J. V. Van Huysse, 1996, FEBS letters.

J. Lingrel, T. Kuntzweiler, G. Scheiner‐Bobis, 2020, Encyclopedia of Molecular Pharmacology.

Amelioration of PXR-mediated CYP3A4 induction by mGluR2 modulators.

Roy J. Vaz, Hong Shen, T. Kuntzweiler, 2018, Bioorganic & medicinal chemistry letters.

Asp804 and Asp808 in the Transmembrane Domain of the Na,K-ATPase α Subunit Are Cation Coordinating Residues*

J. Lingrel, T. Kuntzweiler, J. Argüello, 1996, The Journal of Biological Chemistry.