S. Vyskocil

发表

An inhibitor of NEDD8-activating enzyme as a new approach to treat cancer

Amanda Doucette, Mansoureh Rezaei, Alice McDonald, 2009, Nature.

Axially chiral 1,1′-binaphthyls with non-identical groups in 2,2′-positions. Synthesis of the enantiomerically pure 2-hydroxy-2′-thiol and substituted 2-amino-2′-thiols

S. Vyskocil, M. Polášek, P. Kočovský, 1997 .

Transition metal catalysed synthesis of tetrahydro derivatives of [5]-, [6]- and [7]helicene

S. Vyskocil, D. Šaman, I. Stará, 1999 .

ENANTIOSELECTIVE [2+2+2] CYCLOISOMERISATION OF ALKYNES IN THE SYNTHESIS OF HELICENES: THE SEARCH FOR EFFECTIVE CHIRAL LIGANDS

S. Vyskocil, P. Guiry, G. Lloyd‐Jones, 2011 .

Synthesis and catalytic activity of spaced ferrocene oxazolines

S. Vyskocil, I. Císařová, P. Štěpnička, 2003 .

Identification of Novel Carbocyclic Pyrimidine Cyclic Dinucleotide STING Agonists for Antitumor Immunotherapy Using Systemic Intravenous Route.

Adnan O. Abu-Yousif, M. Mizutani, Courtney A. Cullis, 2021, Journal of medicinal chemistry.

Synthesis of 3-hexahelicenol and its transformation to 3-hexahelicenylamines, diphenylphosphine, methyl carboxylate, and dimethylthiocarbamate.

S. Vyskocil, D. Šaman, I. Stará, 2003, The Journal of organic chemistry.

Substrate-assisted inhibition of ubiquitin-like protein-activating enzymes: the NEDD8 E1 inhibitor MLN4924 forms a NEDD8-AMP mimetic in situ.

Ping Li, Hua Liao, M. Rolfe, 2010, Molecular cell.

Palladium(II) Complexes of 2-Dimethylamino-2‘- diphenylphosphino-1,1‘-binaphthyl (MAP) with Unique P,Cσ-Coordination and Their Catalytic Activity in Allylic Substitution, Hartwig−Buchwald Amination, and Suzuki Coupling

S. Vyskocil, I. Císařová, V. Langer, 1999 .

Synthesis of alpha-amino acids via asymmetric phase transfer-catalyzed alkylation of achiral nickel(II) complexes of glycine-derived Schiff bases.

S. Vyskocil, M. North, I. Císařová, 2003, Journal of the American Chemical Society.

Catalytic enantioselective synthesis of 18F-fluorinated alpha-amino acids under phase-transfer conditions using (S)-NOBIN.

S. Ametamey, S. Vyskocil, P. Schubiger, 2004, Nuclear medicine and biology.

Synthesis of a Potent NAE Inhibitor: Pevonedistat

S. Vyskocil, S. Langston, H. Mizutani, 2016 .

On the ‘Novel two-phase oxidative cross-coupling of the two-component molecular crystal of 2-naphthol and 2-naphthylamine’

S. Vyskocil, M. Polášek, P. Kočovský, 1998 .

Non-symmetrically substituted 1,1'-binaphthyls in enantioselective catalysis.

S. Vyskocil, P. Kočovský, Pavel Kocovský, 2003, Chemical reviews.

The SN2 Reaction in the Solid State. An Unusual, BAl2 Aminolysis of an Ester Group in Crystalline (±)-2-Amino-2‘-hydroxy-3‘-(methoxycarbonyl)- 1,1‘-binaphthyl Elucidated by X-ray Diffraction and Isotopic Labeling. New Experimental Evidence for Linearity in SN2 Substitution

S. Vyskocil, D. Zax, V. Langer, 1996 .

Diastereoisomeric cationic pi-allylpalladium-(P,C)-MAP and MOP complexes and their relationship to streochemical memory effects in allylic alkylation.

S. Vyskocil, C. Butts, P. Kočovský, 2000, Chemistry.

Transition metal catalysis in organic synthesis: reflections, chirality and new vistas

S. Vyskocil, P. Kočovský, G. Lloyd‐Jones, 1999 .

Synthesis of 2-amino-2′-diphenylphosphino-1,1′-binaphthyl (MAP) and its accelerating effect on the Pd(0)-catalyzed N-arylation

S. Vyskocil, P. Kočovský, M. Smrčina, 1998 .

Derivatives of 2-Amino-2‘-diphenylphosphino-1,1‘-binaphthyl (MAP) and Their Application in Asymmetric Palladium(0)-Catalyzed Allylic Substitution†

S. Vyskocil, P. Kočovský, V. Hanuš, 1998 .

Synthesis and Resolution of Racemic 2-Amino-2'-hydroxy-1,1'-binaphthyl

S. Vyskocil, P. Kočovský, J. Poláková, 1996 .

Synthesis of enantiomerically pure binaphthyl derivatives. Mechanism of the enantioselective, oxidative coupling of naphthols and designing a catalytic cycle

S. Vyskocil, P. Kočovský, J. Poláková, 1993 .

Enantiomerically enriched (R)- and (S)-α-methylphenylalanine via asymmetric PTC C-alkylation catalysed by NOBIN

S. Vyskocil, Y. Belokon’, H. Kagan, 1999 .

Synthesis of N-Alkylated and N-Arylated Derivatives of 2-Amino-2‘-hydroxy-1,1‘-binaphthyl (NOBIN) and 2,2‘-Diamino-1,1‘-binaphthyl and Their Application in the Enantioselective Addition of Diethylzinc to Aromatic Aldehydes†

S. Vyskocil, P. Kočovský, V. Hanuš, 1998 .

Selective Cross-Coupling of 2-Naphthol and 2-Naphthylamine Derivatives. A Facile Synthesis of 2,2',3-Trisubstituted and 2,2',3,3'-Tetrasubstituted 1,1'-Binaphthyls

T. A. Claxton, S. Vyskocil, A. Abbott, 1994 .

Copper(II)-mediated oxidative coupling of 2-aminonaphthalene homologues. Competition between the straight dimerization and the formation of carbazoles.

S. Vyskocil, V. Langer, P. Kočovský, 2001, The Journal of organic chemistry.

Synthesis of 2-hydroxy-8'-(hydroxymethyl)-1,1'-binaphthalene (iso-homo-binol). A new structural pattern in the binaphthyl realm

S. Vyskocil, P. Kočovský, W. Mitchell, 2003 .

Synthesis of C2-Symmetrical [1,1'-Binaphthalene]-2,2'-diamines with Additional Chelating Groups Attached to the Nitrogen Atoms as Potential Ligands for Asymmetric Catalysis

S. Vyskocil, P. Kočovský, P. Maloň, 2000 .

Total synthesis and structural elucidation of azaspiracid-1. Final assignment and total synthesis of the correct structure of azaspiracid-1.

Yoichi M. A. Yamada, K. Nicolaou, S. Vyskocil, 2006, Journal of the American Chemical Society.

Asymmetric Michael reaction of diethyl malonate with crotonaldehyde catalyzed by chiral aminocarboxylates, amino alcoholates, and amino phenolates

S. Vyskocil, A. Peregudov, V. I. Maleev, 2001 .

2H-quadrupolar coupling-based analysis of stereochemical and regiochemical memory in the Pd-catalysed allylic alkylation of iso-cinnamyl type substrates employing the chiral monophosphine ligands ‘MOP’ and ‘MAP’

S. Vyskocil, P. Kočovský, G. Lloyd‐Jones, 2003 .

Total synthesis and structural elucidation of azaspiracid-1. Synthesis-based analysis of originally proposed structures and indication of their non-identity to the natural product.

K. Nicolaou, S. Vyskocil, F. Bernal, 2006, Journal of the American Chemical Society.

Structural revision and total synthesis of azaspiracid-1, part 1: intelligence gathering and tentative proposal.

Yoichi M. A. Yamada, K. Nicolaou, S. Vyskocil, 2004, Angewandte Chemie.

Structural revision and total synthesis of azaspiracid-1, part 2: definition of the ABCD domain and total synthesis.

Yoichi M. A. Yamada, K. Nicolaou, S. Vyskocil, 2004, Angewandte Chemie.

Total synthesis of the proposed azaspiracid-1 structure, part 1: construction of the enantiomerically pure C1-C20, C21-C27, and C28-C40 fragments.

K. Nicolaou, S. Vyskocil, F. Bernal, 2003, Angewandte Chemie.

Total synthesis of the proposed azaspiracid-1 structure, part 2: coupling of the C1-C20, C21-C27, and C28-C40 fragments and completion of the synthesis.

K. Nicolaou, S. Vyskocil, T. Ling, 2003, Angewandte Chemie.

On the “Novel Two-Phase Oxidative Cross-Coupling of the Two-Component Molecular Crystal of 2-Naphthol and 2-Naphthylamine”.

S. Vyskocil, M. Polášek, P. Kočovský, 1998 .

Highly Efficient Catalytic Synthesis of α‐Amino Acids under Phase‐Transfer Conditions with a Novel Catalyst/Substrate Pair

S. Vyskocil, M. North, Y. Belokon’, 2001 .

2,8'-disubstituted-1,1'-binaphthyls: a new pattern in chiral ligands.

S. Vyskocil, I. Císařová, M. Polášek, 2002, Chemistry.

Non-Symmetrically Substituted 1,1′-Binaphthyls in Enantioselective Catalysis

S. Vyskocil, P. Kočovský, M. Smrčina, 2003 .

Design and optimization of potent and orally bioavailable tetrahydronaphthalene Raf inhibitors.

Yuan Tian, Hongbo Zeng, Mansoureh Rezaei, 2011, Journal of medicinal chemistry.

Weak intra- and intermolecular interactions in a binaphthol imine: an experimental charge-density study on (+/-)-8'-benzhydrylideneamino-1,1'-binaphthyl-2-ol.

H. Senn, S. Vyskocil, P. Kočovský, 2009, Acta crystallographica. Section B, Structural science.

Structural Revision and Total Synthesis of Azaspiracid‐1. Part 2. Definition of the ABCD Domain and Total Synthesis.

Yoichi M. A. Yamada, K. Nicolaou, S. Vyskocil, 2004 .