T. Gilmore

发表

Inhibition of p38 MAP kinase by utilizing a novel allosteric binding site

L. Tong, S. Pav, C. Pargellis, 2002, Nature Structural Biology.

Pyrazole urea-based inhibitors of p38 MAP kinase: from lead compound to clinical candidate.

J. Madwed, L. Tong, S. Pav, 2002, Journal of medicinal chemistry.

Inhibition of p38 MAP kinase by utilizing a novel allosteric binding site

Liang Tong, Eugene R. Hickey, John W. Regan, 2002 .

Discovery and characterization of the N-phenyl-N'-naphthylurea class of p38 kinase inhibitors.

K. Qian, J. Madwed, C. Pargellis, 2009, Bioorganic & medicinal chemistry letters.

The kinetics of binding to p38MAP kinase by analogues of BIRB 796.

C. Pargellis, P. Cirillo, T. Gilmore, 2003, Bioorganic & medicinal chemistry letters.

Antisense and small-molecule modulation of diacylglycerol acyltransferase

I. Enyedy, T. Gilmore, B. Hubbard, 2007 .

Discovery of diamide compounds as diacylglycerol acyltransferase 1 (DGAT1) inhibitors.

T. Gilmore, R. Streeper, B. Wang, 2016, Bioorganic & medicinal chemistry letters.

Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores.

T. Gilmore, J. Regan, C. Torcellini, 2011, Bioorganic & medicinal chemistry letters.

Nonsteroidal dissociated glucocorticoid agonists containing azaindoles as steroid A-ring mimetics.

T. Gilmore, C. Torcellini, Alison J Kukulka, 2010, Journal of medicinal chemistry.

Discovery and SAR study of novel dihydroquinoline-containing glucocorticoid receptor agonists.

John R. Proudfoot, Richard M. Nelson, J. Proudfoot, 2006, Bioorganic & medicinal chemistry letters.

Discovery and SAR study of novel dihydroquinoline containing glucocorticoid receptor ligands.

Richard M Nelson, J. Proudfoot, T. Gilmore, 2006, Bioorganic & medicinal chemistry letters.

Structure-activity relationships of the p38alpha MAP kinase inhibitor 1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)naph- thalen-1-yl]urea (BIRB 796).

J. Madwed, C. Pargellis, P. Cirillo, 2003, Journal of medicinal chemistry.

A strain of Fujinami sarcoma virus which is temperature-sensitive in protein phosphorylation and cellular transformation

T. Pawson, G. Martin, T. Gilmore, 1980, Cell.

Discovery of an Orally Bioavailable Benzimidazole Diacylglycerol Acyltransferase 1 (DGAT1) Inhibitor That Suppresses Body Weight Gain in Diet-Induced Obese Dogs and Postprandial Triglycerides in Humans.

T. Gilmore, V. Tedesco, B. Hubbard, 2017, Journal of medicinal chemistry.