D. Kovalskyy

发表

Recognition of the HIV capsid by the TRIM5α restriction factor is mediated by a subset of pre-existing conformations of the TRIM5α SPRY domain.

D. Kovalskyy, D. Ivanov, 2014, Biochemistry.

The small‐molecule 3G11 inhibits HIV‐1 reverse transcription

D. Kovalskyy, D. Ivanov, Baek Kim, 2017, Chemical biology & drug design.

Role of Protein Phosphatase 1 in Dephosphorylation of Ebola Virus VP30 Protein and Its Targeting for the Inhibition of Viral Transcription*

V. S. Naumchik, Tatiana Ammosova, S. Nekhai, 2014, The Journal of Biological Chemistry.

1E7‐03, a low MW compound targeting host protein phosphatase‐1, inhibits HIV‐1 transcription

K. Kehn-Hall, S. Nekhai, A. Üren, 2014, British journal of pharmacology.

Phenyl-1-Pyridin-2yl-Ethanone-Based Iron Chelators Increase IκB-α Expression, Modulate CDK2 and CDK9 Activities, and Inhibit HIV-1 Transcription

S. Nekhai, F. Kashanchi, D. Kovalskyy, 2014, Antimicrobial Agents and Chemotherapy.

Effect of mimetic CDK9 inhibitors on HIV-1-activated transcription.

Z. Klase, S. Nekhai, F. Kashanchi, 2013, Journal of molecular biology.

Small Molecules Targeted to a Non-Catalytic “RVxF” Binding Site of Protein Phosphatase-1 Inhibit HIV-1

Tatiana Ammosova, S. Nekhai, K. Jeang, 2012, PloS one.

Activation of HIV-1 with Nanoparticle-Packaged Small-Molecule Protein Phosphatase-1-Targeting Compound

S. Nekhai, D. Kovalskyy, E. Akala, 2015, Scientia pharmaceutica.

Mononuclear π-complexes of Pd(II) and Pt(II) with 1-allyl-3-(2-hydroxyethyl)thiourea: Synthesis, structure, molecular docking, DNA binding ability and genotoxic activity

D. Kovalskyy, V. Pekhnyo, M. Platonov, 2021, Polyhedron.

Structural basis of RNA cap modification by SARS-CoV-2

R. Hromas, D. Kovalskyy, L. Martínez-Sobrido, 2020, Nature Communications.

Conformational Changes of the Multispecific Transporter Organic Anion Transporter 1 (OAT1/SLC22A6) Suggests a Molecular Mechanism for Initial Stages of Drug and Metabolite Transport

I. Tsigelny, V. Kouznetsova, D. Kovalskyy, 2011, Cell Biochemistry and Biophysics.

Structural bioinformatics in post-genomic era

D. Kovalskyy, A. Kornelyuk, K. Odynets, 2004 .

Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling

P. Schmieder, W. Birchmeier, U. Heinemann, 2021, Magnetic resonance.

Phenyl-1-Pyridin-2yl-Ethanone-Based Iron Chelators Increase I (cid:2) B- (cid:3) Expression, Modulate CDK2 and CDK9 Activities, and Inhibit HIV-1 Transcription

S. Nekhai, F. Kashanchi, D. Kovalskyy, 2014 .

Identification of novel small molecule inhibitors of adenovirus gene transfer using a high throughput screening approach.

D. Kovalskyy, E. Kalkman, A. Parker, 2013, Journal of controlled release : official journal of the Controlled Release Society.

Reactivation of latent HIV-1 provirus via targeting protein phosphatase-1

S. Nekhai, F. Kashanchi, A. Üren, 2015, Retrovirology.

B Cell Endosomal RAB7 Promotes TRAF6 K63 Polyubiquitination and NF-κB Activation for Antibody Class-Switching

P. Casali, Hui Yan, D. Kovalskyy, 2020, The Journal of Immunology.

Inhibition of FoxM1-Mediated DNA Repair by Imipramine Blue Suppresses Breast Cancer Growth and Metastasis

J. Arbiser, Yidong Chen, M. Hanes, 2016, Clinical Cancer Research.

Effect of transcription inhibition and generation of suppressive viral non-coding RNAs

F. Kashanchi, D. Kovalskyy, M. Weinberg, 2019, Retrovirology.

The improvement of the algorithm for order parameter calculation (S2) from molecular dynamics simulation using the correlation motion function.

D. Kovalskyy, A. Kornelyuk, O. Ivanova, 2006, Biophysical chemistry.

A molecular dynamics study of the structural stability of HIV‐1 protease under physiological conditions: The role of Na+ ions in stabilizing the active site

D. Kovalskyy, A. Kornelyuk, A. E. Mark, 2004, Proteins.

Targeting the Non-catalytic RVxF Site of Protein Phosphatase-1 With Small Molecules for Ebola Virus Inhibition

Tatiana Ammosova, S. Nekhai, A. Üren, 2019, Front. Microbiol..

Novel Potent Orthosteric Antagonist of ASIC1a Prevents NMDAR-Dependent LTP Induction.

D. Kovalskyy, E. Isaeva, O. Ievglevskyi, 2015, Journal of medicinal chemistry.

Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loading with syndecan and EpCAM cargo

D. Kovalskyy, P. Roche, S. Betzi, 2020, Journal of extracellular vesicles.

Targeting Tat–TAR RNA Interaction for HIV-1 Inhibition

S. Nekhai, D. Kovalskyy, N. Kumari, 2021, Viruses.

Targeting Tat-TAR RNA Interaction for HIV-1 Inhibition

S. Nekhai, D. Kovalskyy, N. Kumari, 2021 .

Molecular dynamics simulation study of effect of the conservative Leu10→Ile mutation on intramolecular mobility of HIV-1 protease

D. Kovalskyy, A. Kornelyuk, V. M. Dubina, 2004 .