G. Quéléver

发表

N-acyl substituted 7-amino-4-chloroisocoumarin: a peptide degradation model via an imide mechanism.

F. Bihel, J. Kraus, C. Garino, 2004, Bioorganic & medicinal chemistry letters.

Naphthyl and coumarinyl biarylpiperazine derivatives as highly potent human beta-secretase inhibitors. Design, synthesis, and enzymatic BACE-1 and cell assays.

T. Iwatsubo, J. Kraus, B. Maigret, 2006, Journal of medicinal chemistry.

Structural characterization of poly(amino)ester dendrimers and related impurities by electrospray tandem mass spectrometry.

G. Quéléver, Aura Tintaru, Ling Peng, 2010, Rapid communications in mass spectrometry : RCM.

Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new beta-amyloid peptide production inhibitors and their activities on various classes of protease.

O. Pourquié, F. Bihel, J. Kraus, 2003, Bioorganic & medicinal chemistry.

Direct synthesis of 5-aryltriazole acyclonucleosides via Suzuki coupling in aqueous solution

G. Quéléver, Fanqi Qu, Ruizhi Zhu, 2007 .

Synthesis of poly(aminoester) dendrimers via 'click' chemistry in combination with the divergent and convergent strategies

G. Quéléver, Ling Peng, P. Moreno, 2015 .

C-S coupling using a mixed-ligand Pd catalyst: a highly effective strategy for synthesizing arylthio-substituted heterocycles.

G. Quéléver, Ling Peng, Fanqi Qu, 2013, Chemistry.

Enhanced delivery of gamma-secretase inhibitor DAPT into the brain via an ascorbic acid mediated strategy.

C. Melon, C. Garino, G. Quéléver, 2005, Organic & biomolecular chemistry.

Substituted thiazolamide coupled to a redox delivery system: a new gamma-secretase inhibitor with enhanced pharmacokinetic profile.

M. Wolfe, F. Bihel, J. Kraus, 2005, Organic & biomolecular chemistry.

A "click" chemistry constructed affinity system for 2-oxoglutaric acid receptors and binding proteins.

G. Quéléver, Ling Peng, Yang Wang, 2014, Organic & biomolecular chemistry.

Design of β-Secretase Inhibitors by Introduction of a Mandelyl Moiety in DAPT Analogues

J. Kraus, C. Garino, G. Quéléver, 2005 .

1,1'-Xylyl bis-1,4,8,11-tetraaza cyclotetradecane: a new potential copper chelator agent for neuroprotection in Alzheimer's disease. Its comparative effects with clioquinol on rat brain copper distribution.

J. Kraus, C. Garino, G. Quéléver, 2006, Bioorganic & medicinal chemistry letters.

New 2-bromomethyl-8-substituted-benzo[c]chromen-6-ones. Synthesis and biological properties.

F. Bihel, J. Kraus, J. Boucher, 2005, Bioorganic & medicinal chemistry letters.

Design of potential new HIV protease inhibitors: enantioconvergent synthesis of new pyrrolidin-3-ol, and pyrrolidin-3-one peptide conjugates

F. Bihel, J. Courcambeck, J. Kraus, 2001 .

Importance of size-to-charge ratio in construction of stable and uniform nanoscale RNA/dendrimer complexes.

Cheng-Cai Zhang, Dai-Wen Pang, Ling Peng, 2007, Organic & biomolecular chemistry.

New 2-bromomethyl-8-substituted-benzo[c]chromen-6-ones. Synthesis and biological properties.

F. Bihel, J. Kraus, J. Boucher, 2005, Bioorganic & medicinal chemistry letters.

Synthesis of new 7-membered α-phenylthio cyclic oxamides: HIV inhibitors

G. Priem, J. Kraus, G. Quéléver, 1998 .

BACE-1 inhibitory activities of new substituted phenyl-piperazine coupled to various heterocycles: chromene, coumarin and quinoline.

J. Kraus, C. Garino, G. Quéléver, 2006, Bioorganic & medicinal chemistry letters.

Novel cyclized Pifithrin-α p53 inactivators: synthesis and biological studies

J. Kraus, C. Garino, G. Quéléver, 2005 .

New antiviral nucleoside prodrugs await application.

J. Kraus, C. Garino, F. Souard, 2003, Current medicinal chemistry.

Simple coupling reaction between amino acids and weakly nucleophilic heteroaromatic amines.

J. Kraus, C. Garino, G. Quéléver, 2004, Journal of combinatorial chemistry.

Conformational sensitivity of conjugated poly(ethylene oxide)-poly(amidoamine) molecules to cations adducted upon electrospray ionization - a mass spectrometry, ion mobility and molecular modeling study.

S. Pricl, G. Quéléver, P. Posocco, 2014, Analytica chimica acta.

Syntheses of new unsymmetrical bispolyazamacrocycles

J. Kraus, G. Quéléver, M. Camplo, 1998 .

Microwave promoted C–O coupling for synthesizing O-aryloxytriazole nucleoside analogues

J. Iovanna, G. Quéléver, Ling Peng, 2015 .

Pd-catalyzed oxidative C-H alkenylation for synthesizing arylvinyltriazole nucleosides.

G. Quéléver, Ling Peng, Fanqi Qu, 2015, Organic & biomolecular chemistry.

Prospects for the resistance to HIV protease inhibitors: current drug design approaches and perspectives.

Jean-Louis Kraus, J. Kraus, C. Garino, 2005, Current pharmaceutical design.

Novel cyclized Pifithrin-alpha p53 inactivators: synthesis and biological studies.

J. Kraus, C. Garino, G. Quéléver, 2005, Bioorganic & medicinal chemistry letters.

Tri-N-Boc-tetraazamacrocycle-nucleoside conjugates: synthesis and anti-HIV activities.

J. Chermann, J. Kraus, G. Quéléver, 1998, Nucleosides & nucleotides.

Tri‐N‐Boc‐tetraazamacrocycle—Nucleoside Conjugates: Synthesis and Anti‐HIV Activities.

J. Chermann, J. Kraus, G. Quéléver, 2010 .

Are p53 inhibitors potentially useful therapeutics?

J. Kraus, C. Garino, G. Quéléver, 2005 .

Syntheses of new modified Phe-Pro peptides. Use of proline replacements in potential HIV inhibitors.

J. Chermann, J. Kraus, G. Quéléver, 1998, Bioorganic & medicinal chemistry letters.

Direct Synthesis of 5-Aryltriazole Acyclonucleosides via Suzuki Coupling in Aqueous Solution.

G. Quéléver, Fanqi Qu, Ruizhi Zhu, 2007 .

Electrospray tandem mass spectrometry of poly(amino)ester dendrimers: Dissociation rules and structural characterization of defective molecules

G. Quéléver, Aura Tintaru, Ling Peng, 2011 .