Shunichirou Tsutsumi

Design and synthesis of novel DFG-out RAF/vascular endothelial growth factor receptor 2 (VEGFR2) inhibitors: 3. Evaluation of 5-amino-linked thiazolo[5,4-d]pyrimidine and thiazolo[5,4-b]pyridine derivatives.

Biching Sang, J. Yano, M. Hirose, 2012, Bioorganic & medicinal chemistry.

Characterization and evaluation of miconazole salts and cocrystals for improved physicochemical properties.

T. Kojima, Y. Ikeda, Shunichirou Tsutsumi, 2011, International journal of pharmaceutics.

Design and synthesis of novel DFG-out RAF/vascular endothelial growth factor receptor 2 (VEGFR2) inhibitors: 2. Synthesis and characterization of a novel imide-type prodrug for improving oral absorption.

M. Okaniwa, T. Miyazaki, T. Imada, 2012, Bioorganic & medicinal chemistry.

Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH2 (TAK-448), with Highly Potent Testosterone-Suppressive Activity and Excellent Water Solubility.

Y. Ikeda, Shunichirou Tsutsumi, M. Yamaguchi, 2016, Journal of medicinal chemistry.

Design and synthesis of novel DFG-out RAF/vascular endothelial growth factor receptor 2 (VEGFR2) inhibitors. 1. Exploration of [5,6]-fused bicyclic scaffolds.

H. Oki, Biching Sang, J. Yano, 2012, Journal of medicinal chemistry.

Discovery of a selective kinase inhibitor (TAK-632) targeting pan-RAF inhibition: design, synthesis, and biological evaluation of C-7-substituted 1,3-benzothiazole derivatives.

Tomoyasu Ishikawa, Akito Nakamura, Terufumi Takagi, 2013, Journal of medicinal chemistry.

Establishment of cocrystal cocktail grinding method for rational screening of pharmaceutical cocrystals.

Y. Ikeda, Shunichirou Tsutsumi, Katsuhiko Yamamoto, 2012, International journal of pharmaceutics.

High-throughput cocrystal slurry screening by use of in situ Raman microscopy and multi-well plate.

Katsuhiko Yamamoto, Takashi Kojima, Toshiya Moriwaki, 2010, International journal of pharmaceutics.