R. Amici

发表

Structure-based drug design to the discovery of new 2-aminothiazole CDK2 inhibitors.

Anna Vulpetti, E. Casale, A. Vulpetti, 2006, Journal of molecular graphics & modelling.

3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 1. Lead finding.

Anna Vulpetti, Antonella Isacchi, Enrico Pesenti, 2004, Journal of medicinal chemistry.

Synthesis and biological evaluation of N-hydroxyphenylacrylamides and N-hydroxypyridin-2-ylacrylamides as novel histone deacetylase inhibitors.

A. Mai, S. Minucci, C. Mercurio, 2010, Journal of medicinal chemistry.

Chiral Resolution and Pharmacological Characterization of the Enantiomers of the Hsp90 Inhibitor 2‐Amino‐7‐[4‐fluoro‐2‐(3‐pyridyl)phenyl]‐4‐methyl‐7,8‐dihydro‐6H‐quinazolin‐5‐one Oxime

S. Minucci, C. Mercurio, R. Amici, 2014, ChemMedChem.

Synthesis, biological characterization and molecular modeling insights of spirochromanes as potent HDAC inhibitors.

S. Minucci, C. Mercurio, L. Moretti, 2016, European journal of medicinal chemistry.

Cdc7 kinase inhibitors: pyrrolopyridinones as potential antitumor agents. 1. Synthesis and structure-activity relationships.

R. Bosotti, A. Isacchi, A. Montagnoli, 2008, Journal of medicinal chemistry.

3-Amino-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles: a new class of CDK2 inhibitors.

J. Bischoff, C. Mercurio, A. Vulpetti, 2006, Bioorganic & medicinal chemistry letters.

Nitrile oxide cycloaddition of non-activated alkynes: a novel approach to the synthesis of neuroactive isoxazoles

P. Pevarello, R. Amici, M. Varasi, 1993 .

Cinnamic anilides as new mitochondrial permeability transition pore inhibitors endowed with ischemia-reperfusion injury protective effect in vivo.

S. Minucci, P. Pelicci, R. Amici, 2014, Journal of Medicinal Chemistry.

Optimization of 6,6-dimethyl pyrrolo[3,4-c]pyrazoles: Identification of PHA-793887, a potent CDK inhibitor suitable for intravenous dosing.

A. Isacchi, E. Casale, J. Bischoff, 2010, Bioorganic & medicinal chemistry.

6‐Substituted Pyrrolo[3,4‐c]pyrazoles: An Improved Class of CDK2 Inhibitors

C. Mercurio, A. Vulpetti, D. Ballinari, 2007, ChemMedChem.

REDUCTIVE ALKYLATION OF a-AMINOAMIDES

P. Pevarello, R. Amici, M. Varasi, 1996 .

Sodium channel activity and sigma binding of 2-aminopropanamide anticonvulsants.

C. Caccia, P. Pevarello, R. Amici, 1999, Bioorganic & medicinal chemistry letters.