Rajeshwar Singh

发表

2-Aminoquinazoline inhibitors of cyclin-dependent kinases.

D. W. Fry, E. Dobrusin, Y. Bathini, 2005, Bioorganic & medicinal chemistry letters.

3-Acylamino-azetidin-2-one as a novel class of cysteine proteases inhibitors.

E. Purisima, R. Ménard, Rajeshwar Singh, 2003, Bioorganic & medicinal chemistry letters.

Synthesis and antibacterial activity of the C-7 side chain of 3-aminoquinazolinediones.

H. D. Showalter, M. Huband, M. Shapiro, 2008, Bioorganic & medicinal chemistry letters.

First and Second Generation γ-Secretase Modulators (GSMs) Modulate Amyloid-β (Aβ) Peptide Production through Different Mechanisms

A. Sabirsh, Rajeshwar Singh, S. Parpal, 2012, The Journal of Biological Chemistry.

6-Acylamino-penam derivatives: synthesis and inhibition of cathepsins B, L, K, and S.

E. Purisima, R. Ménard, Rajeshwar Singh, 2002, Bioorganic & medicinal chemistry letters.

Design and synthesis of 6-substituted amino-4-oxa-1-azabicyclo[3,2,0]heptan-7-one derivatives as cysteine proteases inhibitors.

E. Purisima, R. Ménard, Rajeshwar Singh, 2002, Bioorganic & medicinal chemistry letters.

The reaction of metal fluorides with unsym-azetidinone disulfides and 2.beta.-(halomethyl)penams. The 3.beta.-fluoro-3.alpha.-methylcephams

Rajeshwar Singh, R. Micetich, P. Payne, 1987 .

Quinazolinone-based fungal efflux pump inhibitors. Part 1: Discovery of an (N-methylpiperazine)-containing derivative with activity in clinically relevant Candida spp.

Rajeshwar Singh, N. Iqbal, M. Dudley, 2004, Bioorganic & medicinal chemistry letters.

A facile synthesis of substituted 3-amino-1H-quinazoline-2,4-diones

J. Rubin, H. D. Showalter, Rajeshwar Singh, 2005 .

3-aminoquinazolinediones as a new class of antibacterial agents demonstrating excellent antibacterial activity against wild-type and multidrug resistant organisms.

J. Domagala, H. D. Showalter, J. Bronstein, 2006, Journal of medicinal chemistry.

Synthesis and structural-activity relationships of 3-hydroxyquinazoline-2,4-dione antibacterial agents.

J. Domagala, H. D. Showalter, S. Gracheck, 2004, Bioorganic & medicinal chemistry letters.

Synthesis of substituted quinazolines

Y. Bathini, Rajeshwar Singh, R. Micetich, 2002 .

Structure-activity relationships of 3-aminoquinazolinediones, a new class of bacterial type-2 topoisomerase (DNA gyrase and topo IV) inhibitors.

J. Domagala, H. D. Showalter, S. Gracheck, 2007, Bioorganic & medicinal chemistry letters.

Synthesis and Antibacterial Activity of 7-Hydrazinoquinolones.

Rajeshwar Singh, R. Micetich, M. P. Singh, 1998 .

Quinazolinone fungal efflux pump inhibitors. Part 3: (N-methyl)piperazine variants and pharmacokinetic optimization.

Rajeshwar Singh, N. Iqbal, M. Dudley, 2007, Bioorganic & medicinal chemistry letters.

Quinazolinone fungal efflux pump inhibitors. Part 2: In vitro structure-activity relationships of (N-methyl-piperazinyl)-containing derivatives.

Rajeshwar Singh, N. Iqbal, M. Dudley, 2004, Bioorganic & medicinal chemistry letters.

Substituted 1,2,4-triazoles as complexing ligands—I Ni(II), Co(II), Cu(II), Zn(II), Pd(II), Cd(II) and Pb(II) complexes with 4-amino-3,5-dimercapto-1,2,4-triazole

Rajeshwar Singh, L. Mishra, J. Srivastava, 1977 .

Synthesis and in vitro antimicrobial activity of 3-heteroarylsulphonylmethyl cephems: a new class of cephalosporins

M. Singh, Rajeshwar Singh, R. Micetich, 1995 .

Synthesis and structure—activity relationship of C-3 substituted triazolylthiomethyl cephems

M. Singh, Rajeshwar Singh, R. Micetich, 1996 .

Identification of a novel boron-containing antibacterial agent (AN0128) with anti-inflammatory activity, for the potential treatment of cutaneous diseases.

S. Benkovic, K. R. Maples, Rajeshwar Singh, 2006, Bioorganic & medicinal chemistry letters.

Structure-activity relationships of 6-(aminomethylphenoxy)-benzoxaborole derivatives as anti-inflammatory agent.

K. Jarnagin, J. Nieman, Rajeshwar Singh, 2013, Bioorganic & medicinal chemistry letters.

Discovery of a Novel Class of Boron-Based Antibacterials with Activity against Gram-Negative Bacteria

J. Nieman, S. Cusack, D. Livermore, 2013, Antimicrobial Agents and Chemotherapy.

Boron‐based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center

K. Jarnagin, J. Nieman, K. R. Maples, 2012, FEBS letters.

2-Aminoquinazoline inhibitors of cyclin-dependent kinases.

D. W. Fry, E. Dobrusin, Y. Bathini, 2005, Bioorganic & medicinal chemistry letters.

Studies on morpholine complex of palladium(II)

Rajeshwar Singh, E. Singh, R. Singh, 1972 .

New 9β-lanostane-type triterpenic and 13,14-seco-steroidal esters from the roots of Artemisia scoparia

Rajeshwar Singh, M. Ali, Surandra Kumar Sharma, 1996 .

Synthesis of the novel antibacterial 6,8-dihydroxy-7-propyl-9H-pyrrolo[1,2-b][1,3]-benzoxazin-9-one

J. Domagala, Rajeshwar Singh, R. Micetich, 2000 .

Bacterial two-component signalling as a therapeutic target in drug design. Inhibition of NRII by the diphenolic methanes (bisphenols).

J. Domagala, M. Cummings, D. Alessi, 1998, Advances in experimental medicine and biology.

Boron‐based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center

K. Jarnagin, J. Nieman, K. R. Maples, 2012, FEBS letters.

First and Second Generation γ-Secretase Modulators (GSMs) Modulate Amyloid-β (Aβ) Peptide Production through Different Mechanisms

A. Sabirsh, Rajeshwar Singh, S. Parpal, 2012, The Journal of Biological Chemistry.

with Activity against Gram-negative Bacteria

J. Nieman, S. Cusack, D. Livermore, 2013 .