B. Baratte

发表

Crystal structure of a human cyclin-dependent kinase 6 complex with a flavonol inhibitor, fisetin.

Laurent Meijer, L. Meijer, U. Schulze-Gahmen, 2005, Journal of medicinal chemistry.

3,6-Diamino-4-(2-halophenyl)-2-benzoylthieno[2,3-b]pyridine-5-carbonitriles are selective inhibitors of Plasmodium falciparum glycogen synthase kinase-3.

L. Meijer, L. Pearl, N. Pressburger, 2013, Journal of medicinal chemistry.

Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation

S. Knapp, P. Bonnet, A. Chaikuad, 2020, Journal of enzyme inhibition and medicinal chemistry.

Screening for antimitotic compounds using the cdc25 tyrosine phosphatase, an activator of the mitosis-inducing p34cdc2/cyclin Bcdc13 protein kinase.

L. Meijer, D. Beach, D. Beach, 1992, Anticancer research.

Anti-mitotic properties of indirubin-3′-monoxime, a CDK/GSK-3 inhibitor: induction of endoreplication following prophase arrest

L. Meijer, G. Eisenbrand, B. Baratte, 2001, Oncogene.

Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129

B. Baratte, S. Ruchaud, G. Burgaud, 2017, Marine drugs.

Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies.

B. Baratte, S. Ruchaud, B. Josselin, 2019, Bioorganic & medicinal chemistry.

Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration.

P. Le Pape, B. Baratte, S. Ruchaud, 2018, Bioorganic & medicinal chemistry letters.

Pax6 expression patterns in Lampetra fluviatilis and Scyliorhinus canicula embryos suggest highly conserved roles in the early regionalization of the vertebrate brain

B. Baratte, M. Lepage, S. Mazan, 2002, Brain Research Bulletin.

Exploration of 7-azaindole-coumaranone hybrids and their analogues as protein kinase inhibitors.

B. Baratte, S. Ruchaud, Richard M. Beteck, 2021, Chemico-biological interactions.

Neurymenolide A, a Novel Mitotic Spindle Poison from the New Caledonian Rhodophyta Phacelocarpus neurymenioides

B. Baratte, S. Ruchaud, C. Payri, 2019, Marine drugs.

Betulin, a Newly Characterized Compound in Acacia auriculiformis Bark, Is a Multi-Target Protein Kinase Inhibitor

M. Dimanche-Boitrel, M. Rousselot, B. Baratte, 2021, Molecules.

Constituents of Acacia nilotica (L.) Delile with Novel Kinase Inhibitory Activity

B. Baratte, S. Ruchaud, S. Bach, 2017 .

Phenytoin inhibits necroptosis

D. Green, A. Degterev, S. Bornstein, 2018, Cell Death & Disease.

Structure Activity Relationship Studies around DB18, a Potent and Selective Inhibitor of CLK Kinases

B. Baratte, S. Ruchaud, N. Levoin, 2022, Molecules.

Streptomyces hygroscopicus UFPEDA 3370: A valuable source of the potent cytotoxic agent nigericin and its evaluation against human colorectal cancer cells.

C. Peixoto, B. Baratte, A. Wisniewski, 2020, Chemico-biological interactions.

From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines

B. Baratte, E. Limanton, S. Ruchaud, 2018, Molecules.

From simple quinoxalines to potent oxazolo[5,4-f]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3).

Carlos Roca, C. Pérez, Ana Martínez, 2019, Organic & biomolecular chemistry.

The Canadian Prairie Plant Thermopsis rhombifolia Contains Luteolin, a Flavone that Inhibits Cyclin Dependent Kinase 9 and Arrest Cells in the G1-Phase of the Cell Cycle

F. Sautel, B. Baratte, R. Golsteyn, 2020 .

Comparison between Conventional and Nonconventional Methods for the Synthesis of Some 2-Oxazolidinone Derivatives and Preliminary Investigation of Their Inhibitory Activity Against Certain Protein Kinases

B. Baratte, S. Ruchaud, S. Bach, 2019, Russian Journal of Organic Chemistry.

Fused Systems Based on 2‐Aminopyrimidines: Synthesis Combining Deprotolithiation‐in situ Zincation with N‐Arylation Reactions and Biological Properties

O. Ivashkevich, B. Baratte, V. Dorcet, 2017 .

Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases

B. Baratte, J. Bazureau, S. Ruchaud, 2015, Molecules.

Biological Evaluation of Arylsemicarbazone Derivatives as Potential Anticancer Agents

B. Baratte, S. Ruchaud, M. Hernandes, 2019, Pharmaceuticals.

Synthesis, biological evaluation and molecular modeling studies of imidazo[1,2-a]pyridines derivatives as protein kinase inhibitors.

O. Lozach, B. Baratte, S. Ruchaud, 2016, European journal of medicinal chemistry.

Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases

F. Gouilleux, B. Baratte, F. McCarthy, 2021, Molecules.

Regorafenib analogues and their ferrocenic counterparts: synthesis and biological evaluation

L. Corcos, C. Le Jossic-Corcos, B. Baratte, 2020 .

Plasmodium falciparum glycogen synthase kinase-3: molecular model, expression, intracellular localisation and selective inhibitors.

Laurent Meijer, Virginie Thomas, Conrad Kunick, 2004, Biochimica et biophysica acta.

In vitro identification of imidazo[1,2-a]pyrazine-based antileishmanial agents and evaluation of L. major casein kinase 1 inhibition.

P. Le Pape, B. Baratte, N. Rachidi, 2020, European journal of medicinal chemistry.

Phenytoin inhibits necroptosis

D. Green, A. Degterev, S. Bornstein, 2018, Cell Death & Disease.

Tamoxifen inhibits CDK5 kinase activity by interacting with p35/p25 and modulates the pattern of tau phosphorylation.

K. Kosik, I. Landrieu, P. Colas, 2015, Chemistry & biology.

Structure and expression of three Emx genes in the dogfish Scyliorhinus canicula: functional and evolutionary implications.

D. Jaillard, J. Plouhinec, T. Sauka-Spengler, 2002, Developmental biology.

Roscovitine Targets, Protein Kinases and Pyridoxal Kinase*[boxs]

Lin Tang, Hervé Galons, Olivier Lozach, 2005, Journal of Biological Chemistry.

Tamoxifen Inhibits CDK 5 Kinase Activity by Interacting with p 35 / p 25 and Modulates the Pattern of Tau Phosphorylation Graphical

K. Kosik, I. Landrieu, P. Colas, 2015 .

Synthesis and biological evaluation of selected 7H-pyrrolo[2,3-d]pyrimidine derivatives as novel CDK9/CyclinT and Haspin inhibitors.

B. Baratte, S. Ruchaud, Richard M. Beteck, 2021, Chemico-biological interactions.

Molecular cloning and sequencing of the α-tubulin gene from Schistosoma mansoni

A. Capron, C. Dissous, B. Baratte, 1991 .

Molecular cloning and sequencing of the alpha-tubulin gene from Schistosoma mansoni.

A. Capron, C. Dissous, B. Baratte, 1991, Molecular and biochemical parasitology.

Purification of GSK-3 by affinity chromatography on immobilized axin.

F. Costantini, L. Meijer, A. Borgne, 2000, Protein expression and purification.

Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazines.

P. Le Pape, B. Baratte, S. Ruchaud, 2015, European journal of medicinal chemistry.

Functionalization of 9-thioxanthone at the 1-position: From arylamino derivatives to [1]benzo(thio)pyrano[4,3,2-de]benzothieno[2,3-b]quinolines of biological interest.

B. Baratte, V. Dorcet, R. Duval, 2019, Bioorganic chemistry.

Kinase-Based Screening of Marine Natural Extracts Leads to the Identification of a Cytotoxic High Molecular Weight Metabolite from the Mediterranean Sponge Crambe tailliezi

P. Colas, B. Baratte, S. Ruchaud, 2019, Marine drugs.

Molecular cloning and characterisation of p15(CDK-BP), a novel CDK-binding protein.

L. Meijer, B. Baratte, P. Léopold, 2002, Biochimica et biophysica acta.

Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinase.

B. Baratte, S. Ruchaud, T. Roisnel, 2020, Bioorganic & medicinal chemistry.

Suc1: cdc2 affinity reagent or essential cdk adaptor protein?

B. Baratte, L. Vogel, 1996, Progress in cell cycle research.

Isolation and characterization of authentic Phe-Met-Arg-Phe-NH2 and the novel Phe-Thr-Arg-Phe-NH2 peptide from Nereis diversicolor.

B. Baratte, P. Bulet, H. Gras-masse, 1991, European journal of biochemistry.

Sibiriline, a new small chemical inhibitor of receptor‐interacting protein kinase 1, prevents immune‐dependent hepatitis

P. Vandenabeele, M. Dimanche-Boitrel, B. Baratte, 2017, The FEBS journal.

Otx1 gene‐controlled morphogenesis of the horizontal semicircular canal and the origin of the gnathostome characteristics

D. Jaillard, P. Janvier, B. Baratte, 2000, Evolution & development.

Leucettines, a class of potent inhibitors of cdc2-like kinases and dual specificity, tyrosine phosphorylation regulated kinases derived from the marine sponge leucettamine B: modulation of alternative pre-RNA splicing.

L. Meijer, S. Knapp, O. Fedorov, 2011, Journal of medicinal chemistry.

6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury

P. Vandenabeele, M. Dimanche-Boitrel, B. Baratte, 2017, Scientific Reports.

Imidazo[1,2-a]quinazolines as novel, potent EGFR-TK inhibitors: Design, synthesis, bioactivity evaluation, and in silico studies.

B. Baratte, R. Esmaeili, A. Foroumadi, 2023, Bioorganic chemistry.

Characterization of Brachyury genes in the dogfish S. canicula and the lamprey L. fluviatilis. Insights into gastrulation in a chondrichthyan.

T. Sauka-Spengler, B. Baratte, M. Lepage, 2003, Developmental biology.

From Synthetic Simplified Marine Metabolite Analogues to New Selective Allosteric Inhibitor of Aurora B Kinase.

B. Baratte, J. Bignon, S. Ruchaud, 2021, Journal of medicinal chemistry.

6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury

P. Vandenabeele, M. Dimanche-Boitrel, B. Baratte, 2017, Scientific Reports.

New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis.

S. Knapp, A. Joerger, B. Baratte, 2019, European journal of medicinal chemistry.

Structure and expression of an Otx5-related gene in the dogfish Scyliorhinus canicula: evidence for a conserved role of Otx5 and Crx genes in the specification of photoreceptors

T. Sauka-Spengler, B. Baratte, D. Shi, 2001, Development Genes and Evolution.

Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity.

S. Knapp, A. Chaikuad, B. Baratte, 2022, European journal of medicinal chemistry.

Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration.

P. Le Pape, B. Baratte, S. Ruchaud, 2018, Bioorganic & medicinal chemistry letters.

Discovery of simplified benzazole fragments derived from the marine benzosceptrin B as necroptosis inhibitors involving the receptor interacting protein Kinase-1.

B. Baratte, S. Ruchaud, B. Iorga, 2020, European journal of medicinal chemistry.