B. McKeever

发表

Crystal Structure of Inhibitor-Bound Human 5-Lipoxygenase-Activating Protein

Jilly F. Evans, Shihua Xu, A. Ferguson, 2007, Science.

Positions of His‐64 and a bound water in human carbonic anhydrase II upon binding three structurally related inhibitors

J J Baldwin, J. Springer, G. M. Smith, 1994, Protein science : a publication of the Protein Society.

Modeling aided design of potent glycogen phosphorylase inhibitors.

R. Myers, B. McKeever, K. Chapman, 2005, Journal of molecular graphics & modelling.

Synthesis and antiviral activity of a series of HIV-1 protease inhibitors with functionality tethered to the P1 or P1' phenyl substituents: X-ray crystal structure assisted design.

P. Darke, W. Schleif, J. Quintero, 1992, Journal of Medicinal Chemistry.

New isomeric classes of topically active ocular hypotensive carbonic anhydrase inhibitors: 5-substituted thieno[2,3-b]thiophene-2-sulfonamides and 5-substituted thieno[3,2-b]thiophene-2-sulfonamides.

M. Murcko, J. Springer, P. Mallorga, 1991, Journal of medicinal chemistry.

Crystallographic analysis of a complex between human immunodeficiency virus type 1 protease and acetyl-pepstatin at 2.0-A resolution.

R. Dixon, J. Springer, P. Darke, 1991, The Journal of biological chemistry.

Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole core.

K. Fan, R. Gregg, Suresh B. Singh, 2016, Bioorganic & medicinal chemistry letters.

Discovery of a Novel, Orally Efficacious Liver X Receptor (LXR) β Agonist.

K. Fan, R. Gregg, Zhijie Liu, 2016, Journal of medicinal chemistry.

New Renin Inhibitor VTP-27999 Alters Renin Immunoreactivity and Does Not Unfold Prorenin

B. McKeever, A. Danser, M. Schalekamp, 2013, Hypertension.

Biphenyl/diphenyl ether renin inhibitors: filling the S1 pocket of renin via the S3 pocket.

R. Bentley, C. Doe, Suresh B. Singh, 2011, Bioorganic & medicinal chemistry letters.

Three-dimensional structure of aspartyl protease from human immunodeficiency virus HIV-1

M. Navia, J. Springer, P. Darke, 1989, Nature.

Structure-based design of β-site APP cleaving enzyme 1 (BACE1) inhibitors for the treatment of Alzheimer's disease.

Shankar Venkatraman, S. Venkatraman, Suresh B. Singh, 2013, Journal of medicinal chemistry.

Identification of spirooxindole and dibenzoxazepine motifs as potent mineralocorticoid receptor antagonists.

Suresh B. Singh, B. McKeever, Andrew P. Marcus, 2016, Bioorganic & medicinal chemistry.

Amino acid substitution of arginine 80 in 17beta-hydroxysteroid dehydrogenase type 3 and its effect on NADPH cofactor binding and oxidation/reduction kinetics.

R. Sheridan, B. McKeever, W. Geissler, 2002, Biochimica et biophysica acta.

Preliminary crystallographic data for protein S, a development-specific protein of Myxococcus xanthus.

S. Inouye, M. Inouye, B. McKeever, 1980, The Journal of biological chemistry.