R. B. Bakr

发表

Novel Phenolic Compounds as Potential Dual EGFR and COX-2 Inhibitors: Design, Semisynthesis, in vitro Biological Evaluation and in silico Insights

Atiah H. Almalki, M. Abdelgawad, A. Musa, 2021, Drug design, development and therapy.

Sulfonamide-based 4-anilinoquinoline derivatives as novel dual Aurora kinase (AURKA/B) inhibitors: Synthesis, biological evaluation and in silico insights.

M. Abdelgawad, Sami I. Alzarea, R. B. Bakr, 2020, Bioorganic & medicinal chemistry.

DESIGN AND SYNTHESIS OF NEW EGFR- TYROSINE KINASE INHIBITORS CONTAINING PYRAZOLO[3,4-d]PYRIMIDINE CORES AS ANTICANCER AGENTS

R. B. Bakr, Eman K. A. Abdelall, M. Abdel-Hamid, 2012 .

Efficient and Recoverable Bio-Organic Catalyst Cysteine for Synthesis, Docking Study, and Antifungal Activity of New Bio-Active 3,4-Dihydropyrimidin-2(1H)-ones/thiones Under Microwave Irradiation

R. B. Bakr, A. Kadry, Nadia A. A. Elkanzi, 2022, ACS omega.

Design, Synthesis, Molecular Docking of Novel Substituted Pyrimidinone Derivatives as Anticancer Agents

R. B. Bakr, A. F. El-Farargy, A. Ghoneim, 2020, Polycyclic Aromatic Compounds.

Docking Study, Synthesis, and Anti-Inflammatory Potential of Some New Pyridopyrimidine-Derived Compounds

M. Abdelgawad, A. Musa, M. Ghoneim, 2022, Journal of inflammation research.

New 1,2,3-Triazole-Containing Hybrids as Antitumor Candidates: Design, Click Reaction Synthesis, DFT Calculations, and Molecular Docking Study

R. B. Bakr, H. El‐Sheshtawy, Nadia Ali Ahmed Elkanzi, 2021, Molecules.

Design, Synthesis, Molecular Modeling Study, and Antimicrobial Activity of Some Novel Pyrano[2,3‐ b ]pyridine and Pyrrolo[2,3‐ b ]pyrano[2.3‐ d ]pyridine Derivatives

R. B. Bakr, Nadia Ali Ahmed Elkanzi, A. Ghoneim, 2018, Journal of Heterocyclic Chemistry.

Green Design, Synthesis, and Molecular Docking Study of Novel Quinoxaline Derivatives with Insecticidal Potential against Aphis craccivora

R. B. Bakr, W. Arafa, Hamud A. Altaleb, 2022, ACS omega.

Optimization of pyrazolo[1,5-a]pyrimidine based compounds with pyridine scaffold: Synthesis, biological evaluation and molecular modeling study

M. Abdelgawad, A. Musa, M. Ghoneim, 2022, Arabian Journal of Chemistry.

Pyrimidine and fused pyrimidine derivatives as promising protein kinase inhibitors for cancer treatment

R. B. Bakr, Khaled R. A. Abdellatif, R. Bakr, 2020, Medicinal Chemistry Research.

Thiochromene candidates: design, synthesis, antimicrobial potential and in silico docking study

R. B. Bakr, I. H. E. Azab, Nadia A. A. Elkanzi, 2021, Journal of the Iranian Chemical Society.

New advances in synthesis and clinical aspects of pyrazolo[3,4-d]pyrimidine scaffolds.

R. B. Bakr, Khaled R. A. Abdellatif, R. Bakr, 2018, Bioorganic chemistry.

Novel Β-lactams and Thiazolidinone Derivatives from 1,4-dihydroquinoxaline Schiff’s Base: Synthesis, Antimicrobial Activity and Molecular Docking Studies

R. B. Bakr, H. Hrichi, Nadia Ali Ahmed Elkanzi, 2020, Chemistry Journal of Moldova.

Design, synthesis and biological evaluation of some novel benzothiazole/benzoxazole and/or benzimidazole derivatives incorporating a pyrazole scaffold as antiproliferative agents.

M. Abdelgawad, R. B. Bakr, H. Omar, 2017, Bioorganic chemistry.

Synthesis and studies molecular docking of some new thioxobenzo[g]pteridine derivatives and 1,4-dihydroquinoxaline derivatives with glycosidic moiety

R. B. Bakr, A. Ghoneim, Nadia Ali Ahmed Elkanzi, 2018, Journal of Taibah University for Science.

Design, synthesis and antitumor activity of novel pyrazolo[3,4-d]pyrimidine derivatives as EGFR-TK inhibitors.

M. Abdelgawad, R. B. Bakr, Wafaa R. Mohamed, 2016, Bioorganic chemistry.

Novel indan-1, 3-diones derivatives: design, green synthesis, effect against tomato damping-off disease caused by Fusarium oxysporum and in silico molecular docking study

R. B. Bakr, W. Arafa, Nadia A. A. Elkanzi, 2022, Arabian Journal of Chemistry.

Preparation of some novel thiazolidinones, imidazolinones, and azetidinone bearing pyridine and pyrimidine moieties with antimicrobial activity

R. B. Bakr, Nadia Ali Ahmed Elkanzi, R. Bakr, 2020 .

Design, Synthesis, and In Silico Molecular Docking Study of Some Novel Thiochromene Derivatives with Antimicrobial Potential

R. B. Bakr, I. H. El Azab, Nadia A. A. Elkanzi, 2022, Polycyclic Aromatic Compounds.

Synthesis and Anticancer Activity of Some New Pyrazolo[3,4-d]pyrimidin-4-one Derivatives

M. Abdelgawad, R. B. Bakr, R. Ahmed, 2014, Molecules.

Antioxidant, Antimicrobial, and Molecular Docking Studies of Novel 1, 4-naphthoquinone Derivatives

R. B. Bakr, H. Hrichi, Nadia Ali Ahmed Elkanzi, 2021 .

Synthesis, in vitro evaluation and molecular docking of new pyrazole derivatives bearing 1,5,10,10a-tetrahydrobenzo[g]quinoline-3-carbonitrile moiety as potent antibacterial agents

R. B. Bakr, H. Hrichi, O. Hendawy, 2020, Journal of the Iranian Chemical Society.

New pyrimidine-benzoxazole/benzimidazole hybrids: Synthesis, antioxidant, cytotoxic activity, in vitro cyclooxygenase and phospholipase A2-V inhibition.

M. Abdelgawad, R. B. Bakr, W. Ahmad, 2019, Bioorganic chemistry.

Novel pyrimidine-pyridine hybrids: Synthesis, cyclooxygenase inhibition, anti-inflammatory activity and ulcerogenic liability.

M. Abdelgawad, R. B. Bakr, Amany A. Azouz, 2018, Bioorganic chemistry.

DDDT_A_310820 2325..2337

Atiah H. Almalki, M. Abdelgawad, A. Musa, 2021 .

Pyrimidine and fused pyrimidine derivatives as promising protein kinase inhibitors for cancer treatment

R. B. Bakr, Khaled R. A. Abdellatif, R. Bakr, 2020 .

Synthesis of Chalcones Derivatives and Their Biological Activities: A Review

R. B. Bakr, H. Hrichi, Wassila Derafa, 2022, ACS omega.

Targeting tumor cells with pyrazolo[3,4-d]pyrimidine scaffold: A literature review on synthetic approaches, structure activity relationship, structural and target-based mechanisms

M. Abdelgawad, A. Musa, R. B. Bakr, 2022, Arabian Journal of Chemistry.

Phthalazone tethered 1,2,3-triazole conjugates: In silico molecular docking studies, synthesis, in vitro antiproliferative, and kinase inhibitory activities.

M. Abdelgawad, A. Musa, M. Ghoneim, 2023, Bioorganic chemistry.