M. Bols

发表

Binding of serotonin to the human serotonin transporter. Molecular modeling and experimental validation.

L. Çelik, S. Sinning, K. Severinsen, 2008, Journal of the American Chemical Society.

β-Cyclodextrin as a mimetic of the natural GFP-chromophore environment

M. Bols, M. Cacciarini, M. Nielsen, 2012 .

QSAR studies and pharmacophore identification for arylsubstituted cycloalkenecarboxylic acid methyl esters with affinity for the human dopamine transporter.

S. Sinning, M. Bols, O. Wiborg, 2007, Bioorganic & medicinal chemistry.

Efficient synthesis of isofagomine and noeuromycin.

M. Bols, J. Andersch, 2001, Chemistry.

Synthesis and biological evaluation of potent glycosidase inhibitors: 4-deoxy-4,4-difluoroisofagomine and analogues

F. Qing, M. Bols, Xingang Zhang, 2009 .

Mechanisms of glycosylation reactions studied by low-temperature nuclear magnetic resonance.

M. Bols, Tobias Gylling Frihed, C. Pedersen, 2015, Chemical reviews.

β-Mannosylation with 4,6-benzylidene protected mannosyl donors without preactivation.

M. Bols, Tobias Gylling Frihed, Mads Heuckendorff, 2015, Chemical communications.

β-Selective mannosylation with a 4,6-silylene-tethered thiomannosyl donor.

M. Bols, J. Bendix, Mads Heuckendorff, 2014, Organic letters.

Conformationally armed 3,6-tethered glycosyl donors: synthesis, conformation, reactivity, and selectivity.

M. Bols, Mads Heuckendorff, C. Pedersen, 2013, The Journal of organic chemistry.

Influence of O6 in mannosylations using benzylidene protected donors: stereoelectronic or conformational effects?

G. A. van der Marel, M. Bols, M. Walvoort, 2013, The Journal of organic chemistry.

Synthesis of Shld Derivatives, Their Binding to the Destabilizing Domain, and Influence on Protein Accumulation in Transgenic Plants.

M. Meldal, M. Bols, M. Petersen, 2019, Journal of medicinal chemistry.

Hydrolysis of Toxic Natural Glucosides Catalyzed by Cyclodextrin Dicyanohydrins

M. Bols, E. H. Nielsen, J. Bjerre, 2008 .

Synthesis of L-Hexoses.

M. Bols, Tobias Gylling Frihed, C. Pedersen, 2015, Chemical reviews.

Silicon-Tethered Reactions

M. Bols, T. Skrydstrup, 1995 .

Processing Glucosidase Inhibition by 1-Azafagomine

M. Bols, A. Takatsuki, M. Muroi, 2000, Bioscience, biotechnology, and biochemistry.

Hydroxymethylation of aldonolactones and a chemical synthesis of 3-deoxy-3-fluoro-D-fructose

M. Bols, W. Szarek, Helle Grubbe, 1992 .

Combinatorial Chemistry of Piperidine Based Carbohydrate Mimics

M. Bols, J. Nielsen, M. Willert, 1997 .

An Inexpensive and Scalable Synthesis of Shld.

M. Bols, F. Jørgensen, 2018, The Journal of organic chemistry.

A Free-Energy Relationship between the Rate of Acidic Hydrolysis of Glycosides and the pKa of Isofagomines

M. Bols, Henrik H. Jensen, Laila Lyngbye, 2001 .

Imino- and azasugar protonation inside human acid β-glucosidase, the enzyme defective in Gaucher disease.

M. Bols, A. Morrone, C. Matassini, 2020, Angewandte Chemie.

Imino‐ and Azasugar Protonation Inside Human Acid β‐Glucosidase, the Enzyme that is Defective in Gaucher Disease

M. Bols, A. Morrone, C. Matassini, 2020, Angewandte Chemie.

Recognition of Peptides by Cyclodextrin Trimers

M. Bols, Lavinia G. Marinescu, Tobias Gylling Frihed, 2011 .

Synthesis of monofluorinated isofagomine analogues and evaluation as glycosidase inhibitors

F. Qing, M. Bols, Lavinia G. Marinescu, 2011 .

Stereoelectronic substituent effects in polyhydroxylated piperidines and hexahydropyridazines.

M. Bols, Henrik H. Jensen, A. Jensen, 2002, Chemistry.

Synthesis, inhibition and binding of simple non-nitrogen inhibitors of monoamine transporters.

S. Sinning, M. Bols, O. Wiborg, 2007, Bioorganic & medicinal chemistry.

Cyclodextrin ketones as oxidation catalysts: investigation of bridged derivatives.

M. Bols, Lavinia G. Marinescu, T. H. Fenger, 2009, Organic & biomolecular chemistry.

Aglycon mimicking: Glycoside bond cleavage transition state mimics based on hydroxypyrrolidine inhibitors

M. Sierks, M. Bols, I. Lundt, 1995 .

Total Synthesis of Five Lipoteichoic acids of Clostridium difficile.

D. Schwudke, H. Heine, M. Bols, 2014, Chemistry.

1‐Azafagomine: A Hydroxyhexahydropyridazine That Potently Inhibits Enzymatic Glycoside Cleavage

M. Bols, R. Hazell, I. Thomsen, 2001 .

Cyclodextrin Ketones with the Catalytic Group at the Secondary Rim and Their Effectiveness in Enzyme‐Like Epoxidation of Stilbenes

M. Bols, Lavinia G. Marinescu, T. H. Fenger, 2011 .

Investigation of the slow inhibition of almond beta-glucosidase and yeast isomaltase by 1-azasugar inhibitors: evidence for the 'direct binding' model.

M. Bols, I. Plesner, T. Hardlei, 2000, The Biochemical journal.

Effects of 4-deoxy-L-threo-pentose, a novel carbohydrate, on neural cell proteoglycan synthesis and function.

R. Riopelle, A. Lyon, K. Dow, 1992, Biochimica et biophysica acta.

Efficient stereocontrolled glycosidation of secondary sugar hydroxyls by silicon tethered intramolecular glycosidation

M. Bols, 1993 .

High dopamine transporter selectivity can be displayed by remarkably simple non-nitrogen containing inhibitors.

S. Sinning, M. Bols, O. Wiborg, 2007, Bioorganic & medicinal chemistry letters.

Synthesis of 3-C-hydroxymethyl- and 3-deoxyisofagomine and investigation of their binding to β-glucosidase

M. Bols, J. Duus, B. Petersen, 2000 .

Synthesis of All EightL-Glycopyranosyl Donors Using CH Activation

M. Bols, Tobias Gylling Frihed, C. Pedersen, 2014 .

Synthesis of all eight L-glycopyranosyl donors using C-H activation.

M. Bols, Tobias Gylling Frihed, C. Pedersen, 2014, Angewandte Chemie.

Isofagomine lactams, synthesis and enzyme inhibition.

M. Bols, Xifu Liang, Huizhen Liu, 2003, Organic & biomolecular chemistry.

Accurate determination of rate constants of very slow, tight-binding competitive inhibitors by numerical solution of differential equations, independently of precise knowledge of the enzyme concentration.

M. Bols, I. Plesner, A. Bülow, 2001, Analytical biochemistry.

Simple synthesis of (R)-Carnitine from d-Galactono-1,4-lactone

M. Bols, C. Pedersen, I. Lundt, 1992 .

Synthesis of Isofagomine Derivatives as New Fluorescence pH Indicators/Glycosidase Inhibitors

M. Bols, B. Laursen, Sidsel A Bogh, 2020 .

Evaluation of isofagomine and its derivatives as potent glycosidase inhibitors.

M. Sierks, M. Bols, T. Skrydstrup, 1996, Biochemistry.

Steric effects are not the cause of the rate difference in hydrolysis of stereoisomeric glycosides.

M. Bols, Henrik H. Jensen, 2003, Organic letters.

SYNTHETIC STUDIES OF FLUORINATED ANALOGUES OF 1-AZAFAGOMINE : REMARKABLE NUCLEOPHILIC SUBSTITUTION OF FLUORINE BY HYDRAZINE

M. Bols, I. Thomsen, B. V. Ernholt, 1997 .

Enzyme inhibition by iminosugars: analysis and insight into the glycosidase-iminosugar dependency of pH.

F. Qing, M. Bols, C. Pedersen, 2013, Bioorganic & medicinal chemistry.

Recent developments of transition-state analogue glycosidase inhibitors of non-natural product origin.

Mikael Bols, M. Bols, Xifu Liang, 2002, Chemical reviews.

1.21 – Glycosidase Inhibitors: Structure, Activity, Synthesis, and Medical Relevance

M. Bols, F. Ortega-Caballero, Ó. López, 2007 .

Synthesis of the 2‐Deoxyisomaltose Analogue of Acarbose by an Improved Route to Chiral Valieneamines

M. Bols, T. Tagmose, 2006 .

Carbohydrate Building Blocks

M. Bols, 1995 .

Easy access to L-mannosides and L-galactosides by using C-H activation of the corresponding 6-deoxysugars.

M. Bols, Tobias Gylling Frihed, Mads Heuckendorff, 2012, Angewandte Chemie.

Substitution of α-azido ethers with Grignard reagents and its use in combinatorial chemistry

M. Bols, Mukulesh Baruah, 2002 .

Superarming of glycosyl donors by combined neighboring and conformational effects.

A. Madsen, M. Bols, A. Demchenko, 2013, Organic letters.

Going to extremes: "super" armed glycosyl donors in glycosylation chemistry.

M. Bols, Henrik H. Jensen, C. Pedersen, 2007, Chemistry.

"Super armed" glycosyl donors: conformational arming of thioglycosides by silylation.

M. Bols, L. U. Nordstrøm, C. Pedersen, 2007, Journal of the American Chemical Society.

Stereoelectronic substituent effects.

Mikael Bols, M. Bols, Henrik Helligsø Jensen, 2006, Accounts of chemical research.

Conformationally armed glycosyl donors: reactivity quantification, new donors and one pot reactions.

M. Bols, Lavinia G. Marinescu, C. Pedersen, 2008, Chemical communications.

Glycosyl donors in “unusual” conformations – influence on reactivity and selectivity

M. Bols, Lavinia G. Marinescu, C. Pedersen, 2011 .

Silylated Sugars – Synthesis and Properties

M. Bols, Tobias Gylling Frihed, M. Pedersen, 2021, Synlett.

The disarming effect of the 4,6-acetal group on glycoside reactivity: torsional or electronic?

M. Bols, L. U. Nordstrøm, Henrik H. Jensen, 2004, Journal of the American Chemical Society.

Equatorial contra axial polar substituents. The relation of a chemical reaction to stereochemical substituent constants.

M. Bols, Xifu Liang, Henrik H. Jensen, 2002, The Journal of organic chemistry.

Direct experimental evidence for the high chemical reactivity of α- and β-xylopyranosides adopting a (2,5)B conformation in glycosyl transfer.

J. Marrot, M. Bols, M. Sollogoub, 2011, Chemistry.

Synthesis and investigation of L-fuco- and D-glucurono-azafagomine

M. Bols, Henrik H. Jensen, R. Hazell, 2002 .

Synthesis of 3-substituted isofagomine analogues using an unusual syn hydrogenation reaction

M. Bols, P. Bach, A. Lohse, 2000 .

Chemoenzymatic Synthesis of Enantiopure 1-Azafagomine

M. Bols, Xifu Liang, 1999 .

Synthesis of labelled 1-azafagomine

M. Bols, S. Hansen, 1999 .

Radical azidonation of aldehydes.

M. Bols, Lavinia G. Marinescu, Jacob Thinggaard, 2003, The Journal of organic chemistry.

Noeuromycin, a glycosyl cation mimic that strongly inhibits glycosidases.

M. Bols, Xifu Liang, H. Søhoel, 2001, Journal of the American Chemical Society.

Garner's aldehyde

M. Bols, Xifu Liang, J. Andersch, 2002 .

A new and convenient benzyloxyalkylating agent induced by samarium diiodide

M. Bols, T. Skrydstrup, J. Beau, 1996 .

Taming of the DIBAL Promoted Debenzylation of α‐Cyclodextrin. Kinetics, Substituent Effects and Efficient Synthesis of Lings Tetrol

M. Bols, Victor Friis, 2022, Chemistry.

C–H Functionalization on Carbohydrates

M. Bols, Tobias Gylling Frihed, C. Pedersen, 2016 .

New cup-shaped α-cyclodextrin derivatives and a study of their catalytic properties in oxidation reactions

M. Bols, Lavinia G. Marinescu, Ó. López, 2007 .

Very high rate enhancement of benzyl alcohol oxidation by an artificial enzyme.

M. Bols, Lavinia G. Marinescu, 2006, Angewandte Chemie.

Artificial glycosyl phosphorylases.

M. Bols, F. Ortega-Caballero, B. Christensen, 2005, Chemistry.

Four orders of magnitude rate increase in artificial enzyme-catalyzed aryl glycoside hydrolysis.

M. Bols, F. Ortega-Caballero, J. Bjerre, 2005, The Journal of organic chemistry.

Artificial Epoxidase II. Synthesis of Cyclodextrin Ketoesters and Epoxidation of Alkenes

M. Bols, B. Christensen, C. Rousseau, 2005 .

Remarkable supramolecular catalysis of glycoside hydrolysis by a cyclodextrin cyanohydrin.

M. Bols, F. Ortega-Caballero, B. Christensen, 2005, Journal of the American Chemical Society.

Substrate control through per-O-methylation of cyclodextrin acids.

M. Bols, T. H. Fenger, 2010, Chemical communications.

Amino–Acetone-Bridged Cyclodextrins ― Artificial Alcohol Oxidases

M. Bols, Lavinia G. Marinescu, A. Fernández-Mayoralas, 2010 .

Silicon-Tethered Reactions

M. Bols, T. Skrydstrup, 1995 .

Synthesis of the first pseudosugar-C-disaccharide. A potential antigen for eliciting glycoside-bond forming antibodies with catalytic groups

M. Sierks, M. Bols, I. Lundt, 1995 .

Glycosyl Fluorides as Intermediates in BF3·OEt2‐Promoted Glycosylation with Trichloroacetimidates

M. Bols, C. Pedersen, M. Nielsen, 2017 .

Quantifying the electronic effects of carbohydrate hydroxy groups by using aminosugar models.

M. Bols, C. Pedersen, J. Olsen, 2011, Chemistry.

Simple Synthesis of beta-D-Glucosyl Esters.

M. Bols, G. Widmalm, L. Hubert-Pfalzgraf, 1993 .

Synthesis of isofagomine, a novel glycosidase inhibitor

M. Sierks, M. Bols, T. Skrydstrup, 1994 .

Radical substitution with azide: TMSN3-PhI(OAc)2 as a substitute of IN3.

M. Bols, Lavinia G. Marinescu, C. Pedersen, 2005, Organic & biomolecular chemistry.

1-Aza Sugars, Apparent Transition State Analogues of Equatorial Glycoside Formation/Cleavage

M. Bols, 1998 .

SYNTHESIS OF TRIBUTYLTINMETHYLATED SUGARS, BUILDING BLOCKS FOR TETHERED REACTIONS

M. Bols, O. Hindsgaul, H. C. Hansen, 1996 .

Selenoureido-iminosugars: A new family of multitarget drugs.

J. Fernández-Bolaños, M. Bols, J. Padrón, 2016, European journal of medicinal chemistry.

Zinc and Copper Complexes of Methylated Di- and Tetraaminocyclodextrins

M. Bols, Julia Warren, 2019, European Journal of Organic Chemistry.

Artificial Metallooxidases from Cyclodextrin Diacids.

M. Bols, Bo Wang, 2017, Chemistry.

Synthesis of Cyclodextrins with Carboxylic Acids at the Secondary Rim and an Evaluation of Their Properties as Chemzymes for Glycoside Hydrolysis

M. Bols, Lavinia G. Marinescu, Emil Lindbäck, 2012 .

Cyclodextrin derivatives that display Enzyme Catalysis

M. Bols, Lavinia G. Marinescu, 2009 .

Cyclodextrin-based artificial oxidases with high rate accelerations and selectivity

M. Bols, Emil Lindbäck, C. Pedersen, 2014 .

Artificial enzyme activity from cyclodextrins with cyanohydrins on the secondary rim

M. Bols, C. Pedersen, You Zhou, 2013 .

Synthesis of Tin‐Containing Cyclodextrins as Potential Enzyme Models

M. Bols, Lavinia G. Marinescu, C. Pedersen, 2012 .

Two Diastereomeric Artificial Enzymes with Different Catalytic Activity

M. Bols, Emil Lindbäck, C. Pedersen, 2012 .

Simple cyclodextrin aldehydes as excellent artificial oxidases

M. Bols, T. H. Fenger, 2011 .

Substantial Spatial Flexibility and Hydrogen Bonding within the Catalysis Exerted by Cyclodextrin Artificial Glycosidases

M. Bols, J. Bjerre, 2010 .

Cyclodextrin Aldehydes are Oxidase Mimics

M. Bols, J. Bjerre, Thomas Hauch Fenger, 2009, Chembiochem : a European journal of chemical biology.

Selective discrimination of cyclodextrin diols using cyclic sulfates.

M. Bols, Lavinia G. Marinescu, C. Rousseau, 2009, Organic letters.

Synthesis of an 1-azaglucose analogue with ring-oxygen retained

M. Bols, P. Bach, 1999 .

Determination of protonation states of iminosugar–enzyme complexes using photoinduced electron transfer† †Electronic supplementary information (ESI) available: NMR spectra of new compounds, experimental details and Fig. S1–S5 (19 pages). See DOI: 10.1039/c7sc01540b Click here for additional data fil

M. Bols, B. Laursen, J. Navarro Poulsen, 2017, Chemical science.

A fluorescence study of isofagomine protonation in β-glucosidase.

M. Bols, B. Laursen, K. Kilså, 2015, Organic & biomolecular chemistry.

Synthesis of 5-azacastanospermine, a conformationally restricted azafagomine analogue.

M. Bols, X. Liang, K. Søndergaard, 2001, Chemistry.

Synthesis of furan 4'-thio-C-nucleosides, their methylsulfonium and sulfoxide derivatives. Evaluation as glycosidase inhibitors

J. Fernández-Bolaños, M. Bols, I. Maya, 2003 .

Silyl-protective groups influencing the reactivity and selectivity in glycosylations

M. Bols, C. Pedersen, 2017, Beilstein journal of organic chemistry.

Intramolecular Glycosidation: Stereocontrolled Synthesis of alpha-Glucosides from a 2-O-Alkoxysilyl Thioglucoside.

E. Pedersen, O. Buchardt, M. Bols, 1993 .

Investigation of the base promoted tandem syn-elimination–Favorskii rearrangement of levoglucosan sulfonates

M. Bols, R. Hazell, I. Thomsen, 2002 .

New branched carbohydrate building block from a tandem elimination-Farvorski rearrangement

M. Bols, 1998 .

Synthesis of 6-deoxy-6-phenylisofagomine derivatives

M. Bols, A. Lohse, 1997 .

Synthesis of kojitriose using silicon-tethered glycosidation.

M. Bols, 1996, Acta chemica Scandinavica.

Long Range Intramolecular Glycosidation

M. Bols, H. C. Hansen, 1994 .

Application of intramolecular glycosidation to the stereocontrolled synthesis of disaccharides containing α-gluco and α-galacto linkages

M. Bols, 1993 .

Stereocontrolled synthesis of α-glucosides by intramolecular glycosidation

M. Bols, 1992 .

Synthesis of All Eight Stereoisomeric 6‐Deoxy‐L‐hexopyranosyl Donors – Trends in Using Stereoselective Reductions or Mitsunobu Epimerizations

M. Bols, Tobias Gylling Frihed, C. Pedersen, 2014 .

Chemoenzymatic synthesis of isogalactofagomine.

M. Bols, A. Lohse, X. Liang, 2000, The Journal of organic chemistry.

A New Intramolecular Reaction for the Regioselective Debenzylation or Protection of Alcohols.

M. Bols, J. Madsen, 1998, Angewandte Chemie.

Synthesis and evaluation of sulfonium analogues of isofucofagomine as glycosidase inhibitors

J. Fernández-Bolaños, M. Bols, Victor Ulgar, 2002 .

Safe radical azidonation using polystyrene supported diazidoiodate(I)

M. Bols, Lavinia G. Marinescu, C. Pedersen, 2005 .

Combinatorial synthesis of benztropine libraries and their evaluation as monoamine transporter inhibitors.

S. Sinning, M. Bols, O. Wiborg, 2004, Organic & biomolecular chemistry.

Substitution of α‐Azido Ethers with Grignard Reagents and Its Use in Combinatorial Chemistry.

M. Bols, Mukulesh Baruah, 2002 .

Synthesis and Thermotropic Phase Behavior of Four Glycoglycerolipids

M. Bols, T. Pomorski, M. Cárdenas, 2013, Molecules.

Effective synthesis of negatively charged cyclodextrins. Selective access to phosphate cyclodextrins

M. Bols, Ó. López, 2008 .

Artificial enzymes, “Chemzymes”: current state and perspectives

M. Bols, Lavinia G. Marinescu, C. Rousseau, 2008, Applied Microbiology and Biotechnology.

1-Azaribofuranoside analogues as designed inhibitors of purine nucleoside phosphorylase. Synthesis and biological evaluation.

M. Bols, S. Hansen, 1998, Acta chemica Scandinavica.

Synthesis of Some Trifluoromethylated Cyclodextrin Derivatives and Analysis of Their Properties as Artificial Glycosidases and Oxidases

M. Bols, Lavinia G. Marinescu, T. H. Fenger, 2007 .

Synthesis of 5‐Bromomethylfurfural from Cellulose as a Potential Intermediate for Biofuel

M. Bols, Nitee Kumari, C. Pedersen, 2011 .

3-Deoxy-glucosone is an intermediate in the formation of furfurals from D-glucose.

M. Bols, T. Sølling, H. Jadhav, 2011, ChemSusChem.

Conversion of d-glucose into 5-hydroxymethylfurfural (HMF) using zeolite in [Bmim]Cl or tetrabutylammonium chloride (TBAC)/CrCl2

Esben Taarning, M. Bols, C. Pedersen, 2012 .

Preparation of 2,3-Epoxyaldonolactones and their Conversion into 2-Fluoro-2-deoxy-aldonolactones and -sugars.

D. Aksnes, M. Bols, H. Tønnesen, 1990 .

Conformationally superarmed S-ethyl glycosyl donors as effective building blocks for chemoselective oligosaccharide synthesis in one pot.

M. Bols, J. P. Yasomanee, A. Demchenko, 2017, Organic & biomolecular chemistry.

Solution-phase combinatorial synthesis using multicomponent Grignard reagents

M. Bols, Xifu Liang, 2002 .

Influence of monosaccharide derivatives on liver cell glycosaminoglycan synthesis: 3-deoxy-D-xylo-hexose (3-deoxy-D-galactose) and methyl (methyl 4-chloro-4-deoxy-beta-D-galactopyranosid) uronate.

M. Bols, W. Szarek, W. Zou, 1995, Biochimica et biophysica acta.

Quantifying electronic effects of common carbohydrate protecting groups in a piperidine model system.

M. Bols, Mads Heuckendorff, C. Pedersen, 2010, Chemistry.

An isofagomine analogue with an amidine at the pseudoanomeric position.

J. Fernández-Bolaños, M. Bols, S. Sauer, 2011, Organic letters.

SYNTHESIS OF A RIBOFURANOSYL CATION MIMIC

Martin Felix Jørgensen, M. Bols, M. Persson, 1996 .

Synthesis of a new potent α-fucosidase inhibitor

M. Bols, T. Tagmose, Anja Hansen, 1996 .

On the nature of the electronic effect of multiple hydroxyl groups in the 6-membered ring - the effects are additive but steric hindrance plays a role too.

M. Bols, C. Pedersen, 2017, Organic & biomolecular chemistry.

Super arming of a glycosyl donor using a molecular lever

M. Bols, C. Pedersen, K. Kowalska, 2016 .

Stereochemical substituent effects: investigation of the cyano, amide and carboxylate group

M. Bols, C. Pedersen, 2005 .

Conformational effects on glycoside reactivity: study of the high reactive conformer of glucose.

M. Bols, C. McDonnell, R. Hazell, 2004, Journal of the American Chemical Society.

A Large Difference in the Thermodynamics of Binding of Isofagomine and 1-Deoxynojirimycin to β-Glucosidase

M. Bols, A. Bülow, and Igor W. Plesner, 2000 .

A uronic acid analogue of isofagomine lactam as a nanomolar glucuronidase inhibitor

J. Fernández-Bolaños, M. Bols, Emil Lindbäck, 2012 .

Slow inhibition of almond beta-glucosidase by azasugars: determination of activation energies for slow binding.

M. Bols, I. Plesner, A. Bülow, 2001, Biochimica et biophysica acta.

Isogalactofagomine lactam. A neutral nanomolar galactosidase inhibitor

M. Bols, Xifu Liang, H. Søhoel, 2001 .

Synthesis of 1-azagalactofagomine, a potent galactosidase inhibitor

M. Bols, Henrik H. Jensen, 2001 .

Synthesis of (±)-isofagomine and its stereoisomers from arecoline

M. Bols, S. Hansen, 2000 .

Synthesis and deconvolution of the first combinatorial library of glycosidase inhibitors.

M. Bols, K. Lundgren, K. B. Jensen, 1999, Bioorganic & medicinal chemistry.

THE FIRST COMBINATORIAL LIBRARY OF AZASUGAR GLYCOSIDASE INHIBITORS

M. Bols, K. B. Jensen, A. Lohse, 1999 .

Anomer‐Selective Glycosidase Inhibition by 2‐N‐Alkylated 1‐Azafagomines

M. Bols, Oscar Lopez Lopez, 2007, Chembiochem : a European journal of chemical biology.

Synthesis of a New Potent α‐Fucosidase Inhibitor.

M. Bols, T. Tagmose, Anja Hansen, 2010 .

Recent Developments of Transition‐State Analogue Glycosidase Inhibitors of Non‐Natural Product Origin

M. Bols, Xifu Liang, Henrik H. Jensen, 2010 .

The C-4 Configuration as a Probe for the Study of Glycosidation Reactions

M. Bols, T. Olszewski, A. Bülow, 2004 .

The influence of neighboring group participation on the hydrolysis of 2-O-substituted methyl glucopyranosides.

M. Bols, Mads Heuckendorff, C. Pedersen, 2011, Organic Letters.

Going to Extremes: “Super” Armed Glycosyl Donors in Glycosylation Chemistry

M. Bols, Henrik H. Jensen, C. Pedersen, 2007 .

Exploring the relationship between the conformation and pKa: can a pKa value be used to determine the conformational equilibrium?

M. Bols, S. Sauer, Christian Marcus Pedersen, 2015, Organic & biomolecular chemistry.

Rhamnosylation: diastereoselectivity of conformationally armed donors.

M. Bols, Mads Heuckendorff, C. Pedersen, 2012, The Journal of organic chemistry.

On the electronic effects of OH groups. Synthesis and investigation of tetrahydroxylated azabicycloheptanes.

M. Bols, Henrik H. Jensen, C. Pedersen, 2005, Organic & biomolecular chemistry.

A study of anhydrocelluloses--is a cellulose structure with residues in a 1C4-conformation more prone to hydrolysis?

M. Bols, C. Pedersen, V. Jadhav, 2011, Organic & biomolecular chemistry.

Synthesis and biological evaluation of glycosidase inhibitors: gem-difluoromethylenated nojirimycin analogues.

F. Qing, M. Bols, F. Ortega-Caballero, 2006, Journal of medicinal chemistry.

Enantiospecific synthesis of 1-azafagomine.

M. Bols, R. Hazell, K. B. Jensen, 2000, Chemistry.

Synthesis and Chemistry of Noeuromycin and Isofagomine Analogues

M. Bols, Xifu Liang, J. Andersch, 2004 .

Active Site Protonation of 1‐Azafagomine in Glucosidases Studied by Solid‐State NMR Spectroscopy

N. Nielsen, M. Bols, M. Bjerring, 2007 .

Synthesis and Chemistry of Noeuromycin and Isofagomine Analogues.

M. Bols, Xifu Liang, J. Andersch, 2005 .

Isogalactofagomine Lactam. A Neutral Nanomolar Galactosidase Inhibitor.

M. Bols, Xifu Liang, Helmer Soehoel, 2001 .

Synthesis of 1‐Azagalactofagomine, a Potent Galactosidase Inhibitor.

M. Bols, Henrik H. Jensen, 2001 .

Synthesis of (.+-.)-Isofagomine and Its Stereoisomers from Arecoline.

M. Bols, S. Hansen, 2000 .

Azafagomine hydrazones: an argument against a “Flat” transition state in glycoside cleavage

M. Bols, S. Hansen, 2000 .

Specific Glycosidase Activity Isolated from a Random Phage Display Antibody Library

M. Sierks, M. Bols, G. Goud, 2001, Biotechnology progress.

Aziridines as a structural motif to conformational restriction of azasugars.

J. Fernández-Bolaños, M. Bols, Vinni H. Lillelund, 2003, Organic & biomolecular chemistry.

The role of the active site Zn in the catalytic mechanism of the GH38 Golgi α-mannosidase II: Implications from noeuromycin inhibition

D. Kuntz, M. Bols, D. Rose, 2006 .

Preparation of 2-, 3-, and 4-deoxy derivatives of L-rhamnose, and derivatives of 2-azido-2-deoxy-L-rhamnose and 2,6-dideoxy-2-fluoro-L-glucose, for use in glycosylation reactions.

M. Bols, E. Ottosen, I. Lundt, 1991, Carbohydrate research.

A study of the DIBAL-promoted selective debenzylation of α-cyclodextrin protected with two different benzyl groups

M. Bols, Naser Yousefi, Morten L Zimmermann, 2022, Beilstein journal of organic chemistry.

Isofagomine, Noeuromycin and other 1‐Azasugars, Iminosugar‐Related Glycosidase Inhibitors

M. Bols, Ó. López, 2008 .

beta-Selectivity of Sterically Hindered Acyl Chlorides in the Acylation of 2,3,4,6-Tetra-O-benzyl-alpha-D-glucopyranose.

B. Roos, M. Bols, Harri Setälä, 1993 .

An artificial enzyme that catalyzes hydrolysis of aryl glycosides

M. Bols, C. Rousseau, N. Nielsen, 2004 .

A bioisosteric oligosaccharide mimetic based on isofagomine-type monomers

M. Bols, J. Duus, Xifu Liang, 2001 .

Difluoromethylenated polyhydroxylated pyrrolidines: facile synthesis, crystal structure and biological evaluation.

F. Qing, M. Bols, Jun Xu, 2009, Future medicinal chemistry.

ALPHA - OR BETA -AMINO POLYHYDROXY ACIDS FROM THE REACTION OF BROMODEOXYALDONOLACTONES WITH LIQUID AMMONIA

M. Bols, I. Lundt, 1991 .

α- or β-Amino Polyhydroxy Acids from the Reaction of Bromodeoxyaldonolactones with Liquid Ammonia.

M. Bols, I. Lundt, 1991 .

Cyclodextrins containing an acetone bridge. Synthesis and study as epoxidation catalysts.

M. Bols, B. Christensen, T. E. Petersen, 2004, Organic & biomolecular chemistry.

The Grignard Reaction of Cyclodextrin‐6‐aldehydes Revisited: A Study of the Stereoselectivity Upon Addition of Organometallic Reagents to Aldehydes and Ketones

M. Bols, Lavinia G. Marinescu, Emil Lindbäck, 2010 .

Synthesis of L‐Hexoses

M. Bols, Tobias Gylling Frihed, C. Pedersen, 2015 .

An Azido-Hanessian Reaction

M. Bols, Mukulesh Baruah, 2002 .

Radical Azidonation of Benzylic Positions with Iodonium Azide.

M. Bols, Christel Viuf, 2001, Angewandte Chemie.

Binding and Orientation of Tricyclic Antidepressants within the Central Substrate Site of the Human Serotonin Transporter*

L. Çelik, S. Sinning, K. Severinsen, 2009, The Journal of Biological Chemistry.

alpha-Amino Polyhydroxy Tetronic and Pentonic Acids from Bromodeoxyaldonolactones.

I. Pelczer, M. Bols, H. Lönnberg, 1988 .

Two- and three dimensional combinatorial chemistry from multicomponent Grignard reagents.

S. Sinning, M. Bols, O. Wiborg, 2004, Journal of combinatorial chemistry.

Supramolecular oxidation of anilines using hydrogen peroxide as stoichiometric oxidant.

M. Bols, Lavinia G. Marinescu, C. Rousseau, 2005, Journal of the American Chemical Society.

Short synthesis of piperidine based hexopyranose minics. A remarkable example of syn hydrogenation

M. Bols, P. Bach, A. Lohse, 1999 .

Cyclodextrin‐Based Artificial Enzymes: Synthesis and Function

M. Bols, C. Pedersen, 2013 .

Attachment of cyclodextrin acids to PEGA resin and study of binding with fluorescence microscopy.

M. Meldal, M. Bols, Bo Wang, 2021, Bioorganic & Medicinal Chemistry Letters.

Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12.

M. Meldal, M. Bols, M. Roux, 2020, ACS combinatorial science.

Methane capture with α-cyclodextrins

M. Bols, J. Bendix, H. Bordallo, 2023, New Journal of Chemistry.

Artificial enzymes based on cyclodextrin with phenol as the catalytic group

M. Bols, Emil Lindbäck, C. Pedersen, 2012 .

Radical azidonation of aldehydes.

M. Bols, Lavinia G. Marinescu, Jacob Thinggaard, 2003, The Journal of organic chemistry.

Intramolecular Glycosidation Reactions

G. Hart, B. Ernst, M. Bols, 2008 .

The structure of afragilimycin A.

M. Bols, A. Ocaktan, N. Andersen, 1991, The Journal of antibiotics.

Binding and Orientation of Tricyclic Antidepressants within the Central Substrate Site of the Human Serotonin Transporter*

L. Çelik, S. Sinning, K. Severinsen, 2009, The Journal of Biological Chemistry.

Stereoelectronic substituent effects in polyhydroxylated piperidines and hexahydropyridazines.

M. Bols, Henrik H. Jensen, A. Jensen, 2002, Chemistry.

Quantifying electronic effects of common carbohydrate protecting groups in a piperidine model system.

M. Bols, Mads Heuckendorff, C. Pedersen, 2010, Chemistry.

Conformationally armed glycosyl donors: reactivity quantification, new donors and one pot reactions.

M. Bols, Lavinia G. Marinescu, C. Pedersen, 2008, Chemical communications.

Binding of serotonin to the human serotonin transporter. Molecular modeling and experimental validation.

L. Çelik, S. Sinning, K. Severinsen, 2008, Journal of the American Chemical Society.

Radical Azidonation of Benzylic Positions with Iodonium Azide.

M. Bols, Christel Viuf, 2001, Angewandte Chemie.

Inhibition of collagenase by aranciamycin and aranciamycin derivatives.

L. Binderup, M. Bols, P. Rasmussen, 1992, Journal of medicinal chemistry.