G. Giacomelli

发表

Formic Acid: A Promising Bio‐Renewable Feedstock for Fine Chemicals

M. Mura, L. D. Luca, G. Giacomelli, 2012 .

Solution‐Phase Synthesis of Mixed Amide Libraries by Simultaneous Addition of Functionalities (SPSAF) to a Diketopiperazine Tetracarboxylic Acid Scaffold Monitored by GC Analysis of Isobutyl Alcohol

G. Giacomelli, A. Porcheddu, M. Taddei, 2000 .

NEW 1,3,5-TRIAZINE DERIVATIVES AS TEMPLATES FOR THE HOMOGENEOUS PHASE SYNTHESIS OF CHEMICAL LIBRARIES

G. Giacomelli, A. Porcheddu, M. Falorni, 1998 .

Synthesis of Oximes and Hydroxamic Acids

G. Giacomelli, A. Porcheddu, 2010 .

Mild and highly selective formyl protection of primary hydroxyl groups.

G. Giacomelli, A. Porcheddu, L. De Luca, 2002, The Journal of organic chemistry.

1,3,5-Triazines

G. Giacomelli, A. Porcheddu, Giampaolo Giacomelli, 2008 .

New Oxazole‐Based Conformationally Restricted Peptidomimetics: Design and Synthesis of Pseudopeptides

G. Giacomelli, A. Porcheddu, G. Dettori, 2000 .

Microwave‐Assisted Solution‐Phase Synthesis of 1,4,5‐Trisubstituted Pyrazoles

G. Giacomelli, A. Porcheddu, M. Taddei, 2003 .

NEW 1,3,5-TRIAZINE DERIVATIVES AS TEMPLATES FOR THE HOMOGENEOUS PHASE SYNTHESIS OF CHEMICAL LIBRARIES

G. Giacomelli, A. Porcheddu, M. Falorni, 1998 .

A Practical and Efficient Approach to PNA Monomers Compatible with Fmoc-Mediated Solid-Phase Synthesis Protocols†

M. Carta, G. Giacomelli, A. Porcheddu, 2008 .

A microwave assisted synthesis of benzoxazoles from carboxylic acids

G. Giacomelli, Giammario Nieddu, 2013 .

An Insight of the Reactions of Amines with Trichloroisocyanuric Acid.

L. D. Luca, G. Giacomelli, L. Luca, 2004 .

Chiral ligands containing heteroatoms. 10. 1-(2-pyridyl)alkylamines as chiral catalysts in the addition of diethylzinc to aldehydes: temperature dependence on the enantioselectivity.

G. Giacomelli, M. Falorni, S. Conti, 1992 .

Alkylmetal asymmetric reduction. 18. Starting materials in the preparation of new chiral reducing agents: synthetic approach to primary alkyl halides derived from (+)-camphor

G. Giacomelli, M. Falorni, L. Lardicci, 1986 .

Peptide nucleic acids (PNAs), a chemical overview.

G. Giacomelli, A. Porcheddu, 2005, Current medicinal chemistry.

Simple one-flask method for the preparation of hydroxamic acids.

G. Giacomelli, A. Porcheddu, M. Salaris, 2003, Organic letters.

Synthesis of Optically Active α-Amino Acids Containing Pyrazolyl Ring as Substituent

L. D. Luca, G. Giacomelli, A. Porcheddu, 2000 .

New pyrazole containing bicarboxylic α-amino acids: mimics of the cis amide bond

L. D. Luca, G. Giacomelli, A. Porcheddu, 1999 .

Chiral ligands containing heteroatoms:13. Optically active 4-(2′-pyridyl)-1,3-oxazolidines: An improved synthesis of 2-(2′-pyridyl)-2-aminoalcohols

G. Giacomelli, S. Cossu, M. Falorni, 1994 .

Synthesis of (−)-(S)-3-sec-butyl- and (+)-(S)-5-sec-butyl-2(1H)-pyridinone

G. Giacomelli, G. Chelucci, 1990 .

Trichloroisocyanuric/TEMPO oxidation of alcohols under mild conditions: a close investigation.

G. Giacomelli, A. Porcheddu, L. De Luca, 2003, The Journal of organic chemistry.

A "catch and release" strategy for the parallel synthesis of 2,4,5-trisubstituted pyrimidines.

G. Giacomelli, A. Porcheddu, L. De Luca, 2004, Journal of combinatorial chemistry.

Preparation of pyrazole and isoxazole libraries on cellulose beads: a new cheap and versatile biopolymer

L. D. Luca, G. Giacomelli, A. Porcheddu, 2003 .

Beckmann rearrangement of oximes under very mild conditions.

G. Giacomelli, A. Porcheddu, L. De Luca, 2002, The Journal of organic chemistry.

Synthesis of 1-Substituted 2-((2S)-2-Pyrrolidinyl)pyridine from L- Proline.

G. Giacomelli, M. Falorni, G. Chelucci, 1990 .

Synthesis of (2R, 5S)- and (2S, 5S)-2-carboxy-1,4-diaza-[4.3.0]bicyclononane as building blocks for the synthesis of new potential HIV protease inhibitors

G. Giacomelli, A. Porcheddu, M. Falorni, 1996 .

Chiral ligands containing heteroatoms. 11. Optically active 2-hydroxymethyl piperazincs as catalysts in the enantioselective addition of diethylzinc to benzaldehyde

G. Giacomelli, M. Falorni, M. Satta, 1993 .

Angeli-Rimini's reaction on solid support: a new approach to hydroxamic acids.

G. Giacomelli, A. Porcheddu, 2006, The Journal of organic chemistry.

Synthesis of 1-alkyl-4-imidazolecarboxylates: a catch and release strategy.

G. Giacomelli, A. Porcheddu, L. De Luca, 2005, Journal of combinatorial chemistry.

Microwave-assisted synthesis of isonitriles: a general simple methodology.

G. Giacomelli, A. Porcheddu, M. Salaris, 2005, The Journal of organic chemistry.

Alkyl metal asymmetric reduction. 11. The reaction of α,β-unsaturated ketones with β-branched trialkylaluminium compounds.

G. Giacomelli, A. Caporusso, L. Lardicci, 1981 .

Parallel synthesis of trisubstituted formamidines: a facile and versatile procedure.

G. Giacomelli, A. Porcheddu, Ivana Piredda, 2009, Journal of combinatorial chemistry.

An easy and convenient synthesis of Weinreb amides and hydroxamates.

G. Giacomelli, M. Taddei, L. De Luca, 2001, The Journal of organic chemistry.

[1,3,5]-Triazine: A Versatile Heterocycle in Current Applications of Organic Chemistry

L. D. Luca, G. Giacomelli, A. Porcheddu, 2004 .

Alkylmetal asymmetric reduction. 13. A sterically crowded chiral organoaluminum compound as a reducing agent of ketones

G. Giacomelli, L. Lardicci, F. Palla, 1984 .

Alkylmetal asymmetric reduction. 9. Asymmetric reduction of alkyl phenyl ketones by sterically hindered chiral organoaluminum compounds

G. Giacomelli, A. Caporusso, R. Menicagli, 1978 .

Alkyl metal asymmetric reduction. VII. Temperature dependence of the stereoselectivity of alkyl phenyl ketone reductions by chiral organoaluminum compounds

G. Giacomelli, R. Menicagli, L. Lardicci, 1975 .

Alkyl metal asymmetric reduction. Part VIII. Stereoselectivity of the reduction of alkyl phenyl ketones by optically active aliphatic Grignard reagents

G. Giacomelli, A. Caporusso, L. Lardicci, 1975 .

Alkyl metal asymmetric reduction. VI. Alkyl phenyl ketone reductions by dialkylzinc compounds. Dynamic and stereochemical aspects

G. Giacomelli, R. Santi, L. Lardicci, 1974 .

Alkyl metal asymmetric reduction. V. Reduction of alkyl methyl ketones by chiral organoaluminum compounds

G. Giacomelli, R. Menicagli, L. Lardicci, 1974 .

Alkyl metal asymmetric reduction. III. Stereochemistry of alkyl phenyl ketone reductions by chiral organoaluminum compounds

G. Giacomelli, R. Menicagli, L. Lardicci, 1973 .

Solid-phase synthesis of isoxazole-based amino acids: a new scaffold for molecular diversity.

G. Giacomelli, L. De Luca, A. Riu, 2001, Journal of Organic Chemistry.

A facile approach to the synthesis of chiral 2-substituted benzofurans.

G. Giacomelli, L. De Luca, Giammario Nieddu, 2007, The Journal of organic chemistry.

Dicobalt hexacarbonyl derivatives of chiral acetylenes

G. Giacomelli, I. Horváth, M. Kajtár, 1995 .

Microwave-promoted selective mono-N-alkylation of anilines with tertiary amines by heterogeneous catalysis.

G. Giacomelli, A. Porcheddu, L. De Luca, 2011, Chemistry.

A mild and efficient alternative to the classical Swern oxidation.

G. Giacomelli, A. Porcheddu, L. De Luca, 2001, The Journal of organic chemistry.

Cellulose beads: a new versatile solid support for microwave- assisted synthesis. Preparation of pyrazole and isoxazole libraries.

G. Giacomelli, A. Porcheddu, M. Taddei, 2003, Journal of combinatorial chemistry.

An Easy Microwave‐Assisted Synthesis of Sulfonamides Directly from Sulfonic Acids.

L. D. Luca, G. Giacomelli, 2008 .

An efficient route to alkyl chlorides from alcohols using the complex TCT/DMF.

G. Giacomelli, A. Porcheddu, L. De Luca, 2002, Organic letters.

Synthesis of new α-amino- acids containing the isoxazole moiety

G. Giacomelli, M. Falorni, E. Spanu, 1998 .

Microwave-assisted synthesis of isonitriles: a general simple methodology.

G. Giacomelli, A. Porcheddu, M. Salaris, 2005, The Journal of organic chemistry.

A method for generating nitrile oxides from nitroalkanes: a microwave assisted route for isoxazoles

L. D. Luca, G. Giacomelli, A. Porcheddu, 2003 .

Synthesis of chiral pyrazoles and isoxazoles as constrained amino acids

G. Giacomelli, M. Falorni, Anton Mario Spanedda, 1998 .

Chiral ligands containing heteroatoms. 6. 1-(2-Pyridylmethyl)pyrrolidine in the chiral catalysis of addition of diethylzinc to benzaldehyde.

G. Giacomelli, M. Falorni, G. Chelucci, 1990 .

Microwave-Assisted Synthesis of N-Monosubstituted Urea Derivatives

L. D. Luca, G. Giacomelli, A. Porcheddu, 2010 .

A very mild and chemoselective oxidation of alcohols to carbonyl compounds.

G. Giacomelli, A. Porcheddu, L. De Luca, 2001, Organic letters.

Chiral ligands containing heteroatoms.7. An investigation on the stereochemistry of the ketone reductions by chiral diamines/tin hydride systems.

N. Culeddu, G. Giacomelli, M. Falorni, 1991 .

1,3,5-Triazine: A Versatile Heterocycle in Current Applications of Organic Chemistry

L. D. Luca, G. Giacomelli, A. Porcheddu, 2005 .

Chiral ligands containing heteroatoms. 15.1 cyclic β-amino alcohols as chiral inductors for enantioselective reductions of ketones

G. Giacomelli, M. Falorni, C. Collu, 1996 .

A New, Simple Procedure for the Synthesis of Formyl Amides

L. D. Luca, G. Giacomelli, A. Porcheddu, 2004 .

A Mild and Inexpensive Procedurefor the Synthesis of N,N′-Di-Boc-Protected Guanidines

L. D. Luca, G. Giacomelli, A. Porcheddu, 2009 .

Alkylmetal asymmetric reduction. XVI: tris(cis-myrtanyl)gallium: an unusual organometallic compound as enantioselective reducing agent of ketones

G. Giacomelli, M. Falorni, L. Lardicci, 1985 .

Alkylmetal asymmetric reduction. 12. Optically active phenylalkanes from organoaluminum derivatives and aliphatic ketones

G. Giacomelli, L. Lardicci, 1982 .

Nucleophile Cleavable Linker Units

G. Giacomelli, A. Porcheddu, 2009 .

Synthesis of new oxazole-containing peptidomimetics

G. Giacomelli, G. Dettori, M. Falorni, 1998 .

One-pot synthesis of amides from aldehydes and amines via C-H bond activation.

G. Giacomelli, A. Porcheddu, Roberta Cadoni, 2012, Organic letters.

Chiral acetylenes as synthetic intermediates. 4. Synthesis and chiroptical properties of optically active .alpha.,.beta.-acetylenic ketones

C. Rosini, G. Giacomelli, A. Caporusso, 1983 .

Chiral ligands containing heteroatoms. III. Enantioselective ketone reductions using tin(II) organometallic systems from chiral piperazines

G. Giacomelli, M. Falorni, M. Marchetti, 1989 .

Chiral ligands containing heteroatoms. 8. 2-[(2s)-2-pyrrolidinyl]pyridine as a novel catalyst in the enantioselective addition of diethylzinc to aldehydes

G. Giacomelli, M. Falorni, G. Chelucci, 1991 .

Optically active beryllium and aluminium alkyls as new asymmetric reduction agents: action on alkyl phenyl ketones

G. Giacomelli, R. Menicagli, L. Lardicci, 1971 .

A new supported reagent for the photochemical generation of radicals in solution.

G. Giacomelli, M. Taddei, L. De Luca, 2001, Organic letters.

Optically active organometallic derivatives in asymmetric reactions: chiral aluminum 2-methylbutoxide in the reduction of methyl ethyl ketone

G. Giacomelli, R. Menicagli, L. Lardicci, 1973 .

Synthesis of C2-symmetry 2,2′-bipyridine and 1,10-phenanthroline chiral ligands bearig the 6,6-dimethylnorpinan-2-aryl group

G. Giacomelli, M. Falorni, G. Chelucci, 1992 .

Metal catalysis in organic reactions. Part 4. Stereospecificity in the dimerization and cyclotrimerization of chiral alk-1-ynes

G. Giacomelli, A. Caporusso, L. Lardicci, 1977 .

Some recent approaches to the synthesis of 2-substituted benzofurans.

G. Giacomelli, A. Porcheddu, L. De Luca, 2009, Current medicinal chemistry.

An easy microwave-assisted synthesis of sulfonamides directly from sulfonic acids.

G. Giacomelli, L. De Luca, 2008, The Journal of organic chemistry.

ALKYL METAL ASYMMETRIC REDUCTION PART 7, TEMPERATURE DEPENDENCE OF THE STEREOSELECTIVITY OF ALKYL PHENYL KETONE REDUCTIONS BY CHIRAL ORGANOALUMINIUM COMPOUNDS

G. Giacomelli, R. Menicagli, L. Lardicci, 1975 .

Nickel-catalyzed stereodifferentiating displacement reaction between prochiral 1-alkenes and optically active organoaluminium solvates.

G. Giacomelli, L. Lardicci, L. Bertero, 1981 .

On the reactivity of organometallic compounds towards functional substrates

G. Giacomelli, A. Caporusso, L. Lardicci, 1974 .

ALKYL METAL ASYMMETRIC REDUCTION PART 3, THE STEREOCHEMISTRY OF ALKYL PHENYL KETONE REDUCTIONS BY CHIRAL ORGANOALUMINIUM COMPOUNDS

G. Giacomelli, R. Menicagli, L. Lardicci, 1973 .

A Mild Procedure for the Preparation of 3-Aryl-4-formylpyrazoles

L. D. Luca, G. Giacomelli, A. Porcheddu, 2004 .

Chiral ligands containing heteroatoms. 14. 1,3-oxazolidinyl methanols as chiral catalysts in the enantioselective addition of diethylzinc to aldehydes

G. Giacomelli, M. Falorni, S. Conti, 1996 .

Metal catalysis in organic reactions. 16. Conjugate reduction of .alpha.,.beta.-unsaturated ketones by trialkylalane-nickel systems

G. Giacomelli, A. Caporusso, L. Lardicci, 1982 .

Metal catalysis in organic reactions. X. Nickel-catalyzed dimerization of 1-alkynes to 1,3-dialkylbutenynes

G. Giacomelli, A. Caporusso, F. Marcacci, 1979 .

The transition metal-catalyzed displacement reaction between organometallic compounds and olefins

G. Giacomelli, P. Pino, L. Lardicci, 1971 .

Alkyl metal asymmetric reduction. II. Steric control of a δ-chiral center in the reduction of achiral ketones.☆

G. Giacomelli, R. Menicagli, L. Lardicci, 1972 .

Chiral discrimination in the isomerization of racemic 1-olefins by an optically active organoaluminium–nickel system

G. Giacomelli, R. Menicagli, L. Lardicci, 1979 .

Metal catalysis in organic reactions. 16. Conjugate reduction of .alpha.,.beta.-unsaturated ketones by trialkylalane-nickel systems

G. Giacomelli, A. Caporusso, L. Lardicci, 1982 .

Alkylmetal Asymmetric Reduction. Part 17. Stereochemical Course of Ketone Reduction by β-Branched Alkyl Derivatives of Beryllium and Aluminum.

C. Rosini, G. Giacomelli, M. Falorni, 1986 .

Absolute configuration of optically active propargyl alcohols: a circular dichroism approach

C. Rosini, G. Giacomelli, P. Salvadori, 1984 .

Optically active 4-oxaroline derivatives: New useful chiral synthons derived from serine and threonine

G. Giacomelli, S. Cossu, M. Falorni, 1995 .

Optically Active 4-Oxaproline Derivatives: New Useful Chiral Synthons Derived from Serine and Threonine.

G. Giacomelli, S. Cossu, M. Falorni, 1995 .

Chiral acetylenes as synthetic intermediates—II

G. Giacomelli, C. Bertucci, A. Caporusso, 1978 .

Chiral acetylenes as synthetic intermediates—II: Optically active 1,4-dialkylbuta-1,3-dienes: synthesis and conformational studies

G. Giacomelli, C. Bertucci, A. Caporusso, 1978 .

Chiral Ligands Containing Heteroatoms. Part 9. General Procedures for the Synthesis of Optically Active 1-(2-Pyridyl)alkylamines from α -Amino Acids.

G. Giacomelli, M. Falorni, G. Chelucci, 1993 .

A Simple Method for the Reduction of Carboxylic Acids to Aldehydes or Alcohols Using H(2) and Pd/C.

G. Giacomelli, A. Porcheddu, M. Taddei, 1999, The Journal of organic chemistry.

Synthesis of Optically Active α-Amino Acids Containing Pyrazolyl Ring as Substituent.

G. Giacomelli, A. Porcheddu, M. Falorni, 2010 .

New Pyrazole Containing Bicarboxylic α‐Amino Acids: Mimics of the cis Amide Bond.

G. Giacomelli, A. Porcheddu, M. Falorni, 2000 .

New cellulose-supported reagent: a sustainable approach to guanidines.

G. Giacomelli, A. Porcheddu, A. Chighine, 2004, Organic letters.

Metal catalysis in organic reactions. 12. Asymmetric induction phenomena in the isomerization of racemic 1-alkenes by chiral aluminum solvate-nickel systems

G. Giacomelli, R. Menicagli, L. Lardicci, 1981 .

4-(4,6-Dimethoxy[1,3,5]triazin-2-yl)-4-methyl-morpholinium Chloride (DMTMM): A Valuable Alternative to PyBOP for Solid Phase Peptide Synthesis

G. Giacomelli, A. Porcheddu, M. Taddei, 2000 .

A new diketopiperazine tetra-carboxylic acid as template for the homogeneous phase synthesis of chemical libraries

G. Giacomelli, M. Taddei, M. Falorni, 1997 .

Mild and highly selective formyl protection of primary hydroxyl groups.

G. Giacomelli, A. Porcheddu, L. De Luca, 2002, Journal of Organic Chemistry.

A Method for Generating Nitrile Oxides from Nitroalkanes: A Microwave Assisted Route for Isoxazoles.

G. Giacomelli, A. Porcheddu, L. Luca, 2003 .

Chiral Ligands Containing Heteroatoms; 12.1 Synthesis of Optically Active 2-Amino-2-(2′-pyridyl)-1-alkanols from β-Hydroxy-α-amino Acids

G. Giacomelli, S. Cossu, M. Falorni, 1995 .

Unusual reactivity of 4-carboxyamido-2-oxazoline systems: new synthesis of optically active n-sulphonyl derivatives.

G. Giacomelli, S. Cossu, M. Falorni, 1994 .

ASYMMETRIC ISOMERIZATION OF ALLYL ALCOHOLS WITH RHODIUM(I)-CHIRAL PHOSPHINE COMPLEXES

G. Giacomelli, C. Botteghi, 1977 .