H. Ohno

发表

siRNA delivery into tumor cells by lipid-based nanoparticles composed of hydroxyethylated cholesteryl triamine.

Y. Maitani, N. Fujii, Y. Hattori, 2013, International journal of pharmaceutics.

Enhanced plasmid DNA transfer into tumor cells by nanoparticle composed of cholesteryl triamine and diamine.

Y. Maitani, N. Fujii, Y. Hattori, 2013, Biological & pharmaceutical bulletin.

Convergent synthesis of (-)-quinocarcin based on the combination of Sonogashira coupling and gold(I)-catalyzed 6-endo-dig hydroamination.

N. Fujii, H. Ohno, S. Oishi, 2013, Chemistry.

Palladium-catalyzed medium-ring formation for construction of the core structure of laurencia oxacycles: synthetic study of laurendecumallene B.

N. Fujii, H. Ohno, S. Oishi, 2013, Organic letters.

Palladium(0)-catalyzed synthesis of medium-sized heterocycles by using bromoallenes as an allyl dication equivalent.

H. Ohno, H. Hamaguchi, Miyo Ohata, 2004, Journal of the American Chemical Society.

Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation.

N. Fujii, H. Ohno, S. Oishi, 2015, Chemistry.

Intramolecular C ? X Bond Formation between CX or X ? H and Alkynes

H. Ohno, 2013 .

Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182.

M. Matsuoka, N. Fujii, H. Ohno, 2013, Bioorganic & medicinal chemistry.

Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles.

M. Matsuoka, N. Fujii, H. Ohno, 2012, Organic & biomolecular chemistry.

Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents.

M. Matsuoka, N. Fujii, H. Ohno, 2012, Bioorganic & medicinal chemistry.

Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents.

M. Matsuoka, Takayuki Kato, N. Fujii, 2013, Bioorganic & medicinal chemistry letters.

Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus.

M. Matsuoka, H. Tsujimoto, N. Fujii, 2009, Bioorganic & medicinal chemistry.

Total synthesis of odoamide, a novel cyclic depsipeptide, from an Okinawan marine cyanobacterium.

N. Fujii, H. Ohno, S. Oishi, 2016, Organic & biomolecular chemistry.

Synthesis of IB-01212 by multiple N-methylations of peptide bonds.

N. Fujii, H. Ohno, S. Oishi, 2014, Bioorganic & medicinal chemistry.

Production of IgG1-based bispecific antibody without extra cysteine residue via intein-mediated protein trans-splicing

K. Tsumoto, T. Ise, H. Kamada, 2021, Scientific Reports.

Azido‐Alkynes in Gold(I)‐Catalyzed Indole Syntheses

H. Ohno, S. Inuki, Junpei Matsuoka, 2021, Chemical record.

Access to Indole-Fused Benzannulated Medium-Sized Rings through Gold(I)-Catalyzed Cascade Cyclization of Azido-Alkynes.

H. Ohno, S. Oishi, A. Hashmi, 2021, Chemistry.

Concise synthesis of indole-fused 1,4-diazepines through copper(I)-catalyzed domino three-component coupling-cyclization-N-arylation under microwave irradiation.

N. Fujii, H. Ohno, S. Oishi, 2008, Organic letters.

Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization.

H. Ohno, Tetsuaki Tanaka, Mio Yamamoto, 2005, Angewandte Chemie.

Synthesis of Triazolo- and Oxadiazolopiperazines by Gold(I)-Catalyzed Domino Cyclization: Application to the Design of a Mitogen Activated Protein (MAP) Kinase Inhibitor.

H. Ohno, M. Ohue, S. Oishi, 2018, Organic letters.

Vinylaziridines in Organic Synthesis

H. Ohno, 2006 .

A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase

K. Kitaura, G. Tsujimoto, H. Fukada, 2011, Molecular and Cellular Biochemistry.

An azoreductase, aerobic NADH-dependent flavoprotein discovered from Bacillus sp.: functional expression and enzymatic characterization

S. Taguchi, H. Ohno, T. Ooi, 2007, Applied Microbiology and Biotechnology.

Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors.

G. Tsujimoto, N. Fujii, H. Ohno, 2013, Organic & biomolecular chemistry.

Effect of cationic lipid in cationic liposomes on siRNA delivery into the lung by intravenous injection of cationic lipoplex

Y. Hattori, H. Ohno, H. Onishi, 2018, Journal of drug targeting.

Effect of cationic lipid type in cationic liposomes for siRNA delivery into the liver by sequential injection of chondroitin sulfate and cationic lipoplex

Y. Hattori, H. Ohno, H. Onishi, 2018, Journal of Drug Delivery Science and Technology.

Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions.

N. Fujii, H. Ohno, S. Oishi, 2007, Angewandte Chemie.

Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors.

K. Kitaura, K. Matsuno, A. Asai, 2011, Journal of medicinal chemistry.

Cu(II)-mediated oxidative intermolecular ortho C-H functionalisation using tetrahydropyrimidine as the directing group.

N. Fujii, H. Ohno, S. Oishi, 2009, Chemical communications.

Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor.

N. Fujii, H. Ohno, S. Oishi, 2016, Chemical & pharmaceutical bulletin.

Total Synthesis of Dictyodendrins A-F by the Gold-Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole.

Y. Miyamoto, M. Oka, H. Ohno, 2020, Chemistry.

Radical cyclization by ipso substitution of the methoxy group: considerable effect of HMPA on samarium-mediated cyclization.

H. Ohno, Tetsuaki Tanaka, Hiroki Iwasaki, 2003, The Journal of organic chemistry.

Samarium(II)-mediated spirocyclization by intramolecular aryl radical addition onto an aromatic ring.

H. Ohno, N. Tsutsui, Tetsuaki Tanaka, 2008, The Journal of organic chemistry.

The first samarium(II)-mediated aryl radical cyclisation onto an aromatic ring.

H. Ohno, Tetsuaki Tanaka, Hiroki Iwasaki, 2004, Chemical communications.

The first samarium(II)-mediated stereoselective spirocyclization onto an aromatic ring.

H. Ohno, Tetsuaki Tanaka, R. Wakayama, 2002, Chemical communications.

Activation of Neuropeptide FF Receptors by Kisspeptin Receptor Ligands.

G. Tsujimoto, S. Ohkura, N. Inoue, 2011, ACS medicinal chemistry letters.

Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase.

N. Fujii, H. Ohno, S. Oishi, 2008, Journal of medicinal chemistry.

Gold(I)-Catalyzed Cascade Cyclization Reactions of Allenynes for the Synthesis of Fused Cyclopropanes and Acenaphthenes.

H. Ohno, S. Oishi, S. Inuki, 2019, Angewandte Chemie.

Gold(I)-Catalyzed Cascade Cyclization Reactions of Allenynes for the Synthesis of Fused Cyclopropanes and Acenaphthenes.

H. Ohno, S. Oishi, S. Inuki, 2019, Angewandte Chemie.

Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity.

M. Matsuoka, N. Fujii, H. Ohno, 2008, Journal of medicinal chemistry.

Design and synthesis of amidine-type peptide bond isosteres: application of nitrile oxide derivatives as active ester equivalents in peptide and peptidomimetics synthesis.

N. Fujii, H. Ohno, M. Nomizu, 2011, Organic & biomolecular chemistry.

Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists.

G. Tsujimoto, N. Fujii, H. Ohno, 2012, Bioconjugate chemistry.

Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres.

N. Fujii, H. Ohno, T. Furuya, 2012, Journal of medicinal chemistry.

Potent CXCR4 antagonists containing amidine type Peptide bond isosteres.

M. Matsuoka, N. Fujii, H. Ohno, 2011, ACS medicinal chemistry letters.

Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors.

A. Asai, J. Sawada, N. Fujii, 2014, Bioorganic & medicinal chemistry.

Synthesis and Application of Fluorescein‐ and Biotin‐Labeled Molecular Probes for the Chemokine Receptor CXCR4

G. Tsujimoto, M. Matsuoka, N. Fujii, 2008, Chembiochem : a European journal of chemical biology.

Synthesis and applications of vinylaziridines and ethynylaziridines.

H. Ohno, 2014, Chemical reviews.

Direct synthesis of aryl-annulated [c]carbazoles by gold(i)-catalysed cascade reaction of azide-diynes and arenes.

H. Ohno, S. Oishi, Misaki Kobayashi, 2018, Chemical science.

Structure‐activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists

N. Fujii, H. Ohno, S. Oishi, 2008, Biopolymers.

Enantioselective Synthesis of Allenes

K. Tomioka, H. Ohno, Y. Nagaoka, 2008 .

Structure-activity relationship study on small peptidic GPR54 agonists.

N. Fujii, H. Ohno, S. Oishi, 2006, Bioorganic & medicinal chemistry.

Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants

M. Matsuoka, A. Asai, N. Fujii, 2010 .

Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: synthesis and bioevaluation of alpha-helical anti-HIV peptide analogues.

M. Matsuoka, T. Narumi, N. Fujii, 2009, Organic & biomolecular chemistry.

Construction of linked nitrogen heterocycles by palladium(0)-catalyzed intramolecular domino cyclization of 2-alkynylaziridines bearing a 2-aminoethyl group via ring expansion with isocyanate.

N. Fujii, H. Ohno, S. Oishi, 2010, The Journal of organic chemistry.

Direct construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes.

N. Fujii, H. Ohno, S. Oishi, 2015, Organic letters.

Structure‐Activity Relationships of Pyrazine‐Based CK2 Inhibitors: Synthesis and Evaluation of 2,6‐Disubstituted Pyrazines and 4,6‐Disubstituted Pyrimidines

Takafumi Hara, G. Tsujimoto, N. Fujii, 2008, Archiv der Pharmazie.

Concise site-specific synthesis of DTPA-peptide conjugates: application to imaging probes for the chemokine receptor CXCR4.

H. Saji, N. Fujii, H. Kimura, 2011, Bioorganic & medicinal chemistry.

Structure-activity relationship study on polyglutamine binding peptide QBP1.

N. Fujii, H. Ohno, T. Toda, 2009, Bioorganic & medicinal chemistry.

Synthesis of jaspine B regioisomers through palladium-catalyzed stereoselective tetrahydrofuran formation: Insight into the ligand recognition of sphingosine kinases

N. Fujii, H. Ohno, I. Nakanishi, 2018 .

Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B.

N. Fujii, H. Ohno, I. Nakanishi, 2017, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres.

M. Matsuoka, T. Narumi, N. Fujii, 2010, Organic & biomolecular chemistry.

Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach.

M. Matsuoka, H. Nagasawa, N. Fujii, 2008, Bioorganic & medicinal chemistry letters.

Structure of human protein kinase CK2 alpha 2 with a potent indazole-derivative inhibitor.

K. Kitaura, G. Tsujimoto, T. Kinoshita, 2009, Acta crystallographica. Section F, Structural biology and crystallization communications.

Small interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes

Y. Hattori, H. Ohno, H. Onishi, 2017, Journal of liposome research.

Design and synthesis of fluorescent probes for GPR54.

N. Fujii, H. Ohno, A. Hirasawa, 2014, Bioorganic & medicinal chemistry.

Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists.

N. Fujii, H. Ohno, T. Noguchi, 2013, Bioorganic & medicinal chemistry.

Synthesis and application of an Nδ-acetyl-Nδ-hydroxyornithine analog: identification of novel metal complexes of deferriferrichrysin.

N. Fujii, H. Ohno, Y. Hata, 2012, Bioorganic & medicinal chemistry.

Development of Mirror-Image Screening Systems for XIAP BIR3 Domain Inhibitors.

N. Fujii, H. Ohno, S. Oishi, 2019, Bioconjugate chemistry.

Recent Progress in Palladium-Catalyzed Cascade Cyclizations for Natural Product Synthesis

H. Ohno, S. Inuki, 2018, Synthesis.

Recent Advances in the Construction of Polycyclic Compounds by Palladium-Catalyzed Atom-Economical Cascade Reactions

H. Ohno, 2013 .

Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors.

T. Kinoshita, N. Fujii, H. Ohno, 2016, Bioorganic & medicinal chemistry.

Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles.

H. Ohno, S. Oishi, Junpei Matsuoka, 2017, Angewandte Chemie.

Novel anti-flavivirus drugs targeting the nucleolar distribution of core protein.

K. Mizuguchi, Tsuyoshi Esaki, C. Nagao, 2019, Virology.

Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides.

N. Fujii, H. Ohno, S. Oishi, 2015, Organic letters.

Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines.

N. Fujii, H. Ohno, S. Oishi, 2014, Organic letters.

The Role of Acetylides in Dual Gold Catalysis: A Mechanistic Investigation of the Selectivity Difference in the Naphthalene Synthesis from Diynes

H. Ohno, F. Rominger, A. Hashmi, 2014 .

Gold‐Catalyzed Cascade Reactions of Alkynes for Construction of Polycyclic Compounds

H. Ohno, 2013 .

Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes.

N. Fujii, H. Ohno, S. Oishi, 2012, The Journal of organic chemistry.

Gold(I)-catalyzed polycyclizations of polyenyne-type anilines based on hydroamination and consecutive hydroarylation cascade.

N. Fujii, H. Ohno, S. Oishi, 2011, The Journal of organic chemistry.

Gold‐Catalyzed Intramolecular Alkyne Cycloisomerization Cascade: Direct Synthesis of Aryl‐Annulated[a]carbazoles from Aniline‐Substituted Diethynylarenes

N. Fujii, H. Ohno, S. Oishi, 2010 .

Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds.

M. Matsuoka, N. Fujii, H. Ohno, 2015, Organic & biomolecular chemistry.

Chem. Pharm. Bull. 53(10) 1211—1226 (2005)

H. Ohno, 2005 .

Efficient synthesis of aminomethylated azaindoles and corresponding pyrrole-fused derivatives by copper-catalyzed domino multicomponent coupling and cyclization

N. Fujii, H. Ohno, S. Oishi, 2012 .

Direct synthesis of fused indoles by gold-catalyzed cascade cyclization of diynes.

N. Fujii, H. Ohno, S. Oishi, 2011, The Journal of organic chemistry.

Rapid access to 3-(aminomethyl)isoquinoline-fused polycyclic compounds by copper-catalyzed four-component coupling, cascade cyclization, and oxidation.

N. Fujii, T. Watabe, H. Ohno, 2009, The Journal of organic chemistry.

Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines.

N. Fujii, H. Ohno, S. Oishi, 2010, Organic letters.

Palladium-catalyzed direct synthesis of carbazoles via one-pot N-arylation and oxidative biaryl coupling: synthesis and mechanistic study.

N. Fujii, H. Ohno, S. Oishi, 2009, The Journal of organic chemistry.

One‐Pot Synthesis of Carbazoles by Palladium‐Catalyzed N‐Arylation and Oxidative Coupling.

N. Fujii, H. Ohno, S. Oishi, 2008 .

Direct synthesis of highly fused perimidines by copper(I)-catalyzed hydroamination of 2-ethynylbenzaldehydes

N. Fujii, H. Ohno, S. Oishi, 2011 .

Palladium-catalyzed sp(3) CH activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines.

N. Fujii, H. Ohno, S. Oishi, 2008, Organic letters.

Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides.

T. Narumi, N. Fujii, H. Ohno, 2007, Organic letters.

One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling.

Satoshi Ueda, Shinya Oishi, N. Fujii, 2007, Chemical communications.

A convenient synthesis of activated enantiomerically pure 2-ethynylaziridines

N. Fujii, H. Ohno, T. Ibuka, 1998 .

Construction of Quaternary Carbon Stereocenter of α-Tertiary Amine through Remote C-H Functionalization of Tris Derivatives: Enantioselective Total Synthesis of Myriocin.

H. Ohno, S. Oishi, S. Inuki, 2019, Organic letters.

Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/D-ring system.

H. Ohno, Tetsuaki Tanaka, K. Murakami, 2006, Chemical & pharmaceutical bulletin.

The first total synthesis of (+/-)-scopadulin, an antiviral aphidicolane diterpene.

H. Ohno, T. Murata, K. Murakami, 2001, Organic letters.

Efficient one-step conversion of primary aliphatic amines into primary alcohols: application to a model study for the total synthesis of (+/-)-scopadulin.

H. Ohno, S. Rahman, N. Maezaki, 2000, Organic letters.

Evaluation of scopadulciol-related molecules for their stimulatory effect on the cytotoxicity of acyclovir and ganciclovir against Herpes simplex virus type 1 thymidine kinase gene-transfected HeLa cells.

K. Hayashi, Toshimitsu Hayashi, H. Ohno, 2004, Chemical & pharmaceutical bulletin.

A model study for the total synthesis of (±)-scopadulin: stereoselective construction of the A/B ring system with desired functionalities

H. Ohno, Tetsuaki Tanaka, K. Murakami, 2001 .

Total synthesis of (+/-)-stemodinone via an efficient ring-exchange strategy.

H. Ohno, K. Murakami, S. Rahman, 2001, The Journal of organic chemistry.

Synthesis of fused and linked bicyclic nitrogen heterocycles by palladium-catalyzed domino cyclization of propargyl bromides.

N. Fujii, H. Ohno, S. Oishi, 2010, Chemistry.

Gold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines.

H. Ohno, W. Hiller, N. Krause, 2016, Organic & biomolecular chemistry.

Palladium-catalyzed reductive ring opening with formic acid of aziridines bearing an α,β-unsaturated ester group

A. Otaka, H. Tamamura, N. Fujii, 1997 .

Gold-catalyzed three-component annulation: efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones.

N. Fujii, H. Ohno, S. Oishi, 2012, Organic letters.

Total Synthesis of Zephycarinatines via Photocatalytic Reductive Radical ipso ‐Cyclization

A. Ichimura, H. Ohno, S. Oishi, 2020, Angewandte Chemie.

Total Synthesis of Zephycarinatines via Photocatalytic Reductive Radical ipso-Cyclization.

A. Ichimura, H. Ohno, S. Oishi, 2020, Angewandte Chemie.

Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: diastereoselective access to bicyclic nitrogen heterocycles.

H. Ohno, Tetsuaki Tanaka, Tsuyoshi Mizutani, 2005, Angewandte Chemie.

Kinesin spindle protein (KSP) inhibitors with 2,3-fused indole scaffolds.

A. Asai, J. Sawada, N. Fujii, 2010, Journal of medicinal chemistry.

Heck-type cyclization of oxime ethers: stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2007, Angewandte Chemie.

Wurster's Blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV/Vis/NIR and fluorescence.

N. Fujii, H. Ohno, Ryo Katoono, 2014, Chemistry, an Asian journal.

Construction of nitrogen heterocycles bearing an aminomethyl group by copper-catalyzed domino three-component coupling-cyclization.

N. Fujii, H. Ohno, S. Oishi, 2009, The Journal of organic chemistry.

Efficient synthesis of pyrimido[1,2-c] [1,3]benzothiazin-6-imines and related tricyclic heterocycles by S(N)Ar-type C-S, C-N, or C-O bond formation with heterocumulenes.

N. Fujii, H. Ohno, S. Oishi, 2010, The Journal of organic chemistry.

Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation.

N. Fujii, H. Ohno, S. Oishi, 2014, Chemical communications.

Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group.

N. Fujii, H. Ohno, S. Oishi, 2015, Organic letters.

Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds.

Kazuo Kitaura, Shinya Oishi, Gozoh Tsujimoto, 2012, Journal of medicinal chemistry.

Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation.

N. Fujii, H. Ohno, S. Oishi, 2008, Chemical communications.

Palladium(0)-catalyzed tandem cyclization of allenenes: direct construction of tricyclic heterocycles through aromatic C--H activation.

H. Ohno, H. Hamaguchi, Tetsuaki Tanaka, 2005, Chemistry.

A novel samarium(II)-mediated tandem spirocyclization onto an aromatic ring

H. Ohno, M. Yamashita, N. Tsutsui, 2011 .

Total synthesis of (-)-quinocarcin by gold(I)-catalyzed regioselective hydroamination.

Shinya Oishi, Hiroaki Chiba, N. Fujii, 2012, Angewandte Chemie.

2-ethynylaziridines as chiral carbon nucleophiles: stereoselective synthesis of 1,3-amino alcohols with three stereocenters via allenylindium reagents bearing a protected amino group.

H. Ohno, H. Hamaguchi, T. Tanaka, 2001, The Journal of organic chemistry.

Nonbiomimetic total synthesis of indole alkaloids using alkyne-based strategies.

H. Ohno, S. Inuki, 2021, Organic & biomolecular chemistry.

Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group.

N. Fujii, H. Ohno, S. Oishi, 2015, Angewandte Chemie.

A Thermodynamic Preference of Chiral N-Methanesulfonyl and N-Arenesulfonyl 2,3-cis-3-Alkyl-2-Vinylaziridines over Their 2,3-Trans-Isomers: Useful Palladium(0)-Catalyzed Equilibration Reactions for the Synthesis of (E)-Alkene Dipeptide Isosteres

Y. Miwa, H. Tamamura, N. Fujii, 1997 .

Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres.

T. Narumi, N. Fujii, H. Ohno, 2007, Biopolymers.

Development of useful reactions based on the novel reactivities of allenic compounds and their application to tandem cyclizations.

H. Ohno, 2005, Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan.

Sterically congested chiral activated aziridines: Synthesis of both 2,3-cis- and 2,3-trans-2-alkenyl-3-alkylaziridines from common intermediates

Y. Miwa, N. Fujii, H. Ohno, 1999 .

Regiospecific ring-opening reactions of β-aziridinyl α,β-enoates with acids: application to the stereoselective synthesis of a couple of diastereoisomeric (E)-alkene dipeptide isosteres from a single β-aziridinyl α,β-enoate and to the convenient preparation of amino alcohols bearing α,β-unsaturated

A. Otaka, H. Tamamura, N. Fujii, 2000 .

Palladium-Catalyzed Reductive Ring Opening with Formic Acid of Aziridines Bearing an α,β-Unsaturated Ester Group.

A. Otaka, H. Tamamura, N. Fujii, 1998 .

A 2,3-cis-selective synthesis of aziridines bearing a vinyl group from allyl methyl carbonates and allyl mesylates

H. Tamamura, N. Fujii, H. Ohno, 1998 .

Palladium(0)-Catalyzed Isomerization Reactions of Aziridines Bearing an alpha,beta-Unsaturated Ester Group: A Thermodynamic Preference for Chiral Alkyl (2E)-4,5-cis-4,5-Epimino-N-(alkyl- or arylsulfonyl) 2-Enoates over the Other Three Stereoisomers.

Y. Miwa, H. Tamamura, N. Fujii, 1997, The Journal of organic chemistry.

Design and synthesis of a novel class of CK2 inhibitors: application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles.

G. Tsujimoto, N. Fujii, H. Ohno, 2012, Organic & biomolecular chemistry.

Potassium carbonate-promoted stereospecific 5-endo-trig cyclization of unactivated allenes in the absence of any transition metals.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2006, Organic letters.

Facile synthesis of 1,2,3,4-tetrahydro-beta-carbolines by one-pot domino three-component indole formation and nucleophilic cyclization.

N. Fujii, H. Ohno, S. Oishi, 2009, Organic letters.

Reactions of N-Arylsulfonyl-2,3-cis- and N-Arylsulfonyl-2,3-trans-3-alkyl-2-vinylaziridines with Organocopper Reagents: Importance of 2,3-cis-Stereochemistry in Controlling Regio- and Stereoselectivity.

N. Fujii, H. Ohno, H. Aoyama, 1998, The Journal of organic chemistry.

Development of useful reactions involving tandem cyclizations based on the novel reactivities of allenic compounds.

H. Ohno, 2005, Chemical & pharmaceutical bulletin.

Stereodivergent synthesis of chiral 2-alkenylaziridines: palladium(0)-catalyzed 2,3-cis-selective aziridination and base-mediated 2,3-trans-selective aziridination.

N. Fujii, H. Ohno, Y. Takemoto, 2004, Chemical & pharmaceutical bulletin.

Asymmetric synthesis of β2,3-amino acids by InI–Pd(0)-promoted metalation and addition of chiral 2-vinylaziridines

N. Fujii, H. Ohno, Y. Takemoto, 2002 .

[Development of aziridination and azetizination reactions of amino allenes using a palladium catalyst].

H. Ohno, 2001, Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan.

Stereoselective synthesis of chiral 2,3-cis-2-ethynylaziridines by base-mediated intramolecular amination of bromoallenes.

H. Ohno, H. Hamaguchi, Tetsuaki Tanaka, 2001, Organic letters.

Stereoselective synthesis of nonracemic 1,3-amino alcohols from chiral 2-vinylaziridines by InI–Pd(0)-promoted metalation

N. Fujii, H. Ohno, Y. Takemoto, 2001 .

Umpolung of Chiral 2‐Ethynylaziridines: Indium(I)‐Mediated Stereoselective Synthesis of Nonracemic 1,3‐Amino Alcohols Bearing Three Chiral Centers, Catalyzed by Palladium(0).

H. Ohno, H. Hamaguchi, Tetsuaki Tanaka, 2000 .

Stereoselective Synthesis of Chiral Amino Allenes by Organocopper-Mediated anti-SN2′-Substitution Reaction of Chiral Ethynylaziridines

N. Fujii, H. Ohno, Y. Takemoto, 2000 .

SYNTHESIS OF CHIRAL AMINO ALLENES VIA AN ORGANOCYANOCUPRATE-MEDIATED RING-OPENING REACTION OF ENANTIOPURE ETHYNYLAZIRIDINES

Y. Miwa, N. Fujii, H. Ohno, 1999 .

Convenient syntheses of chiral 3-substituted 2-ethynylaziridines

N. Fujii, H. Ohno, Y. Takemoto, 1999 .

Convenient synthesis of spiroindole derivatives via palladium-catalyzed cyclization of propargyl chlorides

N. Fujii, H. Ohno, S. Oishi, 2015 .

Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates.

N. Fujii, H. Ohno, S. Oishi, 2010, The Journal of organic chemistry.

Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides.

N. Fujii, H. Ohno, Miyo Ohata, 2008, Organic letters.

Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization.

N. Fujii, H. Ohno, S. Oishi, 2009, The Journal of organic chemistry.

First Palladium-Catalyzed Aziridination Reaction of Amino Allenes.

Y. Miwa, N. Fujii, H. Ohno, 1999, The Journal of organic chemistry.

Concise Synthesis of Indole-Fused 1,4-Diazepines Through Copper(I)-Catalyzed Domino Three-Component Coupling—Cyclization—N-Arylation under Microwave Irradiation.

N. Fujii, H. Ohno, S. Oishi, 2008 .

Enantioselective total synthesis of (+)-lysergic acid, (+)-lysergol, and (+)-isolysergol by palladium-catalyzed domino cyclization of allenes bearing amino and bromoindolyl groups.

N. Fujii, H. Ohno, S. Oishi, 2011, The Journal of organic chemistry.

Gold(I)-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring-Fused Indoles and Propellane-Type Indolines.

H. Ohno, S. Oishi, S. Inuki, 2020, The Journal of organic chemistry.

Gold-catalyzed hydroarylation of allenes: a highly regioselective carbon-carbon bond formation producing six-membered rings.

N. Fujii, H. Ohno, S. Oishi, 2007, Organic letters.

Palladium‐Catalyzed Construction of Polycyclic Heterocycles by an Alkyne Insertion and Direct Arylation Cascade.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2011 .

Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization.

N. Fujii, H. Ohno, S. Oishi, 2016, Organic letters.

A highly regio- and stereoselective formation of bicyclo[4.2.0]oct-5-ene derivatives through thermal intramolecular [2 + 2] cycloaddition of allenes.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2007, The Journal of organic chemistry.

Novel synthesis of chiral terminal allenes via palladium(0)-catalyzed reduction of mesylates of 2-bromoalk-2-en-1-ols bearing a protected amino group, using diethylzinc

N. Fujii, H. Ohno, S. Oishi, 2000 .

Palladium-catalyzed regio- and stereoselective synthesis of N-protected 2,4-dialkylated azacyclobutanes from amino allenes

N. Fujii, H. Ohno, Y. Takemoto, 1999 .

Formal total synthesis of (+)-lysergic acid via zinc(II)-mediated regioselective ring-opening reduction of 2-alkynyl-3-indolyloxirane.

N. Fujii, H. Ohno, S. Oishi, 2011, The Journal of organic chemistry.

Recent Advances in the Construction of Polycyclic Compounds by Palladium-Catalyzed Atom-Economical Cascade Reactions

H. Ohno, 2013 .

Novel Synthesis of Azocine, Azepine, Oxocine, and Oxepine Derivatives by Palladium-catalyzed Medium-Ring Formation from Bromoallenes

H. Ohno, H. Hamaguchi, Miyo Ohata, 2003 .

Dual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes.

N. Fujii, H. Ohno, F. Rominger, 2014, Chemistry.

Gold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds.

H. Ohno, S. Oishi, S. Inuki, 2018, Organic letters.

Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists.

N. Fujii, H. Ohno, S. Oishi, 2007, Organic & biomolecular chemistry.

Gold-Catalyzed Atom-Economical Cascade Reactions of Alkynes for Ring Formation

N. Fujii, H. Ohno, S. Oishi, 2014 .

Purification and characterization of an Aspergillus oryzae-produced carboxylesterase that catalyzes O-deacetylation of a fully acetylated O-glucoside of N-phenylacetohydroxamic acid.

H. Ohno, T. Uematsu, T. Yoshioka, 1997, European journal of biochemistry.

Chemo- and stereoselectivity in titanium-mediated regioselective ring-opening reaction of epoxides at the more substituted carbon

H. Ohno, Tetsuaki Tanaka, Y. Kobayashi, 2005 .

Regio- and stereoselectivity in reactions of 2,3-cis- and trans-3-alkyl-2-vinylaziridines with organocopper reagents: Importance of 2,3-cis-stereochemistry in controlling selectivity

A. Otaka, H. Tamamura, N. Fujii, 1997 .

Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid-phase synthesis of a cyclic pentapeptide mimetic

T. Narumi, N. Fujii, H. Ohno, 2008 .

Total synthesis of (+/-)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group.

N. Fujii, H. Ohno, S. Oishi, 2008, Organic letters.

Redox-induced Conformational Changes in 1,3-Propylene- and m-Xylylenebis[5-(10-butyl-5,10-dihydrobenzo[a]indolo[2,3-c]carbazole)]: Twin-BIC Donors that Form Sandwich-like Dimeric Cations Exhibiting NIR Absorption

H. Ohno, Ryo Katoono, K. Fujiwara, 2016 .

Double C-H functionalization in sequential order: direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2012, Chemistry.

Selective Synthesis of Nonracemic 3-Pyrrolines and 2,3-cis-2-Vinylaziridines from (Z)-Amino Allylic Alcohols: A New Synthetic Route to Chiral 3,4-Dehydroproline

H. Ohno, Y. Takemoto, T. Ibuka, 1999 .

Lewis-acid-mediated ring-exchange reaction of dihydrobenzofurans and its application to the formal total synthesis of (−)-quinocarcinamide

N. Fujii, H. Ohno, S. Oishi, 2012 .

Asymmetric Construction of Quaternary Carbon Centers by Titanium-Mediated Stereospecific Allylation of 2,3-Epoxy Alcohol Derivatives.

H. Ohno, Tetsuaki Tanaka, K. Hiramatsu, 2004 .

Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne.

N. Fujii, H. Ohno, Y. Yoshida, 2016, The Journal of organic chemistry.

Bromoallenes as allyl dication equivalents in the presence or absence of palladium(0): direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes.

N. Fujii, H. Ohno, H. Hamaguchi, 2007, Chemistry.

Bromoallenes as allyl dication equivalents in the absence of palladium(0): synthesis of bicyclic sulfamides by tandem cyclization of bromoallenes.

H. Ohno, H. Hamaguchi, Shohei Kosaka, 2005, Angewandte Chemie.

Heck-Type Cyclization of Oxime Ethers: Stereoselective Carbon—Carbon Bond Formation with Aryl Halides to Produce Heterocyclic Oximes.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2007 .

Palladium(0)-catalyzed stereoselective cyclization of allenenes: divergent synthesis of pyrrolidines and 3-azabicyclo[3.1.0]hexanes from single allenenes.

H. Ohno, Tetsuaki Tanaka, Y. Kadoh, 2004, The Journal of organic chemistry.

Novel synthesis of 3-azabicyclo[3.1.0]hexanes by unusual palladium(0)-catalyzed cyclopropanation of allenenes.

H. Ohno, Tetsuaki Tanaka, Y. Kadoh, 2003, Organic letters.

Palladium(0)-catalyzed tandem cyclization of allenenes.

H. Ohno, Tetsuaki Tanaka, Kumiko Miyamura, 2003, Angewandte Chemie.

Palladium-catalyzed sp(3) CH activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines.

N. Fujii, H. Ohno, S. Oishi, 2008, Organic letters.

Synthesis of allenes from allylic alcohol derivatives bearing a bromine atom using a palladium(0)/diethylzinc system.

N. Fujii, H. Ohno, S. Oishi, 2002, The Journal of organic chemistry.

Fe(ii)-Complexation of tripodal hexapeptide ligands with three bidentate triazolylpyridines: induction of metal-centred chirality by peptide macrocyclization.

T. Kameda, N. Fujii, H. Ohno, 2017, Dalton transactions.

Synthesis and functional analysis of deferriferrichrysin derivatives: application to colorimetric pH indicators.

N. Fujii, H. Ohno, Y. Hata, 2013, Bioorganic & medicinal chemistry.

Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle.

T. Kameda, H. Ohno, S. Oishi, 2018, Inorganic Chemistry.

Head-to-tail macrocyclization of cysteine-free peptides using an o-aminoanilide linker.

N. Fujii, H. Ohno, S. Oishi, 2018, Bioorganic & medicinal chemistry letters.

Layered compounds. XLI. Tricarbonylchromium complexes of multilayered [2.2]paracyclophanes☆

H. Ohno, T. Otsubo, Y. Sakata, 1977 .

Synthesis and biological evaluation of the [d-MeAla(11)]-epimer of coibamide A.

A. Hau, N. Fujii, H. Ohno, 2015, Bioorganic & medicinal chemistry letters.

Synthesis of pachastrissamine (jaspine B) and its derivatives by the late-stage introduction of the C-2 alkyl side-chains using olefin cross metathesis

N. Fujii, H. Ohno, S. Oishi, 2013 .

Improved method of an unusual conversion of aliphatic amines into alcohols

H. Ohno, Tetsuaki Tanaka, S. Rahman, 2001 .

Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C.

N. Fujii, H. Ohno, S. Oishi, 2011, Bioorganic & medicinal chemistry.

Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B).

N. Fujii, H. Ohno, S. Oishi, 2010, The Journal of organic chemistry.

Studies on the Chemical Synthesis of Potential Antimetabolites. 36. Synthesis and Some Biochemical Properties of (±)1-Deazaaristeromycin

H. Ohno, A. Nomura, Y. Mizuno, 1984 .

Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of bromoallenes.

N. Fujii, H. Ohno, S. Oishi, 2009, Organic letters.

Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-SN2' reactions and their use in the preparation of low-molecule CXCR4 antagonists.

K. Kitaura, A. Otaka, H. Tamamura, 2006, The Journal of organic chemistry.

Palladium-catalysed biscyclisation of allenic bromoalkenes through a zipper-mode cascade.

N. Fujii, H. Ohno, S. Oishi, 2008, Chemical communications.

Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes.

N. Fujii, H. Ohno, T. Noguchi, 2013, Bioorganic & medicinal chemistry letters.

Construction of the Pyrrolo[2,3- d]carbazole Core of Spiroindoline Alkaloids by Gold-Catalyzed Cascade Cyclization of Ynamide.

H. Ohno, S. Oishi, H. Kumagai, 2019, The Journal of organic chemistry.

The Effects of a Selective CK2 Inhibitor on Anti-glomerular Basement Membrane Glomerulonephritis in Rats.

G. Tsujimoto, H. Ohno, A. Hirasawa, 2015, Biological & pharmaceutical bulletin.

Unusual radical ipso-substitution reaction of an aromatic methoxy group induced by tris(trimethylsilyl)silane-AIBN or SmI2

H. Ohno, Tetsuaki Tanaka, N. Maezaki, 2000 .

Evaluation of Small Interfering RNA Delivery into Cells by Reverse Transfection in Suspension with Cationic Liposomes

Y. Hattori, H. Ohno, H. Onishi, 2017 .

Synthesis of Grb2 SH2 Domain Proteins for Mirror-Image Screening Systems.

N. Fujii, H. Ohno, T. Noguchi, 2017, Bioconjugate chemistry.

Total Synthesis of Dictyodendrins A-F by the Gold-Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole.

Y. Miyamoto, M. Oka, H. Ohno, 2020, Chemistry.

Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold.

H. Ohno, Y. Yoshida, S. Oishi, 2017, Organic letters.

Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation.

S. Ohkura, T. Yamamura, F. Matsuda, 2014, Journal of medicinal chemistry.

Stereoselective Synthesis of 2-Alkenylaziridines and 2-Alkenylazetidines by Palladium-Catalyzed Intramolecular Amination of α- and β-Amino Allenes

N. Fujii, H. Ohno, Y. Takemoto, 2001 .

Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins.

M. Matsuoka, N. Fujii, H. Ohno, 2009, Bioorganic & medicinal chemistry.

Development and application of fluorescent SDF-1 derivatives.

G. Tsujimoto, M. Matsuoka, N. Fujii, 2012, Future medicinal chemistry.

The effects of 5‐OP‐RU stereochemistry on its stability and MAIT‐MR1 axis

S. Yamasaki, H. Ohno, S. Oishi, 2020, Chembiochem : a European journal of chemical biology.

Design of Coibamide A Mimetics with Improved Cellular Bioactivity

H. Ohno, S. Oishi, K. McPhail, 2021, ACS medicinal chemistry letters.

Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: disclosing the importance of side-chain and backbone functionalities.

Stephen C Peiper, Satoshi Ueda, Shinya Oishi, 2007, Journal of medicinal chemistry.

Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2007, Organic letters.

Zipper‐Mode Double C—H Activation: Palladium‐Catalyzed Direct Construction of Highly Fused Heterocyclic Systems.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2008 .

Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility.

Shinya Oishi, Shinya Nakamura, Tomoki Takeuchi, 2014, ACS medicinal chemistry letters.

Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: identification of novel peptidic inhibitors.

Shinya Oishi, Hiroyuki Osada, Masato Kaneda, 2013, Bioorganic & medicinal chemistry letters.

Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates.

T. Narumi, N. Fujii, H. Ohno, 2008, The Journal of organic chemistry.

siRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes.

E. Yonemochi, K. Kawano, N. Fujii, 2015, Biological & pharmaceutical bulletin.

A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres.

T. Narumi, A. Otaka, N. Fujii, 2006, Chemical communications.

A Novel One‐Pot Reaction Involving Organocopper‐Mediated Reduction/Transmetalation/Asymmetric Alkylation, Leading to the Diastereoselective Synthesis of Functionalized (Z)‐Fluoroalkene Dipeptide Isosteres.

T. Narumi, A. Otaka, N. Fujii, 2007 .

Total Synthesis of (+)-Polyoxamic Acid via Visible-Light-Mediated Photocatalytic β-Scission and 1,5-Hydrogen Atom Transfer of Glucose Derivative.

H. Ohno, S. Oishi, S. Inuki, 2020, The Journal of organic chemistry.

Development of novel NK3 receptor antagonists with reduced environmental impact.

S. Ohkura, F. Matsuda, N. Fujii, 2016, Bioorganic & medicinal chemistry.

Synthesis of the Src SH2 domain and its application in bioassays for mirror-image screening

N. Fujii, H. Ohno, T. Noguchi, 2017 .

Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction.

N. Fujii, H. Ohno, T. Noguchi, 2017, Bioorganic & medicinal chemistry letters.

Selective synthesis of cis-2-vinyl-3-alkylaziridines and 3-pyrrolines from common intermediates (Z)-4-N-arylsulfonylaminoalk-2-en-1-ols

N. Fujii, H. Ohno, Y. Takemoto, 1999 .

Selective synthesis of cis-2-vinyl-3-alkylaziridines and 3-pyrrolines from common intermediates (Z)-4-N-arylsulfonylaminoalk-2-en-1-ols

N. Fujii, H. Ohno, Y. Takemoto, 1999 .

Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold.

M. Matsuoka, N. Fujii, H. Ohno, 2015, Bioorganic & medicinal chemistry.

Screening of a virtual mirror-image library of natural products.

N. Fujii, H. Ohno, T. Noguchi, 2016, Chemical communications.

X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitution.

K. Kitaura, M. Matsuoka, T. Nakatsu, 2009, Journal of molecular biology.

Structure–activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists

S. Ohkura, T. Yamamura, F. Matsuda, 2015 .

Scaffold hopping of fused piperidine-type NK3 receptor antagonists to reduce environmental impact.

H. Ohno, S. Oishi, S. Inuki, 2019, Bioorganic & medicinal chemistry.

Title Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C

N. Fujii, H. Ohno, S. Oishi, 2019 .

Gold(I)-Catalyzed Benzylic C(sp3)-H Functionalizations: Divergent Synthesis of Indole[a]- and [b]-Fused Polycycles.

H. Ohno, S. Inuki, Norihito Arichi, 2022, Angewandte Chemie.

5,10-Dihydrobenzo[a]indolo[2,3-c]carbazole: A Highly Fluorescent Disk-shaped Electron Donor Exhibiting Dual UV–vis–NIR and Fluorescence Spectral Changes upon Electrolysis

N. Fujii, H. Ohno, Ryo Katoono, 2013 .

The Synthesis of Alkaloids Using Transition-Metal-Catalyzed Intramolecular Amination Reactions

N. Fujii, H. Ohno, S. Oishi, 2013, Synlett.

Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group.

M. Matsuoka, N. Fujii, H. Ohno, 2009, Bioorganic & medicinal chemistry.

Samarium(II)-promoted radical spirocyclization onto an aromatic ring.

H. Ohno, Tetsuaki Tanaka, Hiroki Iwasaki, 2003, The Journal of organic chemistry.

Umpolung of chiral 2-ethynylaziridines: Indium(I)-mediated stereoselective synthesis of nonracemic 1,3-amino alcohols bearing three chiral centers, catalyzed by palladium(0)

Ohno, H. Ohno, H. Hamaguchi, 2000, Organic letters.

Cu(II)-Mediated Oxidative Intermolecular ortho C—H Functionalization Using Tetrahydropyrimidine as the Directing Group.

N. Fujii, H. Ohno, S. Oishi, 2009 .

Development of a 1:1-binding biparatopic anti-TNFR2 antagonist by epitope selection

K. Namba, K. Tsumoto, T. Ise, 2022, bioRxiv.

Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid-phase synthesis of a cyclic pentapeptide mimetic

T. Narumi, N. Fujii, H. Ohno, 2008 .

Development of novel CXC chemokine receptor 7 (CXCR7) ligands: selectivity switch from CXCR4 antagonists with a cyclic pentapeptide scaffold.

N. Heveker, N. Fujii, H. Ohno, 2015, Journal of medicinal chemistry.

Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations.

K. Kitaura, T. Narumi, A. Otaka, 2006, The Journal of organic chemistry.

Synthesis of IB-01212 by multiple N-methylations of peptide bonds.

N. Fujii, H. Ohno, S. Oishi, 2014, Bioorganic & medicinal chemistry.

Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor.

N. Fujii, H. Ohno, S. Oishi, 2016, Chemical & pharmaceutical bulletin.

Identification of minimal sequence for HIV-1 fusion inhibitors.

M. Matsuoka, A. Otaka, N. Fujii, 2008, Bioorganic & Medicinal Chemistry.

A Novel Oxazolidine Linker for the Synthesis of Peptide Aldehydes

N. Fujii, H. Ohno, S. Oishi, 2007, International Journal of Peptide Research and Therapeutics.

Double C-H functionalization in sequential order: direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade.

N. Fujii, H. Ohno, Tetsuaki Tanaka, 2012, Chemistry.

Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines.

N. Fujii, H. Ohno, S. Oishi, 2014, Organic letters.

Synthesis and applications of vinylaziridines and ethynylaziridines.

H. Ohno, 2014, Chemical reviews.

Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates.

N. Fujii, H. Ohno, S. Oishi, 2010, Journal of Organic Chemistry.

Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization.

H. Ohno, Tetsuaki Tanaka, Mio Yamamoto, 2005, Angewandte Chemie.

Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes.

N. Fujii, H. Ohno, S. Oishi, 2012, The Journal of organic chemistry.

Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne.

N. Fujii, H. Ohno, Y. Yoshida, 2016, The Journal of organic chemistry.

Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization.

N. Fujii, H. Ohno, S. Oishi, 2009, The Journal of organic chemistry.

Bromoallenes as synthetic equivalents of allyl dications: synthesis of medium-sized nitrogen heterocycles through the cyclization of bromoallenes in the presence of a palladium(0) catalyst and an alcohol.

H. Ohno, H. Hamaguchi, Miyo Ohata, 2003, Angewandte Chemie.

A highly cis-selective synthesis of 2-ethynylaziridines by intramolecular amination of chiral bromoallenes: improvement of stereoselectivity based on the computational investigation.

H. Ohno, K. Ando, H. Hamaguchi, 2002, Journal of the American Chemical Society.

Selective Synthesis of Nonracemic 3-Pyrrolines and 2,3-cis-2-Vinylaziridines from (Z)-Amino Allylic Alcohols: A New Synthetic Route to Chiral 3,4-Dehydroproline

H. Ohno, Y. Takemoto, T. Ibuka, 1999 .

Rhodium(I)- or Iridium(I)-Mediated Equilibrated Reactions of Activated 2,3-cis- and trans-3-Alkyl-2-vinylaziridines

H. Ohno, T. Ibuka, N. Mimura, 1998 .

Synthesis of fused and linked bicyclic nitrogen heterocycles by palladium-catalyzed domino cyclization of propargyl bromides.

N. Fujii, H. Ohno, S. Oishi, 2010, Chemistry.

Structure − Activity Relationship Study on Odoamide: Insights into the Bioactivities of Aurilide-Family Hybrid Peptide − Polyketides

N. Fujii, H. Ohno, S. Oishi, 2018 .

Development of a novel fusion inhibitor against T-20-resistant HIV-1.

M. Matsuoka, A. Otaka, N. Fujii, 2009, Advances in experimental medicine and biology.

Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors.

G. Tsujimoto, N. Fujii, H. Ohno, 2013, Organic & biomolecular chemistry.