S. Gerritz

发表

Influenza Nucleoprotein: Promising Target for Antiviral Chemotherapy

C. Cianci, S. Gerritz, Carol Deminie, 2012, Antiviral chemistry & chemotherapy.

9 – The Role of NMR in the Analysis of Chemical Libraries

S. Gerritz, A. Sefler, 2004 .

Identification and biochemical analyses of selective CB2 agonists.

Caitlin E. Scott, S. Gerritz, Litao Zhang, 2019, European journal of pharmacology.

Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptor.

Kathryn E. Livingston, A. Christopoulos, M. Banks, 2015, Journal of medicinal chemistry.

Editorial overviewCombinatorial chemistry: Rumors of the demise of combinatorial chemistry are greatly exaggerated

S. Gerritz, A. Merritt, 2003 .

Identification and biochemical analyses of selective CB 2 agonists

Ogawa, Caitlin E. Scott, S. Gerritz, 2019 .

Discovery and optimization of (R)-prolinol-derived agonists of the Growth Hormone Secretagogue receptor (GHSR).

R. Stoffel, S. Gerritz, D. Gordon, 2008, Bioorganic & medicinal chemistry letters.

Discovery of Selective Cannabinoid CB2 Receptor Agonists by High-Throughput Screening

Caitlin E. Scott, M. Banks, S. Gerritz, 2018, SLAS discovery : advancing life sciences R & D.

Regulated Induced Proximity Targeting Chimeras (RIPTACs): a Novel Heterobifunctional Small Molecule Therapeutic Strategy for Killing Cancer Cells Selectively

C. Crews, S. Gerritz, J. Mousseau, 2023, bioRxiv.

Solid-phase synthesis of a library based on biphenyl-containing trypsin-like serine protease inhibitors.

D. Cheney, S. Gerritz, M. Sofia, 2009, Bioorganic & medicinal chemistry letters.

Solid-phase synthesis of trisubstituted guanidines

D. Drewry, S. Gerritz, J. A. Linn, 1997 .

Solid phase synthesis of 1,3,5-trisubstituted pyridin-2-ones

S. Gerritz, D. Heyer, A. L. Handlon, 1999 .

Solid phase synthesis of 1,5-disubstituted pyrazole-4-hydroxamic acids and pyrazole-4-carboxamides via direct amidation of β-ketoesters

S. Gerritz, M. Sofia, W. Zhai, 2012 .

Highly selective reducing agents. Reduction of nitrobenzene to aniline in the presence of aldehydes, alkyl halides, and acid halides.

P. L. Gaus, S. Gerritz, Patrick M. Jeffries, 1989 .

Solid phase synthesis of novel pyrrolidinedione analogs as potent HIV-1 integrase inhibitors.

N. Meanwell, Zeyu Lin, S. Gerritz, 2010, Journal of combinatorial chemistry.

A facile one-step synthesis of 5-chloro-imidazo[1,5-a]quinazoline by microwave irradiation

S. Gerritz, Guo Li, R. Kakarla, 2009 .

Optimization of focused chemical libraries using recursive partitioning.

Andrew Rusinko, David H Drewry, S Stanley Young, 2002, Combinatorial chemistry & high throughput screening.

Discovery and Optimization of Novel Pyrazolopyrimidines as Potent and Orally Bioavailable Allosteric HIV-1 Integrase Inhibitors.

K. Kish, G. Trainor, N. Meanwell, 2020, Journal of medicinal chemistry.

A fast and efficient bromination of isoxazoles and pyrazoles by microwave irradiation

S. Gerritz, Guo Li, R. Kakarla, 2007 .

Discovery of pyrazine carboxamide CB1 antagonists: the introduction of a hydroxyl group improves the pharmaceutical properties and in vivo efficacy of the series.

Ying Wang, Samuel W Gerritz, William R Ewing, 2007, Bioorganic & medicinal chemistry letters.

Attachment of unreactive amines to the solid support: synthesis of phenyl-substituted anilines, 2-aminopyridines, and 2-aminopyrimidines.

S. Gerritz, M. Sofia, Shirong Zhu, 2003, Journal of combinatorial chemistry.

Solid-phase synthesis and anti-infective activity of a combinatorial library based on the natural product anisomycin.

Y. Shu, K. S. Lam, S. Gerritz, 2005, Bioorganic & medicinal chemistry letters.

Inhibition of influenza virus replication via small molecules that induce the formation of higher-order nucleoprotein oligomers

Eric T Baldwin, Samuel W Gerritz, Michael Sinz, 2011, Proceedings of the National Academy of Sciences.

A Novel Small Molecule Inhibitor of Hepatitis C Virus Entry

M. Poss, N. Meanwell, C. Mazzucco, 2010, PLoS pathogens.

Macrocyclic prolinyl acyl guanidines as inhibitors of β-secretase (BACE).

A. Good, J. Macor, C. Albright, 2015, Bioorganic & medicinal chemistry letters.

Biochemical and behavioral effects of PDE10A inhibitors: Relationship to target site occupancy

M. Seager, J. Macor, S. Gerritz, 2016, Neuropharmacology.

A High-Throughput Screen for Receptor Protein Tyrosine Phosphatase–γ Selective Inhibitors

M. Banks, C. Albright, S. Gerritz, 2011, Journal of biomolecular screening.

Discovery of positive allosteric modulators and silent allosteric modulators of the μ-opioid receptor

M. Banks, S. Gerritz, J. Traynor, 2013, Proceedings of the National Academy of Sciences.

Quantitative techniques for the comparison of solid supports.

S. Gerritz, 2001, Current opinion in chemical biology.

Identification and Preclinical Pharmacology of the γ-Secretase Modulator BMS-869780

J. Macor, M. Ahlijanian, Joseph L. Cantone, 2014, International journal of Alzheimer's disease.

Small molecule receptor protein tyrosine phosphatase γ (RPTPγ) ligands that inhibit phosphatase activity via perturbation of the tryptophan-proline-aspartate (WPD) loop.

V. Goldfarb, B. Beno, J. Macor, 2011, Journal of medicinal chemistry.

Probing the Reactivity of Solid Supports via Hammett Relationships

W. Zuercher, S. Gerritz, R. Trump, 2000 .

High-Throughput Screening and Rapid Inhibitor Triage Using an Infectious Chimeric Hepatitis C Virus

B. Beno, J. Leet, C. Mazzucco, 2012, PloS one.

Small-molecule pyrimidine inhibitors of the cdc2-like (Clk) and dual specificity tyrosine phosphorylation-regulated (Dyrk) kinases: development of chemical probe ML315.

Thomas C. Coombs, D. Auld, M. Shen, 2013, Bioorganic & medicinal chemistry letters.

Two general routes to 1,4-disubstituted-2,3,4,5-tetrahydro- 1H-3-benzazepines.

S. Gerritz, D. Uehling, S. Nanthakumar, 2000, Organic letters.

Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptor.

Kathryn E. Livingston, A. Christopoulos, M. Banks, 2015, Journal of medicinal chemistry.

Rapid Compound Integrity Assessment for High-Throughput Screening Hit Triaging

Peter Chase, Wilson Z Shou, Harold N Weller, 2020, SLAS discovery : advancing life sciences R & D.

Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the μ-Opioid Receptor

Marta Filizola, Paola Bisignano, Yi Shang, 2015, J. Chem. Inf. Model..