A. Carta

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Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives.

E. Laurini, M. Fermeglia, S. Pricl, 2015, European journal of medicinal chemistry.

Inhibitors of Yellow Fever Virus replication based on 1,3,5-triphenyl-4,5-dihydropyrazole scaffold: Design, synthesis and antiviral evaluation.

R. Loddo, A. Carta, I. Delogu, 2017, European journal of medicinal chemistry.

Structure-based selectivity optimization of piperidine-pteridine derivatives as potent Leishmania pteridine reductase inhibitors.

A. Cavalli, P. Michels, V. Hannaert, 2012, Journal of medicinal chemistry.

Solid Lipid Nanoparticles as Formulative Strategy to Increase Oral Permeation of a Molecule Active in Multidrug-Resistant Tuberculosis Management

L. Ferraro, S. Piras, P. Giunchedi, 2020, Pharmaceutics.

[1,2,3]Triazolo[4,5-h]quinolones. A new class of potent antitubercular agents against multidrug resistant Mycobacterium tuberculosis strains.

S. Cannas, S. Zanetti, A. Carta, 2007, Bioorganic & medicinal chemistry letters.

Synthesis and antimycobacterial activity of 3-aryl-, 3-cyclohexyl- and 3-heteroaryl- substituted-2-(1H(2H)-benzotriazol-1(2)-yl)prop-2-enenitriles, prop-2-enamides and propenoic acids. II.

A. Carta, P. Sanna, L. Gherardini, 2002, Farmaco.

Phytochemical Compositions and Biological Activities of Essential Oils from the Leaves, Rhizomes and Whole Plant of Hornstedtia bella Škorničk

S. Zanetti, P. Rappelli, P. Cappuccinelli, 2020, Antibiotics.

5,6-Dichloro-2-Phenyl-Benzotriazoles: New Potent Inhibitors of Orthohantavirus

R. Loddo, S. Piras, P. Corona, 2020, Viruses.

Determination of amphetamine-derived designer drugs in human urine by SPE extraction and capillary electrophoresis with mass spectrometry detection.

A. Carta, A. Pau, B. Asproni, 2005, Journal of chromatography. B, Analytical technologies in the biomedical and life sciences.

Antiviral Activity of Benzotriazole Based Derivatives

R. Loddo, S. Piras, P. Corona, 2020 .

Supercritical fluid extraction and GC detection of p,p1-DDE and PCB congeners in some samples of dying species from Sardinia

A. Carta, G. Chessa, G. Boatto, 2003 .

Screening Method for Five Commonly Used Amphetamines in Urine by NMR Spectroscopy

N. Culeddu, A. Carta, M. Porcu, 2014 .

Quinoxaline 1,4-dioxide: a versatile scaffold endowed with manifold activities.

P. Corona, A. Carta, M. Loriga, 2005, Current medicinal chemistry.

Antibiotics and Carbohydrate-Containing Drugs Targeting Bacterial Cell Envelopes: An Overview

S. Sestito, S. Piras, A. Carta, 2022, Pharmaceuticals.

Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives

D. Schuster, V. Temml, S. Piras, 2021, Molecules.

Reactions of benzotriazoles with diethyl ethoxymethylenemalonate; ethylation and michael addition. Comparison with other esters and N-heterocycles

A. Bacchi, A. Carta, G. Pelizzi, 1997 .

Design, synthesis, and biological screening of a series of 4′-fluoro-benzotriazole-acrylonitrile derivatives as microtubule-destabilising agents (MDAs)

L. Bagella, S. Piras, A. Carta, 2022, Journal of enzyme inhibition and medicinal chemistry.

Inhibition of Enterovirus A71 by a Novel 2-Phenyl-Benzimidazole Derivative

S. Sestito, R. Loddo, S. Piras, 2021, Viruses.

Quinoxaline‐based efflux pump inhibitors restore drug susceptibility in drug‐resistant nontuberculous mycobacteria

S. Piras, P. Corona, A. Carta, 2022, Archiv der Pharmazie.

Human Enterovirus B: Selective Inhibition by Quinoxaline Derivatives and Bioinformatic RNA-Motif Identification as New Targets

S. Piras, G. Sanna, A. Carta, 2022, Pharmaceuticals.

Synthesis, anti-mycobacterial, anti-trichomonas and anti-candida in vitro activities of 2-substituted-6,7-difluoro-3-methylquinoxaline 1,4-dioxides.

S. Zanetti, L. Sechi, A. Carta, 2004, European journal of medicinal chemistry.

Role of ethanol-derived acetaldehyde in operant oral self-administration of ethanol in rats

M. Rosas, E. Acquas, A. Carta, 2015, Psychopharmacology.

Synthesis and in vitro antitumor activity of new quinoxaline derivatives.

P. Corona, A. Carta, M. Loriga, 2009, European journal of medicinal chemistry.

Validated LC-MS-MS Method for Multiresidual Analysis of 13 Illicit Phenethylamines in Amniotic Fluid.

A. Carta, C. Trignano, G. Boatto, 2016, Journal of analytical toxicology.

LC-MS/MS analysis of acetaminophen and caffeine in amniotic fluid

A. Carta, C. Trignano, G. Boatto, 2015 .

Novel substituted quinoxaline 1,4-dioxides with in vitro antimycobacterial and anticandida activity.

S. Zanetti, L. Sechi, A. Carta, 2002, European journal of medicinal chemistry.

Chemistry, biological properties and SAR analysis of quinoxalinones.

S. Piras, A. Carta, G. Loriga, 2006, Mini reviews in medicinal chemistry.

Synthesis and in vitro evaluation of the anti-viral activity of N-[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl]alkylcarboxamides.

M. Ferrone, M. Fermeglia, S. Pricl, 2006, Medicinal chemistry (Shariqah (United Arab Emirates)).

Synthesis of variously substituted 3-phenoxymethyl quinoxalin-2-ones and quinoxalines capable to potentiate in vitro the antiproliferative activity of anticancer drugs in multi-drug resistant cell lines.

R. Loddo, S. Piras, P. la Colla, 2006, Medicinal chemistry (Shariqah (United Arab Emirates)).

Synthesis of 3,6,7-substituted-quinoxalin-2-ones for evaluation of antimicrobial and anticancer activity. Part 2.

S. Zanetti, L. Sechi, A. Carta, 1999, Farmaco.

Design, Synthesis, Antiviral Evaluation, and SAR Studies of New 1-(Phenylsulfonyl)-1H-Pyrazol−4-yl-Methylaniline Derivatives

R. Loddo, A. Carta, I. Delogu, 2019, Front. Chem..

Synthesis and antiproliferative activity of 3-aryl-2-[1H(2H)-benzotriazol-1(2)-yl]acrylonitriles variously substituted: Part 4.

R. Loddo, A. Carta, B. Busonera, 2004, Farmaco.

Synthesis and antiproliferative activity of 3-aryl-2-(1H-benzotriazol-1-yl)acrylonitriles. Part III.

R. Loddo, A. Carta, M. La Colla, 2002, European journal of medicinal chemistry.

Synthesis of Two Novel Tricyclic Rings:Triazolo[4,5-g]quinolines and Pyrido[2,3-g]quinoxalines Derived from 6,7-Diaminoquinolines

A. Carta, G. Paglietti, P. Sanna, 2000 .

Synthesis and evaluation for biological activity of 3-alkyl and 3-halogenoalkyl-quinoxalin-2-ones variously substituted. Part 4.

R. Loddo, A. Carta, M. Loriga, 2002, Farmaco.

A New synthesis of triazolo[4,5-g]quinolines and unexpected ring reduced products by treatment with hydrazine hydrate

A. Carta, G. Paglietti, 2004 .

5-acetyl-2-arylbenzimidazoles as antiviral agents. Part 4.

P. Corona, G. Sanna, G. Giliberti, 2012, European journal of medicinal chemistry.

Benzotriazole: An overview on its versatile biological behavior

I. Briguglio, S. Piras, P. Corona, 2014, European Journal of Medicinal Chemistry.

Synthesis and antitubercular activity of 3-aryl substituted-2-[1H(2H)benzotriazol-1(2)-yl]acrylonitriles.

A. Carta, M. Nikookar, P. Sanna, 2000, European journal of medicinal chemistry.

Design, synthesis, and preliminary in vitro and in silico antiviral activity of [4,7]phenantrolines and 1-oxo-1,4-dihydro-[4,7]phenantrolines against single-stranded positive-sense RNA genome viruses.

M. Ferrone, M. Fermeglia, S. Pricl, 2007, Bioorganic & medicinal chemistry.

Biological Activities of Essential Oils from Leaves of Paramignya trimera (Oliv.) Guillaum and Limnocitrus littoralis (Miq.) Swingle

S. Zanetti, P. Rappelli, P. Cappuccinelli, 2020, Antibiotics.

Inhibition of RNA Helicases of ssRNA+ Virus Belonging to Flaviviridae, Coronaviridae and Picornaviridae Families

I. Briguglio, S. Piras, P. Corona, 2010, International journal of medicinal chemistry.

3-Aryl-2-[1H-benzotriazol-1-yl]acrylonitriles: a novel class of potent tubulin inhibitors.

E. Laurini, M. Fermeglia, S. Pricl, 2011, European journal of medicinal chemistry.

Novel substituted quinoxaline 1,4-dioxides with in vitro antimycobacterial and anticandida activity.

Giuseppe Paglietti, S. Zanetti, L. Sechi, 2002, European journal of medicinal chemistry.

Synthesis and in vitro antitumor activity of new quinoxaline derivatives.

P. Corona, A. Carta, M. Loriga, 2009, European journal of medicinal chemistry.

Triazolopyridinyl-acrylonitrile derivatives as antimicrotubule agents: Synthesis, in vitro and in silico characterization of antiproliferative activity, inhibition of tubulin polymerization and binding thermodynamics.

E. Laurini, M. Fermeglia, S. Pricl, 2017, European journal of medicinal chemistry.

Synthesis and anti-mycobacterial activities of triazoloquinolones.

S. Zanetti, I. Briguglio, S. Piras, 2011, European journal of medicinal chemistry.

Synthesis and Antiproliferative Activity of 3-Aryl-2-(1H-benzotriazol-1-yl)acrylonitriles (III). Part 3.

R. Loddo, A. Carta, M. Palomba, 2003 .

Novel functionalized pyrido[2,3-g]quinoxalinones as antibacterial, antifungal and anticancer agents.

S. Zanetti, A. Carta, D. Usai, 2001, Farmaco.

Preparation and biological evaluation of 6/7-trifluoromethyl(nitro)-, 6,7-difluoro-3-alkyl (aryl)-substituted-quinoxalin-2-ones. Part 3.

S. Zanetti, L. Sechi, A. Carta, 1999, Farmaco.

1,2,3-triazolo[4,5-h]quinolines. III. Preparation and antimicrobial evaluation of 4-ethyl-4,7-dihydro-1(2)-R-1(2)H triazolo[4,5-h]quinolin-7-one-6-carboxylic acids as anti-infectives of the urinary tract.

S. Zanetti, G. Fadda, A. Carta, 1990, Farmaco.

Synthesis and Antiproliferative Activity of 3-Aryl-2-[1H(2H)-benzotriazol-1(2)-yl]acrylonitriles Variously Substituted. Part 4.

R. Loddo, A. Carta, B. Busonera, 2004 .

Synthesis and Biological Evaluation of Triazolo[4,5- g ]quinolines, Imidazo[4,5- g ]quinolines and Pyrido[2,3- g ]quinoxaline. Part II

A. Carta, G. Paglietti, P. Caredda, 2003 .

13C-NMR as useful tool for unambiguous identification of ring substituted N1(2)(3)-alkylbenzotriazole isomers

A. Carta, F. Sparatore, G. Paglietti, 2001 .

Synthesis of substituted 2-ethoxycarbonyl- and 2-carboxyquinoxalin-3-ones for evaluation of antimicrobial and anticancer activity.

S. Zanetti, L. Sechi, A. Carta, 1998, Farmaco.

Structural Elucidation of Isomeric Methyl (E)-3-[5-Aminobenzotriazol-1(2)(3)-yl]propenoates by NMR Spectroscopy

H. Molinari, A. Carta, P. Sanna, 1997 .

Synthesis of substituted 2-ethoxycarbonyl- and 2-carboxyquinoxalin-3-ones for evaluation of antimicrobial and anticancer activity.

S. Zanetti, L. Sechi, A. Carta, 1998, Farmaco.

Quinoxalin-2-ones. Part 5. Synthesis and antimicrobial evaluation of 3-alkyl-, 3-halomethyl- and 3-carboxyethylquinoxaline-2-ones variously substituted on the benzo-moiety.

S. Zanetti, L. Sechi, A. Carta, 2003, Farmaco.

2-[N-Alkyl(R-phenyl)-aminomethyl]-3-phenyl-7-trifluoromethylquinoxalines as anticancer agents inhibitors of folate enzymes.

Maria Paola Costi, I. Briguglio, S. Piras, 2014, European journal of medicinal chemistry.

Novel 3-benzoyl-2-piperazinylquinoxaline derivatives as potential antitumor agents

Maria Paola Costi, S. Piras, A. Carta, 2006 .

Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines.

I. Briguglio, R. Loddo, S. Piras, 2014, European journal of medicinal chemistry.

Quinoline tricyclic derivatives. Design, synthesis and evaluation of the antiviral activity of three new classes of RNA-dependent RNA polymerase inhibitors.

I. Briguglio, S. Piras, P. Corona, 2011, Bioorganic & medicinal chemistry.

Activity and molecular modeling of a new small molecule active against NNRTI-resistant HIV-1 mutants.

M. Fermeglia, S. Pricl, R. Loddo, 2009, European journal of medicinal chemistry.

Synthesis of Two Novel Tricyclic Rings: Triazolo[4,5-g]quinolines and Pyrido[2,3-g]quinoxalines Derived from 6,7-Diaminoquinolines.

A. Carta, G. Paglietti, P. Sanna, 2000 .

Synthesis, anti‐Mycobacterial, anti‐Trichomonas and anti‐Candida in vitro Activities of 2‐Substituted‐6,7‐difluoro‐3‐methylquinoxaline 1,4‐Dioxides.

S. Zanetti, L. Sechi, A. Carta, 2004 .

Improvement of thymol properties by complexation with cyclodextrins: in vitro and in vivo studies.

P. Giunchedi, E. Gavini, A. Carta, 2014, Carbohydrate polymers.

Evaluation of the effect of hydroxypropyl-β-cyclodextrin on topical administration of milk thistle extract.

P. Giunchedi, E. Gavini, A. Carta, 2013, Carbohydrate polymers.

Antiviral activities of 5-chlorobenzotriazole derivatives

R. Loddo, S. Piras, P. Corona, 2018, Monatshefte für Chemie - Chemical Monthly.

A combined in silico/in vitro approach unveils common molecular requirements for efficient BVDV RdRp binding of linear aromatic N-polycyclic systems.

E. Laurini, M. Fermeglia, S. Pricl, 2016, European journal of medicinal chemistry.

Enhancement of antimicrobial activity of pump inhibitors associating drugs.

S. Zanetti, S. Piras, P. Corona, 2019, Journal of infection in developing countries.

Synthesis of Linear Azolo and Pyrido Quinolines from Quinoline Derivatives

S. Piras, P. Corona, A. Carta, 2008 .

Synthesis, Antitumor and Antiviral In Vitro Activities of New Benzotriazole-Dicarboxamide Derivatives

R. Loddo, S. Piras, P. Corona, 2021, Frontiers in Chemistry.

Design, synthesis and antitubercular activity of 4-alkoxy-triazoloquinolones able to inhibit the M. tuberculosis DNA gyrase.

S. Zanetti, E. Laurini, Suzana Aulic, 2019, European journal of medicinal chemistry.

Synthesis of Substituted Aminoquinolines as Useful Intermediates for Preparation of Aromatic N-Tricyclic Systems

P. Corona, A. Carta, M. Palomba, 2006 .

Benzimidazole-2-Phenyl-Carboxamides as Dual-Target Inhibitors of BVDV Entry and Replication

R. Loddo, S. Piras, A. Carta, 2022, Viruses.

Preliminary anti-Coxsackie activity of novel 1-[4-(5,6-dimethyl(H)-1H(2H)-benzotriazol-1(2)-yl)phenyl]-3-alkyl(aryl)ureas.

R. Loddo, S. Piras, P. Corona, 2019, Medicinal chemistry.

Dichloro-Phenyl-Benzotriazoles: A New Selective Class of Human Respiratory Syncytial Virus Entry Inhibitors

E. Laurini, Suzana Aulic, M. Fermeglia, 2019, Front. Chem..

Quinoxaline derivatives as new inhibitors of coxsackievirus B5.

E. Laurini, M. Fermeglia, S. Pricl, 2017, European journal of medicinal chemistry.

Synthesis and anti-picornaviridae in vitro activity of a new class of helicase inhibitors the N,N'-bis[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl] alkyldicarboxamides.

M. Ferrone, M. Fermeglia, S. Pricl, 2007, Medicinal chemistry (Shariqah (United Arab Emirates)).

In vitro activity of new quinoxalin 1,4-dioxide derivatives against strains of Mycobacterium tuberculosis and other mycobacteria.

S. Cannas, S. Zanetti, L. Sechi, 2005, International journal of antimicrobial agents.

Choleretic activity of 3-[ring substituted benzotriazol-1(2)-yl]alkanoic and alkenoic acids.

A. Carta, F. Sparatore, G. Paglietti, 1994, Farmaco.

Propolis as lipid bioactive nano-carrier for topical nasal drug delivery.

R. Cavalli, P. Giunchedi, E. Gavini, 2015, Colloids and surfaces. B, Biointerfaces.

2-Carboxyquinoxalines kill mycobacterium tuberculosis through noncovalent inhibition of DprE1.

Maria Paola Costi, S. Cole, L. Chiarelli, 2015, ACS chemical biology.

In vitro activity of quinoxaline 1,4-dioxides derivatives against enterococci clinical strains

S. Zanetti, A. Carta, D. Usai, 2004 .

Simultaneous determination of ten amphetamine designer drugs in human whole blood by capillary electrophoresis with diode array detection.

A. Carta, A. Sanna, G. Boatto, 2005, Biomedical chromatography : BMC.

SAR and Anti-Mycobacterial Activity of Quinolones and Triazoloquinolones: An Update

I. Briguglio, S. Piras, P. Corona, 2012 .

A Lead-Based Fragment Library Screening of the Glycosyltransferase WaaG from Escherichia coli

D. Daley, A. Carta, Jonas Ståhle, 2022, Pharmaceuticals.

Enantiomeric separation of 13 new amphetamine-like designer drugs by capillary electrophoresis, using modified-B-cyclodextrins.

I. Briguglio, A. Carta, G. Boatto, 2013, Chirality.

2-Arylbenzimidazoles as antiviral and antiproliferative agents--Part 2.

R. Loddo, P. Corona, P. la Colla, 2009, Medicinal chemistry (Shariqah (United Arab Emirates)).

2-Arylbenzimidazoles as antiviral and antiproliferative agents. Part 1.

R. Loddo, P. la Colla, A. Carta, 2008, Medicinal chemistry (Shariqah (United Arab Emirates)).

Styrylbenzimidazoles. Synthesis and biological activity - part 3.

R. Loddo, P. Corona, G. Giliberti, 2010, Medicinal chemistry (Shariqah (United Arab Emirates)).

Determinazione analitica di designer drugs amfetamino simili in matrici complesse

A. Carta, 2016 .

Determination of phenol and o-cresol by GC/MS in a fatal poisoning case.

A. Carta, D. Serra, A. Pau, 2004, Forensic science international.

Structure-based selectivity optimization of piperidine-pteridine derivatives as potent Leishmania pteridine reductase inhibitors.

A. Cavalli, P. Michels, V. Hannaert, 2012, Journal of medicinal chemistry.

Design, Synthesis, and Antiviral Activities of New Benzotriazole-Based Derivatives

R. Loddo, S. Piras, P. Corona, 2023, Pharmaceuticals.

5-acetyl-2-arylbenzimidazoles as antiviral agents. Part 4.

P. Corona, G. Sanna, G. Giliberti, 2012, European journal of medicinal chemistry.