B. Ilien

发表

Pirenzepine Promotes the Dimerization of Muscarinic M1 Receptors through a Three-step Binding Process*

J. Galzi, Y. Mély, P. Didier, 2009, The Journal of Biological Chemistry.

RF-amide neuropeptides and their receptors in Mammals: Pharmacological properties, drug development and main physiological functions.

F. Bihel, F. Simonin, B. Ilien, 2016, Pharmacology & therapeutics.

FLUORESCENr MIJSCARINIC EGFP-hM 1 CHIMERJC RECEPTORS: DESIGN, LICiAND BINDING AND FUNCTIONAL, PR.OPERTIES

C. Weill, B. Ilien, M. Goeldner, 1999 .

Fluorescent muscarinic EGFP-hM1 chimeric receptors: design, ligand binding and functional properties.

J. Galzi, C. Weill, B. Ilien, 1999, Journal of receptor and signal transduction research.

Synthesis and purification of highly tritiated aryldiazonium photoprobes for cholinergic binding sites

B. Ilien, M. Goeldner, F. Sobrio, 1996 .

Fluorescent derivatives of AC-42 to probe bitopic orthosteric/allosteric binding mechanisms on muscarinic M1 receptors.

Esther Kellenberger, Marcel Hibert, Jean-Luc Galzi, 2012, Journal of medicinal chemistry.

Fluorescent pirenzepine derivatives as potential bitopic ligands of the human M1 muscarinic receptor.

J. Galzi, I. Parrot, B. Ilien, 2004, Journal of medicinal chemistry.

On the Use of Nonfluorescent Dye Labeled Ligands in FRET-Based Receptor Binding Studies

J. Galzi, B. Ilien, P. Klotz, 2005 .

Direct and energy-transfer photolabelling of brain muscarinic acetylcholine receptors.

B. Ilien, C. Hirth, 1989, European journal of biochemistry.

Muscarinic acetylcholine receptor: thermodynamic analysis of the interaction of agonists and antagonists.

J. Gies, B. Ilien, Y. Landry, 1986, Biochimica et biophysica acta.

Solubilized serotonin receptors from rat and dog brain

B. Ilien, P. Laduron, A. Schotte, 1982, FEBS letters.

Solubilization of serotonin receptors from rat frontal Cortex.

B. Ilien, P. Laduron, H. Gorissen, 1980, Biochemical pharmacology.

Differentiation of solubilized dopamine receptors from spirodecanone binding sites in rat striatum

B. Ilien, P. Laduron, G. Aerts, 1980, FEBS letters.

Endogenous mammalian RF-amide peptides, including PrRP, kisspeptin and 26RFa, modulate nociception and morphine analgesia via NPFF receptors

T. Sorg, H. Meziane, F. Bihel, 2013, Neuropharmacology.

On the use of nonfluorescent dye labeled ligands in FRET-based receptor binding studies.

J. Galzi, B. Ilien, P. Klotz, 2005, Journal of medicinal chemistry.

A mu-opioid receptor-filter assay. Rapid estimation of binding affinity of ligands and reversibility of long-lasting ligand-receptor complexes.

J. Galzi, B. Ilien, A. Méjean, 1988, Biochemical pharmacology.

Identification of an N-acylated-DArg-Leu-NH2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia.

F. Bihel, F. Simonin, M. Schmitt, 2021, Journal of medicinal chemistry.

RF313, an orally bioavailable neuropeptide FF receptor antagonist, opposes effects of RF-amide-related peptide-3 and opioid-induced hyperalgesia in rodents

T. Sorg, H. Meziane, F. Bihel, 2017, Neuropharmacology.

Assessment of Morphine-induced Hyperalgesia and Analgesic Tolerance in Mice Using Thermal and Mechanical Nociceptive Modalities

F. Simonin, B. Ilien, Safia Ayachi, 2014, Journal of visualized experiments : JoVE.

Separation of three cyclic-nucleotide-phosphodiesterases from bovine aorta.

A. Stierlé, B. Ilien, C. Lugnier, 1978, Biochemical and biophysical research communications.

Exploration of the Orthosteric/Allosteric Interface in Human M1 Muscarinic Receptors by Bitopic Fluorescent Ligands

Esther Kellenberger, Jean-Luc Galzi, E. Kellenberger, 2013, Molecular Pharmacology.

Analytical Subcellular Fractionation of Rat Cortex: Resolution of Serotonergic Nerve Endings and Receptors

B. Ilien, P. Laduron, P. Janssen, 1983, Journal of neurochemistry.

Covalent labeling of muscarinic acetylcholine receptors by tritiated aryldiazonium photoprobes.

C. Weill, B. Ilien, M. Goeldner, 1997, Biochemical pharmacology.

A rapid and versatile method to label receptor ligands using "click" chemistry: Validation with the muscarinic M1 antagonist pirenzepine.

J. Galzi, B. Ilien, D. Bonnet, 2006, Bioconjugate chemistry.

New photoaffinity labels for rat brain muscarinic acetylcholine receptors.

B. Ilien, A. Méjean, C. Hirth, 1989, Biochemical pharmacology.

Solubilization of muscarinic acetylcholine receptors from mammalian brain: an analytical approach.

B. Ilien, P. Laduron, G. Aerts, 1981, Analytical biochemistry.

Characterization of solubilized serotonin (S2) receptors in rat brain.

B. Ilien, P. Laduron, H. Gorissen, 1982, Molecular pharmacology.

Pharmacological and structural integrity of muscarinic M2 acetylcholine receptors produced in Sf9 insect cells.

C. Guenet, C. Weill, B. Ilien, 1997, European journal of pharmacology.

Time-resolved FRET binding assay to investigate hetero-oligomer binding properties: proof of concept with dopamine D1/D3 heterodimer.

D. Rognan, J. Pin, A. Mann, 2015, ACS chemical biology.

Sodium‐potassium ATPase inhibition potentiates compound 48/80‐induced histamine secretion from mast cells

N. Frossard, B. Ilien, Y. Landry, 1984, British journal of pharmacology.

Fluorescence resonance energy transfer to probe human M1 muscarinic receptor structure and drug binding properties

J. Galzi, J. Bourguignon, B. Ilien, 2003, Journal of neurochemistry.

Photoactivatable opiate derivatives as irreversible probes of the mu-opioid receptor.

J. Galzi, B. Ilien, J. Meunier, 1990, Journal of medicinal chemistry.

m‐Sulfonate Benzene Diazonium Chloride: A Powerful Affinity Label for the γ‐Aminobutyric Acid Binding Site from Rat Brain

M. Bouchet, B. Ilien, M. Goeldner, 1992, Journal of neurochemistry.

Solubilization of brain muscarinic, dopaminergic and serotonergic receptors: a critical analysis.

B. Ilien, P. Laduron, 1982, Biochemical pharmacology.

Photoaffinity labelling of the mu-opioid receptor is dependent on the nature of the photosensitive group of carfentanil derivatives.

J. Galzi, B. Ilien, M. Goeldner, 1990, European journal of pharmacology.

A μ-opioid receptor-filter assay: Rapid estimation of binding affinity of ligands and reversibility of long-lasting ligand-receptor complexes

J. Galzi, B. Ilien, M. Goeldner, 1988 .

Pharmacological inhibition of calmodulin-sensitive phosphodiesterases.

B. Ilien, M. Ruckstuhl, Y. Landry, 1982, Journal de pharmacologie.

Functional Characterization and Potential Applications for Enhanced Green Fluorescent Protein‐ and Epitope‐Fused Human M1 Muscarinic Receptors

J. Galzi, S. Chasserot-Golaz, C. Weill, 1999, Journal of neurochemistry.