I. Mándity

发表

FoldamerDB: a database of peptidic foldamers

T. Beke-Somfai, Bilal Nizami, Dorottya Bereczki-Szakál, 2019, Nucleic Acids Res..

Design and Selection of Novel C1s Inhibitors by In Silico and In Vitro Approaches

P. Gál, P. Závodszky, I. Hajdú, 2019, Molecules.

Secondary structure dependent self-assembly of beta-peptides into nanosized fibrils and membranes.

I. Dékány, I. Mándity, F. Fülöp, 2006, Angewandte Chemie.

An overview of peptide and peptoid foldamers in medicinal chemistry

I. Mándity, F. Fülöp, 2015, Expert opinion on drug discovery.

Harnessing the Versatility of Continuous-Flow Processes: Selective and Efficient Reactions.

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2016, Chemical record.

A Domino Ring-Closure Followed by Retro-Diels–Alder Reaction for the Preparation of Pyrimido[2,1-a]isoindole Enantiomers

M. Haukka, I. Mándity, F. Fülöp, 2016 .

Design of peptidic foldamer helices: a stereochemical patterning approach.

I. Mándity, F. Fülöp, Gábor Olajos, 2009, Angewandte Chemie.

Foldameric β-H18/20P Mixed Helix Stabilized by Head-to-Tail Contacts: A Way to Higher-Order Structures

I. Mándity, F. Fülöp, T. Martinek, 2013 .

α,β‐ und α,α,β,β‐Peptidfoldamere basierend auf cis‐β‐Aminocyclopentancarbonsäure

I. Mándity, F. Fülöp, C. Cabrele, 2012 .

Unique α,β- and α,α,β,β-peptide foldamers based on cis-β-aminocyclopentanecarboxylic acid.

I. Mándity, F. Fülöp, C. Cabrele, 2012, Angewandte Chemie.

Rapid, simple, and efficient deprotection of benzyl/benzylidene protected carbohydrates by utilization of flow chemistry

I. Mándity, F. Fülöp, R. Leino, 2011 .

Continuous-flow azide–alkyne cycloadditions with an effective bimetallic catalyst and a simple scavenger system

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2014 .

Electrospray ionization–tandem mass spectrometric study of fused nitrogen‐containing ring systems

I. Mándity, K. Ludányi, Dóra Bogdán, 2022, Journal of mass spectrometry : JMS.

Flow-chemistry enabled efficient synthesis of β-peptides: backbone topology vs. helix formation.

T. Juhász, I. Mándity, S. Béni, 2019, Chemical communications.

ConjuPepDB: a database of peptide–drug conjugates

T. Beke-Somfai, Bilal Nizami, I. Mándity, 2020, Nucleic Acids Res..

Scope and limitation of propylene carbonate as a sustainable solvent in the Suzuki–Miyaura reaction

I. Mándity, K. Ludányi, Z. Varga, 2019, RSC advances.

Carbon dots from citric acid and its intermediates formed by thermal decomposition.

S. Marras, G. Granozzi, I. Mándity, 2019, Chemistry.

Statin‐boosted cellular uptake and endosomal escape of penetratin due to reduced membrane dipole potential

I. Mándity, P. Nagy, F. Zakany, 2020, British journal of pharmacology.

Highly functionalized cyclic β-amino acid moieties as promising scaffolds in peptide research and drug design

I. Mándity, F. Fülöp, L. Kiss, 2017, Amino Acids.

An efficient route for the synthesis of 2-arylthiazino[5,6-b]indole derivatives

I. Mándity, G. Bernáth, L. Fodor, 2007 .

An Efficient Route for the Synthesis of 2‐Arylthiazino[5,6‐b]indole Derivatives.

I. Mándity, G. Bernáth, L. Fodor, 2007 .

Heterogeneous Dipeptide-Catalyzed α-Amination of Aldehydes in a Continuous-Flow Reactor: Effect of Residence Time on Enantioselectivity

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2015 .

Strategic Application of Residence-Time Control in Continuous-Flow Reactors

Ferenc Fülöp, István M Mándity, Sándor B Ötvös, 2015, ChemistryOpen.

N-Acetylation of Amines in Continuous-Flow with Acetonitrile—No Need for Hazardous and Toxic Carboxylic Acid Derivatives

I. Mándity, F. Fülöp, György Orsy, 2020, Molecules.

Highly efficient 1,4-addition of aldehydes to nitroolefins: organocatalysis in continuous flow by solid-supported peptidic catalysts.

I. Mándity, F. Fülöp, Sándor B Otvös, 2012, ChemSusChem.

Effects of the alternating backbone configuration on the secondary structure and self-assembly of beta-peptides.

M. Hollósi, I. Mándity, F. Fülöp, 2006, Journal of the American Chemical Society.

Chain-length-dependent helical motifs and self-association of beta-peptides with constrained side chains.

I. Mándity, F. Fülöp, T. Martinek, 2005, Journal of the American Chemical Society.

Accelerated Synthesis of Protected Peptides in a Continuous‐Flow Fixed‐Bed Reactor

I. Mándity, F. Fülöp, Aliz Szloszár, 2017 .

Continuous-flow solid-phase peptide synthesis: a revolutionary reduction of the amino acid excess.

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2014, ChemSusChem.

Direct amide formation in a continuous-flow system mediated by carbon disulfide

I. Mándity, F. Fülöp, György Orsy, 2020, Catalysis Science & Technology.

Asymmetric aldol reaction in a continuous-flow reactor catalyzed by a highly reusable heterogeneous peptide

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2012 .

Highly Selective Continuous-Flow Synthesis of Potentially Bioactive Deuterated Chalcone Derivatives.

Y. Wu, F. Chang, I. Mándity, 2015, ChemPlusChem.

Continuous-Flow retro-Diels-Alder Reaction: A Process Window for Designing Heterocyclic Scaffolds

I. Mándity, F. Fülöp, Márta Palkó, 2018, European Journal of Organic Chemistry.

Stereocontrolled synthesis of five diastereomers of trimethyl 3-aminocyclopentane-1,2,4-tricarboxylates

I. Mándity, F. Fülöp, R. Sillanpää, 2013 .

Building β-peptide H10/12 foldamer helices with six-membered cyclic side-chains: fine-tuning of folding and self-assembly.

I. Mándity, F. Fülöp, T. Martinek, 2010, Organic letters.

Sculpting the beta-peptide foldamer H12 helix via a designed side-chain shape.

I. Mándity, F. Fülöp, T. Martinek, 2009, Chemical communications.

Exploiting aromatic interactions for β-peptide foldamer helix stabilization: a significant design element.

I. Mándity, F. Fülöp, L. Fülöp, 2014, Chemistry.

Membrane active Janus-oligomers of β3-peptides

V. Urlacher, J. Mihály, Gergely Kohut, 2020, Chemical science.

Homochirality of β‐Peptides: A Significant Biomimetic Property of Unnatural Systems

I. Mándity, F. Fülöp, G. Paragi, 2017, ChemistryOpen.

Alkyne-azide cycloadditions with copper powder in a high-pressure continuous-flow reactor: high-temperature conditions versus the role of additives.

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2013, Chemistry, an Asian journal.

Sustainable synthesis of N-methylated peptides in a continuous-flow fixed bed reactor

I. Mándity, F. Fülöp, Aliz Szloszár, 2018, Journal of Flow Chemistry.

VCD studies on cyclic peptides assembled from L‐α‐amino acids and a trans‐2‐aminocyclopentane‐ or trans‐2‐aminocyclohexane carboxylic acid

K. Gaus, Z. Majer, M. Hollósi, 2010, Journal of peptide science : an official publication of the European Peptide Society.

Physicochemical Profiling of Baicalin Along with the Development and Characterization of Cyclodextrin Inclusion Complexes

I. Antal, I. Mándity, B. Noszál, 2019, AAPS PharmSciTech.

An ω-3, but Not an ω-6 Polyunsaturated Fatty Acid Decreases Membrane Dipole Potential and Stimulates Endo-Lysosomal Escape of Penetratin

I. Mándity, P. Fülöp, P. Nagy, 2021, Frontiers in Cell and Developmental Biology.

Statin-boosted cellular uptake of penetratin due to reduced membrane dipole potential

I. Mándity, P. Nagy, F. Zakany, 2020, bioRxiv.

A comparative assessment of two kynurenic acid analogs in the formalin model of trigeminal activation: a behavioral, immunohistochemical and pharmacokinetic study

G. Veres, Á. Párdutz, L. Vécsei, 2016, Journal of Neural Transmission.

Continuous-flow retro-Diels–Alder reaction: an efficient method for the preparation of pyrimidinone derivatives

I. Mándity, F. Fülöp, Márta Palkó, 2018, Beilstein journal of organic chemistry.

Species-specific acid-base characterization of carnosine and homocarnosine using nuclear magnetic resonance

A. Mirzahosseini, Nikolett Varró, I. Mándity, 2022, Chemical Physics Letters.

Deciphering metal ion preference and primary coordination sphere robustness of a designed zinc finger with high‐resolution mass spectrometry

J. Jänis, J. Valjakka, I. Mándity, 2017, Protein science : a publication of the Protein Society.

Kynurenic acid and its analogue can alter the opioid receptor G-protein signaling after acute treatment via NMDA receptor in rat cortex and striatum

G. Veres, L. Vécsei, I. Mándity, 2017, Journal of the Neurological Sciences.

Highly selective deuteration of pharmaceutically relevant nitrogen-containing heterocycles: a flow chemistry approach

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2011, Molecular Diversity.

Physico-chemical characterization and in vitro/in vivo evaluation of loratadine:dimethyl-β-cyclodextrin inclusion complexes.

I. Mándity, P. Sipos, P. Szabó-Révész, 2011, Journal of pharmaceutical and biomedical analysis.

Safe and Efficient Continuous-Flow Synthesis and Batchwise Hydrolysis of Ethyl 5-Acetyl-1 H -pyrazole-3-carboxylate: A Key Synthon of Darolutamide

G. Keserű, I. Mándity, Balázs Volk, 2022, Synthesis.

An overview of peptide and peptoid foldamers in medicinal chemistry.

I. Mándity, F. Fülöp, 2015, Expert opinion on drug discovery.

Efficient continuous-flow synthesis of novel 1,2,3-triazole-substituted β-aminocyclohexanecarboxylic acid derivatives with gram-scale production

I. Mándity, Sándor B. Ötvös, F. Fülöp, 2013, Beilstein journal of organic chemistry.

Highly functionalized cyclic β-amino acid moieties as promising scaffolds in peptide research and drug design

I. Mándity, F. Fülöp, L. Kiss, 2017, Amino Acids.

Synthesis of conformationally constrained, orthogonally protected 3-azabicyclo[3.2.1]octane β-amino esters

I. Mándity, L. Kiss, E. Forró, 2010 .

Effect of the Lipid Landscape on the Efficacy of Cell-Penetrating Peptides

I. Mándity, P. Nagy, Z. Varga, 2023, Cells.

Continuous-Flow Synthesis of Thioureas, Enabled by Aqueous Polysulfide Solution

G. Keserű, P. Ábrányi‐Balogh, I. Mándity, 2021, Molecules.

Continuous-flow catalytic deuterodehalogenation carried out in propylene carbonate

I. Mándity, F. Fülöp, György Orsy, 2019, Green Chemistry.

Foldameric probes for membrane interactions by induced β-sheet folding.

I. Mándity, T. Martinek, Z. Hegedüs, 2016, Chemical communications.

A covalent strategy to target intrinsically disordered proteins: Discovery of novel tau aggregation inhibitors.

L. Wittner, B. Davis, G. Keserű, 2022, European journal of medicinal chemistry.

Evaluation of the therapeutic efficacy of 213Bi-labelled DOTA-conjugated alpha-melanocyte stimulating hormone peptide analogues in melanocortin-1 receptor positive preclinical melanoma model.

G. Nagy, I. Mándity, F. Bruchertseifer, 2023, International journal of pharmaceutics.

Stimuli-Responsive Membrane Anchor Peptide Nanofoils for Tunable Membrane Association and Lipid Bilayer Fusion

J. Andréasson, J. Mihály, T. Beke-Somfai, 2022, ACS applied materials & interfaces.

In Vivo evaluation of newly synthesized 213Bi-conjugated alpha-melanocyte stimulating hormone (α-MSH) peptide analogues in melanocortin-1 receptor (MC1-R) positive experimental melanoma model.

G. Nagy, I. Mándity, F. Bruchertseifer, 2023, Journal of pharmaceutical and biomedical analysis.