C. Cavallaro

发表

Molecular Diversity in Lead Discovery: From Quantity to Quality

D. Schnur, C. Cavallaro, A. Tebben, 2005 .

Ligand and Target Discovery by Fragment-Based Screening in Human Cells

Stephen R. Johnson, B. Cravatt, B. Correia, 2017, Cell.

A statistical-based approach to assessing the fidelity of combinatorial libraries encoded with electrophoric molecular tags. Development and application of tag decode-assisted single bead LC/MS analysis.

W. Egan, J. Reader, M. Orlowski, 2000, Journal of combinatorial chemistry.

Microscale purification in support of high-throughput medicinal chemistry.

C. Cavallaro, E. Priestley, Andrew F Donnell, 2021, Chemical communications.

Catalytic dechlorination of polychlorinated biphenyls.

C. Cavallaro, J. Schwartz, Y. Liu, 1995, Environmental science & technology.

The discovery of BMS-457, a potent and selective CCR1 antagonist.

W. Guo, C. Cavallaro, A. Tebben, 2013, Bioorganic & medicinal chemistry letters.

Increasing saturation: development of broadly applicable photocatalytic Csp2–Csp3 cross-couplings of alkyl trifluoroborates and (hetero)aryl bromides for array synthesis

C. Cavallaro, E. Simmons, Melda Sezen-Edmonds, 2021, Reaction Chemistry & Engineering.

Discovery of the CCR1 antagonist, BMS-817399, for the treatment of rheumatoid arthritis.

J. Barrish, C. Cavallaro, A. Tebben, 2014, Journal of medicinal chemistry.

Ni/Photoredox-Catalyzed C(sp2)-C(sp3) Cross-Coupling of Alkyl Pinacolboronates and (Hetero)Aryl Bromides.

C. Cavallaro, E. Simmons, Melda Sezen-Edmonds, 2022, Organic letters.

Discovery and lead optimization of a novel series of CC chemokine receptor 1 (CCR1)-selective piperidine antagonists via parallel synthesis.

J. Chen, S. Mandlekar, C. Cavallaro, 2012, Journal of medicinal chemistry.

Synthesis and structure-activity relationships of novel indazolyl glucocorticoid receptor partial agonists.

A. Doweyko, J. Barrish, S. Nadler, 2013, Bioorganic & medicinal chemistry letters.

4.14 – Library Design: Ligand and Structure-Based Principles for Parallel and Combinatorial Libraries

Dora M. Schnur, Andrew J. Tebben, Cullen L. Cavallaro, 2007 .

Preparation of 2,7-diaminosubstituted-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonitriles by solid-phase synthesis.

F. Chi, C. Cavallaro, A. Purandare, 2008, Journal of combinatorial chemistry.

Allylindium and allylboronic acid pinacolate: Mild reagents for the allylation of resin-bound aldehydes. Application to the solid-phase synthesis of hydroxypropylamines

C. Cavallaro, R. Dolle, T. Herpin, 1999 .

Identification of potent inhibitors of Plasmodium falciparum plasmepsin II from an encoded statine combinatorial library.

I. Gluzman, D. Goldberg, M. Orlowski, 1998, Bioorganic & medicinal chemistry letters.

RAPID PREPARATION OF VARIOUSLY PROTECTED GLYCALS USING TITANIUM(III)

C. Cavallaro, J. Schwartz, R. Spencer, 1999 .

Reduction of Glycosyl Bromides to Anhydroalditols by Titanocene Borohydride.

C. Cavallaro, J. Schwartz, 1996, The Journal of organic chemistry.

A Rapid Synthesis of Pyranoid Glycals from Glycosyl Bromides

C. Cavallaro, J. Schwartz, 1995 .

A Rapid Synthesis of Pyranoid Glycals from Glycosyl Bromides.

C. Cavallaro, J. Schwartz, 1996 .

Synthesis of Differentially Protected Azatryptophan Analogs via Pd2(dba)3/XPhos Catalyzed Negishi Coupling of N-Ts Azaindole Halides with Zinc Derivative from Fmoc-protected tert-Butyl (R)-2-amino-3-iodopropanoate.

A. Mathur, C. Cavallaro, A. Roy, 2020, The Journal of organic chemistry.

Developing Adnectins that target SRC co-activator binding to PXR: a structural approach toward understanding promiscuity of PXR.

Eric T Baldwin, Martin C. Wright, Andrew J Tebben, 2015, Journal of molecular biology.

Substituted Diaryl Ether Compounds as Retinoic Acid-Related Orphan Receptor-γt (RORγt) Agonists.

Zhuyin Li, C. Weigelt, B. Fink, 2021, Bioorganic & medicinal chemistry letters.

Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists.

Zhuyin Li, C. Weigelt, B. Fink, 2020, Bioorganic & medicinal chemistry letters.

Methods for combinatorial and parallel library design.

Dora M Schnur, Brett R Beno, Andrew J Tebben, 2011, Methods in molecular biology.

Discovery and SAR of aryl hydroxy pyrimidinones as potent small molecule agonists of the GPCR APJ.

Michael C. Myers, A. Nayeem, P. Gargalovic, 2020, Bioorganic & medicinal chemistry letters.

Application of lean manufacturing concepts to drug discovery: rapid analogue library synthesis.

Harold N Weller, John G Houston, David S. Nirschl, 2006, Journal of combinatorial chemistry.

Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists.

C. Weigelt, B. Fink, T. Huynh, 2020, Bioorganic & medicinal chemistry letters.