Corinne Fruit

发表

Enantioselective catalytic aziridinations and asymmetric nitrene insertions into CH bonds.

P. Müller, Corinne Fruit, 2003, Chemical reviews.

New family of peptidomimetics based on the imidazole motif.

Corinne Fruit, S. Petit, L. Bischoff, 2010, Organic letters.

Microwave-Assisted Sequential One-Pot Synthesis of 8-Substituted Pyrazolo[1,5-a][1,3,5]triazines

Corinne Fruit, T. Besson, Jonathan Elie, 2021, Molecules.

Synthesis of polyfunctionalized benzo[d]thiazoles as novel anthranilic acid derivatives

Corinne Fruit, T. Besson, Damien Hédou, 2015 .

Microwave-Assisted Synthesis of Potential Bioactive Benzo-, Pyrido- or Pyrazino-thieno[3,2-d]pyrimidin-4-amine Analogs of MPC-6827

C. Corbière, Corinne Fruit, T. Besson, 2020, Pharmaceuticals.

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

L. Meijer, P. Bonnet, Corinne Fruit, 2018, Molecules.

Diaryliodoniums Salts as Coupling Partners for Transition-Metal Catalyzed C- and N-Arylation of Heteroarenes

Corinne Fruit, T. Besson, Alexandra Pacheco-Benichou, 2020, Catalysts.

Three catalysts for activating carbon-hydrogen bonds

Corinne Fruit, 2016, Science.

One-pot synthesis of 2,3-dihydro-pyrrolopyridinones using in situ generated formimines.

Corinne Fruit, F. Marsais, L. Bischoff, 2006, Organic letters.

Relieving DYRK1A repression of MKL1 confers an adult-like phenotype to human infantile megakaryocytes

Ashton T. Brock, P. Gadue, S. Morris, 2022, The Journal of clinical investigation.

Design of silicon-based misonidazole analogues and (18)F-radiolabelling.

Corinne Fruit, P. Vera, F. Marsais, 2009, Nuclear medicine and biology.

Metalation of Pyrazine and Quinoxaline

Corinne Fruit, N. Plé, 2012 .

Pd-catalyzed decarboxylative cross-coupling of 2-carboxyazine N-oxides with various (hetero)aryl halides.

Corinne Fruit, C. Hoarau, C. Schneider, 2014, Chemistry.

Regioselective decarboxylative cross-coupling of carboxy isoquinoline N-oxides.

Corinne Fruit, C. Hoarau, C. Schneider, 2015, The Journal of organic chemistry.

Cu/Pd-Catalyzed C-2–H Arylation of Quinazolin-4(3H)-ones with (Hetero)aryl Halides

Corinne Fruit, Sylvain Laclef, T. Besson, 2015 .

Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts

Corinne Fruit, T. Besson, 2021, Pharmaceuticals.

Ligand-free Pd-catalyzed and copper-assisted C-H arylation of quinazolin-4-ones with aryl iodides under microwave heating.

Corinne Fruit, Sylvain Laclef, T. Besson, 2015, Organic letters.

Aminomethylation of lithiated nicotinamide: access to new pyridolactams

Corinne Fruit, F. Marsais, Rabah Azzouz, 2008 .

Efficient diastereoselective intermolecular rhodium-catalyzed C-H amination.

P. Müller, Corinne Fruit, P. Dauban, 2006, Angewandte Chemie.

Anionic, in situ generation of formaldehyde: a very useful and versatile tool in synthesis.

Corinne Fruit, F. Marsais, L. Bischoff, 2007, Organic letters.

Synthesis of Benzo-Fused 11H-Pyrido[2,1-b]quinazolin-11-ones by a Buchwald–Hartwig Coupling/Pyridine Dearomatization Sequence in Eucalyptol

Corinne Fruit, T. Besson, S. Berteina‐Raboin, 2020 .

Diastereoselective rhodium-catalyzed nitrene transfer starting from chiral sulfonimidamide-derived iminoiodanes

G. Bernardinelli, P. Müller, Corinne Fruit, 2005 .

Synthesis of Bioactive 2-(Arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff Reaction or Cu- Catalyzed Intramolecular C-S Bond Formation

L. Meijer, N. Loaëc, Corinne Fruit, 2016, Molecules.

Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases

L. Meijer, N. Loaëc, Corinne Fruit, 2016, Molecules.

Recent Developments in Microwave-Assisted Metal-Catalyzed C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications

Corinne Fruit, T. Besson, 2016 .

Orthogonal Palladium‐Catalyzed Direct C−H Bond Arylation of Heteroaromatics with Aryl Halides

Corinne Fruit, C. Hoarau, C. Schneider, 2016 .

Copper-Catalyzed C–H Arylation of Fused-Pyrimidinone Derivatives Using Diaryliodonium Salts

Corinne Fruit, T. Besson, I. Kostakis, 2020, Catalysts.

Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides.

Corinne Fruit, T. Besson, Marine Harari, 2016, Organic letters.

Cu/Pd‐Catalyzed C‐2—H Arylation of Quinazolin‐4(3H)‐ones with (Hetero)aryl Halides.

Corinne Fruit, Sylvain Laclef, T. Besson, 2016 .

Conception of DYRK1A kinase inhibitors via metal-catalyzed C–H arylation, inspired by fragment-growing studies

L. Meijer, P. Bonnet, Corinne Fruit, 2018, Proceedings of 4th International Electronic Conference on Medicinal Chemistry.

Synthesis of 2-Cyanobenzothiazoles via Pd-Catalyzed/Cu-Assisted C-H Functionalization/Intramolecular C-S Bond Formation from N-Arylcyanothioformamides

Corinne Fruit, T. Besson, Alexandra Pacheco-Benichou, 2022, Molecules.

Syntheses and metalation of pyridazinecarboxamides and thiocarboxamides. Diazines. Part 32

Corinne Fruit, A. Turck, N. Plé, 2002 .

An efficient approach to new dihydroxyquinolizidines

Corinne Fruit, T. Tite, F. Marsais, 2010 .

A concise synthesis of lentiginosine derivatives using a pyridinium formation via the Mitsunobu reaction.

Corinne Fruit, F. Marsais, Rabah Azzouz, 2008, The Journal of organic chemistry.

Syntheses of N-diazinyl thiocarboxamides and of thiazolodiazines. Metalation studies. Diazines XXXIII

Corinne Fruit, A. Turck, N. Plé, 2002 .

Metalation of Pyrazinethiocarboxamides. Metalation of Diazines XXVI

Corinne Fruit, A. Turck, N. Plé, 1999 .

Intramolecular Asymmetric Amidations of Sulfonamides and Sulfamates Catalyzed by Chiral Dirhodium(II) Complexes

P. Müller, Corinne Fruit, 2004 .

Aminoacid-derived mercaptoimidazoles.

Corinne Fruit, F. Marsais, S. Petit, 2009, Organic & biomolecular chemistry.

Asymmetric transfer of nitrenes catalyzed by chiral dirhodium(II) using aromatic sulfamate esters

P. Müller, Corinne Fruit, 2004 .

Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors: a survey of recent patent literature

Y. Hérault, L. Meijer, Thu Lan Nguyen, 2017, Expert opinion on therapeutic patents.

DYRK1A regulates B cell acute lymphoblastic leukemia through phosphorylation of FOXO1 and STAT3.

Y. Goo, S. Izraeli, Q. Wen, 2021, The Journal of clinical investigation.

Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4-f]quinazolin-9(8H)-one, a Promising Inhibitor of DYRK1A

L. Meijer, Corinne Fruit, J. Crispino, 2019, Pharmaceuticals.

A new route to Septorin via controlled metalations of pyrazines. Diazines XXX

Corinne Fruit, A. Turck, N. Plé, 2001 .

Regioselective opening of N-Cbz glutamic and aspartic anhydrides with carbon nucleophiles

Corinne Fruit, Corinne Fruit, F. Marsais, 2006 .

Enantioselective Catalytic Aziridinations and Asymmetric Nitrene Insertions into CH Bonds

P. Mueller, Corinne Fruit, 2003 .

On the racemisation of aspartic anhydride during its preparation

Corinne Fruit, F. Buron, F. Marsais, 2007 .

An efficient protocol for the preparation of pyridinium and imidazolium salts based on the Mitsunobu reaction

Corinne Fruit, F. Marsais, S. Petit, 2008 .