A. Di Giorgio

发表

Recent progresses in aminoglycoside conjugation for RNA targeting: antimicrobials and beyond.

M. Duca, Klára Aradi, A. Di Giorgio, 2020, Chemistry.

Modulation of oncogenic miRNA biogenesis using functionalized polyamines

N. Tourasse, M. Duca, C. Staedel, 2018, Scientific Reports.

Inhibition of Patched Drug Efflux Increases Vemurafenib Effectiveness against Resistant BrafV600E Melanoma

D. Douguet, C. Bertolotto, V. Biou, 2020, Cancers.

Fluorescent labeling of human mesenchymal stem cells by thiophene fluorophores conjugated to a lipophilic carrier.

G. Barbarella, M. Duca, A. Di Giorgio, 2010, Chemical communications.

Exploring the impact of the side-chain length on peptide/RNA binding events.

M. Andreola, A. Di Giorgio, S. Azoulay, 2017, Physical chemistry chemical physics : PCCP.

Short peptide nucleic acids (PNA) inhibit hepatitis C virus internal ribosome entry site (IRES) dependent translation in vitro.

F. Zoulim, D. Durantel, A. Di Giorgio, 2008, Antiviral research.

The aminoglycoside streptomycin triggers ferroptosis in tumor initiating cells

C. Planque, M. Duca, A. Di Giorgio, 2022, bioRxiv.

Exploring Heterocycle-Spermine Conjugates as Modulators of Oncogenic microRNAs Biogenesis

M. Duca, A. Di Giorgio, P. Uriac, 2018, ACS Omega.

Polyamide amino acids: a new class of RNA ligands.

A. Di Giorgio, S. Azoulay, N. Patino, 2009, Chemical communications.

Unveiling RNA‐Binding Properties of Verapamil and Preparation of New Derivatives as Inhibitors of HIV‐1 Tat‐TAR Interaction

M. Duca, A. Di Giorgio, S. Azoulay, 2020 .

Ribosome-targeting antibiotics as inhibitors of oncogenic microRNAs biogenesis: Old scaffolds for new perspectives in RNA targeting.

M. Duca, A. Di Giorgio, T. Tran, 2015, Bioorganic & medicinal chemistry.

A cyclic PNA-based compound targeting domain IV of HCV IRES RNA inhibits in vitro IRES-dependent translation.

F. Zoulim, R. Terreux, A. Di Giorgio, 2005, Bioorganic & medicinal chemistry.

Solid-phase synthesis and thermal denaturation study of cyclic PNAs targeting the HIV-1 TAR RNA loop.

A. Di Giorgio, M. Mehiri, G. Upert, 2007, Bioorganic & medicinal chemistry letters.

Thermodynamic studies of a series of homologous HIV-1 TAR RNA ligands reveal that loose binders are stronger Tat competitors than tight ones

A. Di Giorgio, P. Clayette, S. Azoulay, 2013, Nucleic acids research.

Differentiation of Cancer Stem Cells by Using Synthetic Small Molecules: Toward New Therapeutic Strategies against Therapy Resistance

M. Duca, A. Di Giorgio, S. Azoulay, 2020, ChemMedChem.

Small-molecule approaches toward the targeting of oncogenic miRNAs: roadmap for the discovery of RNA modulators.

M. Duca, A. Di Giorgio, T. Tran, 2016, Future medicinal chemistry.

Synthetic small-molecule RNA ligands: future prospects as therapeutic agents.

M. Duca, A. Di Giorgio, A. D. Giorgio, 2019, MedChemComm.

Polyamide amino acids trimers as TAR RNA ligands and anti-HIV agents.

A. Di Giorgio, P. Clayette, S. Azoulay, 2010, Bioorganic & medicinal chemistry.

AZT and AZT-monophosphate Prodrugs Incorporating HIV-protease Substrate Fragment: Synthesis and Evaluation as Specific Drug Delivery Systems

A. Di Giorgio, M. Mehiri, A. Aubertin, 2006, Antiviral chemistry & chemotherapy.

Involvement of Phosphodiesterase 2A Activity in the Pathophysiology of Fragile X Syndrome.

B. Bardoni, V. Trezza, T. Maurin, 2018, Cerebral cortex.

Building of neomycin-nucleobase-amino acid conjugates for the inhibition of oncogenic miRNAs biogenesis.

M. Duca, C. Staedel, A. Di Giorgio, 2018, Organic & biomolecular chemistry.

Oncogenic MicroRNAs Biogenesis as a Drug Target: Structure-Activity Relationship Studies on New Aminoglycoside Conjugates.

M. Duca, C. Staedel, A. Di Giorgio, 2016, Chemistry.

Inhibition of HIV Replication by Cyclic and Hairpin PNAs Targeting the HIV-1 TAR RNA Loop

A. Di Giorgio, G. Upert, Alok K Upadhyay, 2012, Journal of nucleic acids.

Design and Implementation of Synthetic RNA Binders for the Inhibition of miR-21 Biogenesis.

M. Duca, A. Di Giorgio, D. Vo, 2021, ACS medicinal chemistry letters.

Modulation of oncogenic miRNA biogenesis using functionalized polyamines

N. Tourasse, M. Duca, C. Staedel, 2018, Scientific Reports.

Synthesis of Bleomycin-Inspired RNA Ligands Targeting the Biogenesis of Oncogenic miRNAs.

M. Verreault, C. Di Giorgio, M. Duca, 2023, Journal of Medicinal Chemistry.

A "ready-to-use" fluorescent-labelled-cysteine-TBTP (4-thiobutyltriphenylphosphonium) synthon to investigate the delivery of non-permeable PNA (peptide nucleic acids)-based compounds to cells.

A. Di Giorgio, A. Doglio, M. Mehiri, 2007, Bioorganic chemistry.

Synthesis and cellular uptake of a fluorescently labeled cyclic PNA-based compound.

A. Di Giorgio, A. Doglio, R. Condom, 2004, Bioorganic & medicinal chemistry letters.