P. Uriac

发表

Modulation of oncogenic miRNA biogenesis using functionalized polyamines

N. Tourasse, M. Duca, C. Staedel, 2018, Scientific Reports.

Induction of Intracellular Calcium Concentration by Environmental Benzo(a)pyrene Involves a β2-Adrenergic Receptor/Adenylyl Cyclase/Epac-1/Inositol 1,4,5-Trisphosphate Pathway in Endothelial Cells*

O. Fardel, D. Lagadic-Gossmann, P. Uriac, 2011, The Journal of Biological Chemistry.

Stictic acid derivatives from the lichen Usnea articulata and their antioxidant activities.

J. Elix, P. Uriac, J. Boustie, 2007, Journal of natural products.

Heterocyclisations de sels d'iminium provenant de quelques β-amino-β-lactames et de leurs derivés GEM-difonctionnels

P. Uriac, J. Huet, L. Toupet, 1992 .

Effect of polyamine homologation on the transport and biological properties of heterocyclic amidines.

J. Delcros, P. Uriac, V. Eifler-Lima, 2006, Journal of medicinal chemistry.

Polyamine sulfonamides with NMDA antagonist properties are potent calmodulin antagonists and cytotoxic agents.

J. Delcros, J. Moulinoux, P. Uriac, 1998, The international journal of biochemistry & cell biology.

Recognition of enantiomers with chiral molecular tweezers derived from (+)- or (―)-usnic acid

P. Uriac, P. D. Weghe, S. Tomasi, 2010 .

Novel chiral molecular tweezer from (+)-usnic acid.

P. Uriac, L. Toupet, A. Bondon, 2009, Organic letters.

Irreversible inhibitors of the proline racemase unveil innovative mechanism of action as antibacterial agents against Clostridioides difficile

A. Blondel, P. Minoprio, P. Uriac, 2021, Chemical biology & drug design.

Synthesis of a laterally branched polyamine from alpha-methylene-gamma-butyrolactone.

P. Uriac, J. Renault, Mickaël Jean, 2005, Organic letters.

Reactivity of 5-alkynyl-3,4-dihydro-2H-pyrroles with Au(III): Route to vinylgold(III) complexes, aurocycles by cyclisation of these complexes and ML complexes

P. Uriac, T. Roisnel, A. Bondon, 2019, Journal of Organometallic Chemistry.

Electrophilic carbon transfer in gold catalysis: synthesis of substituted chromones

P. Uriac, J. Renault, N. Gouault, 2011 .

Cycloisomerization of γ- and δ-acetylenic acids catalyzed by gold(I) chloride

P. Uriac, P. D. Weghe, L. Toupet, 2007 .

Methylene furanone derivatives and the use thereof as a photoprotective or antioxidant agent

P. Uriac, S. Poigny, Y. Brunel, 2008 .

Separation of a mixture of paraconic acids from Cetraria islandica (L.) Ach. employing a fluorous tag—catch and release strategy

P. Uriac, J. Boustie, David Horhant, 2007 .

Synthesis of New Quinoxaline Derivatives by Reductive Cyclization of Various 1-(2-Nitrophenyl)-2-cyanoamines

P. Uriac, J. Hurvois, T. Renaud, 2001 .

Synthesis of substituted pyrrolin-4-ones from amino acids in mild conditions via a gold-catalyzed approach.

P. Uriac, N. Gouault, M. Le Roch, 2009, The Journal of organic chemistry.

Synthesis of 1-arylidene-2,3-dihydro-1H-inden-2-ols through a tandem carbopalladation/Suzuki-Miyaura sequence

P. Uriac, P. D. Weghe, Estelle Marchal, 2008 .

Exploring Heterocycle-Spermine Conjugates as Modulators of Oncogenic microRNAs Biogenesis

M. Duca, A. Di Giorgio, P. Uriac, 2018, ACS Omega.

Targeting the polyamine transport system with benzazepine- and azepine-polyamine conjugates.

J. Delcros, P. Uriac, S. Tomasi, 2010, Journal of medicinal chemistry.

Synthesis of 3-substituted indolizidines from amino-ynones derivatives

P. Uriac, T. Roisnel, J. Renault, 2016 .

From Aspartic Acid to Dihydropyridone-2-carboxylates: Access to Enantiopure 6-Substituted 4-Oxo- and 4-Hydroxypipecolic Acid Derivatives

P. Uriac, L. Toupet, J. Renault, 2013 .

Gold-mediated synthesis and functionalization of chiral halopyridones.

P. Uriac, L. Toupet, S. Tomasi, 2013, The Journal of organic chemistry.

Solid phase organic synthesis of polyamine derivatives and initial biological evaluation of their antitumoral activity.

J. Delcros, P. Uriac, B. Carboni, 1998, Bioorganic & medicinal chemistry letters.

Oxidation of 2,3- and 2,5-dihydro-1H-1-benzazepines by hydride transfer to an iminium ion: Synthesis of 3H-1-benzazepines

P. Uriac, L. Toupet, S. Sinbandhit, 1996 .

Reactivity of N‐Boc‐Protected Amino‐Ynones in the Presence of Zinc Chloride: Formation of Acetylenic Cyclic Imines and Their Palladium Complexes

P. Uriac, T. Roisnel, P. Jéhan, 2015 .

Unexpected formation of aryl ketones by palladium-catalyzed coupling of aryl bromides with vinylic acetates.

P. Uriac, M. Capet, P. van de Weghe, 2007, Organic letters.

Relationship between cytotoxicity and DNA-binding affinity of amidine derivatives of tetrahydroquino[4,3-b][1]benzazepines and tetrahydrobenzo[k]naphthyridines

P. Uriac, V. Eifler-Lima, J. Huet, 1995 .

Enantiospecific synthesis of pyridinones as versatile intermediates toward asymmetric piperidines.

P. Uriac, N. Gouault, M. Le Roch, 2011, Organic letters.

Synthesis of substituted pyrrolin-4-ones from amino acids in mild conditions via a gold-catalyzed approach.

P. Uriac, N. Gouault, M. Le Roch, 2009, The Journal of organic chemistry.

Methanesulfonic Acid Mediated Cyclization and Meyer–Schuster Rearrangement of γ‐Amino‐ynones: Access to Enantiopure Pyrrolidine Exocyclic Vinylogous Amides

P. Uriac, T. Roisnel, J. Renault, 2014 .

ELECTROSYNTHESIS OF ALPHA -AMINONITRILES : ANODIC CYANATION OF N-SUBSTITUTED TETRAHYDROQUINOLINES AND N-PHENYLPIPERIDINES

E. L. Gall, P. Uriac, L. Toupet, 1997 .

Synthesis of New Quinoxaline Derivatives by Reductive Cyclization of Various 1-(2-Nitrophenyl)-2-cyanoamines.

P. Uriac, J. Hurvois, T. Renaud, 2002 .

Molecular Tweezers: Synthesis and Formation of Host–Guest Complexes

P. Uriac, P. D. Weghe, N. Levoin, 2010 .

Study of the self-association of molecular tweezers bearing two different arms: influence of the stereoelectronic effects of the arm substituents

P. Uriac, A. Bondon, S. Ferron, 2019, Journal of Inclusion Phenomena and Macrocyclic Chemistry.

Dissymmetric Molecular Tweezers in Host–Guest Complexes: Internal or External Complexation?

P. Uriac, D. Jacquemin, L. Toupet, 2015 .

Molecular Tweezers in Host–Guest Complexes: A Computational Study through a DFT-D Approach

P. Uriac, D. Jacquemin, P. D. Weghe, 2012 .

1-Benzazepine derivatives acting as ATP-dependent potassium-channels antagonists

P. Uriac, J. Huet, C. Advenier, 1995 .

Toxicity and osmoprotective activities of analogues of glycine betaine obtained by solid phase organic synthesis towards Sinorhizobium meliloti.

P. Uriac, T. Bernard, B. Carboni, 1999, Bioorganic & medicinal chemistry letters.

Preparation and characterization of copper(II) and nickel(II) complexes of a new chiral salen ligand derived from (+)-usnic acid.

P. Uriac, L. Toupet, S. Tomasi, 2008, Dalton transactions.

Synthesis and cytotoxic activities of usnic acid derivatives.

J. Delcros, P. Uriac, J. Boustie, 2008, Bioorganic & medicinal chemistry.

Anodic Cyanation of N‐Substituted 1‐Benzazepines: Synthesis of the Corresponding α‐Aminonitriles

E. L. Gall, P. Uriac, L. Toupet, 1997 .

1-Benzazepine Derivatives Acting as ATP-Dependent Potassium-Channels Antagonists.

P. Uriac, J. Huet, C. Advenier, 1995 .

Effect of spermine conjugation on the cytotoxicity and cellular transport of acridine.

J. Delcros, I. S. Blagbrough, P. Uriac, 2002, Journal of medicinal chemistry.

13C NMR spectra of 2,3‐dihydro‐1H‐benzo[b]azepines: Differentiation of diastereomers

P. Uriac, J. Huet, 1983 .

Parallel supported synthesis of polyamine-imidazole conjugates.

P. Uriac, S. Picard, J. Renault, 2004, Organic Letters.

Designed mono- and di-covalent inhibitors trap modeled functional motions for Trypanosoma cruzi proline racemase in crystallography

F. Saul, A. Blondel, P. Minoprio, 2018, PLoS neglected tropical diseases.

Combined Approaches for Drug Design Points the Way to Novel Proline Racemase Inhibitor Candidates to Fight Chagas’ Disease

A. Blondel, P. Minoprio, P. Uriac, 2013, PloS one.

Solid-phase combinatorial synthesis of polyamine derivatives using aminoalcohol building blocks

P. Uriac, J. Renault, M. Lebranchu, 2001 .

N-alkylation of N1-mesitylenesulphonylputrescine with N-(4-bromobutyl)phthalimide: A Parallel Approach Using Multipin Solid-phase Synthesis

P. Uriac, S. Tomasi, J. Renault, 2000 .

Antibacterial activity of glycine betaine analogues: involvement of osmoporters.

M. Jebbar, P. Uriac, T. Bernard, 2004, Bioorganic & medicinal chemistry letters.

Fluorous scavenger for parallel preparation of tertiary sulfonamides leading to secondary amines

P. Uriac, Emmanuel Baslé, J. Renault, 2007 .

Rearrangement of 2,5-dihydro-1H-benz[b]azepines by alkoxides

P. Uriac, J. Huet, J. Bonnic, 1984 .

Synthesis and evaluation of amides surrogates of dopamine D3 receptor ligands.

J. Schwartz, P. Uriac, N. Levoin, 2010, Bioorganic & medicinal chemistry letters.

A solid phase parallel synthesis of diverse amides as dopamine D3 receptor ligands

H. Stark, P. Uriac, N. Levoin, 2008 .

Solid phase synthesis of sulphonamides: novel ligands of 5‐HT6 receptors

S. Rault, F. Dauphin, P. Uriac, 2001, The Journal of pharmacy and pharmacology.

A chemotaxonomic study of the Xanthoparmelia pulla group in Algeria

P. Uriac, J. Boustie, P. Jéhan, 2019, Herzogia.

A novel solid-phase reductive alkylation route to acridine and dansyl polyamine conjugates

I. S. Blagbrough, P. Uriac, S. Tomasi, 1999 .

Pharmacomodulation of a Sulfamide 5-HT6 Receptor Ligand

S. Rault, F. Dauphin, P. Uriac, 2004, Journal of enzyme inhibition and medicinal chemistry.

Intramolecular transesterification of depsides yields fluorescent 1H-isochromen-1-ones: Application as a chemical probe for lichen determination.

P. Uriac, P. Jéhan, X. Guillory, 2022, Phytochemistry.

1H NMR and computational studies of the conformations in solution of one host/guest complex formed with an usnic acid tweezer and 2,4,7-trinitro-9-fluorenone (TNF)

P. Uriac, D. Jacquemin, E. Hitti, 2016 .

A DFT-D evaluation of the complexation of a molecular tweezer with small aromatic molecules

Denis Jacquemin, Jérôme Graton, P. Uriac, 2012 .

Ring expansion of some 4-aminoazetidin-2-ones into 4-amino-5-iminopyrrolidin-2-ones

P. Uriac, J. Huet, L. Toupet, 1993 .

Modulation of oncogenic miRNA biogenesis using functionalized polyamines

N. Tourasse, M. Duca, C. Staedel, 2018, Scientific Reports.

Solid-phase synthesis of polyfunctionalized natural products: application to usnic acid, a bioactive lichen compound.

C. Lainé, P. Uriac, S. Picard, 2006, Journal of combinatorial chemistry.

Prodrugs as new therapies against Chagas disease: In vivo synergy between Trypanosoma cruzi proline racemase inhibitors and benznidazole: TcPRAC inhibitor prodrugs against Chagas disease.

A. Blondel, P. Minoprio, P. Uriac, 2021, Journal of Global Antimicrobial Resistance.