S. Akai

发表

In vivo distribution of liposome-encapsulated hemoglobin determined by positron emission tomography.

N. Harada, H. Tsukada, D. Fukumoto, 2009, Artificial organs.

Novel amphiphilic probes for [18F]-radiolabeling preformed liposomes and determination of liposomal trafficking by positron emission tomography.

N. Harada, H. Tsukada, N. Oku, 2007, Journal of medicinal chemistry.

Could London Dispersion Force Control Regioselective (2 + 2) Cyclodimerizations of Benzynes? YES: Application to the Synthesis of Helical Biphenylenes.

Tomonari Murakami, Y. Shigeta, H. Tokiwa, 2021, Journal of the American Chemical Society.

Dynamic Kinetic Resolution for Asymmetric Synthesis

S. Akai, Gamal A. I. Moustafa, Gamal A I Moustafa, 2019, Kinetic Control in Synthesis and Self-Assembly.

Hydrolase-Catalyzed Dynamic Kinetic Resolution of Racemic Alcohols

S. Akai, 2017 .

Dynamic Kinetic Resolution of Racemic Allylic Alcohols via Hydrolase–Metal Combo Catalysis: An Effective Method for the Synthesis of Optically Active Compounds

S. Akai, 2014 .

One-Pot Generation of Benzynes from Phenols: Formation of Primary Anilines by the Deoxyamination of Phenols.

S. Akai, Takashi Ikawa, Shigeaki Masuda, 2020, Chemistry.

Trifluoromethanesulfonyloxy-group-directed regioselective (3 + 2) cycloadditions of benzynes for the synthesis of functionalized benzo-fused heterocycles.

H. Tokiwa, S. Akai, Takashi Ikawa, 2015, Organic & biomolecular chemistry.

Generation of 3-borylbenzynes, their regioselective Diels–Alder reactions, and theoretical analysis

Y. Kita, H. Tokiwa, S. Akai, 2013 .

Experimental and Theoretical Studies on Regiocontrol of Benzyne Reactions Using Silyl and Boryl Directing Groups

H. Tokiwa, S. Akai, Takashi Ikawa, 2012 .

Spatial effects of oxovanadium-immobilized mesoporous silica on racemization of alcohols and application in lipase-catalyzed dynamic kinetic resolution

Katsuya Kato, S. Akai, Takashi Ikawa, 2016 .

Cobalt-Catalyzed Intermolecular Markovnikov Hydroamination of Nonactivated Olefins: N2-Selective Alkylation of Benzotriazole.

S. Akai, Kenzo Yahata, Y. Kaneko, 2020, Organic letters.

1,3- and 1,4-Benzdiyne equivalents for regioselective synthesis of polycyclic heterocycles

S. Akai, Takashi Ikawa, A. Takagi, 2016, Chemical science.

Enantiodivergent Synthesis of Axially Chiral Biphenyls from σ-Symmetric 1,1'-Biphenyl-2,6-diol Derivatives by Single Lipase-Catalyzed Acylative and Hydrolytic Desymmetrization

H. Aoyama, S. Akai, Kengo Kasama, 2020 .

Synthesis of various kinds of isoflavones, isoflavanes, and biphenyl-ketones and their 1,1-diphenyl-2-picrylhydrazyl radical-scavenging activities.

S. Akai, Y. Terao, H. Goto, 2009, Chemical & pharmaceutical bulletin.

Diversity Oriented Synthesis of Allocolchicinoids with Fluoro and/or Oxygen Substituent(s) on the C‐Ring from a Single Common Intermediate

K. Tsujikawa, S. Akai, Takashi Ikawa, 2016 .

RECENT PROGRESS IN THE SYNTHESIS OF p-QUINONES AND p-DIHYDRO-QUINONES THROUGH OXIDATION OF PHENOL DERIVATIVES. A REVIEW

Y. Kita, S. Akai, 1998 .

ortho-Selective nucleophilic addition of amines to 3-borylbenzynes: synthesis of multisubstituted anilines by the triple role of the boryl group.

S. Akai, Takashi Ikawa, A. Takagi, 2013, Organic & biomolecular chemistry.

Nucleophilic deoxyfluorination of catechols.

S. Akai, Hiroyuki Nemoto, T. Nishiyama, 2011, Organic letters.

A Penicillium sp. F33 metabolite and its synthetic derivatives inhibit acetyl-CoA:1-O-alkyl-sn-glycero-3-phosphocholine acetyltransferase (a key enzyme in platelet-activating factor biosynthesis) and carrageenan-induced paw edema in mice.

T. Miyase, A. Ikari, Y. Yamazaki, 2013, Biochemical pharmacology.

Improved In Vivo Delivery of Small RNA Based on the Calcium Phosphate Method

Shogo Kobayashi, H. Yamamoto, S. Akai, 2021, Journal of personalized medicine.

A brief and regiospecific synthesis of the late-stage intermediate to 11-deoxyanthracyclinones

Y. Kita, S. Akai, M. Sasho, 1984 .

1-Ethoxyvinyl 2-furoate, an efficient acyl donor for the lipase-catalyzed enantioselective desymmetrization of prochiral 2,2-disubstituted propane-1,3-diols and meso-1,2-diols

Y. Kita, S. Akai, T. Naka, 2000 .

Continuous‐Flow Dynamic Kinetic Resolution of Racemic Alcohols by Lipase–Oxovanadium Cocatalysis

C. Plass, Niklas Adebar, H. Gröger, 2020 .

1-alkoxyvinyl esters: renaissance of half-century-old acyl donors with potential applicability.

Y. Kita, S. Akai, 2004, Chemical record.

[Development of novel asymmetric reactions oriented to next-generation enzymatic organic syntheses].

S. Akai, 2003, Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan.

Recent Advances in Pummerer Reactions

Y. Kita, S. Akai, 2006 .

Heteropolyacid-catalyzed direct deoxygenation of propargyl and allyl alcohols.

S. Akai, M. Egi, T. Kawai, 2012, The Journal of organic chemistry.

Heteropoly compound catalyzed synthesis of both Z- and E-α,β-unsaturated carbonyl compounds.

S. Akai, M. Egi, T. Kawai, 2011, Angewandte Chemie.

Reusable and Durable Immobilized-Cationic Gold(I) Catalysts for Environmentally Benign Bond-Forming Reactions

S. Akai, K. Azechi, M. Egi, 2011 .

Enzyme-catalyzed asymmetrization of 2,2-disubstituted 1,3-propanediols using 1-ethoxyvinyl esters

Y. Kita, S. Akai, T. Naka, 1997 .

A new synthetic strategy for heteroanthracyclines: Total synthesis of D-ring thiophene analogs of daunomycin

Y. Kita, S. Akai, R. Okunaka, 1987 .

Cationic gold(I)-mediated intramolecular cyclization of 3-alkyne-1,2-diols and 1-amino-3-alkyn-2-ols: a practical route to furans and pyrroles.

S. Akai, K. Azechi, M. Egi, 2009, Organic letters.

Concise synthesis of multisubstituted isoquinolines from pyridines by regioselective Diels-Alder reactions of 2-silyl-3,4-pyridynes.

S. Akai, Takashi Ikawa, T. Nishiyama, 2014, Chemistry.

Enantiospecific synthesis and cytotoxicity evaluation of ligudentatol: a programmed aromatization approach to the 2,3,4-trisubstituted phenolic motif via visible-light-mediated group transfer radical cyclization.

H. Aoyama, S. Akai, M. Arai, 2014, Chemistry, an Asian journal.

ortho-Selective nucleophilic addition of primary amines to silylbenzynes: synthesis of 2-silylanilines.

Y. Ishikawa, S. Fujii, Y. Kita, 2011, Angewandte Chemie.

Regiocomplementary cycloaddition reactions of boryl- and silylbenzynes with 1,3-dipoles: selective synthesis of benzo-fused azole derivatives.

Y. Ishikawa, S. Fujii, H. Tokiwa, 2013, The Journal of organic chemistry.

Direct Nucleophilic Substitution of Alcohols Using an Immobilized Oxovanadium Catalyst

S. Akai, Kenzo Yahata, K. Kanomata, 2021, European Journal of Organic Chemistry.

One-Pot Generation of Functionalized Benzynes from Readily Available 2-Hydroxyphenylboronic Acids.

S. Akai, Takashi Ikawa, A. Takagi, 2020, The Journal of organic chemistry.

2-(Trimethylsilyl)phenyl Trimethylsilyl Ethers as Stable and Readily Accessible Benzyne Precursors.

S. Akai, H. Nakajima, Takashi Ikawa, 2017, The Journal of organic chemistry.

An effective and selective conjugate propargylation reaction of stannylallenes to .alpha.,.beta.-unsaturated carbonyl compounds and .alpha.-nitro olefins

Y. Kita, S. Akai, S. Matsuda, 1990 .

Coupling Reaction between Aldehydes and Non-Activated Hydrocarbons via the Reductive Radical-Polar Crossover Pathway.

S. Akai, S. Sakurai, Kenzo Yahata, 2020, Organic letters.

Enantiodivergent preparation of optically active oxindoles having a stereogenic quaternary carbon center at the C3 position via the lipase-catalyzed desymmetrization protocol: effective use of 2-furoates for either enzymatic esterification or hydrolysis.

Y. Kita, S. Akai, T. Tsujino, 2004, The Journal of organic chemistry.

Total Synthesis of (±)-γ-Rubromycin on the Basis of Two Aromatic Pummerer-Type Reactions†

Ikumi Kuriwaki, T. Dohi, Y. Kita, 2007 .

Asymmetric Total Synthesis of Fredericamycin A.

Y. Kita, S. Akai, S. Kitagaki, 1999, Angewandte Chemie.

Efficient intramolecular cyclizations of phenoxyethynyl diols into multisubstituted α,β-unsaturated lactones.

S. Akai, Kaori Shimizu, Y. Ota, 2013, Organic letters.

Transition Metal-Catalyzed Intramolecular Cyclization of Propargyl Alcohols and Their Derivatives for the Synthesis of Highly Substituted Five-Membered Oxygen Heterocycles

S. Akai, M. Egi, 2015 .

Facile and efficient syntheses of carboxylic anhydrides and amides using (trimethylsilyl)ethoxyacetylene

Y. Kita, S. Akai, M. Yoshigi, 1986 .

Ammonium Salt-Accelerated Hydrazinolysis of Unactivated Amides: Mechanistic Investigation and Application to a Microwave Flow Process

Y. Hamashima, S. Akai, Y. Shimizu, 2019, Organic Process Research & Development.

Development of a highly efficient single-mode microwave applicator with a resonant cavity and its application to continuous flow syntheses

T. Okamoto, H. Egami, Y. Hamashima, 2015 .

Acid-Promoted Rearrangement of Cyclic α,β-Epoxy Acylates: Stereoselective Synthesis of Spirocyclanes and Quaternary Carbon Centers

M. Kondo, Y. Kita, S. Akai, 1997 .

Asymmetric synthesis of chiral spirocyclanes: A new route to the optically active spiro[cyclopentane-1,1′-indan]-2,5-dione system

Y. Kita, S. Akai, S. Kitagaki, 1996 .

Asymmetric synthesis of chiral spirocyclanes: Selective formation of 2-acyloxy-1-oxospiro[4.n]alkanes by regio- and stereoselective rearrangement of α,β-epoxy acylates in bicyclo[n.3.0]alkane systems

Yutaka Yoshida, Hiromichi Fujioka, M. Kondo, 1995 .

Flow Synthesis of (3R)- and (3S)-(E)-1-Iodohexa-1,5-dien-3-ol: Chiral Building Blocks for Natural Product Synthesis

S. Akai, T. Oishi, S. Katsuragi, 2018, Chemistry Letters.

Lipase-catalyzed domino kinetic resolution of alpha-hydroxynitrones/intramolecular 1,3-dipolar cycloaddition: a concise asymmetric total synthesis of (-)-rosmarinecine.

Y. Kita, S. Akai, Yukiko Kanao, 2005, Chemical communications.

Regioselective Synthesis of 2,3,5-Trisubstituted Indoles from p-Sulfinyl-aniline by Dual Use of the Sulfinyl Group

Y. Kita, N. Kawashita, S. Akai, 2002 .

Chemistry of silylketenes: a simple preparation of α-silyl-α-stannylacetic esters and their stereoselective Reformatsky-type reaction with aldehydes or aldimines

Y. Kita, S. Akai, S. Kitagaki, 1992 .

A short and efficient synthesis of 11-deoxyanthracyclinones: strong base-induced cycloaddition of the suitably substituted tetrahydrohomophthalic anhydride

Y. Kita, S. Akai, M. Sasho, 1985 .

Synthesis of biaryl compounds through three-component assembly: ambidentate effect of the tert-butyldimethylsilyl group for regioselective Diels-Alder and Hiyama coupling reactions.

Y. Kita, S. Akai, Takashi Ikawa, 2008, Angewandte Chemie.

A highly convergent strategy for the synthesis of 4-demethoxydaunomycinone and daunohycinone: A novel synthesis of C4-acetoxylated homophthalic anhydrides

Y. Kita, S. Akai, M. Sasho, 1986 .

Anthracyclinone syntheses using strong base induced cycloaddition of homophthalic anhydrides and related compounds

Y. Kita, S. Akai, M. Sasho, 1984 .

Central-axial-central chirality transfer: asymmetric synthesis of highly substituted indenes bearing a stereogenic quaternary carbon center from optically active propargyl alcohols.

S. Akai, Kaori Shimizu, Y. Ota, 2015, Chemical communications.

1-Ethoxyvinyl acetate as a novel, highly reactive, and reliable acyl donor for enzymatic resolution of alcohols

Y. Kita, S. Akai, T. Naka, 1996 .

One-pot synthesis of optically active allyl esters via lipase-vanadium combo catalysis.

Y. Kita, S. Akai, M. Egi, 2010, Organic letters.

Enantioselective total synthesis of a potent antitumor antibiotic, fredericamycin A.

Y. Kita, S. Akai, S. Kitagaki, 2001, Journal of the American Chemical Society.

AN EFFICIENT SYNTHESIS OF ALPHA -SILYLACETATES HAVING VARIOUS TYPES OF FUNCTIONAL GROUPS IN THE MOLECULES

Y. Kita, S. Akai, J. Sekihachi, 1990 .

A domino process for benzyne preparation: dual activation of o-(trimethylsilyl)phenols by nonafluorobutanesulfonyl fluoride.

S. Akai, Takashi Ikawa, A. Takagi, 2011, Organic letters.

Reaction of ynolate anions derived from silylketenes with electrophiles: a facile preparation of silyl ynol ethers and functionalized silylketenes

Y. Kita, S. Akai, Kouzou Matsumoto, 1996 .

Asymmetric total synthesis of fredericamycin A: an intramolecular cycloaddition pathway.

Y. Kita, S. Akai, H. Fujioka, 2005, Chemistry.

AN EFFICIENT PREPARATION OF PERI-HYDROXY DIHYDROQUINONE DERIVATIVES THROUGH A PUMMERER-TYPE REARRANGEMENT OF SILYLENE-PROTECTED PERI-HYDROXY AROMATIC SULFOXIDES

Kenji Takahashi, Y. Kita, S. Akai, 1996 .

Protecting-group-free catalytic asymmetric total synthesis of (−)-rosmarinecine

Y. Kita, S. Akai, Yukiko Kanao, 2012 .

Total synthesis of a new inhibitor of superoxide anion generation, opc-15161

Y. Kita, S. Akai, H. Fujioka, 1991 .

Total Synthesis of 11-Deoxyanthracyclines: 4-Demethoxy-11-deoxydaunomycin, 11-Deoxydaunomycin, and Their Analogues

Y. Kita, S. Akai, M. Sasho, 1988 .

An efficient, regiospecific synthesis of 4-demethoxydaunomycinone and daunomycinone.

Y. Kita, S. Akai, M. Sasho, 1987 .

Preparation and regioselective Diels-Alder reactions of borylbenzynes: synthesis of functionalized arylboronates.

Y. Kita, S. Akai, Takashi Ikawa, 2010, Angewandte Chemie.

Lipase-catalyzed asymmetric synthesis of naphtho[2,3-c]furan-1(3H)-one derivatives by a one-pot dynamic kinetic resolution/intramolecular Diels-Alder reaction: Total synthesis of (-)-himbacine.

S. Akai, M. Egi, Koji Sugiyama, 2017, Bioorganic & medicinal chemistry.

Mo-Au combo catalysis for rapid 1,3-rearrangement of propargyl alcohols into alpha,beta-unsaturated carbonyl compounds.

S. Akai, Y. Yamaguchi, M. Egi, 2008, Organic letters.

Total synthesis of (-)-agelastatin A: an SH2' radical azidation strategy.

H. Aoyama, S. Akai, Izuru Tsuchimochi, 2018, Chemical communications.

Regioselective, Directed Meta Acylation of Aromatic Compounds

S. Buchwald, S. Akai, A. Peat, 1998 .

Regioselective, nucleophilic carbon–carbon bond formation at the C4-position of indoles initiated by the aromatic Pummerer-type reaction

Ikumi Kuriwaki, Y. Kita, N. Kawashita, 2006 .

Highly regioselective nucleophilic carbon-carbon bond formation on furans and thiophenes initiated by pummerer-type reaction.

Ikumi Kuriwaki, Y. Kita, N. Kawashita, 2004, Organic letters.

Lipase-Catalyzed Dynamic Kinetic Resolution of C1 - and C2 -Symmetric Racemic Axially Chiral 2,2'-Dihydroxy-1,1'-biaryls.

S. Akai, Yasuhiro Oki, Gamal A I Moustafa, 2018, Angewandte Chemie.

Chemo- and regioselective cross-dehydrogenative coupling reaction of 3-hydroxycarbazoles with arenols catalyzed by a mesoporous silica-supported oxovanadium

S. Akai, Y. Uetake, S. Takizawa, 2021, RSC advances.

Base-promoted lipase-catalyzed kinetic resolution of atropisomeric 1,1′-biaryl-2,2′-diols

S. Akai, Kengo Kasama, Gamal A I Moustafa, 2019, RSC advances.

Cationic gold(I)-catalyzed intramolecular cyclization of gamma-hydroxyalkynones into 3(2H)-furanones.

S. Akai, Kaori Shimizu, K. Azechi, 2010, The Journal of organic chemistry.

Lipase-catalyzed enantioselective desymmetrization of prochiral 3,3-bis(hydroxymethyl)oxindoles

Y. Kita, S. Akai, T. Tsujino, 2001 .

Lipase-catalyzed domino dynamic kinetic resolution of racemic 3-vinylcyclohex-2-en-1-ols/intramolecular Diels-Alder reaction: one-pot synthesis of optically active polysubstituted decalins.

Y. Kita, S. Akai, Kouichi Tanimoto, 2004, Angewandte Chemie.

Lipase-catalyzed domino kinetic resolution/intramolecular Diels-Alder reaction: one-pot synthesis of optically active 7-oxabicyclo[2.2.1]heptenes from furfuryl alcohols and beta-substituted acrylic acids.

Y. Kita, S. Akai, M. Imanishi, 2002, Chemistry.

An Effective and Selective Conjugate Propargylation Reaction of Stannylallenes to α,β‐Unsaturated Carbonyl Compounds and . alpha.‐Nitro Olefins.

Y. Kita, S. Akai, Y. Tamura, 1991 .

Practical total synthesis of 11-deoxydaunomycinone and the first total synthesis of 11-deoxydaunomycin

Y. Kita, S. Akai, M. Sasho, 1987 .

A mild and facile synthesis of carboxylic anhydrides

Y. Kita, S. Akai, M. Yoshigi, 1985 .

syn-Selective Reformatsky-Type Reaction of α-Silyl-α-stannylacetic Esters with Aldehydes: Stereoselective Synthesis of (E)- and (Z)-α,β-Unsaturated Esters

Y. Kita, S. Akai, S. Kitagaki, 1991 .

A dynamic kinetic resolution of allyl alcohols by the combined use of lipases and [VO(OSiPh3)3].

Y. Kita, S. Akai, Tomoko Yamamoto, 2006, Angewandte Chemie.

A mesoporous-silica-immobilized oxovanadium cocatalyst for the lipase-catalyzed dynamic kinetic resolution of racemic alcohols.

Katsuya Kato, Katsuya Kato, S. Akai, 2013, Angewandte Chemie.

Preparation of Novel Cyclic Hypervalent Idoine(III) Compounds Having Azido, Cyano, and Nitrato Ligands

Y. Kita, S. Akai, M. Egi, 1996 .

Lipase-Catalyzed Kinetic Resolution of C1-Symmetric Heterocyclic Biaryls.

H. Gröger, S. Akai, K. Kanomata, 2022, Chemical & pharmaceutical bulletin.

Dress-up chiral columns for the enantioseparation of amino acids based on fluorous separation

Koichi Inoue, T. Toyo’oka, S. Akai, 2013, Analytical and Bioanalytical Chemistry.

Aryl Boronic Esters Are Stable on Silica Gel and Reactive under Suzuki-Miyaura Coupling Conditions.

H. Sajiki, S. Akai, Takashi Ikawa, 2022, Organic letters.

Efficient lipase-catalyzed enantioselective desymmetrization of prochiral 2,2-disubstituted 1,3-propanediols and meso 1,2-diols using 1-ethoxyvinyl 2-furoate.

Y. Kita, S. Akai, T. Tsujino, 2002, The Journal of organic chemistry.

MPP+ induces necrostatin-1- and ferrostatin-1-sensitive necrotic death of neuronal SH-SY5Y cells

Keisuke Ito, Y. Tsujimoto, S. Akai, 2017, Cell Death Discovery.

Discovery of aromatic components with excellent fragrance properties and biological activities: β-ionols with antimelanogenetic effects and their asymmetric syntheses.

S. Akai, Takashi Ikawa, R. Komaki, 2013, Chemical & pharmaceutical bulletin.

Synthesis of 2,5-dioxygenated pyrazine 4-oxides: total synthesis of a new inhibitor of superoxide anion generation, OPC-15161

Y. Kita, S. Akai, H. Fujioka, 1994 .

Recent Progress on the Lipase-Catalyzed Asymmetric Syntheses

Y. Kita, S. Akai, 2007 .

Dynamic kinetic resolution of a tertiary alcohol.

H. Gröger, S. Akai, Yasuhiro Oki, 2020, Chemical communications.

Synthetic Studies on the Viridin Skeleton through Regio- and Stereoselective Functionalization of the AE-Ring Moiety

S. Akai, G. Itoh, Takashi Ikawa, 2021, Synlett.

Correlation of indoleamine-2,3-dioxigenase 1 inhibitory activity of 4,6-disubstituted indazole derivatives and their heme binding affinity.

S. Akai, T. Uno, Taku Yamashita, 2019, Bioorganic & medicinal chemistry letters.

An efficient synthesis of p-quinones utilizing a novel Pummerer-type rearrangement of p-sulfinylphenols

Y. Kita, S. Akai, Y. Yoshida, 1995 .

Synthesis of Various Kinds of Isoflavones, Isoflavans, and Biphenyl‐Ketones and Their 1,1‐Diphenyl‐2‐picrylhydrazyl Radical‐Scavenging Activities.

S. Akai, Y. Terao, H. Goto, 2009 .

Oxidative Intramolecular (4 + 2) Cycloaddition of Silylene-Protected 2- Pyridone Derivatives - A Short and Efficient Synthesis of the DEF-Ring of Fredericamycin A.

Y. Kita, S. Akai, H. Ueno, 1994 .

Polar cycloaddition of α-acyl-α-chlorosulfides with alkynes. Novel one-step syntheses of furans and 2-furanones

S. Akai, H. Ishibashi, H. Nakagawa, 1984 .

Palladium-Catalyzed One-Pot Cross-Coupling of Phenols Using Nonafluorobutanesulfonyl Fluoride

S. Akai, Takashi Ikawa, K. Saito, 2012, Synlett.

Acid-catalyzed cyclizations of n-vinyl-α-sulfinylacetamides A novel synthetic approach to erythrinane

S. Akai, Y. Tamura, H. Maeda, 1982 .

Ambident effect of a p-sulfinyl group for the introduction of two carbon substituents to phenol rings: a convergent synthesis of diverse benzofuran neolignans.

Y. Kita, S. Akai, Y. Nakamura, 2000, Organic letters.

Synthetic anthracyclines: regiospecific total synthesis of a D-ring pyridine analogue of 11-deoxydaunomycin

Y. Kita, S. Akai, R. Okunaka, 1990 .

A New Synthetic Strategy for Heteroanthracyclines: Total Synthesis of D-Ring Thiophene Analogs (I) and (II) of Daunomycin.

Y. Kita, S. Akai, R. Okunaka, 1988 .

2-[(Neopentyl glycolato)boryl]phenyl Triflates and Halides for Fluoride Ion-Mediated Generation of Functionalized Benzynes

Y. Hamashima, S. Akai, Takashi Ikawa, 2015 .

Dynamic analysis of fluid distribution in the gastrointestinal tract in rats: positron emission tomography imaging after oral administration of nonabsorbable marker, [(18)F]Deoxyfluoropoly(ethylene glycol).

Yasuyoshi Watanabe, Y. Sugiyama, Masaaki Suzuki, 2013, Molecular pharmaceutics.

PUMMERER REACTION INTERMEDIATE AS AN INITIATING FUNCTION FOR CATIONIC OLEFIN CYCLIZATION

S. Akai, H. Ishibashi, Y. Tamura, 1982 .

Synthesis of the erythrinan skeleton by acid-promoted cyclization of N-(3-oxo-1-cyclohexen-1-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-α-(methylsulfinyl)acetamide

S. Akai, Y. Tamura, H. Ishibashi, 1985 .

Synthesis of the Erythrinan Skeleton by Acid-Promoted Cyclization of N-(3-Oxo-1-cyclohexen-1-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-α-(methylsulfinyl)acetamide.

S. Akai, Y. Tamura, H. Ishibashi, 1986 .

Preparation of optically active cycloalkenes bearing all-carbon quaternary stereogenic centres via lipase–oxovanadium combo-catalysed dynamic kinetic resolution

S. Akai, Takashi Ikawa, Koji Sugiyama, 2017 .

PET imaging of brain cancer with positron emitter-labeled liposomes.

H. Tsukada, N. Oku, T. Asai, 2011, International journal of pharmaceutics.

T cell-independent B cell response is responsible for ABC phenomenon induced by repeated injection of PEGylated liposomes.

H. Tsukada, N. Oku, Hiroyuki Koide, 2010, International journal of pharmaceutics.

Efficient Intramolecular Cyclizations of Phenoxyethynyl Diols into Multisubstituted α,β‐Unsaturated Lactones.

S. Akai, Kaori Shimizu, Y. Ota, 2014 .

Synthesis of Fluorinated Aromatic Compounds by One-Pot Benzyne Generation and Nucleophilic Fluorination

S. Akai, Takashi Ikawa, A. Takagi, 2014 .

Regioselective Rearrangement of 4,4-Disubstituted 2-Hydroxycyclohexa-2,5-Dienones under Deoxyfluorination Conditions.

S. Akai, Takashi Ikawa, Takafumi Ide, 2017, The Journal of organic chemistry.

1-Alkoxyvinyl Ester as an Excellent Acyl Donor: Efficient Macrolactone Synthesis.

Y. Kita, S. Akai, Tohru Kamitanaka, 2021, Journal of Organic Chemistry.

Diblock copolymer of bacterial cellulose and poly(methyl methacrylate) initiated by chain-end-type radicals produced by mechanical scission of glycosidic linkages of bacterial cellulose.

T. Iwata, T. Ohura, S. Akai, 2010, Biomacromolecules.

An Efficient p-Thiocyanation of Phenols and Naphtols Using a Reagent combination of Phenyliodine Dichloride and Lead(II) Thiocyanate

Y. Kita, S. Akai, Y. Takeda, 1997 .

Microflow Fluorinations of Benzynes: Efficient Synthesis of Fluoroaromatic Compounds.

S. Akai, Takashi Ikawa, Shigeaki Masuda, 2018, Chemical & pharmaceutical bulletin.

Cobalt-catalyzed Hydroamination of Alkenes with 5-Substituted Tetrazoles: Facile access to 2,5-Disubstituted Tetrazoles and Asymmetric Intermolecular Hydroaminations.

S. Akai, Kenzo Yahata, Y. Kaneko, 2020, Chemical and pharmaceutical bulletin.

Chemistry of Silylketenes : Simple Preparation of Silylallenes by the Reaction of Silyketenes with Phosphorus Ylides

Y. Kita, S. Akai, S. Kitagaki, 1994 .

Chemistry of Silylketenes: Simple Preparation of Silylallenes by the Reaction of Silylketenes with Phosphorus Ylides.

Y. Kita, S. Akai, S. Kitagaki, 1994 .

Cationic gold(I)-mediated intramolecular cyclization of 3-alkyne-1,2-diols and 1-amino-3-alkyn-2-ols: a practical route to furans and pyrroles.

S. Akai, K. Azechi, M. Egi, 2009, Organic letters.

Transition Metal‐Catalyzed Intramolecular Cyclization of Propargyl Alcohols and Their Derivatives for the Synthesis of Highly Substituted Five‐Membered Oxygen Heterocycles

S. Akai, M. Egi, 2015 .

Efficient intramolecular cyclizations of phenoxyethynyl diols into multisubstituted α,β-unsaturated lactones.

S. Akai, Kaori Shimizu, Y. Ota, 2013, Organic Letters.

Mo-Au combo catalysis for rapid 1,3-rearrangement of propargyl alcohols into alpha,beta-unsaturated carbonyl compounds.

S. Akai, Y. Yamaguchi, M. Egi, 2008, Organic letters.

An efficient synthesis of peri-hydroxy aromatic compounds via a strong-base-induced

Y. Kita, S. Akai, H. Fujioka, 2000, The Journal of organic chemistry.

An Efficient Synthesis of peri-Hydroxy Aromatic Compounds: A Strong Base-Induced [4 + 2]Cycloaddition of 4-Phenylthio-Substituted Homophthalic Anhydrides with Various Sulfinyl-Substituted Dienophiles

Y. Kita, S. Akai, Y. Takeda, 1998 .

PET imaging of brain cancer with positron emitter-labeled liposomes.

H. Tsukada, N. Oku, T. Asai, 2011, International journal of pharmaceutics.

Synthesis of biaryl compounds through three-component assembly: ambidentate effect of the tert-butyldimethylsilyl group for regioselective Diels-Alder and Hiyama coupling reactions.

Y. Kita, S. Akai, Takashi Ikawa, 2008, Angewandte Chemie.