V. Delfosse

发表

Combining 'dry' co-crystallization and in situ diffraction to facilitate ligand screening by X-ray crystallography.

G. Labesse, J. Ferrer, F. Hoh, 2015, Acta crystallographica. Section D, Biological crystallography.

Structural and functional evidences for the interactions between nuclear hormone receptors and endocrine disruptors at low doses.

W. Bourguet, V. Delfosse, Marina Grimaldi, 2017, Comptes rendus biologies.

Reporter Cell Lines for the Characterization of the Interactions between Human Nuclear Receptors and Endocrine Disruptors

William Bourguet, Marina Grimaldi, W. Bourguet, 2015, Front. Endocrinol..

Mechanistic insights into the synergistic activation of the RXR–PXR heterodimer by endocrine disruptor mixtures

S. Cianférani, D. Harrus, B. Demeneix, 2020, Proceedings of the National Academy of Sciences.

Specificity of L,D-Transpeptidases from Gram-positive Bacteria Producing Different Peptidoglycan Chemotypes*

L. Rice, J. Mainardi, Arul Marie, 2007, Journal of Biological Chemistry.

Cloning, purification, crystallization and preliminary crystallographic analysis of a penicillin-binding protein homologue from Pyrococcus abyssi.

V. Delfosse, W. Sougakoff, C. Mayer, 2005, Acta crystallographica. Section F, Structural biology and crystallization communications.

Functional analyses of phosphatidylserine/PI(4)P exchangers with diverse lipid species and membrane contexts set unanticipated rules on lipid transfer

G. Drin, W. Bourguet, V. Delfosse, 2021, bioRxiv.

[Towards bisphenols without hormonal effects].

W. Bourguet, V. Delfosse, Marina Grimaldi, 2013, Medecine sciences : M/S.

Mechanisms of endocrine disruption through nuclear receptors and related pathways

W. Bourguet, V. Delfosse, P. Balaguer, 2019, Current Opinion in Endocrine and Metabolic Research.

Unexpected Inhibition of Peptidoglycan LD-Transpeptidase from Enterococcus faecium by the β-Lactam Imipenem*

L. Rice, J. Mainardi, L. Dubost, 2007, Journal of Biological Chemistry.

Insights into the activation mechanism of human estrogen-related receptor γ by environmental endocrine disruptors

A. Barducci, W. Bourguet, V. Delfosse, 2019, Cellular and Molecular Life Sciences.

Structural and mechanistic insights into bisphenols action provide guidelines for risk assessment and discovery of bisphenol A substitutes

Jean-Luc Pons, Gilles Labesse, William Bourguet, 2012, Proceedings of the National Academy of Sciences.

A structural perspective on nuclear receptors as targets of environmental compounds

W. Bourguet, V. Delfosse, P. Balaguer, 2014, Acta Pharmacologica Sinica.

Nuclear receptor profiling of bisphenol-A and its halogenated analogues.

William Bourguet, Marina Grimaldi, W. Bourguet, 2014, Vitamins and hormones.

An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor β (RARβ, NR1B2) Selective Agonist

H. Gronemeyer, W. Bourguet, V. Delfosse, 2015, PloS one.

Synergistic activation of human pregnane X receptor by binary cocktails of pharmaceutical and environmental compounds

J. Pascussi, W. Bourguet, V. Delfosse, 2015, Nature Communications.

Structure-Based and Knowledge-Informed Design of B-Raf Inhibitors Devoid of Deleterious PXR Binding.

G. Labesse, J. Pons, W. Bourguet, 2021, Journal of medicinal chemistry.

Structural and Functional Profiling of Environmental Ligands for Estrogen Receptors

W. Bourguet, V. Delfosse, Marina Grimaldi, 2014, Environmental health perspectives.

Structure of the Archaeal Pab87 Peptidase Reveals a Novel Self-Compartmentalizing Protease Family

M. Delarue, C. Birck, E. Girard, 2009, PloS one.

Structural and Functional Specialization of OSBP-Related Proteins

G. Drin, W. Bourguet, V. Delfosse, 2020, Contact.

Phosphatidylserine transport by ORP/Osh proteins is driven by phosphatidylinositol 4-phosphate

S. Vanni, G. Drin, C. L. Jackson, 2015, Science.

Crystal Structure of a Novel -Lactam-insensitive Peptidoglycan Transpeptidase

J. Mainardi, M. Arthur, L. Gutmann, 2006 .

Crystal structure of a novel beta-lactam-insensitive peptidoglycan transpeptidase.

J. Mainardi, M. Arthur, L. Gutmann, 2006, Journal of molecular biology.

Reporter cell lines to evaluate the selectivity of chemicals for human and zebrafish estrogen and peroxysome proliferator activated γ receptors

W. Bourguet, V. Delfosse, Marina Grimaldi, 2015, Front. Neurosci..

Osh4p exchanges sterols for phosphatidylinositol 4-phosphate between lipid bilayers

D. Douguet, G. Drin, B. Antonny, 2011, The Journal of cell biology.

Riboswitch structure: an internal residue mimicking the purine ligand

Patricia Bouchard, Daniel A. Lafontaine, Pascale Legault, 2009, Nucleic acids research.

Affinity purification of RNA using an ARiBo tag.

P. Legault, V. Delfosse, P. Dagenais, 2012, Methods in molecular biology.

Functional analyses of phosphatidylserine/PI(4)P exchangers with diverse lipid species and membrane contexts reveal unanticipated rules on lipid transfer

G. Drin, W. Bourguet, V. Delfosse, 2021, BMC Biology.

Crystal structure of human ERRg LBD in complex with bisphenol-B

A. Barducci, W. Bourguet, V. Delfosse, 2019 .

Insights into the activation mechanism of human estrogen-related receptor γ by environmental endocrine disruptors

A. Barducci, W. Bourguet, V. Delfosse, 2019, Cellular and Molecular Life Sciences.

Functional analyses of phosphatidylserine/PI(4)P exchangers with diverse lipid species and membrane contexts reveal unanticipated rules on lipid transfer

G. Drin, W. Bourguet, V. Delfosse, 2021, BMC Biology.

Riboswitch structure: an internal residue mimicking the purine ligand

D. Lafontaine, P. Legault, V. Delfosse, 2009, Nucleic acids research.

Surfactant Poloxamer 188 as a New Crystallizing Agent for Urate Oxidase

G. Sciara, C. Cambillau, V. Delfosse, 2009 .

Endocrine disruptors Structural and functional evidences for the interactions between nuclear hormone receptors and endocrine disruptors at low doses

W. Bourguet, V. Delfosse, Marina Grimaldi, 2022 .

A potent agonist-based PROTAC targeting Pregnane X Receptor that delays colon cancer relapse

J. Pascussi, V. Delfosse, S. Gerbal-Chaloin, 2024, bioRxiv.