P. Kessler

发表

Mambalgin-1 Pain-relieving Peptide, Stepwise Solid-phase Synthesis, Crystal Structure, and Functional Domain for Acid-sensing Ion Channel 1a Inhibition*

D. Douguet, G. Mourier, D. Servent, 2015, The Journal of Biological Chemistry.

MiniCD4 protein resistance mutations affect binding to the HIV-1 gp120 CD4 binding site and decrease entry efficiency

Loïc Martin, P. Selhorst, G. Vanham, 2012, Retrovirology.

Interfacial cavity filling to optimize CD4-mimetic miniprotein interactions with HIV-1 surface glycoprotein.

P. Acharya, P. Kwong, Yongping Yang, 2013, Journal of medicinal chemistry.

Unexpected paracrine action of prostate cancer cells harboring a new class of androgen receptor mutation—A new paradigm for cooperation among prostate tumor cells

D. Jacqmin, H. Lang, J. Céraline, 2007, International journal of cancer.

Live-cell one- and two-photon uncaging of a far-red emitting acridinone fluorophore.

J. Vonesch, J. Léonard, J. Nicoud, 2010, Journal of the American Chemical Society.

A snake toxin as a theranostic agent for the type 2 vasopressin receptor

B. Jego, G. Mourier, D. Servent, 2020, Theranostics.

Interfacial cavity filling to optimize CD4-mimetic miniprotein interactions with the HIV-1 surface protein

P. Acharya, P. Kwong, Yongping Yang, 2013 .

MiniCD4 Microbicide Prevents HIV Infection of Human Mucosal Explants and Vaginal Transmission of SHIV162P3 in Cynomolgus Macaques

M. Stefanidou, C. Herrera, Loïc Martin, 2012, PLoS pathogens.

nAChR and α-neurotoxin: New tools for old acquaintances

A. Ménez, P. Kessler, S. Maurin, 1998, Journal of Physiology-Paris.

Unlike for Human Monocytes after LPS Activation, Release of TNF-α by THP-1 Cells Is Produced by a TACE Catalytically Different from Constitutive TACE

J. Vonesch, J. Reimund, C. Muller, 2012, PloS one.

From a Cone Snail Toxin to a Competitive MC4R Antagonist.

G. Mourier, D. Servent, M. Bouvier, 2022, Journal of medicinal chemistry.

Relative Spatial Position of a Snake Neurotoxin and the Reduced Disulfide Bond α(Cys192-Cys193) at the αγ Interface of the Nicotinic Acetylcholine Receptor*

G. Mourier, A. Ménez, D. Servent, 2000, The Journal of Biological Chemistry.

4-diazocyclohexa-2,5-dienones as photoaffinity reagents for proteins

P. Kessler, M. Goeldner, L. Ehret-Sabatier, 1990 .

Late‐Stage Isotopic Carbon Labeling of Pharmaceutically Relevant Cyclic Ureas Directly from CO2

C. Halldin, P. Kessler, M. Schou, 2018, Angewandte Chemie.

A cysteine-linkable, short cleavable photoprobe with dual functionality to explore protein-protein interfaces.

A. Ménez, P. Kessler, F. Teixeira-Clerc, 2003, Bioconjugate chemistry.

Purification of the nicotinic acetylcholine receptor protein by affinity chromatography using a regioselectively modified and reversibly immobilized alpha-toxin from Naja nigricollis.

A. Ménez, A. Brisson, P. Kessler, 1997, Biochimica et biophysica acta.

Synthesis of an acetylcholine receptor-specific toxin derivative regioselectively labeled with an undecagold cluster.

A. Ménez, A. Brisson, P. Kessler, 1994, Bioconjugate chemistry.

SYNTHESIS OF N-PROTECTED SERINE ETHERS AS PRECURSORS OF NEW PHOTOACTIVATABLE AMINO ACIDS CLEAVABLE BY HYDROGENOLYSIS

P. Kessler, C. Hirth, C. Colas, 1994 .

A splicing variant of the androgen receptor detected in a metastatic prostate cancer exhibits exclusively cytoplasmic actions.

J. Céraline, J. Bergerat, P. Kessler, 2007, Endocrinology.

Characterization of the First Animal Toxin Acting as an Antagonist on AT1 Receptor

D. Servent, C. Llorens-Cortes, P. Kessler, 2023, International journal of molecular sciences.

The three‐finger toxin fold: a multifunctional structural scaffold able to modulate cholinergic functions

D. Servent, P. Kessler, P. Marchot, 2017, Journal of neurochemistry.

Synthesis of a Polyhistidine-bearing Amphipol and its Use for Immobilizing Membrane Proteins.

J. Popot, M. Zoonens, F. Giusti, 2015, Biomacromolecules.

Structural and Functional Diversity of Animal Toxins Interacting With GPCRs

D. Servent, P. Kessler, P. Robin, 2022, Frontiers in Molecular Biosciences.

Specific properties of a C-terminal truncated androgen receptor detected in hormone refractory prostate cancer.

J. Céraline, J. Bergerat, P. Kessler, 2008, Advances in experimental medicine and biology.

A Theranostic Agent Combining a Two-Photon-Absorbing Photosensitizer for Photodynamic Therapy and a Gadolinium(III) Complex for MRI Detection.

F. Bolze, P. Kessler, É. Tóth, 2016, Chemistry.

Only Snake Curaremimetic Toxins with a Fifth Disulfide Bond Have High Affinity for the Neuronal α7 Nicotinic Receptor*

D Bertrand, D. Bertrand, A. Ménez, 1997, The Journal of Biological Chemistry.

Heavy Chain-Only IgG2b Llama Antibody Effects Near-Pan HIV-1 Neutralization by Recognizing a CD4-Induced Epitope That Includes Elements of Coreceptor- and CD4-Binding Sites

J. Mascola, I. Georgiev, P. Acharya, 2013, Journal of Virology.

How Do Short Neurotoxins Bind to a Muscular-type Nicotinic Acetylcholine Receptor?*

A. Ménez, P. Kessler, F. Teixeira-Clerc, 2002, The Journal of Biological Chemistry.

Straightforward Selection of Broadly Neutralizing Single-Domain Antibodies Targeting the Conserved CD4 and Coreceptor Binding Sites of HIV-1 gp120

J. Bouchet, P. Kessler, P. Chames, 2012, Retrovirology.

Elicitation of Neutralizing Antibodies Directed against CD4-Induced Epitope(s) Using a CD4 Mimetic Cross-Linked to a HIV-1 Envelope Glycoprotein

D. Montefiori, Klára Sirokmán, A. Carfi, 2012, PloS one.

Straightforward Selection of Broadly Neutralizing Single-Domain

Patrick Chames, Daniel Baty, Francis Barin, 2012 .

Mambalgin-1 pain-relieving peptide locks the hinge between α4 and α5 helices to inhibit rat acid-sensing ion channel 1a

D. Douguet, D. Servent, M. Salinas, 2021, Neuropharmacology.

Design and synthesis of a novel site-directed reducing agent for the disulfide bond involved in the acetylcholine binding site of the AChoR

D. Servent, P. Kessler, C. Hirth, 1994 .

Stabilization of HIV-1 Envelope in the CD4-bound Conformation through Specific Cross-linking of a CD4 Mimetic*

D. Montefiori, R. Guérois, Hocine Madaoui, 2011, The Journal of Biological Chemistry.

Vinexinβ, an atypical “sensor” of retinoic acid receptor γ signaling: union and sequestration, separation, and phosphorylation

J. Vonesch, B. Kieffer, P. Kessler, 2010, FASEB journal : official publication of the Federation of American Societies for Experimental Biology.

Site‐directed disulfide reduction using an affinity reagent: Application on the nicotinic acetylcholine receptor

A. Ménez, D. Servent, P. Kessler, 1995, FEBS letters.

Stabilization of HIV-1 envelope in the CD4-bound conformation through specific cross-linking of a CD4 mimetic.

D. Montefiori, R. Guérois, Hocine Madaoui, 2011, The Journal of Biological Chemistry.

Structural basis for highly effective HIV-1 neutralization by CD4-mimetic miniproteins revealed by 1.5 Å cocrystal structure of gp120 and M48U1.

J. Mascola, P. Acharya, M. Louder, 2013, Structure.

A synthetic delivery vector for mucosal vaccination

A. Meola, F. Rey, E. Tartour, 2023, bioRxiv.

Two-photon excitation in life sciences: neurotransmitter and fluorescence uncaging

Frédéric Bolze, Maurice Goeldner, Attila Losonczy, 2011, BiOS.

Engineered Synthetic STxB for Enhanced Cytosolic Delivery

E. Tartour, L. Johannes, G. Mourier, 2023, Cells.

Straightforward selection of broadly neutralizing single-domain antibodies targeting the conserved CD4 and co-receptor binding sites of HIV-1 gp120

J. Bouchet, P. Kessler, P. Chames, 2012, Retrovirology.

Mambalgin-1 Pain-relieving Peptide, Stepwise Solid-phase Synthesis, Crystal Structure, and Functional Domain for Acid-sensing Ion Channel 1a Inhibition*

D. Douguet, G. Mourier, D. Servent, 2015, The Journal of Biological Chemistry.