J. Tedrow

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Cationic bis(oxazoline) and pyridyl-bis(oxazoline)Cu(II) and Zn(II) Lewis acid catalysts. A comparative study in catalysis of Diels-Alder and aldol reactions

Davidr . Evans, M. Kozlowski, J. Tedrow, 1996 .

New conditions for the synthesis of thiophenes via the Knoevenagel/Gewald reaction sequence. Application to the synthesis of a multitargeted kinase inhibitor

J. Tedrow, D. Barnes, Maureen A. McLaughlin, 2006 .

Development and Execution of a Production-Scale Continuous [2 + 2] Photocycloaddition

Matthew G. Beaver, J. Tedrow, En-Xuan Zhang, 2020 .

Separation and quantitation of eight isomers in a molecule with three stereogenic centers by normal phase liquid chromatography.

J. Tedrow, Laura E Blue, Nilesh H. Joshi, 2018, Journal of chromatography. A.

Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors.

E. Lobenhofer, Kristin L. Andrews, B. Herberich, 2015, ACS medicinal chemistry letters.

Discovery and optimization of anthranilic acid sulfonamides as inhibitors of methionine aminopeptidase-2: a structural basis for the reduction of albumin binding.

Scott A. Erickson, S. Davidsen, A. Petros, 2006, Journal of medicinal chemistry.

Characterization of Two Stable Degradants of Palladium tBuXPhos Catalyst and a Unique Dearomatization Reaction

J. Tedrow, Christopher Wilde, T. Hwang, 2012 .

Diastereoselective magnesium halide-catalyzed anti-aldol reactions of chiral N-acyloxazolidinones.

Davidr . Evans, J. Tedrow, C. W. Downey, 2002, Journal of the American Chemical Society.

Chiral Salen-Aluminum Complexes as Catalysts for Enantioselective Aldol Reactions of Aldehydes and 5-Alkoxyoxazoles: An Efficient Approach to the Asymmetric Synthesis ofsyn andantiβ-Hydroxy-α-amino Acid Derivatives

Davidr . Evans, J. Tedrow, J. Janey, 2001 .

Design and Enabling Development of Hydroxyethylamine-Derived BACE1 Inhibitor

J. Tedrow, W. Zhong, 2016 .

Synergistic nitroreductase/vanadium catalysis enables chemoselective nitro reductions to anilines in the absence of hydrogen gas

Steven M. Mennen, Alan H. Cherney, J. Tedrow, 2022, Current Research in Chemical Biology.

Process Development and Protein Engineering Enhanced Nitroreductase-Catalyzed Reduction of 2-Methyl-5-nitro-pyridine

Steven M. Mennen, Alan H. Cherney, J. Tedrow, 2020 .

Building Complexity and Achieving Selectivity through Catalysis – Case Studies from the Pharmaceutical Pipeline

Matthew G. Beaver, J. Tedrow, R. P. Farrell, 2020, Synlett.

Development of sulfonamide compounds as potent methionine aminopeptidase type II inhibitors with antiproliferative properties.

Scott A. Erickson, K. Comess, A. Vasudevan, 2006, Bioorganic & medicinal chemistry letters.

Direct reductive amination of aldehyde bisulfite adducts induced by 2-picoline borane: application to the synthesis of a DPP-IV inhibitor.

M. Faul, J. Tedrow, R. Larsen, 2013, The Journal of organic chemistry.

Highly Regioselective Halogenation of Pyridine N-Oxide: Practical Access to 2-Halo-Substituted Pyridines.

J. Tedrow, T. Hwang, R. P. Farrell, 2015, Organic letters.

An efficient, regioselective amination of 3,5-disubstituted pyridine N-oxides using saccharin as an ammonium surrogate.

J. Tedrow, R. P. Farrell, M. S. Silva Elipe, 2013, Organic letters.

A General Method for the Synthesis of Enantiomerically Pure β-Substituted, β-Amino Acids through α-Substituted Succinic Acid Derivatives

John J. M. Wiener, Davidr . Evans, J. Tedrow, 1999 .

Magnesium halide-catalyzed anti-aldol reactions of chiral N-acylthiazolidinethiones.

Davidr . Evans, J. Tedrow, C. W. Downey, 2002, Organic letters.

Molecular Complexity as a Driver for Chemical Process Innovation in the Pharmaceutical Industry.

Steven M. Mennen, Sheng Cui, M. Faul, 2019, The Journal of organic chemistry.

New Conditions for the Synthesis of Thiophenes via the Knoevenagel/Gewald Reaction Sequence. Application to the Synthesis of a Multitargeted Kinase Inhibitor (X).

J. Tedrow, D. Barnes, Maureen A. McLaughlin, 2007 .

Reversal of diastereofacial selectivity in hydride reductions of N-tert-butanesulfinyl imines.

M. Faul, J. Tedrow, J. Colyer, 2006, The Journal of organic chemistry.

Xantphos as a Branch-Selective Ligand for the Acyclic sec-Alkyl Negishi Cross-Coupling of Heteroaryl Halides

Steven M. Mennen, Alan H. Cherney, J. Tedrow, 2018, Organometallics.

Copper-catalyzed N-arylation of sulfonamides with aryl bromides under mild conditions

M. Faul, J. Tedrow, M. Ronk, 2012 .

A General Method for the Synthesis of Enantiomerically Pure β‐Substituted, β‐Amino Acids Through α‐Substituted Succinic Acid Derivatives.

John J. M. Wiener, Davidr . Evans, J. Tedrow, 2000 .

Diastereoselective Magnesium Halide‐Catalyzed anti‐Aldol Reactions of Chiral N‐Acyloxazolidinones.

Davidr . Evans, J. Tedrow, C. W. Downey, 2002 .

Magnesium Halide Catalyzed anti-Aldol Reactions of Chiral N-Acylthiazolidinethiones.

Davidr . Evans, J. Tedrow, C. W. Downey, 2002 .

Highly enantioselective syntheses of homopropargylic alcohols and dihydrofurans catalyzed by a bis(oxazolinyl)pyridine-scandium triflate complex.

J. Tedrow, Z. Sweeney, D. Evans, 2001, Journal of the American Chemical Society.

Application of Chiral Mixed Phosphorus/Sulfur Ligands to Palladium-Catalyzed Allylic Substitutions

Davidr . Evans, J. Tedrow, M. R. Gagné, 2000 .

Enantioselective Lewis Acid Catalyzed Michael Reactions of Alkylidene Malonates. Catalysis by C2-Symmetric Bis(oxazoline) Copper(II) Complexes in the Synthesis of Chiral, Differentiated Glutarate Esters

Davidr . Evans, M. Kozlowski, J. Tedrow, 2000 .

C2-SYMMETRIC CU(II) COMPLEXES AS CHIRAL LEWIS ACIDS. CATALYTIC ENANTIOSELECTIVE MICHAEL ADDITION OF SILYLKETENE ACETALS TO ALKYLIDENE MALONATES

Davidr . Evans, M. Kozlowski, J. Tedrow, 1999 .

Highly enantioselective oxonium ylide formation and stevens rearrangement catalyzed by chiral Dirhodium(II) carboxamidates

David C. Forbes, D. C. Forbes, J. Tedrow, 1997 .

Highly selective rhodium-catalyzed conjugate addition reactions of 4-oxobutenamides.

M. Faul, J. Tedrow, Christopher J. Borths, 2007, The Journal of organic chemistry.

Application of chiral mixed phosphorus/sulfur ligands to enantioselective rhodium-catalyzed dehydroamino acid hydrogenation and ketone hydrosilylation processes.

Davidr . Evans, J. Tedrow, K. Campos, 2003, Journal of the American Chemical Society.

An aldol-based approach to the asymmetric synthesis of L-callipeltose, the deoxyamino sugar of L-callipeltoside A.

E. Hu, J. Tedrow, D. Evans, 2001, Organic letters.

Stereoselective synthesis of a MCHr1 antagonist.

M. Martinelli, R. Syed, J. Tedrow, 2007, The Journal of organic chemistry.

A highly enantioselective catalyst for asymmetric hydroformylation of [2.2.1]-bicyclic olefins

M. Martinelli, R. Syed, J. Tedrow, 2005 .

Route Selection and Process Development for the Vanilloid Receptor‐1 Antagonist AMG 517

J. Tedrow, O. Thiel, 2013 .

Development of a Robust and Highly Selective Ru(II)-Catalyzed Dynamic Kinetic Resolution Used to Manufacture AMG 232

J. Tedrow, K. Diker, J. Colyer, 2020 .

A Practical Preparation of Aryl β-Ketophosphonates.

M. Faul, J. Tedrow, R. Larsen, 2009 .

A practical preparation of aryl β-ketophosphonates

M. Faul, J. Tedrow, R. Larsen, 2009 .

Chiral Mixed Phosphorus/Sulfur Ligands for Palladium-Catalyzed Allylic Alkylations and Aminations.

Davidr . Evans, J. Tedrow, M. R. Gagné, 1999, The Journal of organic chemistry.

Accelerated Development of a Scalable Ring-Closing Metathesis to Manufacture AMG 176 Using a Combined High-Throughput Experimentation and Computational Modeling Approach

Yong Xie, Alan H. Cherney, Daniel J. Griffin, 2020 .

Hydrolysis of Phosphoryl Trichloride (POCl3): Characterization, in Situ Detection, and Safe Quenching of Energetic Metastable Intermediates

Michal M. Achmatowicz, J. Tedrow, Jack Hu, 2010 .

Chiral Salen ± Aluminum Complexes as Catalysts for Enantioselective Aldol Reactions of Aldehydes and 5-Alkoxyoxazoles : An Efficient Approach to the Asymmetric Synthesis of syn and anti b-Hydroxy-a-amino Acid Derivatives * *

J. Rebek, Davidr . Evans, J. Tedrow, 2001 .

Reductive Amination Without the Aldehyde: Use of a Ketolactol as an Aldehyde Surrogate

Pingli Liu, J. Tedrow, E. Bunel, 2014, Topics in Catalysis.

Lead optimization of methionine aminopeptidase-2 (MetAP2) inhibitors containing sulfonamides of 5,6-disubstituted anthranilic acids.

Gary T. Wang, Chang H. Park, Jieyi Wang, 2007, Bioorganic & medicinal chemistry letters.

Process development and manufacture of potassium 2-fluoro-6-hydroxyphenyltrifluoroborate

J. Tedrow, Lokesh Pawar, A. T. Parsons, 2019, Tetrahedron.

Synthesis of 2-deoxyxylolactone from glycerol derivatives via highly enantioselective carbon-hydrogen insertion reactions

J. Tedrow, M. Doyle, A. B. Dyatkin, 1994 .

Synthesis of 2-Deoxyxylolactone from Glycerol Derivatives via Highly Enantioselective Carbon-Hydrogen Insertion Reactions.

J. Tedrow, M. Doyle, A. B. Dyatkin, 1994 .

Chlorination at the 8-Position of a Functionalized Quinolone and the Synthesis of Quinolone Antibiotic ABT-492

M. J. Peterson, Elaine C. Lee, J. Tedrow, 2006 .

Development of a Commercial Manufacturing Process for Sotorasib, a First-in-Class KRASG12C Inhibitor

Alan H. Cherney, Matthew G. Beaver, Michael A. Lovette, 2022, Organic Process Research & Development.

Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors.

E. Lobenhofer, B. Herberich, A. Tasker, 2015, ACS Medicinal Chemistry Letters.

Enantioselective Syntheses of 2-Deoxyxylono-1,4-lactone and 2-Deoxyribono-1,4-lactone from 1,3-Dioxan-5-yl Diazoacetates.

J. Tedrow, M. Doyle, A. B. Dyatkin, 1999, The Journal of organic chemistry.