G. Verniest

发表

Synthesis and Reactivity of Spirocarbocycles as Scaffolds for Nucleoside Analogues.

F. De Proft, V. Pande, Jonas Verhoeven, 2020, The Journal of organic chemistry.

Mass spectrometry-based structure elucidation of small molecule impurities and degradation products in pharmaceutical development

Kris Laukens, Youzhong Liu, Thomas De Vijlder, 2019, TrAC Trends in Analytical Chemistry.

Synthesis of gem-difluorinated 1,6-naphthyridine-5,7-diones

J. Thuring, G. Verniest, F. Deroose, 2012 .

Regio- and Diastereoselective Functionalization of 3-Amino-hexahydrooxazoninones

J. Wouters, G. Verniest, C. Menet, 2018, European Journal of Organic Chemistry.

Azepinone-Constrained Amino Acids in Peptide and Peptidomimetic Design

G. Verniest, D. Tourwé, S. Ballet, 2015 .

Nucleophile-directed selective transformation of cis-1-tosyl-2-tosyloxymethyl-3-(trifluoromethyl)aziridine into aziridines, azetidines, and benzo-fused dithianes, oxathianes, dioxanes, and (thio)morpholines.

N. de Kimpe, K. Törnroos, G. Verniest, 2013, Chemistry.

Synthesis of 2-aryl-3-hydroxymethyl-5,5-difluoropiperidines

J. Thuring, G. Verniest, F. Deroose, 2012 .

Morpholinosulfur Trifluoride (Morph‐DAST)‐Mediated Rearrangement in the Fluorination of Cyclic α,α‐Dialkoxy Ketones toward 1,2‐Dialkoxy‐1,2‐difluorinated Compounds

J. Thuring, G. Verniest, N. Kimpe, 2010 .

Synthesis of aminomethylated 4-fluoropiperidines and 3-fluoropyrrolidines.

G. Macdonald, N. de Kimpe, J. Thuring, 2010, Organic & biomolecular chemistry.

Straightforward synthesis of 1-alkyl-2-(trifluoromethyl)aziridines starting from 1,1,1-trifluoroacetone.

N. de Kimpe, G. Verniest, M. D’hooghe, 2011, Organic & biomolecular chemistry.

Synthesis of substituted β-carbolines via gold(III)-catalyzed cycloisomerization of N-propargylamides

A. Padwa, G. Verniest, N. Kimpe, 2010 .

Regio- and stereocontrolled synthesis of novel 3-sulfonamido-2,3,4,5-tetrahydro-1,5-benzothiazepines from 2-(bromomethyl)- or 2-(sulfonyloxymethyl)aziridines.

N. de Kimpe, Michinori Karikomi, G. Verniest, 2008, Organic & biomolecular chemistry.

Synthesis of 3-amino-4-fluoropyrazoles.

N. de Kimpe, J. Thuring, G. Verniest, 2011, The Journal of organic chemistry.

Regio‐ and Stereocontrolled Synthesis of Novel 3‐Sulfonamido‐2,3,4,5‐tetrahydro‐1,5‐benzothiazepines from 2‐(Bromomethyl)‐ or 2‐(Sulfonyloxymethyl)aziridines.

Michinori Karikomi, G. Verniest, M. D’hooghe, 2008 .

New synthesis of 3-fluoropyrroles.

G. Macdonald, N. de Kimpe, J. Thuring, 2009, The Journal of organic chemistry.

New synthesis of fluorinated pyrazoles.

N. de Kimpe, G. Verniest, Riccardo Surmont, 2010, Organic letters.

Direct electrophilic alpha-fluorination of imines: efficient synthesis of mono- and difluoroimines.

N. de Kimpe, G. Verniest, Riccardo Surmont, 2006, Organic letters.

Gold-catalyzed synthesis of 2-aryl-3-fluoropyrroles.

N. de Kimpe, G. Verniest, Riccardo Surmont, 2009, Organic letters.

Synthesis and reactivity of 1-substituted 2-fluoro- and 2,2-difluoroaziridines.

N. de Kimpe, G. Verniest, F. Colpaert, 2007, The Journal of organic chemistry.

Synthesis of 3-substituted 2-fluoro- and 2,2-difluoroaziridines.

N. de Kimpe, G. Verniest, Riccardo Surmont, 2007, Organic letters.

Synthesis of 2-Fluoro-1,4-benzoxazines and 2-Fluoro-1,4-benzoxazepin-5-ones by Exploring the Nucleophilic Vinylic Substitution (S(N)V) Reaction of gem-Difluoroenamides.

Sven Mangelinckx, N. de Kimpe, G. Verniest, 2015, The Journal of organic chemistry.

Improved Arndt-Eistert synthesis of alpha-diazoketones requiring minimal diazomethane in the presence of calcium oxide as acid scavenger.

A. Alcántara, J. Sinisterra, N. de Kimpe, 2010, The Journal of organic chemistry.

Synthesis of 1-alkyl-2-methylazetidin-3-ones and 1-alkyl-2-methylazetidin-3-ols

G. Verniest, A. Salgado, N. Kimpe, 2003 .

Gold- and silver-mediated cycloisomerizations of N-propargylamides.

A. Padwa, G. Verniest, 2008, Organic letters.

Synthesis of 4-substituted 3,3-difluoropiperidines.

G. Macdonald, N. de Kimpe, J. Thuring, 2010, Journal of Organic Chemistry.

Reductive amination of 4 , 5-dimethoxy-9 , 10-dioxo-9 , 10-dihydroanthracene-2-carbaldehyde derived from aloe-emodin Aminación reductiva del 4 , 5-dimetoxi-9 , 10-dioxo-9 , 10-dihidroantraceno-2-carbaldehído derivado de aloe-emodin

G. Verniest, MSc. Yennys Hernández-Molina, DraC. Magaly Casals-Hung, 2019 .

Asymmetric synthesis of alpha-alkylated N-sulfinyl imidates as new chiral building blocks.

Sven Mangelinckx, N. de Kimpe, G. Verniest, 2009, The Journal of organic chemistry.

Synthesis of chlorinated 2-(aminomethyl)- and 2-(alkoxymethyl)pyrroles

G. Verniest, N. Kimpe, S. Claessens, 2005 .

Gold(I)-catalyzed synthesis of dihydrodibenzoquinolizinium salts

G. Verniest, Niels Marien, 2017 .

The behaviour of the natural pyranonaphthoquinone pentalongin in alcoholic solvents

G. Verniest, N. Kimpe, B. Kesteleyn, 2006 .

Synthesis of 2-spiropseudoindoxyls via an intramolecular nitroalkyne redox-dipolar cycloaddition cascade.

G. Verniest, B. Pinter, Ben Brigou, 2015, Organic letters.

Chemoselective Synthesis of N-Substituted α-Amino-α′-chloro Ketones via Chloromethylation of Glycine-Derived Weinreb Amides

A. Alcántara, G. Verniest, Vittorio Pace, 2013 .

Synthesis of Heterocycle‐Bridged Peptidic Macrocycles through 1,3‐Diyne Transformations

G. Verniest, S. Ballet, S. Verlinden, 2016 .

Synthesis of Substituted β-Carbolines via Gold(III)-Catalyzed Cycloisomerization of N-Propargylamides.

A. Padwa, G. Verniest, N. Kimpe, 2010 .

Synthesis of 2-aryl-4-chloropyrroles via ring expansion of 2-aryl-1-chlorocyclopropanecarbaldehydes

G. Verniest, N. Kimpe, T. V. Thienen, 2005 .

New synthesis of fluorinated pyrazoles.

N. de Kimpe, G. Verniest, Riccardo Surmont, 2010, Organic letters.

Synthesis of fused 3-aminoazepinones via trapping of a new class of cyclic seven-membered allenamides with furan.

G. Verniest, D. Tourwé, G. Van Lommen, 2014, Organic letters.

Total synthesis of four naturally occurring 2-azaanthraquinone antibiotics, 6-deoxy-8-methylbostrycoidin, 6-deoxybostrycoidin, 7-O-demethyl-6-deoxybostrycoidin and scorpinone

G. Verniest, N. Kimpe, S. Claessens, 2005 .

Synthesis and Selective N,O-Functionalization of Pyrazolone-Fused 3-Aminoazepinones

G. Verniest, G. Lommen, Ben Schurgers, 2015 .

Synthesis of 5-amino- and 5-hydroxy-3,3-difluoropiperidines.

N. de Kimpe, J. Thuring, G. Verniest, 2010, Organic & biomolecular chemistry.

Metal-Free Cyclization of ortho-Nitroaryl Ynamides and Ynamines towards Spiropseudoindoxyls.

G. Verniest, K. Van Hecke, S. Goderis, 2018, Angewandte Chemie.

Synthesis of 2-Substituted Cyclobutanones as γ-Irradiation Marker Products of Lipid-Containing Foods

C. Stevens, G. Verniest, N. Kimpe, 2004 .

Heteroaryl cross-coupling as an entry toward the synthesis of lavendamycin analogues: a model study.

N. de Kimpe, A. Padwa, G. Verniest, 2010, The Journal of organic chemistry.

Synthesis of 1-alkyl-2-(trifluoromethyl)azetidines and their regiospecific ring opening toward diverse α-(trifluoromethyl)amines via intermediate azetidinium salts.

N. de Kimpe, G. Verniest, M. D’hooghe, 2012, The Journal of organic chemistry.

A Benchmark of Density Functional Approximations For Thermochemistry and Kinetics of Hydride Reductions of Cyclohexanones

X. Deraet, M. Alonso, G. Verniest, 2019, ChemistryOpen.

Synthesis and transformations of pyrrolo[1,2-a][1,3,5]-triazines

Jonas Verhoeven, L. Meerpoel, J. Thuring, 2018, Tetrahedron Letters.

Stereoselective reduction of N-(3-arylcyclobutylidene)amines

G. Verniest, N. Kimpe, S. Claessens, 2006 .

Stereoselective Reductions of 3-Substituted Cyclobutanones: a Comparison Between Experiment and Theory.

X. Deraet, M. Alonso, G. Verniest, 2020, The Journal of organic chemistry.

Preparation of 4'-Spirocyclobutyl Nucleoside Analogues as Novel and Versatile Adenosine Scaffolds.

V. Pande, Jonas Verhoeven, Weimei Sun, 2019, Chemistry.

Regio- and Stereoselective Synthesis of C-4' Spirocyclobutyl Ribofuranose Scaffolds and Their Use as Biologically Active Nucleoside Analogues.

Jonas Verhoeven, L. Meerpoel, J. Thuring, 2021, Organic letters.

Stereodivergent Synthesis of Biologically Active Spironucleoside Scaffolds via Catalytic Cyclopropanation of 4-exo-Methylene Furanosides.

Jonas Verhoeven, L. Meerpoel, J. Thuring, 2021, The Journal of organic chemistry.

Synthesis of Cyclopropyl Pinacol Boronic Esters from Dibromocyclopropanes

Jonas Verhoeven, L. Meerpoel, J. Thuring, 2022, Synlett.

Preparation of Novel 4′-Spirocyclopropyl Nucleoside Analogues

V. Pande, Jonas Verhoeven, L. Meerpoel, 2021, Synlett.

Four-membered heterocycles with a carbon-heteroatom exocyclic double bond at the 3-position: puckering potential and thermodynamic properties.

Michel Waroquier, N. de Kimpe, V. Van Speybroeck, 2007, The journal of physical chemistry. A.

Towards the Design of Optically Active Thiophene S-Oxides using Quantum Chemistry.

M. Alonso, G. Verniest, T. Woller, 2019, Chemistry.

The 1,3‐diyne linker as a rigid “i,i+7” staple for α‐helix stabilization: Stereochemistry at work

J. Martins, G. Verniest, S. Ballet, 2019, Journal of peptide science : an official publication of the European Peptide Society.

Oxidative α,ω-diyne coupling as an approach towards novel peptidic macrocycles.

J. Martins, G. Verniest, D. Tourwé, 2015, Organic & biomolecular chemistry.

New synthesis of semisquaric acid derivatives via chlorinated N-(cyclobutylidene)amines.

N. de Kimpe, K. Törnroos, G. Verniest, 2005, Journal of Organic Chemistry.

New Synthesis of Semisquaric Acid Derivatives via Chlorinated N‐(Cyclobutylidene)amines.

G. Verniest, N. Kimpe, K. Toernroos, 2005 .

The antibacterial prodrug activator Rv2466c is a mycothiol-dependent reductase in the oxidative stress response of Mycobacterium tuberculosis

L. M. Mateos, W. Versées, E. Sancho-Vaello, 2017, The Journal of Biological Chemistry.

Synthesis of 1-Boc-3-fluoroazetidine-3-carboxylic acid.

G. Macdonald, N. de Kimpe, J. Thuring, 2009, The Journal of organic chemistry.

Synthesis of 3-fluoroazetidines.

N. de Kimpe, G. Verniest, G. Duvey, 2006, The Journal of organic chemistry.

Short synthesis of the seed germination inhibitor 3,4,5-trimethyl-2(5H)-furanone.

N. de Kimpe, G. Verniest, Riccardo Surmont, 2010, The Journal of organic chemistry.

Insight into the solvation and isomerization of 3-halo-1-azaallylic anions from ab initio metadynamics calculations and NMR experiments.

T. Verstraelen, Sven Mangelinckx, N. de Kimpe, 2009, Chemistry.

A Survey of Synthetic Routes towards the Pyranonaphthoquinone Antibiotic Pentalongin and Syntheses of the Corresponding Nitrogen Derivatives

G. Verniest, J. Jacobs, N. Kimpe, 2007 .

New entries toward 3,3-difluoropiperidines.

J. Thuring, G. Verniest, Riccardo Surmont, 2008, The Journal of organic chemistry.

Oxidative α,ω-diyne coupling as an approach towards novel peptidic macrocycles.

G. Verniest, D. Tourwé, S. Ballet, 2015, Organic & biomolecular chemistry.

Efficient Synthesis of 3-Alkoxy-4,4-difluoropiperidines

G. Macdonald, J. Thuring, G. Verniest, 2009 .

Synthesis of 4-substituted 3,3-difluoropiperidines.

G. Macdonald, J. Thuring, G. Verniest, 2010, The Journal of organic chemistry.

Synthesis of 5-amino- and 5-hydroxy-3,3-difluoropiperidines.

J. Thuring, G. Verniest, Riccardo Surmont, 2010, Organic & biomolecular chemistry.