E. Gjerstad

In Vitro ADME Profiling Using High-Throughput RapidFire Mass Spectrometry

Lory R Tan, Xiang Wu, Jing Wang, 2012, Journal of biomolecular screening.

Synthesis of a statistically exhaustive fluorescent peptide substrate library for profiling protease specificity.

J. Janc, E. Gjerstad, J. Wheatley, 2000, Bioorganic & medicinal chemistry letters.

Expression and characterization of recombinant ?-tryptase

J. Janc, E. Gjerstad, H. Chan, 2006 .

Factor VIIa inhibitors: improved pharmacokinetic parameters.

J. Janc, Liang Liu, B. Katz, 2006, Bioorganic & medicinal chemistry letters.

Potent 4-amino-5-azaindole factor VIIa inhibitors.

E. Gjerstad, E. Leahy, P. Sprengeler, 2006, Bioorganic & medicinal chemistry letters.

Structure-guided design of peptide-based tryptase inhibitors.

Yang Liu, James W Janc, J. R. Somoza, 2006, Biochemistry.

Optimization of subsite binding to the beta5 subunit of the human 20S proteasome using vinyl sulfones and 2-keto-1,3,4-oxadiazoles: syntheses and cellular properties of potent, selective proteasome inhibitors.

J. Palmer, R. Rydzewski, Leland C. Burrill, 2006, Journal of medicinal chemistry.

Dissecting and designing inhibitor selectivity determinants at the S1 site using an artificial Ala190 protease (Ala190 uPA).

Erik Verner, James W Janc, J. R. Somoza, 2004, Journal of Molecular Biology.