Ann C. Petersen

发表

DNA Compatible Multistep Synthesis and Applications to DNA Encoded Libraries.

L. Orzechowski, R. Goodnow, A. Satz, 2015, Bioconjugate chemistry.

Analysis of Current DNA Encoded Library Screening Data Indicates Higher False Negative Rates for Numerically Larger Libraries.

A. Satz, Ann C. Petersen, R. Hochstrasser, 2017, ACS combinatorial science.

Metabotropic glutamate receptor 5 negative allosteric modulators: discovery of 2-chloro-4-[1-(4-fluorophenyl)-2,5-dimethyl-1H-imidazol-4-ylethynyl]pyridine (basimglurant, RO4917523), a promising novel medicine for psychiatric diseases.

W. Guba, W. Spooren, J. Peters, 2015, Journal of medicinal chemistry.

A Multifaceted Hit-Finding Approach Reveals Novel LC3 Family Ligands.

Melinda M. Mulvihill, D. Stoffler, M. Holliday, 2022, Biochemistry.

DNA-Encoded Library-Derived DDR1 Inhibitor Prevents Fibrosis and Renal Function Loss in a Genetic Mouse Model of Alport Syndrome

B. Kuhn, M. Rudolph, M. Prunotto, 2018, ACS chemical biology.

Evaluation of secondary amide replacements in a series of CCR5 antagonists as a means to increase intrinsic membrane permeability. Part 1: Optimization of gem-disubstituted azacycles.

Jutta Wanner, L. Setti, D. Rotstein, 2010, Bioorganic & medicinal chemistry letters.

Scaffold hopping towards potent and selective JAK3 inhibitors: discovery of novel C-5 substituted pyrrolopyrazines.

Johannes C. Hermann, A. Kuglstatter, A. Lovey, 2014, Bioorganic & medicinal chemistry letters.

Fragment-Based Drug Design of Novel Pyranopyridones as Cell Active and Orally Bioavailable Tankyrase Inhibitors.

Johannes C. Hermann, D. Carvajal, C. Lukacs, 2015, ACS medicinal chemistry letters.

Development of DNA-Compatible Van Leusen Three-Component Imidazole Synthesis.

A. Satz, Ann C. Petersen, Stefanie N. Geigle, 2019, Organic letters.

Exploration of a new series of CCR5 antagonists: multi-dimensional optimization of a sub-series containing N-substituted pyrazoles.

L. Setti, D. Rotstein, Ann C. Petersen, 2010, Bioorganic & medicinal chemistry letters.

Metal impurities cause false positives in high-throughput screening campaigns.

Stephen Gabriel, Binh Vu, Johannes C. Hermann, 2013, ACS medicinal chemistry letters.