J. Praly

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Inhibition of glycogen phosphorylase in the context of type 2 diabetes, with focus on recent inhibitors bound at the active site.

J. Praly, S. Vidal, 2010, Mini reviews in medicinal chemistry.

Synthesis of a C-glucosylated cyclopropylamide and evaluation as a glycogen phosphorylase inhibitor.

E. Jeanneau, J. Praly, S. Vidal, 2008, Bioorganic & medicinal chemistry letters.

Stereoselective Synthesis of Enantiopure Cycloalkylglycines by 1,3-Dipolar Cycloaddition of a Chiral Nitrone to Cycloalkenes

J. Praly, S. Vidal, L. Perrin, 2014 .

Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors.

S. Zographos, N. Oikonomakos, D. Leonidas, 2009, Bioorganic & medicinal chemistry.

Photohalogenation of glycopyranosyl halides: An expedient route to c-1 gem dihalogenated sugars

J. Praly, L. Toupet, L. Brard, 1989 .

NaBH3CN: A Janus Substitute for Tin-Free Radical-Based Reactions

J. Praly, J. Guiard, Yaniss Rahali, 2014 .

NaBH3CN and other systems as substitutes of tin and silicon hydrides in the light or heat-initiated reduction of halosugars: a tunable access to either 2-deoxy sugars or 1,5-anhydro-itols

J. Praly, Z. Toth, Isabelle Bruyère, 2013 .

Glycoarray by DNA-directed immobilization.

J. Vasseur, J. Praly, S. Vidal, 2012, Methods in molecular biology.

Measurement of Enzymatic Activity and Specificity of Human and Avian Influenza Neuraminidases from Whole Virus by Glycoarray and MALDI‐TOF Mass Spectrometry

V. Moulés, B. Lina, O. Ferraris, 2011, Chembiochem : a European journal of chemical biology.

Specific recognition of lectins by oligonucleotide glycoconjugates and sorting on a DNA microarray.

J. Vasseur, J. Praly, S. Vidal, 2009, Chemical communications.

In Search of Glycogen Phosphorylase Inhibitors: 5-Substituted 3-C-Glucopyranosyl-1,2,4-oxadiazoles from β-D-Glucopyranosyl Cyanides upon Cyclization of O-Acylamidoxime Intermediates

J. Praly, S. Vidal, Mahmoud Benltifa, 2006 .

Efficient atropodiastereoselective access to 5,5'-bis-1,2,3-triazoles: studies on 1-glucosylated 5-halogeno 1,2,3-triazoles and their 5-substituted derivatives as glycogen phosphorylase inhibitors.

E. Chrysina, J. Praly, S. Vidal, 2014, Chemistry.

Photolysis of glycopyranosyl azides C-1 substituted by cyano-, amido-, or tetrazolyl-groups

L. Somsák, J. Praly, C. D. Stefano, 2000 .

Multiplexed binding determination of seven glycoconjugates for Pseudomonas aeruginosa lectin I (PA-IL) using a DNA-based carbohydrate microarray.

J. Vasseur, J. Praly, S. Vidal, 2011, Chemical communications.

Synthesis of lactosylated glycoclusters and inhibition studies with plant and human lectins.

A. Imberty, S. E. Matthews, H. Blanchard, 2012, Carbohydrate research.

Probing multivalency for the inhibition of an enzyme: glycogen phosphorylase as a case study

J. Praly, S. Vidal, T. Docsa, 2009 .

1,3-Dipolar cycloaddition reactions on carbohydrate-based templates: synthesis of spiro-isoxazolines and 1,2,4-oxadiazoles as glycogen phosphorylase inhibitors

J. Praly, S. Vidal, Mahmoud Benltifa, 2006 .

Fucosylated pentaerythrityl phosphodiester oligomers (PePOs): automated synthesis of DNA-based glycoclusters and binding to Pseudomonas aeruginosa lectin (PA-IIL).

A. Imberty, J. Vasseur, J. Praly, 2007, Bioconjugate chemistry.

Variations on the SnCl4 and CF3CO2Ag-promoted glycosidation of sugar acetates: a direct, versatile and apparently simple method with either alpha or beta stereocontrol.

J. Praly, S. Vidal, Samy Cecioni, 2009, Carbohydrate research.

Towards α- or β-d-C-glycosyl compounds by tin-catalyzed addition of glycosyl radicals to acrylonitrile and vinylphosphonate, and flexible reduction of tetra-O-acetyl-α-d-glucopyranosyl bromide with cyanoborohydride

J. Praly, Isabelle Bruyère, B. Qin, 2002 .

Synthesis of peracetylated d-galactopyranosylidene dihalides

J. Klett, J. Praly, Jean-Charles Brendlé, 2001 .

C-Glycopyranosyl Arenes and Hetarenes: Synthetic Methods and Bioactivity Focused on Antidiabetic Potential.

L. Somsák, M. Tóth, É. Bokor, 2017, Chemical reviews.

Microwave assisted "click" chemistry for the synthesis of multiple labeled-carbohydrate oligonucleotides on solid support.

J. Vasseur, J. Praly, S. Vidal, 2006, The Journal of organic chemistry.

Selectivity among two lectins: probing the effect of topology, multivalency and flexibility of "clicked" multivalent glycoclusters.

A. Imberty, M. Wimmerová, J. Praly, 2011, Chemistry.

3-Glucosylated 5-amino-1,2,4-oxadiazoles: synthesis and evaluation as glycogen phosphorylase inhibitors

J. Praly, S. Vidal, D. Goyard, 2015, Beilstein journal of organic chemistry.

Synthesis of 1,2,3-triazoles from xylosyl and 5-thioxylosyl azides: evaluation of the xylose scaffold for the design of potential glycogen phosphorylase inhibitors.

E. Chrysina, J. Praly, S. Vidal, 2012, Carbohydrate research.

DNA-based carbohydrate biochips: a platform for surface glyco-engineering.

J. Vasseur, J. Praly, S. Vidal, 2007, Angewandte Chemie.

Synthesis of dodecavalent fullerene-based glycoclusters and evaluation of their binding properties towards a bacterial lectin.

A. Imberty, J. Praly, S. Vidal, 2011, Chemistry.

Synthesis of azido-functionalized carbohydrates for the design of glycoconjugates.

J. Praly, S. Vidal, D. Goyard, 2012, Methods in molecular biology.

Naphthyl Thio- and Carba-xylopyranosides for Exploration of the Active Site of β-1,4-Galactosyltransferase 7 (β4GalT7).

Daniel P. Willen, Magnus T. Johnson, Jonas Ståhle, 2017, Chemistry.

1,3-Dipolar cycloaddition of a chiral nitrone to (E)-1,4-dichloro-2-butene: a new efficient synthesis of (2S,3S,4R)-4-hydroxyisoleucine

E. Jeanneau, J. Praly, M. Msaddek, 2012 .

Non-isosteric C-glycosyl analogues of natural nucleotide diphosphate sugars as glycosyltransferase inhibitors.

J. Praly, S. Vidal, C. Augé, 2006, Bioorganic & medicinal chemistry.

Free-radical and ionic routes towards hydrolytically stable and bioactive C-glycosyl compounds

J. Praly, Guorong Chen, 2008 .

Structure of anomeric glycosyl radicals and their transformations under reductive conditions.

J. Praly, 2000, Advances in carbohydrate chemistry and biochemistry.

Multi-Step Synthesis and Biological Evaluation of Analogues of Insulin Secretagogue (2S,3R,4S)-4-Hydroxyisoleucine

J. Praly, R. Gross, A. Lajoix, 2008 .

Synthetic studies in the 5-thio-D-xylopyranose series part 1 : A ready access to C -hetaryl 5-thio-D-xylopyranosides by electrophilic substitution

R. Faure, J. Praly, G. Descotes, 1998 .

Novel routes to either racemic or enantiopure α-amino-(4-hydroxy-pyrrolidin-3-yl)acetic acid derivatives and biological evaluation of a new promising pharmacological scaffold.

J. Ghersi-Egea, L. Denoroy, S. Parrot, 2015, European journal of medicinal chemistry.

Synthetic studies in the 5-thio-D-xylopyranose series part 2: Coupling of 5-thio-D-xylopyranosyl donors with electron-rich aryl moieties: Access to C-aryl 5-thio-D-xylopyranosides

J. Praly, G. Descotes, V. Barberousse, 1998 .

Radical-mediated bromination of peracetylated 5-thio-d-xylopyranosyl bromides: an easy access to the corresponding anomeric orthothiolactones

J. Praly, M. Bouchu, G. Descotes, 1996 .

An unprecedented access to trifluoromethylthiosugar derivatives from thiocyanate precursors upon treatment with trifluoromethyltrimethylsilane

B. Langlois, J. Praly, M. Bouchu, 1998 .

New 1-C-(5-thio-D-xylopyranosyl) derivatives as potential orally active venous antithrombotics.

J. Praly, B. Boubia, V. Barberousse, 2003, Carbohydrate research.

Synthesis of C-1 spirocyclopropyl sugars from anomeric diazides.

J. Praly, G. Descotes, Z. E. Kharraf, 1990 .

Synthesis, structure and enzymatic evaluation of new spiro oxathiazole sugar derivatives

R. Faure, J. Praly, B. Joseph, 1994 .

beta-D-Galactopyranosyl-thiohydroximates and D-galactopyranosylidene-spiro-oxathiazoles: synthesis and enzymatic evaluation against E. colid-galactosidase.

L. Somsák, J. Praly, L. Kiss, 2005, Carbohydrate research.

Glucose-based spiro-heterocycles as potent inhibitors of glycogen phosphorylase.

G. Batta, L. Somsák, K. Czifrák, 2009, Bioorganic & medicinal chemistry.

Stereoselective synthesis of 1,2,3-triazolyl-functionalized isoxazolidines, via two consecutive 1,3-dipolar cycloadditions, as precursors of unnatural amino acids

J. Praly, S. Vidal, M. Msaddek, 2013 .

Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase.

Eva Bokor, L. Somsák, M. Tóth, 2009, Bioorganic & medicinal chemistry.

Cycloaddition of a chiral nitrone to allylic motifs: an access to enantiopure sugar-based amino acids displaying a stable glycosidic bond and to 4(S)-4-hydroxy-l-ornithine

J. Praly, M. Msaddek, Kaïss Aouadi, 2012 .

Photolysis of methyl 1-azido glucosides : unprecedented expansions of the pyranose ring under high stereocontrol

J. Praly, G. Descotes, C. D. Stefano, 1994 .

Photolysis of sugar anomeric diazides: Sugar-derived tetrazoles as evidences for a major nitrene decomposition pathway

R. Faure, J. Praly, G. Descotes, 1994 .

Synthesis of (benzimidazol-2-yl)aniline derivatives as glycogen phosphorylase inhibitors.

E. Chrysina, J. Praly, F. Ragab, 2016, Bioorganic & medicinal chemistry.

Novel cyclization of D-glucopyranosyl-(Z)-thiohydroximates leading to new anomeric spiro oxathiazole derivatives

J. Praly, B. Joseph, P. Rollin, 1993 .

A Cycloaddition–Cyclization Combined Approach to Enantiopure 3‐Glycinyl‐4‐hydroxypyrrolidines and 3‐Substituted 4‐Hydroxyprolines

J. Praly, Juliane Abdoul-Zabar, M. Msaddek, 2014 .

Stereocontrolled Access to Higher Sugars (Non‐1‐en‐4‐ulopyranosyl Derivatives) and Glycomimetics [3‐(β‐D‐Glycopyranosyl)‐1‐propenes and(3Z)‐4,8‐Anhydro‐nona‐1,3‐dienitols]

Joelle M. R. Gola, J. Praly, Guorong Chen, 2000 .

In the search of glycogen phosphorylase inhibitors : Synthesis of C-D-glycopyranosylbenzo (hydro )quinones-inhibition of and binding to glycogen phosphorylase in the crystal

N. Oikonomakos, D. Leonidas, E. Chrysina, 2007 .

Conversion of glycosyl azides via N-bromoglycosylimines to aldononitriles

A. Fürstner, J. Praly, 1994 .

A stereocontrolled radical access to C-allyl β-D-glycopyranosides from glycopyranosylidene dihalides found en route to C-glycodienes

Joelle M. R. Gola, J. Praly, Guorong Chen, 1997 .

N-Bromosuccinimide-Mediated Transformation of Acetylated 1,5-Anhydro-1-C-phenyl-d-hexitols

J. Praly, G. Descotes, P. Cettour, 1995 .

Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition.

D. Tousch, L. Somsák, E. Chrysina, 2016, European journal of medicinal chemistry.

Synthesis and some transformations of 1-azido-glycopyranosyl cyanides-precursors of anomeric α-amino acids

L. Somsák, J. Praly, Z. Györgydeák, 1996 .

Preparation and photolysis of 1-cyano-glycopyranosyl azides

R. Faure, L. Somsák, J. Praly, 1995 .

Syntheses of “anomeric” gem dihalogenated glucopyranosyl derivatives

J. Praly, G. Descotes, 1987 .

Structure of C-1 substituted glycopyranosyl azides: new insights based on CD measurements

Z. Majer, M. Hollósi, L. Somsák, 1999 .

Structural Identification of Substituted C-1 Spiro Cyclopropyl Sugars.

R. Faure, J. Praly, B. Fenet, 1991 .

Reduction stereoselective d'halogenures de glycosyles par le deuteriure de tributyletain

J. Praly, 1983 .

Glucose-based spiro-oxathiazoles as in vivo anti-hyperglycemic agents through glycogen phosphorylase inhibition.

D. Tousch, L. Somsák, K. Czifrák, 2020, Organic & biomolecular chemistry.

Synthetic studies in the 5-thio-d-xylopyranose seriespart 3: Preparations ofO-phenyl andC-(4-hydroxyphenyl) 5-thio-d-xylopyranosides

J. Praly, G. Descotes, S. Samreth, 1998 .

Conformation of C‐1‐Substituted Pyranos‐1‐yl and Pyranosan‐5‐yl Radicals Evidence for a Quasi‐Homo‐Anomeric Stabilization Effect

L. Somsák, J. Praly, H. Korth, 1990 .

Free radical-mediated addition of peracetylated 1-bromo-β-d-glucopyranosyl chloride to acrylonitrile

J. Praly, G. Descotes, Z. E. Kharraf, 1992 .

Ring‐Closing Olefin Metathesis of 3,3′‐(D‐Glycopyranosylidene)bis(1‐propene) Compounds as a Route to Anomeric Spiro Sugars

Joelle M. R. Gola, J. Praly, Guorong Chen, 2001 .

A stereoselective method for the synthesis of enantiopure 3-substituted 4-hydroxyproline derivatives via 1,3-dipolar cycloadditions

J. Praly, S. Vidal, M. Msaddek, 2016 .

Synthesis and photolysis of protected d-hex-2-ulopyranosyl azides

Pete Haug, J. Praly, G. Descotes, 1996 .

A New Sugar-Derived Tetrahydrothiazepine Obtained by Thermolysis from Peracetylated 5-Thio-D-Xylopyranosyl Azides

J. Praly, G. Hetzer, Michaela Steng, 1999 .

Radical-Mediated Halogenations of Anomerically N-Substituted Glucopyranosyl Derivatives

L. Somsák, J. Praly, G. Descotes, 1992 .

Achieving high affinity towards a bacterial lectin through multivalent topological isomers of calix[4]arene glycoconjugates.

A. Imberty, S. E. Matthews, Ruth Lalor, 2009, Chemistry.

Synthesis of 4-amidomethyl-1-glucosyl-1,2,3-triazoles and evaluation as glycogen phosphorylase inhibitors.

J. Praly, S. Vidal, D. Goyard, 2015, Carbohydrate research.

Rational design and synthesis of optimized glycoclusters for multivalent lectin-carbohydrate interactions: influence of the linker arm.

Michaela Wimmerová, Anne Imberty, Susan E Matthews, 2012, Chemistry.

CuAAC synthesis of resorcin[4]arene-based glycoclusters as multivalent ligands of lectins.

A. Imberty, S. E. Matthews, H. Blanchard, 2011, Organic & biomolecular chemistry.

AFM investigation of Pseudomonas aeruginosa lectin LecA (PA-IL) filaments induced by multivalent glycoclusters.

A. Imberty, S. E. Matthews, D. Sicard, 2011, Chemical communications.

Identification and synthesis of a trisaccharide produced from lactose by transgalactosylation.

J. Praly, B. Fenet, F. Lecroix, 2000, Carbohydrate research.

Synthesis and structure of bromo glycosyl imines readily obtained from protected glycosyl azides

J. Praly, G. Descotes, R. Faure, 1995 .

Synthesis of ν-triazole derivatives from anomeric sugar diazides

J. Kovács, J. Praly, I. Pintér, 1999 .

Unexpected transformation of 2,3,4,6-tetra-O-acetyl-d-glucopyranosylidene 1,1-diazide with triphenylphosphine

J. Kovács, J. Praly, I. Pintér, 1995 .

Mass spectrometric studies of anomeric glycopyranosyl azides.

P. Benke, L. Somsák, J. Praly, 2001, Journal of mass spectrometry : JMS.

Influence of solvent on the magnitude of the anomeric effect

J. Praly, R. Lemieux, R. U. Lemieux, 1987 .

Sugar bromoimino derivatives: New sugar derivatives readily prepared from β-D-glycosyl azides

L. Somsák, J. Praly, G. Descotes, 1992 .

An Unprecedented Practical Preparation of Protected Aldonolactones

J. Praly, Djennane Senni, 1998 .

An improved synthesis of an umbelliferyl 5-thioxylopyranoside, precursor of the antithrombotic drug Iliparcil.

J. Praly, G. Descotes, V. Barberousse, 1999, Carbohydrate research.

N-(4-Substituted-benzoyl)-N'-(β-d-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods.

S. Zographos, N. Oikonomakos, D. Leonidas, 2012, Bioorganic & Medicinal Chemistry.

Analogues of insulin secretagogue (2S,3R,4S)-4-hydroxyisoleucine: synthesis by 1,3-dipolar cycloaddition reactions of chiral nitrones to alkenes

E. Jeanneau, J. Praly, M. Msaddek, 2008 .

Novel design principle validated: glucopyranosylidene-spiro-oxathiazole as new nanomolar inhibitor of glycogen phosphorylase, potential antidiabetic agent.

L. Somsák, K. Czifrák, J. Praly, 2008, Bioorganic & medicinal chemistry letters.

C‐D‐Glucopyranosyl Derivatives of Tocopherols – Synthesis and Evaluation as Amphiphilic Antioxidants

O. Dangles, C. Dufour, J. Praly, 2008 .

Sodium Salt of D-Glucono-1,5-lactone Tosylhydrazone: A Ready Access to a New Glucosylidene Carbene Precursor

L. Somsák, J. Praly, G. Descotes, 1992 .

C-Glycopyranosyl-1,4-benzoquinones and -hydroquinones opening access to C-glycosylated analogs of vitamin E

J. Praly, Guorong Chen, B. Qin, 2005 .

Synthesis and spectroscopic studies of acetylated alkyl 1-azido-D-glucopyranosides

R. Faure, J. Praly, M. Bouchu, 1993 .

C-Glucosylated malonitrile as a key intermediate towards carbohydrate-based glycogen phosphorylase inhibitors.

C. Potamitis, P. Zoumpoulakis, M. Zervou, 2012, Bioorganic & medicinal chemistry.

DNA-directed immobilisation of glycomimetics for glycoarrays application: comparison with covalent immobilisation, and development of an on-chip IC50 measurement assay.

J. Vasseur, J. Praly, S. Vidal, 2009, Biosensors & bioelectronics.

Binding of N‐acetyl‐N ′‐β‐d‐glucopyranosyl urea and N‐benzoyl‐N ′‐β‐d‐glucopyranosyl urea to glycogen phosphorylase b

B. Tóth, S. Zographos, N. Oikonomakos, 2002 .

Binding of N-acetyl-N '-beta-D-glucopyranosyl urea and N-benzoyl-N '-beta-D-glucopyranosyl urea to glycogen phosphorylase b: kinetic and crystallographic studies.

B. Tóth, S. Zographos, N. Oikonomakos, 2002, European journal of biochemistry.

Unprecedented Synthesis of 4‐Ylidene (3 S)‐3‐hydroxy‐1‐aryl (alkyl)‐pyrrolidine‐2,5‐diones Based on 1,3‐Dipolar Cycloaddition of a Sugar‐derived Nitrone toN‐Substituted Maleimides

J. Praly, M. Msaddek, S. Ghannay, 2019, ChemistrySelect.

New synthetic routes toward enantiopure (2S,3R,4R ) -4 -hydroxyisoleucine by 1,3-dipolar cycloaddition of a chiral nitrone to C4 alkenes

E. Jeanneau, J. Praly, M. Msaddek, 2007 .

Cycloadditions of Chiral Nitrones to Racemic 3-Substituted Butenes: A Direct Access with Kinetic Resolution to Enantiopure Dihydroxylated Amino Acids

J. Praly, S. Vidal, M. Msaddek, 2006 .

Synthesis of 5-halogenated 1,2,3-triazoles under stoichiometric Cu(I)-mediated azide-alkyne cycloaddition (CuAAC or 'Click Chemistry').

J. Praly, S. Vidal, D. Goyard, 2012, Carbohydrate Research.

Binding evaluation of fragment-based scaffolds for probing allosteric enzymes.

J. Praly, J. Lancelin, I. Krimm, 2012, Journal of medicinal chemistry.

Unprecedented 3-O-methyl-3-C-trifluoromethyl-d-ribono- (and l-lyxono)-γ-lactones synthesized by nucleophilic trifluoromethylation of d-hexose-derived cyclic ketones

J. Praly, S. Ghannay, Jihed Brahmi, 2016 .

Halogen-substituted (C-β-D-glucopyranosyl)-hydroquinone regioisomers: synthesis, enzymatic evaluation and their binding to glycogen phosphorylase.

S. Zographos, N. Oikonomakos, D. Leonidas, 2011, Bioorganic & medicinal chemistry.