Dingding Gao

发表

A fluorine scan on the Zn2+-binding thiolate side chain of HDAC inhibitor largazole: Synthesis, biological evaluation, and molecular modeling.

Xiaolin Yu, Bingbin Zhang, Xinsheng Lei, 2019, European journal of medicinal chemistry.

Identification and preliminary structure-activity relationships of 1-Indanone derivatives as novel indoleamine-2,3-dioxygenase 1 (IDO1) inhibitors.

Yingxia Li, Dingding Gao, Yingxia Li, 2017, Bioorganic & medicinal chemistry.

Novel fatty acid binding protein 4 (FABP4) inhibitors: virtual screening, synthesis and crystal structure determination.

Weiliang Zhu, Kaixian Chen, Yechun Xu, 2015, European journal of medicinal chemistry.

From hit to lead: Structure-based discovery of naphthalene-1-sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4.

Weiliang Zhu, Qiu-feng Liu, H. Su, 2018, European journal of medicinal chemistry.

Rhodium(III)-Catalyzed Kinetic Resolution of Racemic 1,6-Dienes via Asymmetric Borylative Cyclization.

Cheng-Yu He, Dingding Gao, G. Lin, 2020, Organic letters.

Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor.

Yingxia Li, Dingding Gao, Heyao Wang, 2019, Bioorganic & medicinal chemistry.

Combined treatment with FABP4 inhibitor ameliorates rosiglitazone‐induced liver steatosis in obese diabetic db/db mice

Dingding Gao, He-Yao Wang, Ying-xia Li, 2021, Basic & clinical pharmacology & toxicology.

Optimization of 1H-indazol-3-amine derivatives as potent fibroblast growth factor receptor inhibitors.

Yingxia Li, Dingding Gao, Jing Ai, 2017, Bioorganic & medicinal chemistry letters.

One-Pot Preparation of Bridged Tricyclic and Fused Tetracyclic Scaffolds via Rhodium(III)-Catalyzed Asymmetric Borylative Cyclization

Cheng-Yu He, Dingding Gao, G. Lin, 2020 .

Discovery of 1-Amino-1H-imidazole-5-carboxamide Derivatives as Highly Selective, Covalent Bruton's Tyrosine Kinase (BTK) Inhibitors.

Dingding Gao, Shouning Yang, Chunhua Ma, 2021, Journal of medicinal chemistry.

Novel inhibitors of the STAT3 signaling pathway: an updated patent review (2014-present)

Dingding Gao, Guo-qiang Lin, Feng Wang, 2022, Expert opinion on therapeutic patents.

Copper(I)-catalyzed diastereo- and enantio-selective construction of optically pure exocyclic allenes

Cheng-Yu He, Dingding Gao, G. Lin, 2020, Nature Communications.

Exogenous FABP4 interferes with differentiation, promotes lipolysis and inflammation in adipocytes

H. Su, Dingding Gao, He-Yao Wang, 2019, Endocrine.

Spirobiflavonoid stereoisomers from the endangered conifer Glyptostrobus pensilis and their protein tyrosine phosphatase 1B inhibitory activity.

Jia Li, Dingding Gao, J. Xiong, 2019, Bioorganic & medicinal chemistry letters.

Discovery of Novel Drug-like PHGDH Inhibitors to Disrupt Serine Biosynthesis for Cancer Therapy.

Min Huang, Dingding Gao, Guo-qiang Lin, 2023, Journal of medicinal chemistry.

Synthesis and biological evaluation of novel larotaxel analogues.

Ning Ding, S. Ren, Dingding Gao, 2018, European journal of medicinal chemistry.

Enantioselective [3+2] annulation of isatin-derived MBH-carbonates and 3-nitroindoles enabled by a bifunctional DMAP-thiourea.

Guangbo Ge, Dingding Gao, G. Lin, 2020, Chemical communications.

Access to Aryl-Naphthaquinone Atropisomers via Phosphine-Catalyzed Atroposelective (4+2) Annulations of δ-Acetoxy Allenoates with 2-Hydroxyquinone Derivatives.

Dingding Gao, Wei Liu, Dong Wang, 2019, Angewandte Chemie.

Access to Aryl‐Naphthaquinone Atropisomers by Phosphine‐Catalyzed Atroposelective (4+2) Annulations of δ‐Acetoxy Allenoates with 2‐Hydroxyquinone Derivatives

Dingding Gao, Wei Liu, Dong Wang, 2019, Angewandte Chemie.

Synthesis of Decahydrocyclobuta[ cd ]indene Skeletons: Rhodium(III)‐Catalyzed Hydroarylation and Relay Thiophene‐Promoted Intramolecular [2+2] Cycloaddition

Dingding Gao, G. Lin, Yuhui Wang, 2020 .

One-Pot Preparation of 9,10-Dihydrophenanthrenes Initiated by Rhodium(III)-Catalyzed C-H Activation and Relay Diels-Alder Reaction.

Xiaodi Yang, Dingding Gao, Hao Xu, 2020, Organic letters.

Rational drug design of benzothiazole-based derivatives as potent signal transducer and activator of transcription 3 (STAT3) signaling pathway inhibitors.

Min Huang, Yueyue Zhu, Dingding Gao, 2021, European journal of medicinal chemistry.

Discovery of PHGDH inhibitors by virtual screening and preliminary structure-activity relationship study.

Min Huang, Dingding Gao, G. Lin, 2022, Bioorganic chemistry.

A retrospective overview of PHGDH and its inhibitors for regulating cancer metabolism.

Dingding Gao, Guo-qiang Lin, Jian-wei Zhang, 2021, European journal of medicinal chemistry.

Discovery of 5-(methylthio)pyrimidine derivatives as L858R/T790M mutant selective epidermal growth factor receptor (EGFR) inhibitors.

Wei Zhang, Jian Ding, Lin-jiang Tong, 2016, Bioorganic & medicinal chemistry.

Discovery of 9,10-dihydrophenanthrene derivatives as SARS-CoV-2 3CLpro inhibitors for treating COVID-19

Xiaodi Yang, Guangbo Ge, Dingding Gao, 2021, European Journal of Medicinal Chemistry.

CXCL12/CXCR4 Axis-Targeted Dual-Functional Nano-Drug Delivery System Against Ovarian Cancer

Ruixiang Li, Hongjuan Xie, Dingding Gao, 2020, International journal of nanomedicine.

Design, synthesis and biological evaluation of benzyloxyphenyl-methylaminophenol derivatives as STAT3 signaling pathway inhibitors.

Dingding Gao, Qiang Xiao, Mingming Zhang, 2016, Bioorganic & medicinal chemistry.

Design, synthesis and biological evaluation of novel potent STAT3 inhibitors based on BBI608 for cancer therapy.

Dingding Gao, Guo-qiang Lin, Jian-wei Zhang, 2020, European journal of medicinal chemistry.

Identification of novel STAT3 inhibitors bearing 2-acetyl-7-phenylamino benzofuran scaffold for antitumour study.

Dingding Gao, Guo-qiang Lin, Jian-wei Zhang, 2020, Bioorganic & medicinal chemistry.

From hit to lead: Structure-based discovery of naphthalene-1-sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4

Weiliang Zhu, Yechun Xu, Qiu-feng Liu, 2018 .

Nature-inspired catalytic asymmetric rearrangement of cyclopropylcarbinyl cation

Dingding Gao, Guo-qiang Lin, Jian-wei Zhang, 2023, Science advances.

Thiourea‐Promoted Cascade Dihalogenation‐Cyclization of Cyclohexadienone‐Containing 1,6‐Enynes

Dingding Gao, G. Lin, Jian-wei Zhang, 2023, Advanced Synthesis & Catalysis.

A practical preparation of bicyclic boronates via metal-free heteroatom-directed alkenyl sp2-C‒H borylation

Dingding Gao, G. Lin, Jian-wei Zhang, 2023, Communications chemistry.

Crystal structure of human FABP4 complexed with ligand 4-Fluoro-3-((4-methoxynaphthalene)-1-sulfonamido) benzoic acid

Weiliang Zhu, Yechun Xu, Qiu-feng Liu, 2018 .

Identification of benzo[b]thiophene-1,1-dioxide derivatives as novel PHGDH covalent inhibitors.

Dingding Gao, Shuai Tang, Xinglu Cao, 2024, Bioorganic chemistry.

Discovery of highly potent covalent SARS-CoV-2 3CLpro inhibitors bearing 2-sulfoxyl-1,3,4-oxadiazole scaffold for combating COVID-19.

Jincun Zhao, Dingding Gao, G. Lin, 2023, European journal of medicinal chemistry.

High-throughput modular click chemistry synthesis of catechol derivatives as covalent inhibitors of SARS-CoV-2 3CLpro

Dingding Gao, Tiancheng Ma, Donglan Liu, 2024, Acta Materia Medica.