M. Porcelloni

发表

Benzofused hydroxamic acids: useful fragments for the preparation of histone deacetylase inhibitors. Part 1: hit identification.

M. Binaschi, C. Maggi, D. Fattori, 2013, Bioorganic & medicinal chemistry letters.

Histone deacetylase inhibitors: from bench to clinic.

M. Binaschi, D. Fattori, M. Paris, 2008, Journal of medicinal chemistry.

4-N-Hydroxy-4-[1-(sulfonyl)piperidin-4-yl]-butyramides as HDAC inhibitors.

M. Binaschi, C. Maggi, D. Fattori, 2011, Bioorganic & medicinal chemistry letters.

Application of Chiral Sulfides to Catalytic Asymmetric Aziridination and Cyclopropanation with In Situ Generation of the Diazo Compound.

G. Hynd, M. Porcelloni, M. Ferrara, 2001, Angewandte Chemie.

Effect of sulfide structure on enantioselectivity in catalytic asymmetric epoxidation of aldehydes: mechanistic insights and implications.

M. Porcelloni, V. Aggarwal, L. Dudin, 2004, Proceedings of the National Academy of Sciences of the United States of America.

Catalytic Asymmetric Synthesis of Epoxides from Aldehydes Using Sulfur Ylides with In Situ Generation of Diazocompounds.

G. Hynd, M. Porcelloni, V. Aggarwal, 2001, Angewandte Chemie.

A new protocol for the in situ generation of aromatic, heteroaromatic, and unsaturated diazo compounds and its application in catalytic and asymmetric epoxidation of carbonyl compounds. Extensive studies to map out scope and limitations, and rationalization of diastereo- and enantioselectivities.

G. Hynd, M. Porcelloni, V. Aggarwal, 2003, Journal of the American Chemical Society.

Solid-phase synthesis of unsymmetrical ureas through the use of Kenner safety-catch linker

D. Fattori, M. Porcelloni, P. D’Andrea, 2003 .

Alkyl piperidine and piperazine hydroxamic acids as HDAC inhibitors.

M. Binaschi, C. Maggi, D. Fattori, 2011, Bioorganic & medicinal chemistry letters.

Histone Deacetylase Inhibitors: From Bench to Clinic

M. Binaschi, D. Fattori, M. Paris, 2008 .

hNK2 receptor antagonists. The use of intramolecular hydrogen bonding to increase solubility and membrane permeability.

Cristina Rossi, C. Maggi, D. Fattori, 2011, Bioorganic & medicinal chemistry letters.

α,α‐Cyclopentaneglycine Dipeptides Capped with Biaryls as Tachykinin NK2 Receptor Antagonists

A. Sisto, D. Fattori, A. Ettorre, 2008, ChemMedChem.

Generation of a new class of hNK(2) receptor ligands using the 'fragment approach'.

Andrea Madami, D. Fattori, M. Porcelloni, 2005, Bioorganic & medicinal chemistry letters.

A New Palladium-Catalyzed Intramolecular Allylation to Pyrrolidin-2-ones(1).

B. Pacini, G. Giambastiani, M. Porcelloni, 1998, The Journal of organic chemistry.

A New Palladium-Catalyzed Intramolecular Allylation to Pyrrolidin-2-ones.

B. Pacini, G. Giambastiani, M. Porcelloni, 1998 .

Application of Chiral Sulfides to Catalytic Asymmetric Aziridination and Cyclopropanation with In Situ Generation of the Diazo Compound.

G. Hynd, M. Porcelloni, M. Ferrara, 2001, Angewandte Chemie.