K. Gigstad

发表

Potent histone deacetylase inhibitors derived from 4-(aminomethyl)-N-hydroxybenzamide with high selectivity for the HDAC6 isoform.

C. Blackburn, A. Gould, C. Barrett, 2013, Journal of medicinal chemistry.

Asymmetric catalysis of the Strecker amino acid synthesis by a cyclic dipeptide

M. Lipton, K. Gigstad, M. Iyer, 1996, Amino Acids.

Characterization of a New Series of Non-covalent Proteasome Inhibitors with Exquisite Potency and Selectivity for the 20s Β5-subunit Figure S1 Activities of Compound 1 and Bortezomib in Cells

T. Soucy, E. Olhava, M. Sintchak, 2010 .

Histone deacetylase inhibitors derived from 1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine and related heterocycles selective for the HDAC6 isoform.

C. Blackburn, A. Gould, C. Barrett, 2014, Bioorganic & medicinal chemistry letters.

Design, synthesis, and evaluation of naphthalene-sulfonamide antagonists of human CCR8.

S. Ghosh, T. Ocain, C. Blackburn, 2007, Journal of medicinal chemistry.

Identification of Novel Carbocyclic Pyrimidine Cyclic Dinucleotide STING Agonists for Antitumor Immunotherapy Using Systemic Intravenous Route.

Adnan O. Abu-Yousif, M. Mizutani, Courtney A. Cullis, 2021, Journal of medicinal chemistry.

Optimization of a series of dipeptides with a P3 β-neopentyl asparagine residue as non-covalent inhibitors of the chymotrypsin-like activity of human 20S proteasome

M. Sintchak, L. Dick, J. Blank, 2012 .

Optimization of a series of dipeptides with a P3 threonine residue as non-covalent inhibitors of the chymotrypsin-like activity of the human 20S proteasome.

Jonathan L Blank, Christopher Tsu, Christopher Blackburn, 2010, Bioorganic & medicinal chemistry letters.

N-substituted cis-4a-(3-hydroxyphenyl)-8a-methyloctahydroisoquinolines are opioid receptor pure antagonists.

J. Deschamps, James B. Thomas, S. Mascarella, 2005, Journal of medicinal chemistry.

Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S β5-subunit

T. Soucy, E. Olhava, M. Sintchak, 2010, The Biochemical journal.

A stereoselective synthetic approach to N-alkyl-4β-methyl-5-phenylmorphans

James B. Thomas, S. Mascarella, F. Carroll, 1999 .

N,C-Capped dipeptides with selectivity for mycobacterial proteasome over human proteasomes: role of S3 and S1 binding pockets.

M. Sintchak, L. Dick, C. Nathan, 2013, Journal of the American Chemical Society.

Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S β5-subunit

E. Olhava, K. Gigstad, F. Bruzzese, 2010, Biochemical Journal.