A. Yamani

发表

Views on amyloid hypothesis and secretase inhibitors for treating Alzheimer's disease: progress and problems.

Y. Kiso, J. Nguyen, A. Yamani, 2006, Current pharmaceutical design.

beta-Secretase inhibitors: modification at the P4 position and improvement of inhibitory activity in cultured cells.

Kazuki Saito, Y. Kiso, Y. Hamada, 2006, Bioorganic & medicinal chemistry letters.

Significance of interactions of BACE1-Arg235 with its ligands and design of BACE1 inhibitors with P2 pyridine scaffold.

Y. Kiso, Y. Hamada, S. Ishiura, 2009, Bioorganic & medicinal chemistry letters.

BACE1 inhibitors: optimization by replacing the P1' residue with non-acidic moiety.

Kazuki Saito, Y. Kiso, Y. Hamada, 2008, Bioorganic & medicinal chemistry letters.

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 1: Substitution of the glycine carboxylic acid group.

A. Fairlamb, A. Lambeir, A. Yamani, 2002, Bioorganic & medicinal chemistry letters.

AN EFFICIENT SYNTHESIS OF ORTHOGONALLY PROTECTED SPERMIDINE

A. Yamani, A. Haemers, K. Augustyns, 2002 .

Trypanothione as a target in the design of antitrypanosomal and antileishmanial agents.

A. Yamani, A. Haemers, K. Augustyns, 2001, Current pharmaceutical design.

Novel non-peptidic and small-sized BACE1 inhibitors.

Kazuki Saito, Y. Kiso, Y. Hamada, 2008, Bioorganic & medicinal chemistry letters.

Design of pentapeptidic BACE1 inhibitors with carboxylic acid bioisosteres at P1' and P4 positions.

Y. Kiso, Y. Hamada, Tooru Kimura, 2010, Bioorganic & medicinal chemistry.

Discovery and optimization of novel pyrazole-benzimidazole CPL304110, as a potent and selective inhibitor of fibroblast growth factor receptors FGFR (1-3).

A. Yamani, K. Dzwonek, M. Wieczorek, 2020, European journal of medicinal chemistry.

Identification of small-molecule enhancers of arginine methylation catalyzed by coactivator-associated arginine methyltransferase 1.

E. Novellino, A. Mai, G. Sbardella, 2012, Journal of medicinal chemistry.

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 2: substitution of the glycine part.

A. Fairlamb, A. Lambeir, A. Yamani, 2002, Bioorganic & medicinal chemistry letters.