N. Gaboriaud-Kolar

发表

O. Tsitsilonis, A. Skaltsounis, S. P. Shukla, 2017, European Journal of Medicinal Chemistry.

Indirubin derivatives are potent and selective anti-Trypanosoma cruzi agents

A. Skaltsounis, C. Meira, N. Gaboriaud-Kolar, 2018, Virulence.

Indirubin core structure of glycogen synthase kinase-3 inhibitors as novel chemotype for intervention with 5-lipoxygenase.

O. Werz, A. Skaltsounis, N. Gaboriaud-Kolar, 2014, Journal of medicinal chemistry.

New semi-synthetic analogs of oleuropein show improved anticancer activity in vitro and in vivo.

O. Tsitsilonis, A. Skaltsounis, P. Samara, 2017, European journal of medicinal chemistry.

(WO2011057959) Indole and indazole derivatives as glycogen synthase activators: a patent evaluation

A. Skaltsounis, N. Gaboriaud-Kolar, 2011, Expert opinion on therapeutic patents.

Evaluation of Dual 5-Lipoxygenase/Microsomal Prostaglandin E2 Synthase-1 Inhibitory Effect of Natural and Synthetic Acronychia-Type Isoprenylated Acetophenones.

O. Werz, A. Skaltsounis, A. Rossi, 2017, Journal of natural products.

Oxidative burst inhibitory and cytotoxic indoloquinazoline and furoquinoline alkaloids from Oricia suaveolens.

Norbert Sewald, Krishna Prasad Devkota, M. Choudhary, 2008, Journal of natural products.

Biomimetic Synthesis of Oleocanthal, Oleacein, and Their Analogues Starting from Oleuropein, A Major Compound of Olive Leaves.

A. Skaltsounis, N. Gaboriaud-Kolar, Amos B. Smith, 2020, Journal of natural products.

A domino ring-closing metathesis as a key-step in the synthesis of chiral lactones from d-mannitol

B. Bodo, N. Gaboriaud-Kolar, B. Nay, 2005 .

Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration Analysis

Vassilios Myrianthopoulos, Emmanuel Mikros, Stefan Knapp, 2016, Journal of medicinal chemistry.

Synthesis, cytotoxic activity, and mechanism of action of furo[2,3-c]acridin-6-one and benzo[b]furo[3,2-h]acridin-6-one analogues of psorospermin and acronycine.

B. Pfeiffer, Marie-Christine Lallemand, F. Tillequin, 2008, Journal of medicinal chemistry.

Symphonia globulifera, a Widespread Source of Complex Metabolites with Potent Biological Activities

Marie-Christine Lallemand, N. Gaboriaud-Kolar, S. Michel, 2015, Planta Medica.

Synthesis of novel guttiferone A derivatives: in-vitro evaluation toward Plasmodium falciparum, Trypanosoma brucei and Leishmania donovani.

J. Wansi, Marie-Christine Lallemand, N. Gaboriaud-Kolar, 2013, European journal of medicinal chemistry.

Indirubin Analogues Inhibit Trypanosoma brucei Glycogen Synthase Kinase 3 Short and T. brucei Growth

A. Skaltsounis, E. Mikros, N. Gaboriaud-Kolar, 2019, Antimicrobial Agents and Chemotherapy.

Indirubin derivatives: a patent review (2010 – present)

A. Skaltsounis, N. Gaboriaud-Kolar, K. Vougogiannopoulou, 2015, Expert opinion on therapeutic patents.

A colorful history: the evolution of indigoids.

A. Skaltsounis, N. Gaboriaud-Kolar, Sang-Sik Nam, 2014, Progress in the chemistry of organic natural products.

The Indirubin Derivative 6-Bromoindirubin-3′-Oxime Activates Proteostatic Modules, Reprograms Cellular Bioenergetic Pathways, and Exerts Antiaging Effects

J. Tchoumtchoua, I. Trougakos, A. Skaltsounis, 2017, Antioxidants & redox signaling.

6-bromo-indirubin-3′-oxime (6BIO), a Glycogen synthase kinase-3β inhibitor, activates cytoprotective cellular modules and suppresses cellular senescence-mediated biomolecular damage in human fibroblasts

I. Trougakos, A. Skaltsounis, A. Sklirou, 2017, Scientific Reports.

From Drug Screening to Target Deconvolution: a Target-Based Drug Discovery Pipeline Using Leishmania Casein Kinase 1 Isoform 2 To Identify Compounds with Antileishmanial Activity

Hervé Galons, Laurent Meijer, Olivier Leclercq, 2016, Antimicrobial Agents and Chemotherapy.

Natural-Based Indirubins Display Potent Cytotoxicity toward Wild-Type and T315I-Resistant Leukemia Cell Lines.

R. Jove, A. Skaltsounis, E. Mikros, 2016, Journal of natural products.

Novel Inverse Binding Mode of Indirubin Derivatives Yields Improved Selectivity for DYRK Kinases

Daniel Cappel, Vassilios Myrianthopoulos, Emmanuel Mikros, 2012, ACS medicinal chemistry letters.

Glycogen phosphorylase inhibitors: a patent review (2008 – 2012)

A. Skaltsounis, N. Gaboriaud-Kolar, 2013, Expert opinion on therapeutic patents.

An inhibitor-driven study for enhancing the selectivity of indirubin derivatives towards leishmanial Glycogen Synthase Kinase-3 over leishmanial cdc2-related protein kinase 3

A. Skaltsounis, E. Mikros, Alexandros Alexandratos, 2014, Parasites & Vectors.

Synthesis, cytotoxic activity and mechanism of action of new Psorospermin-Acronycine analogs

Marie-Christine Lallemand, F. Tillequin, S. Boutefnouchet, 2008 .

Identification of indirubin derivatives as anti-trypanosomal agents

N. Gaboriaud-Kolar, L. Skaltsounis, A. Efstathiou, 2014 .

From Drug Screening to Target Deconvolution: a Target-Based Drug Discovery Pipeline Using Leishmania Casein Kinase 1 Isoform 2 To Identify Compounds with Antileishmanial Activity

L. Meijer, A. Skaltsounis, N. Rachidi, 2016, Antimicrobial Agents and Chemotherapy.