D. Tourwé

A. Beck‐Sickinger, P. Schubiger, D. Tourwé, 2007, The quarterly journal of nuclear medicine and molecular imaging : official publication of the Italian Association of Nuclear Medicine (AIMN) [and] the International Association of Radiopharmacology (IAR), [and] Section of the Society of....

Double-stabilized neurotensin analogues as potential radiopharmaceuticals for NTR-positive tumors.

P. Schubiger, D. Tourwé, A. Blanc, 2006, Nuclear medicine and biology.

Conformation of two somatostatin analogues in aqueous solution. Study by NMR methods and circular dichroism.

V. Hruby, W. Kazmierski, D. Tourwé, 1989, European journal of biochemistry.

Morphiceptin and β‐casomorphin‐5 analogues containing a reduced peptide bond: Selective μ‐receptor agonists and a novel μ antagonist, H‐Tyr‐Proψ(CH2‐NH)Phe‐Pro‐Gly‐OH

T. Burks, D. Tourwé, P. Davis, 1992 .

Presence and regulation of insulin-regulated aminopeptidase in mouse macrophages

J. V. Van Ginderachter, D. Laoui, D. Tourwé, 2014, Journal of the renin-angiotensin-aldosterone system : JRAAS.

Structural basis for bifunctional peptide recognition at human δ-Opioid receptor

Anton Barty, Sébastien Boutet, Marc Messerschmidt, 2015, Nature Structural &Molecular Biology.

Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional Compounds.

A. Misicka, P. Kosson, Piotr F. J. Lipiński, 2017, ACS medicinal chemistry letters.

The γ-methyl-E-olefin as isosteric replacement of the peptide bond

D. Tourwé, G. V. Binst, H. Jaspers, 1996 .

Cleromyrine I, a new cyclohexapeptide from clerodendrum myricoides

D. Tourwé, H. Pepermans, G. V. Binst, 1990 .

Synthesis and conformational study of two cyclic analogues of somatostatin containing an AMPA-spacer unit.

D. Tourwé, D. Gondol, C. Wynants, 1987, International journal of peptide and protein research.

Synthesis and conformational study of a cyclic hexapeptide analogue of somatostatin: cyclo(Phe-D-Trp-Lys-Thr-o-AMPA).

D. Tourwé, H. Pepermans, E. M. van den Berg, 1987, International journal of peptide and protein research.

Proton n.m.r. investigation of conformational influence of penicillamine residues on the disulfide ring system of opioid receptor selective somatostatin derivatives.

V. Hruby, W. Kazmierski, D. Tourwé, 2009, International journal of peptide and protein research.

Development and pharmacological characterization of conformationally constrained urotensin II-related peptide agonists.

N. Doucet, B. Folch, M. Létourneau, 2013, Journal of medicinal chemistry.

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia.

L. Gendron, D. Tourwé, P. Sarret, 2019, ACS chemical neuroscience.

Synthesis of sidechain adapted β-turn mimics for modifying the C-terminus of substance P

D. Tourwé, V. Maes, W. D. Borggraeve, 2005 .

Prototypic Opioid Peptidomimetics Based on the Dmt-Aba-Gly Scaffold

S. Salvadori, G. Balboni, D. Tourwé, 2010 .

Benzo- and indoloquinolizine derivatives. 13. Conformation of the perhydrobenzo[c]quinolizines

D. Tourwé, G. V. Binst, G. Laus, 1978 .

Carbon-13 Nuclear Magnectic Resonance Spectroscopy of Quinolizidine Derivatives

D. Tourwé, G. V. Binst, 1978 .

T3P-Promoted, Mild, One-Pot Syntheses of Constrained Polycyclic Lactam Dipeptide Analogues via Stereoselective Pictet-Spengler and Meyers Lactamization Reactions.

D. Tourwé, S. Ballet, Z. Urbańczyk-Lipkowska, 2015, Organic letters.

Fluorescein‐labeled stable neurotensin derivatives

R. Bergmann, D. Tourwé, T. Hanke, 2006, Journal of peptide science : an official publication of the European Peptide Society.

Monitoring of optical isomers of β-methylphenylalanine in opioid peptides

D. Tourwé, A. Péter, G. Tóth, 1994 .

High-performance liquid chromatographic enantioseparation of unusual secondary amino acids on a D-penicillamine-based chiral ligand exchange column.

D. Armstrong, D. Tourwé, A. Péter, 2006, Chirality.

Application of a new chiral derivatizing agent to the enantioseparation of secondary amino acids.

D. Tourwé, A. Péter, G. Tóth, 2002, Journal of chromatography. A.

Enantioseparation by HPLC of imino acids on macrocyclic glycopeptide stationary phases and as their (S)-N-(4-Nitrophenoxycarbonyl)phenylalanine methoxyethyl ester derivatives

D. Armstrong, D. Tourwé, A. Péter, 2002 .

In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera

A. Lipkowski, P. Kosson, P. Schiller, 2012, Molecular Brain.

Conformational restriction of Tyr and Phe side chains in opioid peptides: information about preferred and bioactive side-chain topology.

K. Verschueren, F. Porreca, D. Tourwé, 1996, Biopolymers.

Novel glycated [99mTc(CO)3]-labeled bombesin analogues for improved targeting of gastrin-releasing peptide receptor-positive tumors.

R. Schibli, D. Tourwé, E. García Garayoa, 2008, Bioconjugate chemistry.

Dermorphin tetra- and heptapeptide analogues containing a [3,4] amide bond replacement by a carbon-carbon double and single bond.

S. Salvadori, D. Tourwé, H. Pepermans, 2009, International journal of peptide and protein research.

High-performance liquid chromatographic separation of unusual amino acid enantiomers derivatized with (1S,2S)-1,3-diacetoxy-1-(4-nitrophenyl)-2-propyl-isothiocyanate

F. Fülöp, D. Tourwé, A. Péter, 2000 .

Rapid construction of substituted 3-amino-1,5-benzothiazepin-4(5H)-one dipeptide scaffolds through an Ugi-4CR - Ullmann cross-coupling sequence.

B. Maes, D. Tourwé, S. Ballet, 2018, Organic & biomolecular chemistry.

A novel solid phase approach to Aia‐containing peptides

D. Tourwé, D. Feytens, Magali De Vlaeminck, 2009, Journal of peptide science : an official publication of the European Peptide Society.

Bradykinin analogs containing the 4‐amino‐2‐benzazepin‐3‐one scaffold at the C‐terminus

D. Tourwé, S. Ballet, L. Quartara, 2007, Journal of peptide science : an official publication of the European Peptide Society.

Efficient one-pot synthesis of amino-benzotriazolodiazocinone scaffolds via catalyst-free tandem Ugi-Huisgen reactions.

V. Caveliers, D. Tourwé, S. Ballet, 2016, Organic & biomolecular chemistry.

Efficient synthesis of conformationally constrained, amino-triazoloazepinone-containing di- and tripeptides via a one-pot Ugi-Huisgen tandem reaction.

D. Tourwé, S. Ballet, T. M. A. Barlow, 2014, Organic & biomolecular chemistry.

Using Conformational constraints at position 6 of Angiotensin II to generate compounds with enhanced AT2R selectivity and proteolytic stability.

M. Aguilar, M. D. Del Borgo, D. Tourwé, 2021, Bioorganic & medicinal chemistry letters.

Novel selective human melanocortin-3 receptor ligands: use of the 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one (Aba) scaffold.

V. Hruby, M. Cai, A. Misicka, 2007, Bioorganic & medicinal chemistry letters.

Synthesis of 4-amino-3-oxo-tetrahydroazepino[3,4-b]indoles: new conformationally constrained Trp analogs

A. Misicka, P. Kosson, P. Schiller, 2007 .

Conformational restriction of the Tyr53 side-chain in the decapeptide HE.

C. Rabourdin-Combe, D. Gerlier, H. Dumortier, 2000, The journal of peptide research : official journal of the American Peptide Society.

Rapid Procedure for N-Phthaloylation of α-Amino Carboxamides, α-Amino Alcohols, α-Amino Esters and Dipeptide Derivatives

J. Briand, G. Guichard, D. Tourwé, 2001 .

A New Structural Motif for μ-Opioid Antagonists

P. Kosson, P. Schiller, A. Lipkowski, 2005 .

Synthesis of 1,2,7,7a-tetrahydro-1aH-cyclopropa[b]quinoline-1a-carboxylic acid derivatives, doubly constrained ACC derivatives, by a remarkable cyclopropanation process.

N. de Kimpe, F. Fülöp, D. Tourwé, 2002, The Journal of organic chemistry.

A facile synthesis of 1,2,3,4-tetrahydro-7-hydroxyisoquinoline-3-carboxylic acid, a conformationally constrained tyrosine analogue

M. Lebl, V. Hruby, K. Verschueren, 1992 .

Preservation of hepatocellular functionality in cultures of primary rat hepatocytes upon exposure to 4-Me2N-BAVAH, a hydroxamate-based HDAC-inhibitor.

J. Fraczek, T. Vanhaecke, V. Rogiers, 2011, Toxicology in vitro : an international journal published in association with BIBRA.

Highly stereoselective one-pot construction of trisubstituted tetrahydro-β-carboline-fused diketopiperazines: a synthetic route towards cialis analogues

D. Tourwé, S. Ballet, M. Jida, 2014 .

High-performance liquid chromatographic separation of enantiomers of synthetic amino acids on a ristocetin A chiral stationary phase.

D. Armstrong, D. Tourwé, A. Péter, 2000, Journal of chromatography. A.

Monitoring of optical isomers of some conformationally constrained amino acids with tetrahydroisoquinoline or tetraline ring structures

F. Fülöp, D. Tourwé, A. Péter, 1995 .

New amino acids derived from L-pyroglutamic acid: Synthesis of Trans-4-benzyl-cis-5-phenyl-L-proline, L-α-(2-benzyl-3-phenylpropyl)-glycine and L-α-(3-phenylpropyl)-glycine

D. Tourwé, P. Verheyden, W. Nest, 1998 .

Synthesis of 3,3-dimethylazetidine-2-carboxylic acid and some derivatives

D. Tourwé, N. Kimpe, M. Boeykens, 1998 .

Highly diastereoselective synthesis of 1-carbamoyl-4-aminoindoloazepinone derivatives via the Ugi reaction.

D. Tourwé, S. Ballet, Z. Urbańczyk-Lipkowska, 2013, Organic letters.

Comparison of the separation efficiencies of chirobiotic T and TAG columns in the separation of unusual amino acids.

D. Armstrong, F. Fülöp, D. Tourwé, 2004, Journal of chromatography. A.

Effect of temperature on retention of enantiomers of beta-methyl amino acids on a teicoplanin chiral stationary phase.

D. Armstrong, D. Tourwé, A. Péter, 1998, Journal of chromatography. A.

Amino triazolo diazepines (Ata) as constrained histidine mimics.

G. Vauquelin, D. Tourwé, P. Vanderheyden, 2011, Organic letters.

Convenient synthesis of 3,4-methano-1,2,3, 4-tetrahydroisoquinoline-3-carboxylic acid and its derivatives as doubly constrained nonproteinogenic amino acid derivatives.

N. de Kimpe, F. Fülöp, J. Martins, 2000, The Journal of organic chemistry.

Deltorphin II analogues with 6-hydroxy-2-aminotetralin-2-carboxylic acid in position 1.

Z. Darula, K. Kövér, É. Makó, 2000, Journal of medicinal chemistry.

Synthesis of fused 3-aminoazepinones via trapping of a new class of cyclic seven-membered allenamides with furan.

G. Verniest, D. Tourwé, G. Van Lommen, 2014, Organic letters.

Cyclic Aromatic Amino Acids with Constrained χ(1) and χ (2) Dihedral Angles.

W. Kazmierski, D. Tourwé, G. Tóth, 1999, Methods in molecular medicine.

High-performance liquid chromatographic separation of the enantiomers of unusual alpha-amino acid analogues.

B. Kaptein, Q. Broxterman, D. Armstrong, 2000, Journal of chromatography. A.

Efficient Synthesis of 1-Benzyloxyphenyl-3-phenylacetones

D. Tourwé, W. Lubell, E. Mannekens, 2000 .

New endomorphin analogs with mu-agonist and delta-antagonist properties

E. Navratilova, H. Yamamura, F. Fülöp, 2004 .

Unprecedented sigmatropic rearrangements leading to 2,3-dihydro-1h-2-benzazepine-3-carboxylic acid.

N. de Kimpe, J. Martins, D. Tourwé, 2001, The Journal of organic chemistry.

Synthesis of the diastereomers of β-Me-Tyr and β-Me-Phe and their effect on the biological properties of the delta opioid receptor antagonist TIPP

P. Schiller, N. N. Chung, D. Tourwé, 1995, Letters in Peptide Science.

Chromatographic methods for monitoring the optical isomers of unusual aromatic amino acids

D. Tourwé, A. Péter, G. Tóth, 1998 .

LC Enantioseparation of Tryptophan Analogs on α-Cyclodextrin Stationary Phase

D. Armstrong, D. Tourwé, A. Péter, 2006 .

Indirect high-performance liquid chromatographic separation of stereoisomers of beta-alkyl-substituted amino acids by the application of (S)-N-(4-nitrophenoxycarbonyl)phenylalanine methoxyethyl ester as chiral derivatizing agent.

D. Tourwé, A. Péter, J. Sapi, 2002, Journal of chromatography. A.

Conformationally constrained deltorphin analogs with 2-aminotetralin-2-carboxylic acid in position 3.

Z. Darula, F. Fülöp, D. Tourwé, 1997, Journal of medicinal chemistry.

Monitoring of Deprotection Reactions of Cyclic Somatostatin Analogues by Fast Atom Bombardment Mass Spectrometry

D. Tourwé, G. V. Binst, H. Jaspers, 2010 .

Conformational properties of the pentapeptide fragment [32-36] of the thymic hormone thymopoietin.

K. Hallenga, D. Tourwé, G. Van Binst, 2009, International journal of peptide and protein research.

Molecular Assembly of Multifunctional 99mTc Radiopharmaceuticals Using “Clickable” Amino Acid Derivatives

R. Schibli, B. Spingler, D. Tourwé, 2010, ChemMedChem.

Side reactions in the preparation of 1,2,3,4-tetrahydro-β-carboline-3-carboxylic acid

D. Tourwé, K. Iterbeke, P. Verheyden, 1998, Letters in Peptide Science.

Direct and indirect high-performance liquid chromatographic enantioseparation of β-amino acids

D. Armstrong, F. Fülöp, D. Tourwé, 2004 .

High-Performance Liquid Chromatographic Separation of Stereoisomers of β-Amino Acids and a Comparison of Separation Efficiencies on Chirobiotic T and TAG Columns

D. Armstrong, F. Fülöp, D. Tourwé, 2004 .

Enantiomeric separation of unusual secondary aromatic amino acids

D. Armstrong, D. Tourwé, A. Péter, 1998 .

Confirmation of the E and Z attribution to the isomers of 3‐ethylidene‐1‐azabicyco‐[2,2,2]octane by CMR spectroscopy

D. Tourwé, G. V. Binst, 1972 .

Monitoring of the Chiral Purity of Ψ(E,CH=CH) Dipeptides using 2,3,4,6‐Tetra‐O‐Acetyl‐β‐D‐Glucopyranosyl Isothiocyanate

D. Tourwé, J. Couder, M. Ceusters, 2010 .

Preclinical evaluation of a new, stabilized neurotensin(8--13) pseudopeptide radiolabeled with (99m)tc.

Alain Blanc, D. Tourwé, A. Blanc, 2002, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.

Design, synthesis, pharmacological evaluation, and structure-activity study of novel endomorphin analogues with multiple structural modifications.

K. Kövér, A. Keresztes, D. Tourwé, 2011, Journal of medicinal chemistry.

Synthesis and conformational study of two L-prolyl-L-leucyl-glycinamide analogues with a reduced peptide bond.

D. Tourwé, G. Van Binst, P. Vander Elst, 2009, International journal of peptide and protein research.

Development of a new microwave-assisted cleavable backbone amide linker (BAL): a comparative study.

E. V. Van der Eycken, D. Tourwé, S. Claerhout, 2010, Organic & biomolecular chemistry.

Sedum alkaloids. VI: Resolution enhanced proton NMR and 13C NMR spectroscopic studies on the solution conformation of Sedum acre alkaloids

B. Colau, D. Tourwé, C. Hootele, 1984 .

Benzo‐and Indoloquinolizine Derivatives XVa. Conformational Analysis of 6,7,12,13‐Tetrahydro‐11bH‐Dibenzo[a,f]Quinolizine Derivatives by 1H AND 13C NMR

D. Tourwé, W. Brandt, G. V. Binst, 2010 .

Benzo- and indoloquinolizine derivatives. I. Synthesis of 4b,5,6,7,8,8a,10,11,16,16b-decahydrodibenz[f,h] indolo[2,3-a] quinolizine

D. Tourwé, G. V. Binst, 1972 .

Sedum alkaloids : VIII. solution conformation of sedamine and related bases

D. Tourwé, C. Hootele, F. Halin, 1985 .

An evaluation of microwave heating for the rapid hydrolysis of peptide samples for chiral amino acid analysis.

E. Gerlo, D. Tourwé, E Gerlo, 1993, Peptide research.

The use of time‐averaged 3JHH restrained molecular dynamics (tar‐MD) simulations for the conformational analysis of five‐membered ring systems: Methodology and applications

Koen Augustyns, Pieter M. S. Hendrickx, Francisco Corzana, 2009, J. Comput. Chem..

Benzo- and Indoloquinolizine Compounds. IV. The Use of 13C-H Coupling Constants in the Stereochemical Study of Nitrogen Bridgehead Compounds

D. Tourwé, G. V. Binst, 1973 .

Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics.

P. Schiller, J. Vanden Broeck, A. Lipkowski, 2015, European journal of medicinal chemistry.

Bifunctional Peptide-Based Opioid Agonist-Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic Pain.

F. Simonin, B. Mégarbane, P. Kosson, 2016, Journal of medicinal chemistry.

Liquid chromatographic study of the enzymatic degradation of endomorphins, with identification by electrospray ionization mass spectrometry.

D. Tourwé, A. Péter, G. Tóth, 1999, Journal of chromatography. A.

Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury Mice.

A. Mollica, P. Schiller, J. Streicher, 2017, ACS chemical neuroscience.

PK20, a new opioid-neurotensin hybrid peptide that exhibits central and peripheral antinociceptive effects

P. Kosson, A. Lipkowski, D. Tourwé, 2010, Molecular pain.

Synthesis of a Protected Acetylene Dipeptide Isostere

D. Tourwé, G. V. Binst, M. V. Marsenille, 2010 .

Influence of ring substitution on the conformation and β-turn mimicry of 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one peptide mimetics

A. Keresztes, D. Tourwé, L. Brans, 2009 .

High-performance liquid chromatographic separation of stereoisomers of N-phthaloyl-protected amino acids and dipeptidomimetics.

D. Armstrong, D. Tourwé, S. Ballet, 2007, Journal of separation science.

Analogs of oxytocin containing a modified peptide bond.

M. Lebl, V. Hruby, D. Tourwé, 2009, International journal of peptide and protein research.

Synthesis and binding characteristics of [3H]neuromedin N, a NTS2 receptor ligand

A. Lipkowski, D. Tourwé, S. Ballet, 2016, Neuropeptides.

Synergetic effects of DNA demethylation and histone deacetylase inhibition in primary rat hepatocytes

J. Fraczek, T. Vanhaecke, V. Rogiers, 2012, Investigational New Drugs.

Angiotensin IV displays only low affinity for native insulin‐regulated aminopeptidase (IRAP)

G. Vauquelin, D. Tourwé, G. Tóth, 2012, Fundamental & clinical pharmacology.

The novel histone deacetylase inhibitor 4-Me2N-BAVAH differentially affects cell junctions between primary hepatocytes.

T. Vanhaecke, V. Rogiers, M. Vinken, 2007, Toxicology.

Histone deacetylase inhibitors : Opening a new field of research in the development of alternative methods ?

J. Fraczek, T. Vanhaecke, V. Rogiers, 2006 .

Location of the three disulfide bonds in an antimicrobial peptide from Amaranthus caudatus using mass spectrometry.

L. Wyns, D. Tourwé, P. Verheyden, 2009, The journal of peptide research : official journal of the American Peptide Society.

Inhibition of NF‐κB activation by the histone deacetylase inhibitor 4‐Me2N‐BAVAH induces an early G1 cell cycle arrest in primary hepatocytes

T. Vanhaecke, V. Rogiers, M. Vinken, 2007, Cell proliferation.

Superpotent [Dmt¹] dermorphin tetrapeptides containing the 4-aminotetrahydro-2-benzazepin-3-one scaffold with mixed μ/δ opioid receptor agonistic properties.

D. Weiss, P. Kosson, A. Lipkowski, 2011, Journal of medicinal chemistry.

In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt1-DALDA Analogues.

P. Schiller, A. Lipkowski, B. Brodin, 2014, ACS medicinal chemistry letters.

Amide analogues of TSA: synthesis, binding mode analysis and HDAC inhibition.

V. Rogiers, P. Geerlings, D. Tourwé, 2003, Bioorganic & medicinal chemistry letters.

Benzo‐ and indoloquinolizines: X—application of carbon‐13 n.m.r. to the stereochemistry of the 4b,5,6,7,8,8a,10,11,16,16b‐decahydrodibenz[f,h]indolo[2,3‐a]quinolizine isomers

D. Tourwé, G. V. Binst, E. D. Cock, 1976 .

HPLC enantioseparation of phenylalanine analogs by application of (S)-N-(4-nitrophenoxycarbonyl)phenylalanine methoxyethyl ester as a new chiral derivatizing agent

R. Casimir, D. Tourwé, A. Péter, 2001 .

Oxidative α,ω-diyne coupling as an approach towards novel peptidic macrocycles.

J. Martins, G. Verniest, D. Tourwé, 2015, Organic & biomolecular chemistry.

Synthesis and biological activities of linear and cyclic enkephalin analogues containing a psi (E,CH = CH) or psi (CH2CH2) isosteric replacement.

J. Leysen, T. Burks, H. Yamamura, 2009, International journal of peptide and protein research.

In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera

P. Kosson, P. Schiller, A. Lipkowski, 2012, Molecular Brain.

New analogues of deltorphin C and enkephalin-Val,5,6-Gly7-NH2 with replacement of Phe by βMePhe

D. Tourwé, A. Péter, G. Tóth, 1995 .

Development of potent and proteolytically stable human neuromedin U receptor agonists.

B. Holst, M. Rosenkilde, V. Caveliers, 2018, European journal of medicinal chemistry.

Neuromedin U and Structural Analogs: an Overview of Their Structure, Function and Selectivity.

I. Smolders, D. Tourwé, S. Ballet, 2019, Current medicinal chemistry.

Trifluoromethylated Proline Surrogates as Part of “Pro–Pro” Turn‐Inducing Templates

Samuel L. C. Moors, D. Tourwé, K. Van Hecke, 2019, Chembiochem : a European journal of chemical biology.

Probing opioid receptor-ligand interactions by employment of indolizidin-9-one amino acid as a constrained Gly(2)-Gly(3) surrogate in a leucine-enkephalin mimic.

M. Jurzak, T. Meert, F. Gosselin, 2001, The journal of peptide research : official journal of the American Peptide Society.

Conformation-directed design of cyclic somatostatins containing a βVI-turn mimetic

D. Tourwé, 1995, Letters in Peptide Science.

Cyclic Somatostatins containing α-benzyl-o-AMPA as a cis peptide bond mimic

D. Tourwé, P. Verheyden, J. V. Betsbrugge, 2002 .

Somatostatin analogues containing o-aminomethylphenylacetic acid as a bridge unit

A. Misicka, D. Tourwé, G. V. Binst, 1995, Letters in Peptide Science.

Evidence for the bioactive conformation in a cyclic hexapeptide analogue of somatostatin containing a cis-peptide bond mimic.

D. Tourwé, H. Pepermans, G. Van Binst, 1988, Biochemical and biophysical research communications.

Synthesis and biological activities of cyclic somatostatin analogues containing o-aminomethylphenylalanine as a bridging unit

K. Verschueren, D. Tourwé, G. V. Binst, 1993 .

Screening of amide analogues of Trichostatin A in cultures of primary rat hepatocytes: search for potent and safe HDAC inhibitors

J. Fraczek, T. Vanhaecke, V. Rogiers, 2009, Investigational New Drugs.

A Metabolic Screening Study of Trichostatin A (TSA) and TSA-Like Histone Deacetylase Inhibitors in Rat and Human Primary Hepatocyte Cultures

T. Vanhaecke, V. Rogiers, P. Bachellier, 2007, Journal of Pharmacology and Experimental Therapeutics.

Novel 99mTc-labeled neurotensin analogues with optimized biodistribution properties.

Veronique Maes, D. Tourwé, V. Maes, 2006, Journal of medicinal chemistry.

Hybrid opioid/non-opioid ligands in pain research.

A. Lipkowski, D. Tourwé, S. Ballet, 2014, Current pharmaceutical design.

PEGylation of (99m)Tc-labeled bombesin analogues improves their pharmacokinetic properties.

R. Schibli, D. Tourwé, C. Müller, 2011, Nuclear medicine and biology.

Novel neurotensin analogues for radioisotope targeting to neurotensin receptor-positive tumors.

J. Barbet, A. Gruaz-Guyon, D. Tourwé, 2009, Bioconjugate chemistry.

A stable neurotensin-based radiopharmaceutical for targeted imaging and therapy of neurotensin receptor-positive tumours

D. Tourwé, A. Blanc, V. Maes, 2008, European Journal of Nuclear Medicine and Molecular Imaging.

Azepinone-Containing Tetrapeptide Analogues of Melanotropin Lead to Selective hMC4R Agonists and hMC5R Antagonist.

V. Hruby, S. Schwartz, M. Cai, 2015, ACS medicinal chemistry letters.

Structure-Based Design of Melanocortin 4 Receptor Ligands Based on the SHU-9119-hMC4R Cocrystal Structure†.

R. Stevens, R. Cone, Suwen Zhao, 2020, Journal of medicinal chemistry.

Synthesis and biological activities of psi (CH2NH) pseudopeptide analogues of the C-terminal hexapeptide of neurotensin.

J. Leysen, D. Tourwé, J. Couder, 2009, International journal of peptide and protein research.

Syntheses and reactions of 1-amino-2,2-dialkylcyclopropane-1-carbonitriles and -carboxamides - Potential precursors of ACC derivatives

T. Huybrechts, D. Tourwé, J. Declercq, 1999 .

Novel diastereomeric opioid tetrapeptides exhibit differing pharmacological activity profiles

D. Tourwé, I. Kertész, A. Borsodi, 2007, Brain Research Bulletin.

Opioid Receptor Binding Characteristics and Structure-Activity Studies of Novel Tetrapeptides in the TIPP (Tyr-Tic-Phe-Phe) Series

D. Tourwé, A. Péter, A. Borsodi, 2006, Neurosignals.

New endomorphin analogs with -agonist and -antagonist properties*

E. Navratilova, H. Yamamura, F. Fülöp, 2004 .

Benzo‐ and indoloquinolizine derivatives. VI—configuration and conformation of 4b,5,6,7,8,8a,10,11,16,16b‐decahydrodibenz[f,h]indolo[2,3‐a]quinolizine diastereoisomers. A 270 MHz 1H NMR study

D. Tourwé, G. V. Binst, 1974 .

Benzo‐ and indoloquinolizine derivatives ‐ VIII: A Two‐step carbostyril preparation in the synthesis of dibenzo[a, f]‐and benz[f]indolo[2,3‐a]quinolizines

D. Tourwé, G. V. Binst, 2010 .

Conformational analysis of the dibenzo [a,g]‐quinolizidines by spectroscopic means. II—The use of high resolution 270 MHz proton magnetic resonance

D. Tourwé, T. Kametani, G. V. Binst, 1977 .

A Click Approach to Structurally Diverse Conjugates Containing a Central Di‐1,2,3‐triazole Metal Chelate

R. Schibli, D. Tourwé, L. Brans, 2009, ChemMedChem.

Monitoring the allyl ester deprotection by HR MAS NMR in BAL‐solid phase peptide synthesis

D. Tourwé, R. Willem,, T. Duchène, 2010, Journal of peptide science : an official publication of the European Peptide Society.

Radiolabeled neurotensin analog, 99mTc-NT-XI, evaluated in ductal pancreatic adenocarcinoma patients.

Franz Buchegger, J. Reubi, F. Buchegger, 2003, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.

Maillard Glycation of Peptides Containing the (NαHis)Ac Chelator for 99mTc(CO)3 Labeling

D. Tourwé, V. Maes, 2006, International Journal of Peptide Research and Therapeutics.

Carbohydrated [99mTc(CO)3](NαHis)Ac-Bombesin(7–14) analogs

D. Tourwé, V. Maes, P. Bläuenstein, 2009 .

Toward stable N4-modified neurotensins for NTS1-receptor-targeted tumor imaging with 99mTc.

J. Reubi, D. Tourwé, B. Nock, 2006, Journal of Medicinal Chemistry.

Synthesis and binding properties of endomorphin-2 analogs containing α-hydroxymethyl amino acids

D. Tourwé, A. Olma, 2000, Letters in Peptide Science.

Synthesis and biological activities of linear and cyclic enkephalin analogs containing a Gly3 Ψ(E,CH = CH)Phe4 replacement

T. Burks, H. Yamamura, D. Tourwé, 1990 .

Assignment of the 1H‐nmr resonances of the four rotamers of β‐casomorphin‐5 in DMSO

D. Tourwé, N. Delaet, P. Verheyden, 1991, Biopolymers.

Rat Hepatocyte Suspensions as a Suitable In Vitro Model for Studying the Biotransformation of Histone Deacetylase Inhibitors

T. Vanhaecke, V. Rogiers, D. Tourwé, 2004, Alternatives to laboratory animals : ATLA.

Direct high-performance liquid chromatographic enantioseparation of α-substituted proline analogues on a quinine-derived chiral anion-exchanger stationary phase

W. Lindner, D. Tourwé, A. Péter, 2003 .

HPLC Separation of Enantiomers of α‐Substituted Proline Analogues by the Application of (S)‐N‐(4‐Nitrophenoxy‐carbonyl)phenylalanine Methoxyethyl Ester as Chiral Derivatizing Agent

D. Tourwé, A. Péter, G. Török, 2004 .

Neuropeptide FF receptors as novel targets for limbic seizure attenuation

T. Vanhaecke, P. Boon, F. Bihel, 2015, Neuropharmacology.

Highly potent 4-amino-indolo[2,3-c]azepin-3-one-containing somatostatin mimetics with a range of sst receptor selectivities.

J. Reubi, D. Tourwé, R. Cescato, 2009, Journal of medicinal chemistry.

New tetracyclic tetrahydro-β-carbolines as tryptophan-derived peptidomimetics

A. Misicka, D. Tourwé, Karolina Pulka, 2010, Molecular Diversity.

Application of the organometallic technetium and rhenium tricarbonyl complex on neuropeptide labelling

P. Schubiger, D. Tourwé, A. Blanc, 2001 .

Structural investigations of re‐tricarbonyl labeled neurotensin analogues using 1D and 2D “magic angle spinning” NMR techniques

R. Schibli, P. Schubiger, D. Tourwé, 2001 .

The replacement of His(4) in angiotensin IV by conformationally constrained residues provides highly potent and selective analogues.

G. Vauquelin, D. Tourwé, P. Vanderheyden, 2009, Journal of medicinal chemistry.

Major phase I biotransformation pathways of Trichostatin a in rat hepatocytes and in rat and human liver microsomes.

V. Rogiers, M. Vinken, D. Tourwé, 2002, Drug metabolism and disposition: the biological fate of chemicals.

Conformationally restricted new somatostatin analogs

G. Kéri, O. Csuka, V. Csernus, 1995 .

Radiotracers, tritium labelling of neuropeptides

A. Lipkowski, D. Tourwé, J. Mallareddy, 2012 .

Catabolism of neurotensins. Implications for the design of radiolabeling strategies of peptides.

R. Schibli, P. Schubiger, R. Alberto, 1999, The quarterly journal of nuclear medicine : official publication of the Italian Association of Nuclear Medicine (AIMN) [and] the International Association of Radiopharmacology.

Structure-activity study of the ORL1 antagonist Ac-Arg-D-Cha-Qaa-D-Arg-D-p-ClPhe-NH2.

F. Simonin, D. Tourwé, W. Lubell, 2004, Journal of medicinal chemistry.

Probing opioid receptor interactions with azacycloalkane amino acids. Synthesis of a potent and selective ORL1 antagonist.

F. Simonin, B. Kieffer, Z. Darula, 2002, Journal of medicinal chemistry.

Differential effects of hydroxamate histone deacetylase inhibitors on cellular functionality and gap junctions in primary cultures of mitogen-stimulated hepatocytes.

T. Vanhaecke, V. Rogiers, M. Vinken, 2008, Toxicology letters.

Inhibition of NF‐κB activation by the histone deacetylase inhibitor 4‐Me2N‐BAVAH induces an early G1 cell cycle arrest in primary hepatocytes

T. Vanhaecke, V. Rogiers, M. Vinken, 2007 .

Peptides 1998, Proceedings of the 25th European Peptide Symposium

C. Rabourdin-Combe, D. Gerlier, D. Tourwé, 1999 .

Presence and regulation of insulin-regulated aminopeptidase in mouse macrophages

J. V. Van Ginderachter, D. Tourwé, B. Stijlemans, 2014, Journal of the renin-angiotensin-aldosterone system : JRAAS.