Liyan Yue

发表

Identification of novel small-molecule inhibitors targeting menin-MLL interaction, repurposing the antidiarrheal loperamide.

Z. Chen, Kaixian Chen, Hualiang Jiang, 2016, Organic & biomolecular chemistry.

Small Molecule Inhibitors Targeting New Targets of Protein-Protein Interactions

C. Luo, Linjuan Li, Chen Wang, 2018 .

Identification of novel inhibitors of histone acetyltransferase hMOF through high throughput screening.

Hong Liu, Shien Liu, C. Luo, 2018, European journal of medicinal chemistry.

Functional interplay between the RK motif and linker segment dictates Oct4–DNA recognition

Hualiang Jiang, X. Kong, C. Luo, 2015, Nucleic acids research.

Inhibition of autophagy by a small molecule through covalent modification of LC3.

Kaixian Chen, Hualiang Jiang, Junyan Lu, 2021, Angewandte Chemie.

Discovery of two aminoglycoside antibiotics as inhibitors targeting the menin-mixed lineage leukaemia interface.

Cheng Luo, Fei Ye, Liyan Yue, 2014, Bioorganic & medicinal chemistry letters.

Discovery and biological evaluation of vinylsulfonamide derivatives as highly potent, covalent TEAD autopalmitoylation inhibitors.

Kaixian Chen, Hualiang Jiang, C. Luo, 2019, European journal of medicinal chemistry.

Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues.

Hao Jiang, Cheng Luo, Zhifeng Chen, 2017, Organic & biomolecular chemistry.

Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening

C. Luo, Chuan-peng Liu, Dan Zhang, 2019, Acta Pharmacologica Sinica.

Identification of small molecule inhibitors targeting the SMARCA2 bromodomain from a high-throughput screening assay

Hao Jiang, C. Luo, H. Ding, 2018, Acta Pharmacologica Sinica.

Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening

Kaixian Chen, Hualiang Jiang, C. Luo, 2019, RSC advances.

Covalent Inhibitors Allosterically Block the Activation of Rho Family Proteins and Suppress Cancer Cell Invasion

Kaixian Chen, Hualiang Jiang, C. Luo, 2020, Advanced science.

Discovery of Novel Inhibitors Targeting the Menin-Mixed Lineage Leukemia Interface Using Pharmacophore- and Docking-Based Virtual Screening

Xiaomin Luo, Yuan Xu, Zhifeng Chen, 2016, J. Chem. Inf. Model..

Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors.

Z. Chen, Kaixian Chen, Hualiang Jiang, 2018, Bioorganic & medicinal chemistry.

Identification of small molecule inhibitors targeting the SMARCA2 bromodomain from a high-throughput screening assay

Hao Jiang, C. Luo, H. Ding, 2018, Acta Pharmacologica Sinica.

Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay.

Z. Chen, Kunqian Yu, Kaixian Chen, 2017, MedChemComm.

Identification of novel small-molecule inhibitors targeting menin-MLL interaction, repurposing the antidiarrheal loperamide.

Z. Chen, Kaixian Chen, Hualiang Jiang, 2016, Organic & biomolecular chemistry.